PL1836211T3 - Makrolidy - Google Patents
MakrolidyInfo
- Publication number
- PL1836211T3 PL1836211T3 PL05813939T PL05813939T PL1836211T3 PL 1836211 T3 PL1836211 T3 PL 1836211T3 PL 05813939 T PL05813939 T PL 05813939T PL 05813939 T PL05813939 T PL 05813939T PL 1836211 T3 PL1836211 T3 PL 1836211T3
- Authority
- PL
- Poland
- Prior art keywords
- macrolides
- Prior art date
Links
- 239000003120 macrolide antibiotic agent Substances 0.000 title 1
- 229940041033 macrolides Drugs 0.000 title 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/70—Carbohydrates; Sugars; Derivatives thereof
- A61K31/7042—Compounds having saccharide radicals and heterocyclic rings
- A61K31/7048—Compounds having saccharide radicals and heterocyclic rings having oxygen as a ring hetero atom, e.g. leucoglucosan, hesperidin, erythromycin, nystatin, digitoxin or digoxin
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
- C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
- C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Animal Behavior & Ethology (AREA)
- Molecular Biology (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Biotechnology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Genetics & Genomics (AREA)
- Engineering & Computer Science (AREA)
- Biochemistry (AREA)
- Communicable Diseases (AREA)
- Oncology (AREA)
- Tropical Medicine & Parasitology (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Saccharide Compounds (AREA)
- Cephalosporin Compounds (AREA)
- Polysaccharides And Polysaccharide Derivatives (AREA)
- Tires In General (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (4)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US63809704P | 2004-12-21 | 2004-12-21 | |
| US71753005P | 2005-09-14 | 2005-09-14 | |
| EP05813939A EP1836211B1 (en) | 2004-12-21 | 2005-12-12 | Macrolides |
| PCT/IB2005/003829 WO2006067589A1 (en) | 2004-12-21 | 2005-12-12 | Macrolides |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| PL1836211T3 true PL1836211T3 (pl) | 2010-07-30 |
Family
ID=35809765
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| PL05813939T PL1836211T3 (pl) | 2004-12-21 | 2005-12-12 | Makrolidy |
Country Status (35)
| Country | Link |
|---|---|
| US (1) | US7462600B2 (pl) |
| EP (2) | EP1836211B1 (pl) |
| JP (1) | JP4111994B1 (pl) |
| KR (1) | KR100897678B1 (pl) |
| CN (1) | CN101120011A (pl) |
| AP (1) | AP2007004026A0 (pl) |
| AR (1) | AR052824A1 (pl) |
| AT (1) | ATE459633T1 (pl) |
| AU (1) | AU2005317735B2 (pl) |
| BR (1) | BRPI0519135A2 (pl) |
| CA (1) | CA2591746A1 (pl) |
| CR (1) | CR9202A (pl) |
| DE (1) | DE602005019786D1 (pl) |
| DK (1) | DK1836211T3 (pl) |
| EA (1) | EA011281B1 (pl) |
| ES (1) | ES2339871T3 (pl) |
| GE (1) | GEP20094834B (pl) |
| GT (1) | GT200500378A (pl) |
| HN (1) | HN2005036113A (pl) |
| HR (1) | HRP20100253T1 (pl) |
| IL (1) | IL183661A0 (pl) |
| MA (1) | MA29108B1 (pl) |
| MX (1) | MX2007007598A (pl) |
| NL (1) | NL1030713C2 (pl) |
