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PL1836211T3 - Makrolidy - Google Patents

Makrolidy

Info

Publication number
PL1836211T3
PL1836211T3 PL05813939T PL05813939T PL1836211T3 PL 1836211 T3 PL1836211 T3 PL 1836211T3 PL 05813939 T PL05813939 T PL 05813939T PL 05813939 T PL05813939 T PL 05813939T PL 1836211 T3 PL1836211 T3 PL 1836211T3
Authority
PL
Poland
Prior art keywords
macrolides
Prior art date
Application number
PL05813939T
Other languages
English (en)
Inventor
Louis Stanley Chupak
Mark Edward Flanagan
Takushi Kaneko
Thomas Victor Magee
Mark Carl Noe
Usa Reilly
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=35809765&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=PL1836211(T3) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Publication of PL1836211T3 publication Critical patent/PL1836211T3/pl

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/70Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7042Compounds having saccharide radicals and heterocyclic rings
    • A61K31/7048Compounds having saccharide radicals and heterocyclic rings having oxygen as a ring hetero atom, e.g. leucoglucosan, hesperidin, erythromycin, nystatin, digitoxin or digoxin
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08Hetero rings containing eight or more ring members, e.g. erythromycins
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/02Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Molecular Biology (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Biotechnology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Cephalosporin Compounds (AREA)
  • Polysaccharides And Polysaccharide Derivatives (AREA)
  • Tires In General (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
PL05813939T 2004-12-21 2005-12-12 Makrolidy PL1836211T3 (pl)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US63809704P 2004-12-21 2004-12-21
US71753005P 2005-09-14 2005-09-14
EP05813939A EP1836211B1 (en) 2004-12-21 2005-12-12 Macrolides
PCT/IB2005/003829 WO2006067589A1 (en) 2004-12-21 2005-12-12 Macrolides

Publications (1)

Publication Number Publication Date
PL1836211T3 true PL1836211T3 (pl) 2010-07-30

Family

ID=35809765

Family Applications (1)

Application Number Title Priority Date Filing Date
PL05813939T PL1836211T3 (pl) 2004-12-21 2005-12-12 Makrolidy

Country Status (35)

Country Link
US (1) US7462600B2 (pl)
EP (2) EP1836211B1 (pl)
JP (1) JP4111994B1 (pl)
KR (1) KR100897678B1 (pl)
CN (1) CN101120011A (pl)
AP (1) AP2007004026A0 (pl)
AR (1) AR052824A1 (pl)
AT (1) ATE459633T1 (pl)
AU (1) AU2005317735B2 (pl)
BR (1) BRPI0519135A2 (pl)
CA (1) CA2591746A1 (pl)
CR (1) CR9202A (pl)
DE (1) DE602005019786D1 (pl)
DK (1) DK1836211T3 (pl)
EA (1) EA011281B1 (pl)
ES (1) ES2339871T3 (pl)
GE (1) GEP20094834B (pl)
GT (1) GT200500378A (pl)
HN (1) HN2005036113A (pl)
HR (1) HRP20100253T1 (pl)
IL (1) IL183661A0 (pl)
MA (1) MA29108B1 (pl)
MX (1) MX2007007598A (pl)
NL (1) NL1030713C2 (pl)
NO (1) NO20073367L (pl)
PE (1) PE20060948A1 (pl)
PL (1) PL1836211T3 (pl)
PT (1) PT1836211E (pl)
SI (1) SI1836211T1 (pl)
TN (1) TNSN07233A1 (pl)
TW (1) TW200626608A (pl)
UA (1) UA85937C2 (pl)
UY (1) UY29285A1 (pl)
WO (1) WO2006067589A1 (pl)
ZA (1) ZA200705108B (pl)

Families Citing this family (23)

