UY27625A1 - COMPRESSED NELFINAVIR OF INCREASED DOSE AND METHOD FOR MANUFACTURING IT - Google Patents
COMPRESSED NELFINAVIR OF INCREASED DOSE AND METHOD FOR MANUFACTURING ITInfo
- Publication number
- UY27625A1 UY27625A1 UY27625A UY27625A UY27625A1 UY 27625 A1 UY27625 A1 UY 27625A1 UY 27625 A UY27625 A UY 27625A UY 27625 A UY27625 A UY 27625A UY 27625 A1 UY27625 A1 UY 27625A1
- Authority
- UY
- Uruguay
- Prior art keywords
- nelfinavir
- compressed
- manufacturing
- increased dose
- mixture
- Prior art date
Links
- QAGYKUNXZHXKMR-UHFFFAOYSA-N CPD000469186 Natural products CC1=C(O)C=CC=C1C(=O)NC(C(O)CN1C(CC2CCCCC2C1)C(=O)NC(C)(C)C)CSC1=CC=CC=C1 QAGYKUNXZHXKMR-UHFFFAOYSA-N 0.000 title abstract 5
- 229960000884 nelfinavir Drugs 0.000 title abstract 5
- 238000000034 method Methods 0.000 title abstract 4
- QAGYKUNXZHXKMR-HKWSIXNMSA-N nelfinavir Chemical compound CC1=C(O)C=CC=C1C(=O)N[C@H]([C@H](O)CN1[C@@H](C[C@@H]2CCCC[C@@H]2C1)C(=O)NC(C)(C)C)CSC1=CC=CC=C1 QAGYKUNXZHXKMR-HKWSIXNMSA-N 0.000 title abstract 4
- 238000004519 manufacturing process Methods 0.000 title 1
- 239000000203 mixture Substances 0.000 abstract 3
- 239000011230 binding agent Substances 0.000 abstract 2
- 238000005469 granulation Methods 0.000 abstract 2
- 230000003179 granulation Effects 0.000 abstract 2
- -1 nelfinavir compound Chemical class 0.000 abstract 1
Landscapes
- Medicinal Preparation (AREA)
- Glanulating (AREA)
Abstract
Un comprimido de nelfinavir de dosis elevada que tiene una relación en peso de nelfinavir a aglutinante de aproximadamente 3: 1 a aproximadamente 5: 1. Los comprimidos de nelfinavir de dosis elevada se fabrican en un procedimiento en el que se forma una mezcla granulada de un compuesto de nelfinavir y un aglutinante, en un procedimiento de granulación, y a continuación se elabora para formar los comprimidos. En el procedimiento de granulación se anade humedad y se aplica energía mecánica a la mezcla, y la mezcla se cura sin adición de humedad o aplicación de energía mecánica.A high dose nelfinavir tablet having a weight ratio of nelfinavir to a binder of about 3: 1 to about 5: 1. High dose nelfinavir tablets are manufactured in a process in which a granulated mixture of a nelfinavir compound and a binder, in a granulation procedure, and then made to form the tablets. In the granulation process moisture is added and mechanical energy is applied to the mixture, and the mixture is cured without addition of moisture or application of mechanical energy.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US60735102A | 2002-01-28 | 2002-01-28 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| UY27625A1 true UY27625A1 (en) | 2003-08-29 |
Family
ID=38812730
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| UY27625A UY27625A1 (en) | 2002-01-28 | 2003-01-27 | COMPRESSED NELFINAVIR OF INCREASED DOSE AND METHOD FOR MANUFACTURING IT |
Country Status (1)
| Country | Link |
|---|---|
| UY (1) | UY27625A1 (en) |
-
2003
