ZA200300819B - Imidazole derivatives. - Google Patents
Imidazole derivatives. Download PDFInfo
- Publication number
- ZA200300819B ZA200300819B ZA200300819A ZA200300819A ZA200300819B ZA 200300819 B ZA200300819 B ZA 200300819B ZA 200300819 A ZA200300819 A ZA 200300819A ZA 200300819 A ZA200300819 A ZA 200300819A ZA 200300819 B ZA200300819 B ZA 200300819B
- Authority
- ZA
- South Africa
- Prior art keywords
- imidazol
- cyclobutyl
- cis
- acetylamino
- branched
- Prior art date
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| RU2319693C9 (ru) | 1999-01-13 | 2008-08-20 | Байер Копэрейшн | Производные мочевины (варианты), фармацевтическая композиция (варианты) и способ лечения заболевания, связанного с ростом раковых клеток (варианты) |
| US8124630B2 (en) | 1999-01-13 | 2012-02-28 | Bayer Healthcare Llc | ω-carboxyaryl substituted diphenyl ureas as raf kinase inhibitors |
| ES2377847T3 (es) | 1999-01-13 | 2012-04-02 | Bayer Healthcare Llc | Difenil ureas sustituidas con omega-carboxi arilo como agentes inhibidores de la cinasa p38 |
| EP1478358B1 (fr) | 2002-02-11 | 2013-07-03 | Bayer HealthCare LLC | Tosylate de sorafenib pour le traitement des maladies caractérisées par une angiogénèse anormale |
| US20030216396A1 (en) | 2002-02-11 | 2003-11-20 | Bayer Corporation | Pyridine, quinoline, and isoquinoline N-oxides as kinase inhibitors |
| WO2003106455A1 (fr) | 2002-06-14 | 2003-12-24 | Applied Research Systems Ars Holding N.V. | Derives de cyanure d'azole methylidene et leur utilisation comme modulateurs de proteine kinase |
| US7141561B2 (en) | 2002-07-25 | 2006-11-28 | Sanofi-Aventis Deutschland Gmbh | Substituted diaryl heterocycles, process for their preparation and their use as medicaments |
| DE10233817A1 (de) * | 2002-07-25 | 2004-02-12 | Aventis Pharma Deutschland Gmbh | Substituierte Diarylheterocyclen, Verfahren zu ihrer Herstellung und ihre Verwendung als Arzneimittel |
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| KR101139557B1 (ko) | 2003-07-23 | 2012-04-30 | 바이엘 파마슈티칼스 코포레이션 | 질환 및 상태의 치료 및 예방을 위한 플루오로 치환오메가-카르복시아릴 디페닐 우레아 |
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| EP1885454A2 (fr) | 2005-05-04 | 2008-02-13 | DeveloGen Aktiengesellschaft | Utilisation des inhibiteurs gsk-3 dans la prevention et le traitement des maladies auto-immunes pancreatiques |
| EP2258359A3 (fr) | 2005-08-26 | 2011-04-06 | Braincells, Inc. | Neurogenèse par modulation des récepteurs muscariniques avec sabcomeline |
| CA2620333A1 (fr) | 2005-08-26 | 2007-03-01 | Braincells, Inc. | Neurogenese par modulation du recepteur muscarinique |
| CN101282941A (zh) | 2005-09-22 | 2008-10-08 | 辉瑞产品公司 | 用于治疗神经障碍的咪唑类化合物 |
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| EP2314289A1 (fr) | 2005-10-31 | 2011-04-27 | Braincells, Inc. | Modulation de la neurogenese dont la médiation est assurée par récepteur gaba |
| EA200801716A1 (ru) | 2006-01-18 | 2009-04-28 | Амген Инк. | Тиазольные соединения и их применение |
| US20100216734A1 (en) | 2006-03-08 | 2010-08-26 | Braincells, Inc. | Modulation of neurogenesis by nootropic agents |
| EP2021000A2 (fr) | 2006-05-09 | 2009-02-11 | Braincells, Inc. | Neurogenèse par modulation de l'angiotensine |
| CA2666590C (fr) | 2006-10-21 | 2015-10-06 | Abbott Gmbh & Co. Kg | Composes heterocycliques et leur utilisation comme inhibiteurs de la glycogene synthase kinase 3 |
| WO2009017453A1 (fr) * | 2007-07-30 | 2009-02-05 | Astrazeneca Ab | Nouvelle combinaison thérapeutique d'antipsychotique et d'inhibiteur de gsk3 958 |
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| US5401851A (en) * | 1992-06-03 | 1995-03-28 | Eli Lilly And Company | Angiotensin II antagonists |
| US5760246A (en) * | 1996-12-17 | 1998-06-02 | Biller; Scott A. | Conformationally restricted aromatic inhibitors of microsomal triglyceride transfer protein and method |
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| ZA987385B (en) * | 1997-08-19 | 2000-04-18 | Lilly Co Eli | Growth hormone secretagogues. |
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| WO2000021550A2 (fr) * | 1998-10-13 | 2000-04-20 | President And Fellows Of Harvard College | Methodes et compositions de traitement des maladies neurodegeneratives |
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| EP1106180B1 (fr) * | 1999-12-08 | 2003-11-12 | Centre National de la Recherche Scientifique (CNRS) | Utilisation de l'hymenialdisine et de ses dérivés pour la fabrication de médicaments |
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- 2001-07-25 HR HR20030048A patent/HRP20030048A2/hr not_active Application Discontinuation
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- 2001-07-25 OA OA1200300017A patent/OA12345A/en unknown
- 2001-07-25 EP EP01949833A patent/EP1305295A1/fr not_active Withdrawn
- 2001-07-25 CA CA002418115A patent/CA2418115A1/fr not_active Abandoned
- 2001-07-25 PE PE2001000752A patent/PE20020337A1/es not_active Application Discontinuation
- 2001-07-25 WO PCT/IB2001/001335 patent/WO2002010141A1/fr not_active Ceased
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