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UA95247C2 - Пиримидиновые соединения как модуляторы рецептора серотонина - Google Patents

Пиримидиновые соединения как модуляторы рецептора серотонина

Info

Publication number
UA95247C2
UA95247C2 UAA200801682A UAA200801682A UA95247C2 UA 95247 C2 UA95247 C2 UA 95247C2 UA A200801682 A UAA200801682 A UA A200801682A UA A200801682 A UAA200801682 A UA A200801682A UA 95247 C2 UA95247 C2 UA 95247C2
Authority
UA
Ukraine
Prior art keywords
receptor modulators
serotonin receptor
pyrimidine compounds
serotonin
pyrimidine
Prior art date
Application number
UAA200801682A
Other languages
English (en)
Ukrainian (uk)
Inventor
Курт А. Дворак
Дейл А. Рудольф
Брок Т. Шайрмен
Original Assignee
Янссен Фармацевтика Н.В.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Янссен Фармацевтика Н.В. filed Critical Янссен Фармацевтика Н.В.
Publication of UA95247C2 publication Critical patent/UA95247C2/ru

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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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Abstract

В заявке описаны определенные пиримидиновые соединения, которые являются модуляторами рецептора серотонина, пригодные при лечении расстройств, опосредованных серотонином.
UAA200801682A 2005-08-04 2006-07-27 Пиримидиновые соединения как модуляторы рецептора серотонина UA95247C2 (ru)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US70571905P 2005-08-04 2005-08-04

Publications (1)

Publication Number Publication Date
UA95247C2 true UA95247C2 (ru) 2011-07-25

Family

ID=37400981

Family Applications (1)

Application Number Title Priority Date Filing Date
UAA200801682A UA95247C2 (ru) 2005-08-04 2006-07-27 Пиримидиновые соединения как модуляторы рецептора серотонина

Country Status (16)

Country Link
EP (1) EP1928461B1 (ru)
JP (1) JP5066088B2 (ru)
KR (1) KR101353268B1 (ru)
CN (1) CN101277700B (ru)
AT (1) ATE539753T1 (ru)
AU (1) AU2006278759B2 (ru)
BR (1) BRPI0614397A2 (ru)
CA (1) CA2617760C (ru)
CR (1) CR9791A (ru)
EA (1) EA014495B1 (ru)
IL (2) IL189164A (ru)
NO (1) NO340744B1 (ru)
NZ (1) NZ565334A (ru)
UA (1) UA95247C2 (ru)
WO (1) WO2007019083A1 (ru)
ZA (1) ZA200802010B (ru)

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UA125631C2 (uk) 2016-11-15 2022-05-04 Темпл Юніверсіті-Оф Дзе Коммонвелт Сістем Оф Хайєр Едьюкейшн Нові модулятори 5-гідрокситриптамінового рецептора 7 і спосіб їх застосування
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EP3797108B1 (en) 2018-05-21 2022-07-20 Constellation Pharmaceuticals, Inc. Modulators of methyl modifying enzymes, compositions and uses thereof
KR102282569B1 (ko) * 2019-02-08 2021-07-29 (주)퓨쳐켐 새로운 18F-표지된 친디엔체와 테트라진 화합물과의 IeDDA 반응을 이용한 18F-표지 방법
EP4003532B1 (en) 2019-07-24 2024-09-04 Constellation Pharmaceuticals, Inc. Crystalline forms of 7-chloro-2-(4-(3-methoxyazetidin-1-yl)cyclohexyl)-2,4-dimethyl-n-((6-methyl-4-(methylthio)-2-oxo-1,2-dihydropyridin-3-yl)methyl)benzo[d][1,3]dioxole-5-carboxamide
KR102483492B1 (ko) * 2019-09-02 2023-01-02 한양대학교 에리카산학협력단 2,5-이치환된 피리미딘 유도체 및 이를 포함하는 약학적 조성물
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WO2007019083A1 (en) 2007-02-15
ATE539753T1 (de) 2012-01-15
EA200800525A1 (ru) 2008-06-30
EP1928461A1 (en) 2008-06-11
CR9791A (es) 2010-05-27
ZA200802010B (en) 2009-09-30
JP5066088B2 (ja) 2012-11-07
IL213679A0 (en) 2011-07-31
CA2617760A1 (en) 2007-02-15
CN101277700A (zh) 2008-10-01
NO20081034L (no) 2008-02-28
NZ565334A (en) 2010-12-24
HK1118469A1 (en) 2009-02-13
IL189164A0 (en) 2008-08-07
NO340744B1 (no) 2017-06-12
KR20080033502A (ko) 2008-04-16
BRPI0614397A2 (pt) 2011-03-29
KR101353268B1 (ko) 2014-02-06
CA2617760C (en) 2015-02-17
AU2006278759B2 (en) 2012-08-16
CN101277700B (zh) 2013-02-20
IL189164A (en) 2013-08-29
AU2006278759A1 (en) 2007-02-15
EP1928461B1 (en) 2012-01-04

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