| NO (1) | NO20073367L (pl) |
| PE (1) | PE20060948A1 (pl) |
| PL (1) | PL1836211T3 (pl) |
| PT (1) | PT1836211E (pl) |
| SI (1) | SI1836211T1 (pl) |
| TN (1) | TNSN07233A1 (pl) |
| TW (1) | TW200626608A (pl) |
| UA (1) | UA85937C2 (pl) |
| UY (1) | UY29285A1 (pl) |
| WO (1) | WO2006067589A1 (pl) |
| ZA (1) | ZA200705108B (pl) |
Families Citing this family (23)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US8367669B2 (en) * | 2005-06-15 | 2013-02-05 | Vanderbilt University | Inhibitors of hemeprotein-catalyzed lipid peroxidation |
| US9133212B1 (en) | 2005-06-15 | 2015-09-15 | Vanderbilt University | Inhibitors of hemeprotein-catalyzed lipid peroxidation |
| WO2007025098A2 (en) | 2005-08-24 | 2007-03-01 | Rib-X Pharmaceuticals, Inc. | Triazole compounds and methods of making and using the same |
| DE602008001611D1 (en) * | 2007-03-13 | 2010-08-05 | Pfizer Prod Inc | Makrolide auf erythromycinbasis |
| AU2008227216A1 (en) * | 2007-03-21 | 2008-09-25 | Creative Antibiotics Sweden Ab | Method and means for preventing and inhibiting type III secretion in infections caused by gram-negative bacteria |
| US20110040078A1 (en) * | 2007-10-25 | 2011-02-17 | Siegfried Wolf | Process for the production of telithromycin |
| CN101917850B (zh) | 2007-10-25 | 2016-01-13 | 森普拉制药公司 | 大环内酯类抗菌剂的制备方法 |
| JP5411160B2 (ja) | 2007-12-21 | 2014-02-12 | エフ.ホフマン−ラ ロシュ アーゲー | 複素環式抗ウイルス性化合物 |
| ES2582794T3 (es) | 2009-08-13 | 2016-09-15 | Basilea Pharmaceutica Ag | Nuevos macrólidos y su uso |
| PL2550286T3 (pl) * | 2010-03-22 | 2016-07-29 | Cempra Pharmaceuticals Inc | Krystaliczne postaci makrolidu i ich zastosowanie |
| CN106974913A (zh) | 2011-04-12 | 2017-07-25 | 美国卫生和人力服务部 | 用于治疗或预防疟疾的疟原虫表面阴离子通道抑制剂 |
| CN102558047B (zh) * | 2011-12-14 | 2013-10-30 | 天津药物研究院药业有限责任公司 | 3-甲基喹啉的制备方法 |
| AU2013239696C1 (en) | 2012-03-27 | 2018-11-29 | Cempra Pharmaceuticals, Inc. | Parenteral formulations for administering macrolide antibiotics |
| RU2015103119A (ru) | 2012-07-13 | 2016-08-27 | Ф. Хоффманн-Ля Рош Аг | Антипролиферативные бензо[в]азепин-2-оны |
| KR101663864B1 (ko) * | 2013-04-19 | 2016-10-07 | 영남대학교 산학협력단 | 아미도피리딘올 유도체 또는 이의 약제학적 허용가능한 염을 유효성분으로 함유하는 염증성 장질환의 예방 또는 치료용 약학조성물 |
| TW201534586A (zh) | 2013-06-11 | 2015-09-16 | Orion Corp | 新穎cyp17抑制劑/抗雄激素劑 |
| CN103739643A (zh) * | 2013-12-30 | 2014-04-23 | 华东理工大学 | 利用分子印迹技术对红霉素进行回收分离纯化的方法 |
| CN104230891B (zh) * | 2014-08-27 | 2016-03-30 | 于宗光 | 一种托匹司他的制备方法 |
| JP2019533669A (ja) | 2016-10-04 | 2019-11-21 | バイオファーマティ ソシエテ アノニム | 抗菌活性を有するケトライド |
| KR20220016918A (ko) | 2019-06-04 | 2022-02-10 | 하거 바이오사이언시즈, 엘엘씨 | 오렉신 길항제로서의 이미다졸로 유도체, 조성물 및 방법 |
| EP3972587A4 (en) * | 2019-06-04 | 2023-01-18 | Hager Biosciences, LLC | PYRAZOLE AND IMIDAZOLE DERIVATIVES, COMPOSITIONS AND METHODS AS OREXIN ANTAGONISTS |
| CN111793022A (zh) * | 2020-04-27 | 2020-10-20 | 滁州拜奥生物科技有限公司 | 一种3-甲基喹啉的制备方法 |
| JP2025530768A (ja) * | 2022-09-01 | 2025-09-17 | ヘイガー バイオサイエンシズ,エルエルシー | 神経疾患および精神疾患の治療のための、オレキシン受容体およびカッパオピオイド受容体に対する二重調節剤としてのピラゾール誘導体およびイミダゾール誘導体、組成物、ならびに治療法 |
