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ZA200301039B - Inhibitors of alpha4 mediated cell adhesion. - Google Patents

Inhibitors of alpha4 mediated cell adhesion.

Info

Publication number
ZA200301039B
ZA200301039B ZA200301039A ZA200301039A ZA200301039B ZA 200301039 B ZA200301039 B ZA 200301039B ZA 200301039 A ZA200301039 A ZA 200301039A ZA 200301039 A ZA200301039 A ZA 200301039A ZA 200301039 B ZA200301039 B ZA 200301039B
Authority
ZA
South Africa
Prior art keywords
inhibitors
cell adhesion
mediated cell
alpha4
alpha4 mediated
Prior art date
Application number
ZA200301039A
Other languages
English (en)
Inventor
Takayuki Kawaguchi
Sumihiro Nomura
Mikiko Tsukimoto
Toshiyuki Kume
Ila Sircar
Original Assignee
Tanabe Seiyaku Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Tanabe Seiyaku Co filed Critical Tanabe Seiyaku Co
Publication of ZA200301039B publication Critical patent/ZA200301039B/xx

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    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C233/00—Carboxylic acid amides
    • C07C233/64—Carboxylic acid amides having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings
    • C07C233/81—Carboxylic acid amides having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by carboxyl groups
    • C07C233/82—Carboxylic acid amides having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by carboxyl groups with the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by an acyclic carbon atom
    • C07C233/87—Carboxylic acid amides having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by carboxyl groups with the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by an acyclic carbon atom of a carbon skeleton containing six-membered aromatic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19—Carboxylic acids, e.g. valproic acid
    • A61K31/195—Carboxylic acids, e.g. valproic acid having an amino group
    • A61K31/197—Carboxylic acids, e.g. valproic acid having an amino group the amino and the carboxyl groups being attached to the same acyclic carbon chain, e.g. gamma-aminobutyric acid [GABA], beta-alanine, epsilon-aminocaproic acid or pantothenic acid
    • A61K31/198—Alpha-amino acids, e.g. alanine or edetic acid [EDTA]
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  • Chemical Kinetics & Catalysis (AREA)
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  • Biomedical Technology (AREA)
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  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Rheumatology (AREA)
  • Pulmonology (AREA)
  • Urology & Nephrology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Psychiatry (AREA)
  • Epidemiology (AREA)
  • Vascular Medicine (AREA)
  • Dermatology (AREA)
  • Obesity (AREA)
  • Virology (AREA)
  • Endocrinology (AREA)
  • Emergency Medicine (AREA)
  • Pain & Pain Management (AREA)
  • AIDS & HIV (AREA)
  • Psychology (AREA)
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ZA200301039A 2000-08-31 2001-08-27 Inhibitors of alpha4 mediated cell adhesion. ZA200301039B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US22912800P 2000-08-31 2000-08-31

Publications (1)

Publication Number Publication Date
ZA200301039B true ZA200301039B (en) 2004-02-09

Family

ID=22859926

Family Applications (1)

Application Number Title Priority Date Filing Date
ZA200301039A ZA200301039B (en) 2000-08-31 2001-08-27 Inhibitors of alpha4 mediated cell adhesion.

Country Status (28)

Country Link
US (6) US7026501B2 (xx)
EP (1) EP1315694B1 (xx)
JP (1) JP3899022B2 (xx)
KR (1) KR100528049B1 (xx)
CN (1) CN1229334C (xx)
AR (1) AR034556A1 (xx)
AT (1) ATE292615T1 (xx)
AU (2) AU2001286778B2 (xx)
BR (1) BR0113629A (xx)
CA (1) CA2418054C (xx)
CZ (1) CZ303460B6 (xx)
DE (1) DE60109943T2 (xx)
DK (1) DK1315694T3 (xx)
ES (1) ES2240509T3 (xx)
HK (1) HK1052684B (xx)
HU (1) HUP0302693A3 (xx)
IL (2) IL154305A0 (xx)
MX (1) MXPA03001837A (xx)
MY (1) MY129000A (xx)
NO (1) NO327861B1 (xx)
NZ (1) NZ524043A (xx)
PL (1) PL206656B1 (xx)
PT (1) PT1315694E (xx)
RU (1) RU2250895C2 (xx)
SI (1) SI1315694T1 (xx)
TW (1) TWI224587B (xx)
WO (1) WO2002018320A2 (xx)
ZA (1) ZA200301039B (xx)

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US20050282900A1 (en) 2005-12-22
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CA2418054C (en) 2008-08-05
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US7456217B2 (en) 2008-11-25
US8501809B2 (en) 2013-08-06
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