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UY29285A1 - Macrolidos - Google Patents

Macrolidos

Info

Publication number
UY29285A1
UY29285A1 UY29285A UY29285A UY29285A1 UY 29285 A1 UY29285 A1 UY 29285A1 UY 29285 A UY29285 A UY 29285A UY 29285 A UY29285 A UY 29285A UY 29285 A1 UY29285 A1 UY 29285A1
Authority
UY
Uruguay
Prior art keywords
compounds
methods
macrolidos
famraceutical
intermediates
Prior art date
Application number
UY29285A
Other languages
English (en)
Spanish (es)
Inventor
Takushi Kaneko
Mark Edward Flanagan
Louis Stanley Chupak
Thomas Victor Magee
Mark Carl Noe
Usa Reilly
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=35809765&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=UY29285(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Publication of UY29285A1 publication Critical patent/UY29285A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/70Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7042Compounds having saccharide radicals and heterocyclic rings
    • A61K31/7048Compounds having saccharide radicals and heterocyclic rings having oxygen as a ring hetero atom, e.g. leucoglucosan, hesperidin, erythromycin, nystatin, digitoxin or digoxin
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08Hetero rings containing eight or more ring members, e.g. erythromycins
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/02Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Molecular Biology (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Biotechnology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Polysaccharides And Polysaccharide Derivatives (AREA)
  • Tires In General (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Cephalosporin Compounds (AREA)
UY29285A 2004-12-21 2005-12-21 Macrolidos UY29285A1 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US63809704P 2004-12-21 2004-12-21
US71753005P 2005-09-14 2005-09-14

Publications (1)

Publication Number Publication Date
UY29285A1 true UY29285A1 (es) 2006-07-31

Family

ID=35809765

Family Applications (1)

Application Number Title Priority Date Filing Date
UY29285A UY29285A1 (es) 2004-12-21 2005-12-21 Macrolidos

Country Status (35)

Country Link
US (1) US7462600B2 (ru)
EP (2) EP2233493A1 (ru)
JP (1) JP4111994B1 (ru)
KR (1) KR100897678B1 (ru)
CN (1) CN101120011A (ru)
AP (1) AP2007004026A0 (ru)
AR (1) AR052824A1 (ru)
AT (1) ATE459633T1 (ru)
AU (1) AU2005317735B2 (ru)
BR (1) BRPI0519135A2 (ru)
CA (1) CA2591746A1 (ru)
CR (1) CR9202A (ru)
DE (1) DE602005019786D1 (ru)
DK (1) DK1836211T3 (ru)
EA (1) EA011281B1 (ru)
ES (1) ES2339871T3 (ru)
GE (1) GEP20094834B (ru)
GT (1) GT200500378A (ru)
HN (1) HN2005036113A (ru)
HR (1) HRP20100253T1 (ru)
IL (1) IL183661A0 (ru)
MA (1) MA29108B1 (ru)
MX (1) MX2007007598A (ru)
NL (1) NL1030713C2 (ru)
NO (1) NO20073367L (ru)
PE (1) PE20060948A1 (ru)
PL (1) PL1836211T3 (ru)
PT (1) PT1836211E (ru)
SI (1) SI1836211T1 (ru)
TN (1) TNSN07233A1 (ru)
TW (1) TW200626608A (ru)
UA (1) UA85937C2 (ru)
UY (1) UY29285A1 (ru)
WO (1) WO2006067589A1 (ru)
ZA (1) ZA200705108B (ru)