- 2003-01-27 UY UY27625A patent/UY27625A1/en not_active Application Discontinuation
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| AR036813A1 (en) | PHARMACEUTICAL COMPOSITIONS | |
| AR041370A1 (en) | SOLID PHARMACEUTICAL FORMULATIONS THAT INCLUDE TELMISARTAN AND ITS PREPARATION | |
| AR051618A1 (en) | COMPRESSED BICYCLE AND METHOD | |
| BRPI0707044B8 (en) | water-insoluble matrix tablet and matrix tablet manufacturing process | |
| AR052878A1 (en) | FORMULATION OF DIRECT COMPRESSION AND PROCESS | |
| ES2195308T3 (en) | PHARMACEUTICAL PHENOFIBRATE COMPOSITION THAT PRESENTS A HIGH BIODISPONIBILITY, AND METHOD FOR PREPARATION. | |
| HN2004000319A (en) | "{1,8} NAFTIRIDIN-2-ONAS AND RELATED COMPOUNDS FOR THE TREATMENT OF CHICHOPHRENIA" | |
| ECSP034831A (en) | SUBSTITUTED DERIVATIVES OF 2-PYRIDINE CYCLHEXAN-1,4-DIAMINE | |
| AR011069A1 (en) | AMIDINE COMPOUNDS, PROCESS FOR THEIR PREPARATION, INTERMEDIARY COMPOUNDS, PHARMACEUTICAL FORMULATIONS THAT UNDERSTAND THEM, AND THEIR USE IN THE MANUFACTURE OF A MEDICINAL PRODUCT AS AN INHIBITOR OF NITRIC OXIDE, INDUCIBLE SYNTHESES. | |
| ECSP099320A (en) | Tetrahydropyrrolopyrazine substituted compounds and their application in medicines | |
| AR109263A2 (en) | COMPOSITION INCLUDING MOXIDECTINE | |
| AR025052A1 (en) | DERIVATIVES OF 2-DIALQUILAMINOALQUILBIFENILO SUBSTITUTED, PROCEDURE FOR PREPARATION, MEDICATIONS CONTAINING THESE COMPOUNDS AND THE USE OF THESE COMPOUNDS FOR THE PREPARATION OF MEDICINES. | |
| DOP2002000389A (en) | METHOD FOR MANUFACTURING A PHARMACEUTICAL COMPOSITION OF LOW DOSE THAT HAS A DISTRIBUTION AND POWER OF THE UNIFORM DRUG | |
| AR055907A1 (en) | PROCEDURE FOR MANUFACTURING A BITUMINOUS COATING WITH PRERREVESTIMIENT | |
| AR036085A1 (en) | DOSAGE FORMS AND PROCEDURE FOR MANUFACTURING | |
| ATE377042T1 (en) | FLUORELASTOMER COMPOSITIONS | |
| AR038236A1 (en) | COMPRESSED NELFINAVIR OF INCREASED DOSE AND METHOD TO MANUFACTURE IT | |
| UY27625A1 (en) | COMPRESSED NELFINAVIR OF INCREASED DOSE AND METHOD FOR MANUFACTURING IT | |
| CY1108916T1 (en) | SUBSTITUTED PYROLS, THE UNIONS CONTAINING THEM, THE PREPARATION PROCEDURE AND THEIR USE | |
| BRPI0517032A (en) | compounds, process for their manufacture, pharmaceutical compositions comprising them, method for treating and / or preventing diseases and using such compounds | |
| DOP2003000567A (en) | COMPRESSED NELFINAVIR OF INCREASED DOSE AND METHOD TO MANUFACTURE IT | |
| MXPA02010828A (en) | Pharmaceutical composition in capsules comprising a non-steroidal anti-inflammatory and an opiate analgesic for handling pain. | |
| PL378106A1 (en) | Method for producing a pharmaceutical composition in the form of fibrate-containing tablets and tablets produced by said method | |
| AR053899A1 (en) | FORMULATIONS CONTAINING GLIMEPIRIDA AND / OR ITS SALTS | |
| AR110045A2 (en) | PHARMACEUTICAL COMPOSITIONS |
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| 109 | Application deemed to be withdrawn |
Effective date: 20150421 |