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US8367669B2 (en) * 2005-06-15 2013-02-05 Vanderbilt University Inhibitors of hemeprotein-catalyzed lipid peroxidation
US9133212B1 (en) 2005-06-15 2015-09-15 Vanderbilt University Inhibitors of hemeprotein-catalyzed lipid peroxidation
WO2007025098A2 (en) 2005-08-24 2007-03-01 Rib-X Pharmaceuticals, Inc. Triazole compounds and methods of making and using the same
DE602008001611D1 (en) * 2007-03-13 2010-08-05 Pfizer Prod Inc Makrolide auf erythromycinbasis
AU2008227216A1 (en) * 2007-03-21 2008-09-25 Creative Antibiotics Sweden Ab Method and means for preventing and inhibiting type III secretion in infections caused by gram-negative bacteria
US20110040078A1 (en) * 2007-10-25 2011-02-17 Siegfried Wolf Process for the production of telithromycin
CN101917850B (zh) 2007-10-25 2016-01-13 森普拉制药公司 大环内酯类抗菌剂的制备方法
JP5411160B2 (ja) 2007-12-21 2014-02-12 エフ.ホフマン−ラ ロシュ アーゲー 複素環式抗ウイルス性化合物
ES2582794T3 (es) 2009-08-13 2016-09-15 Basilea Pharmaceutica Ag Nuevos macrólidos y su uso
PL2550286T3 (pl) * 2010-03-22 2016-07-29 Cempra Pharmaceuticals Inc Krystaliczne postaci makrolidu i ich zastosowanie
CN106974913A (zh) 2011-04-12 2017-07-25 美国卫生和人力服务部 用于治疗或预防疟疾的疟原虫表面阴离子通道抑制剂
CN102558047B (zh) * 2011-12-14 2013-10-30 天津药物研究院药业有限责任公司 3-甲基喹啉的制备方法
AU2013239696C1 (en) 2012-03-27 2018-11-29 Cempra Pharmaceuticals, Inc. Parenteral formulations for administering macrolide antibiotics
RU2015103119A (ru) 2012-07-13 2016-08-27 Ф. Хоффманн-Ля Рош Аг Антипролиферативные бензо[в]азепин-2-оны
KR101663864B1 (ko) * 2013-04-19 2016-10-07 영남대학교 산학협력단 아미도피리딘올 유도체 또는 이의 약제학적 허용가능한 염을 유효성분으로 함유하는 염증성 장질환의 예방 또는 치료용 약학조성물
TW201534586A (zh) 2013-06-11 2015-09-16 Orion Corp 新穎cyp17抑制劑/抗雄激素劑
CN103739643A (zh) * 2013-12-30 2014-04-23 华东理工大学 利用分子印迹技术对红霉素进行回收分离纯化的方法
CN104230891B (zh) * 2014-08-27 2016-03-30 于宗光 一种托匹司他的制备方法
JP2019533669A (ja) 2016-10-04 2019-11-21 バイオファーマティ ソシエテ アノニム 抗菌活性を有するケトライド
KR20220016918A (ko) 2019-06-04 2022-02-10 하거 바이오사이언시즈, 엘엘씨 오렉신 길항제로서의 이미다졸로 유도체, 조성물 및 방법
EP3972587A4 (en) * 2019-06-04 2023-01-18 Hager Biosciences, LLC PYRAZOLE AND IMIDAZOLE DERIVATIVES, COMPOSITIONS AND METHODS AS OREXIN ANTAGONISTS
CN111793022A (zh) * 2020-04-27 2020-10-20 滁州拜奥生物科技有限公司 一种3-甲基喹啉的制备方法
JP2025530768A (ja) * 2022-09-01 2025-09-17 ヘイガー バイオサイエンシズ,エルエルシー 神経疾患および精神疾患の治療のための、オレキシン受容体およびカッパオピオイド受容体に対する二重調節剤としてのピラゾール誘導体およびイミダゾール誘導体、組成物、ならびに治療法

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Also Published As

Publication number Publication date
AR052824A1 (es) 2007-04-04
DK1836211T3 (da) 2010-05-17
ATE459633T1 (de) 2010-03-15
TNSN07233A1 (fr) 2008-11-21
NO20073367L (no) 2007-09-05
GEP20094834B (en) 2009-11-25
EA011281B1 (ru) 2009-02-27
PE20060948A1 (es) 2006-10-11
AU2005317735A1 (en) 2006-06-29
CN101120011A (zh) 2008-02-06
KR20070089191A (ko) 2007-08-30
ES2339871T3 (es) 2010-05-26
BRPI0519135A2 (pt) 2008-12-23
WO2006067589A1 (en) 2006-06-29
DE602005019786D1 (de) 2010-04-15
CR9202A (es) 2007-07-16
UY29285A1 (es) 2006-07-31
JP4111994B1 (ja) 2008-07-02
EA200701113A1 (ru) 2007-12-28
HN2005036113A (es) 2010-12-06
EP1836211A1 (en) 2007-09-26
KR100897678B1 (ko) 2009-05-14
UA85937C2 (uk) 2009-03-10
US20060135447A1 (en) 2006-06-22
GT200500378A (es) 2006-11-28
ZA200705108B (en) 2009-01-28
HRP20100253T1 (hr) 2010-06-30
EP2233493A1 (en) 2010-09-29
NL1030713C2 (nl) 2006-12-12
AU2005317735B2 (en) 2009-06-04
IL183661A0 (en) 2007-09-20
PT1836211E (pt) 2010-04-08
JP2008524319A (ja) 2008-07-10
TW200626608A (en) 2006-08-01
MX2007007598A (es) 2007-07-25
MA29108B1 (fr) 2007-12-03
US7462600B2 (en) 2008-12-09
SI1836211T1 (sl) 2010-04-30
EP1836211B1 (en) 2010-03-03
CA2591746A1 (en) 2006-06-29
NL1030713A1 (nl) 2006-06-22
AP2007004026A0 (en) 2007-06-30

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