Family Cites Families (74)
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|---|---|---|---|---|
| US2653899A (en) | 1952-04-14 | 1953-09-29 | Lilly Co Eli | Erythromycin, its salts, and method of preparation |
| US2823203A (en) | 1954-06-24 | 1958-02-11 | Abbott Lab | Method of producing substantially pure erythromycin a |
| US4331803A (en) | 1980-06-04 | 1982-05-25 | Taisho Pharmaceutical Co., Ltd. | Novel erythromycin compounds |
| SI8110592A8 (en) | 1981-03-06 | 1996-06-30 | Pliva Pharm & Chem Works | Process for preparing of n-methyl-11-aza-10-deoxo-10-dihydroerythromycine a and derivatives thereof |
| US4474768A (en) | 1982-07-19 | 1984-10-02 | Pfizer Inc. | N-Methyl 11-aza-10-deoxo-10-dihydro-erytromycin A, intermediates therefor |
| US4742049A (en) | 1986-06-04 | 1988-05-03 | Abbott Laboratories | Semisynthetic erythromycin antibiotics |
| US5075289A (en) | 1988-06-07 | 1991-12-24 | Abbott Laboratories | 9-r-azacyclic erythromycin antibiotics |
| IE70593B1 (en) | 1989-09-29 | 1996-12-11 | Eisai Co Ltd | Biphenylmethane derivative the use of it and pharmacological compositions containing same |
| US5523399A (en) | 1991-12-27 | 1996-06-04 | Taisho Pharmaceutical Co., Ltd. | 5-O-desosaminylerythronolide derivatives |
| US5527780A (en) | 1992-11-05 | 1996-06-18 | Roussel Uclaf | Erythromycin derivatives |
| FR2697524B1 (fr) | 1992-11-05 | 1994-12-23 | Roussel Uclaf | Nouveaux dérivés de l'érythromycine, leur procédé de préparation et leur application comme médicaments. |
| FR2719587B1 (fr) | 1994-05-03 | 1996-07-12 | Roussel Uclaf | Nouveaux dérivés de l'érythromycine, leur procédé de préparation et leur application comme médicaments. |
| US5629322A (en) | 1994-11-15 | 1997-05-13 | Merck & Co., Inc. | Cyclic amidine analogs as inhibitors of nitric oxide synthase |
| FR2727969B1 (fr) | 1994-12-09 | 1997-01-17 | Roussel Uclaf | Nouveaux derives de l'erythromycine, leur procede de preparation et leur application comme medicaments |
| US5747466A (en) | 1995-11-08 | 1998-05-05 | Abbott Laboratories | 3-deoxy-3-descladinose derivatives of erythromycins A and B |
| FR2742757B1 (fr) | 1995-12-22 | 1998-01-30 | Roussel Uclaf | Nouveaux derives de l'erythromycine, leur procede de preparation et leur application comme medicaments |
| WO1997042204A1 (en) | 1996-05-07 | 1997-11-13 | Abbott Laboratories | 6-o-substituted erythromycins and method for making them |
| US5750510A (en) | 1997-04-04 | 1998-05-12 | Abbott Laboratories | 3-descladinose-2,3-anhydroerythromycin derivatives |
| FR2748746B1 (fr) | 1996-05-14 | 1998-08-14 | Hoechst Marion Roussel Inc | Nouveau procede d'isomerisation du radical methyle en 10 de derives de l'erythromycine |
| US6271255B1 (en) | 1996-07-05 | 2001-08-07 | Biotica Technology Limited | Erythromycins and process for their preparation |