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US8367669B2 (en) * 2005-06-15 2013-02-05 Vanderbilt University Inhibitors of hemeprotein-catalyzed lipid peroxidation
US9133212B1 (en) 2005-06-15 2015-09-15 Vanderbilt University Inhibitors of hemeprotein-catalyzed lipid peroxidation
EP3290427A1 (en) 2005-08-24 2018-03-07 Melinta Therapeutics, Inc. Triazole compounds and methods of making and using the same
ATE471943T1 (de) * 2007-03-13 2010-07-15 Pfizer Prod Inc Makrolide auf erythromycinbasis
US20100099674A1 (en) * 2007-03-21 2010-04-22 Innate Pharmaceuticals Ab Method and means for preventing and inhibiting type iii secretion in infections caused by gram-negative bacteria
WO2009055557A1 (en) 2007-10-25 2009-04-30 Cempra Pharmaceuticals, Inc. Process for the preparation of macrolide antibacterial agents
WO2009053259A1 (en) * 2007-10-25 2009-04-30 Sandoz Ag Process for the production of telithromycin
WO2009080534A1 (en) 2007-12-21 2009-07-02 F. Hoffmann-La Roche Ag Heterocyclic antiviral compounds
ES2582794T3 (es) 2009-08-13 2016-09-15 Basilea Pharmaceutica Ag Nuevos macrólidos y su uso
JP5711352B2 (ja) * 2010-03-22 2015-04-30 センプラ ファーマシューティカルズ,インコーポレイテッド マクロライドの結晶形、およびその使用
AU2012242926B2 (en) * 2011-04-12 2016-07-14 The United States Of America, As Represented By The Secretary, Department Of Health And Human Services Plasmodial surface anion channel inhibitors for the treatment or prevention of malaria
CN102558047B (zh) * 2011-12-14 2013-10-30 天津药物研究院药业有限责任公司 3-甲基喹啉的制备方法
US10188674B2 (en) 2012-03-27 2019-01-29 Cempra Pharmaceuticals, Inc. Parenteral formulations for administering macrolide antibiotics
JP6141428B2 (ja) 2012-07-13 2017-06-07 エフ・ホフマン−ラ・ロシュ・アクチェンゲゼルシャフト 抗増殖性ベンゾ[b]アゼピン−2−オン
KR101612179B1 (ko) * 2013-04-19 2016-04-12 영남대학교 산학협력단 아미도피리딘올 유도체 또는 이의 약제학적 허용가능한 염을 유효성분으로 함유하는 암질환 예방 또는 치료용 약학조성물
TW201534586A (zh) 2013-06-11 2015-09-16 Orion Corp 新穎cyp17抑制劑/抗雄激素劑
CN103739643A (zh) * 2013-12-30 2014-04-23 华东理工大学 利用分子印迹技术对红霉素进行回收分离纯化的方法
CN104230891B (zh) * 2014-08-27 2016-03-30 于宗光 一种托匹司他的制备方法
JP2019533669A (ja) * 2016-10-04 2019-11-21 バイオファーマティ ソシエテ アノニム 抗菌活性を有するケトライド
CA3140173A1 (en) * 2019-06-04 2020-12-10 Belew Mekonnen Pyrazole and imidazole derivatives, compositions and methods as orexin antagonists
JP2022534704A (ja) 2019-06-04 2022-08-03 ヘイガー バイオサイエンシズ,エルエルシー オレキシンアンタゴニストとしてのイミダゾロ誘導体、組成物、及び方法
CN111793022A (zh) * 2020-04-27 2020-10-20 滁州拜奥生物科技有限公司 一种3-甲基喹啉的制备方法
AU2023333164A1 (en) * 2022-09-01 2025-04-03 Hager Biosciences, Llc Pyrazole and imidazole derivatives as dual orexin and kappa-opioid receptors modulators, composition, methods for treating neurological and psychiatric disorders

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Also Published As

Publication number Publication date
CA2591746A1 (en) 2006-06-29
KR100897678B1 (ko) 2009-05-14
TNSN07233A1 (fr) 2008-11-21
WO2006067589A1 (en) 2006-06-29
ATE459633T1 (de) 2010-03-15
BRPI0519135A2 (pt) 2008-12-23
ES2339871T3 (es) 2010-05-26
HRP20100253T1 (hr) 2010-06-30
PE20060948A1 (es) 2006-10-11
GEP20094834B (en) 2009-11-25
CN101120011A (zh) 2008-02-06
AP2007004026A0 (en) 2007-06-30
UA85937C2 (ru) 2009-03-10
EA200701113A1 (ru) 2007-12-28
EP1836211A1 (en) 2007-09-26
EP2233493A1 (en) 2010-09-29
ZA200705108B (en) 2009-01-28
AR052824A1 (es) 2007-04-04
JP4111994B1 (ja) 2008-07-02
KR20070089191A (ko) 2007-08-30
CR9202A (es) 2007-07-16
IL183661A0 (en) 2007-09-20
JP2008524319A (ja) 2008-07-10
AU2005317735A1 (en) 2006-06-29
DE602005019786D1 (de) 2010-04-15
NL1030713A1 (nl) 2006-06-22
MX2007007598A (es) 2007-07-25
EA011281B1 (ru) 2009-02-27
PL1836211T3 (pl) 2010-07-30
TW200626608A (en) 2006-08-01
AU2005317735B2 (en) 2009-06-04
EP1836211B1 (en) 2010-03-03
NL1030713C2 (nl) 2006-12-12
GT200500378A (es) 2006-11-28
PT1836211E (pt) 2010-04-08
DK1836211T3 (da) 2010-05-17
HN2005036113A (es) 2010-12-06
NO20073367L (no) 2007-09-05
US7462600B2 (en) 2008-12-09
US20060135447A1 (en) 2006-06-22
SI1836211T1 (sl) 2010-04-30
MA29108B1 (fr) 2007-12-03

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Effective date: 20160606