UA99461C2 - N5-(2-ethoxyethyl)-n3-(2-pyridinyl)-3,5-piperidinedicarboxamide derivatives for use as renin inhibitors - Google Patents
N5-(2-ethoxyethyl)-n3-(2-pyridinyl)-3,5-piperidinedicarboxamide derivatives for use as renin inhibitorsInfo
- Publication number
- UA99461C2 UA99461C2 UAA200913506A UAA200913506A UA99461C2 UA 99461 C2 UA99461 C2 UA 99461C2 UA A200913506 A UAA200913506 A UA A200913506A UA A200913506 A UAA200913506 A UA A200913506A UA 99461 C2 UA99461 C2 UA 99461C2
- Authority
- UA
- Ukraine
- Prior art keywords
- compound
- treatment
- piperidinedicarboxamide
- ethoxyethyl
- pyridinyl
- Prior art date
Links
- 239000002461 renin inhibitor Substances 0.000 title 1
- 229940086526 renin-inhibitors Drugs 0.000 title 1
- 150000001875 compounds Chemical class 0.000 abstract 5
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 abstract 4
- 102100028255 Renin Human genes 0.000 abstract 3
- 108090000783 Renin Proteins 0.000 abstract 3
- 201000010099 disease Diseases 0.000 abstract 3
- 230000000694 effects Effects 0.000 abstract 3
- 238000000034 method Methods 0.000 abstract 2
- 239000008194 pharmaceutical composition Substances 0.000 abstract 2
- 238000004519 manufacturing process Methods 0.000 abstract 1
- 230000001225 therapeutic effect Effects 0.000 abstract 1
Landscapes
- Plural Heterocyclic Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
В заявке описаны соединения формулы I(I),где Rl, R2, R3, R4 и R5 являются такими, как определено в описании,предназначенные для применения при диагностике и лечении теплокровного животного, преимущественно для лечения заболевания (= нарушения), которое зависит от активности ренина; применение соединения этого класса для приготовления фармацевтической композиции, предназначенной для лечения заболевания, которое зависит от активности ренина; применение соединения этого класса для лечения заболевания, которое зависит от активности ренина; фармацевтические композиции соединения этого класса; способ лечения, который включает введение соединения этого класса, и способ его получения.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP07012412 | 2007-06-25 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| UA99461C2 true UA99461C2 (en) | 2012-08-27 |
Family
ID=43618556
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| UAA200913506A UA99461C2 (en) | 2007-06-25 | 2008-06-23 | N5-(2-ethoxyethyl)-n3-(2-pyridinyl)-3,5-piperidinedicarboxamide derivatives for use as renin inhibitors |
Country Status (2)
| Country | Link |
|---|---|
| UA (1) | UA99461C2 (ru) |
| ZA (1) | ZA200908547B (ru) |
-
2008
- 2008-06-23 UA UAA200913506A patent/UA99461C2/ru unknown
-
2009
- 2009-12-02 ZA ZA200908547A patent/ZA200908547B/xx unknown
Also Published As
| Publication number | Publication date |
|---|---|
| ZA200908547B (en) | 2010-09-29 |
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