| FR2751656B1 (fr) | 1996-07-24 | 1998-10-16 | Hoechst Marion Roussel Inc | Nouveaux derives de l'erythromycine, leur procede de preparation et leur application comme medicaments |
| TR199901127T2 (xx) | 1996-09-04 | 1999-07-21 | Abbott Laboratories | Antibakteriyel etkili 6-O-ikameli ketolitler. |
| US5804565A (en) | 1996-09-24 | 1998-09-08 | Taisho Pharmaceutical Co., Ltd. | Erythromycin A derivatives |
| KR20000069138A (ko) * | 1996-11-27 | 2000-11-25 | 우에하라 아끼라 | 에리트로마이신 a 유도체 |
| AU6421398A (en) | 1997-03-24 | 1998-10-20 | Taisho Pharmaceutical Co., Ltd. | Erythromycin a derivatives |
| US6162794A (en) | 1997-05-09 | 2000-12-19 | Pfizer Inc. | Erythromycin derivatives |
| US20020025937A1 (en) | 2000-03-20 | 2002-02-28 | Yong-Jin Wu | 9-oxime erythromycin derivatives |
| EP0895999A1 (en) | 1997-08-06 | 1999-02-10 | Pfizer Products Inc. | C-4" substituted macrolide antibiotics |
| ZA987689B (en) | 1997-09-02 | 1999-02-24 | Abbott Lab | 3-descladinose 6-O substituted erythromycin derivatives |
| US6034069A (en) | 1997-09-30 | 2000-03-07 | Abbott Laboratories | 3-'N-modified 6-O-substituted erythromycin ketolide derivatives having antibacterial activity |
| PA8461401A1 (es) | 1997-10-29 | 2000-05-24 | Pfizer Prod Inc | Derivados de eritromicina triciclicos |
| WO1999021869A1 (en) | 1997-10-29 | 1999-05-06 | Taisho Pharmaceutical Co., Ltd. | Erythromycin a, 11,12-carbamate derivatives |
| HN1998000159A (es) | 1997-10-29 | 1999-02-09 | Monsanto Co | Derivados de 9- amino - 3 ceto eritromicina |
| AP1060A (en) | 1998-01-02 | 2002-04-23 | Pfizer Prod Inc | Novel erythromycin derivatives. |
| AP9801420A0 (en) | 1998-01-02 | 1998-12-31 | Pfizer Prod Inc | Novel macrolides. |
| ATE275151T1 (de) | 1998-03-03 | 2004-09-15 | Pfizer Prod Inc | 3,6-ketal-makrolidantibiotika |
| US5955440A (en) | 1998-03-27 | 1999-09-21 | Abbott Laboratories | Macrolide LHRH antagonists |
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| JP4573925B2 (ja) | 1998-07-09 | 2010-11-04 | アベンティス・ファーマ・ソシエテ・アノニム | 新規のエリスロマイシン誘導体、その製造方法及びその薬剤としての使用 |
| US6387885B1 (en) | 1998-08-26 | 2002-05-14 | Abbott Laboratories | 3′,3′-N-bis-desmethyl-3′-N-cycloalkyl erythromycin derivatives as LHRH antagonists |
| US6020521A (en) | 1998-08-26 | 2000-02-01 | Abbott Laboratories | Macrolide LHRH antagonists |
| US6262030B1 (en) | 1998-11-03 | 2001-07-17 | Pfizer Inc. | Erythromycin derivatives |
| TR200200436T2 (tr) | 1998-11-03 | 2002-06-21 | Pfizer Inc. | Yeni makrolit antibiyotikler |
| TR200102129T2 (tr) | 1998-12-10 | 2002-01-21 | Pfizer Products Inc. | Karbamat ve karbazat ketolid antibiyotikleri. |
| HK1042707A1 (zh) | 1999-01-27 | 2002-08-23 | 辉瑞产品公司 | 酮内酯类抗生素 |
| US6054435A (en) | 1999-03-19 | 2000-04-25 | Abbott Laboratories | 6-O-substituted macrolides having antibacterial activity |
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| AU4354900A (en) * | 1999-04-16 | 2000-11-02 | Kosan Biosciences, Inc. | Ketolide antibacterials |
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| US20020061857A1 (en) | 1999-04-23 | 2002-05-23 | Yong-Jin Wu | 9-amino-3-oxo erythromycin derivatives |
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| CA2451391A1 (en) | 2001-07-03 | 2003-01-16 | Chiron Corporation | C12 modified erythromycin macrolides and ketolides having antibacterial activity |
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-
2005
- 2005-12-12 KR KR1020077014160A patent/KR100897678B1/ko not_active Expired - Fee Related
- 2005-12-12 MX MX2007007598A patent/MX2007007598A/es active IP Right Grant
- 2005-12-12 CN CNA2005800482465A patent/CN101120011A/zh active Pending
- 2005-12-12 ES ES05813939T patent/ES2339871T3/es active Active
- 2005-12-12 CA CA002591746A patent/CA2591746A1/en not_active Abandoned
- 2005-12-12 EP EP05813939A patent/EP1836211B1/en active Active
- 2005-12-12 JP JP2007547694A patent/JP4111994B1/ja not_active Expired - Fee Related
- 2005-12-12 AU AU2005317735A patent/AU2005317735B2/en not_active Ceased
- 2005-12-12 HR HR20100253T patent/HRP20100253T1/hr unknown
- 2005-12-12 WO PCT/IB2005/003829 patent/WO2006067589A1/en not_active Ceased
- 2005-12-12 BR BRPI0519135-1A patent/BRPI0519135A2/pt not_active IP Right Cessation
- 2005-12-12 AP AP2007004026A patent/AP2007004026A0/xx unknown
- 2005-12-12 PL PL05813939T patent/PL1836211T3/pl unknown
- 2005-12-12 PT PT05813939T patent/PT1836211E/pt unknown
- 2005-12-12 DK DK05813939.5T patent/DK1836211T3/da active
- 2005-12-12 EP EP10154783A patent/EP2233493A1/en not_active Withdrawn
- 2005-12-12 DE DE602005019786T patent/DE602005019786D1/de active Active
- 2005-12-12 SI SI200530941T patent/SI1836211T1/sl unknown
- 2005-12-12 EA EA200701113A patent/EA011281B1/ru not_active IP Right Cessation
- 2005-12-12 UA UAA200706959A patent/UA85937C2/uk unknown
- 2005-12-12 GE GEAP200510142A patent/GEP20094834B/en unknown
- 2005-12-12 AT AT05813939T patent/ATE459633T1/de not_active IP Right Cessation
- 2005-12-14 PE PE2005001462A patent/PE20060948A1/es not_active Application Discontinuation
- 2005-12-19 HN HN2005036113A patent/HN2005036113A/es unknown
- 2005-12-20 AR ARP050105370A patent/AR052824A1/es unknown
- 2005-12-20 TW TW094145385A patent/TW200626608A/zh unknown
- 2005-12-20 GT GT200500378A patent/GT200500378A/es unknown
- 2005-12-20 NL NL1030713A patent/NL1030713C2/nl not_active IP Right Cessation
- 2005-12-21 US US11/313,523 patent/US7462600B2/en not_active Expired - Fee Related
- 2005-12-21 UY UY29285A patent/UY29285A1/es not_active Application Discontinuation
-
2007
- 2007-06-04 IL IL183661A patent/IL183661A0/en unknown
- 2007-06-15 ZA ZA200705108A patent/ZA200705108B/xx unknown
- 2007-06-20 TN TNP2007000233A patent/TNSN07233A1/fr unknown
- 2007-06-21 CR CR9202A patent/CR9202A/es not_active Application Discontinuation
- 2007-06-21 MA MA30024A patent/MA29108B1/fr unknown
- 2007-06-29 NO NO20073367A patent/NO20073367L/no not_active Application Discontinuation
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