UA92047C2 - Карбоніламінопіролпіразоли - потужні інгібітори кінази[карбониламинопирролпиразолы - мощные ингибиторы киназы - Google Patents
Карбоніламінопіролпіразоли - потужні інгібітори кінази[карбониламинопирролпиразолы - мощные ингибиторы киназыInfo
- Publication number
- UA92047C2 UA92047C2 UAA200807387A UAA200807387A UA92047C2 UA 92047 C2 UA92047 C2 UA 92047C2 UA A200807387 A UAA200807387 A UA A200807387A UA A200807387 A UAA200807387 A UA A200807387A UA 92047 C2 UA92047 C2 UA 92047C2
- Authority
- UA
- Ukraine
- Prior art keywords
- kinase inhibitors
- pyrrolopyrazoles
- carbonylamino
- potent kinase
- compounds
- Prior art date
Links
- XPBFIMLMVNXIIB-UHFFFAOYSA-N 3-isocyanatopyrrolo[3,2-c]pyrazole Chemical class N1=CC=C2N=NC(N=C=O)=C21 XPBFIMLMVNXIIB-UHFFFAOYSA-N 0.000 title 1
- 229940043355 kinase inhibitor Drugs 0.000 title 1
- 239000003757 phosphotransferase inhibitor Substances 0.000 title 1
- 230000003389 potentiating effect Effects 0.000 title 1
- 150000001875 compounds Chemical class 0.000 abstract 3
- 101000987297 Homo sapiens Serine/threonine-protein kinase PAK 4 Proteins 0.000 abstract 1
- 102100027940 Serine/threonine-protein kinase PAK 4 Human genes 0.000 abstract 1
- 229940045988 antineoplastic drug protein kinase inhibitors Drugs 0.000 abstract 1
- 239000003112 inhibitor Substances 0.000 abstract 1
- 239000000203 mixture Substances 0.000 abstract 1
- 239000003909 protein kinase inhibitor Substances 0.000 abstract 1
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US75334905P | 2005-12-21 | 2005-12-21 | |
| US86493206P | 2006-11-08 | 2006-11-08 | |
| PCT/IB2006/003646 WO2007072153A2 (en) | 2005-12-21 | 2006-12-12 | Carbonylamino pyrrolopyrazoles, potent kinase inhibitors |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| UA92047C2 true UA92047C2 (xx) | 2010-09-27 |
Family
ID=40247953
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| UAA200807387A UA92047C2 (xx) | 2005-12-21 | 2006-12-12 | Карбоніламінопіролпіразоли - потужні інгібітори кінази[карбониламинопирролпиразолы - мощные ингибиторы киназы |
Country Status (5)
| Country | Link |
|---|---|
| CN (1) | CN101346382B (xx) |
| SI (1) | SI1979356T1 (xx) |
| TN (1) | TNSN08274A1 (xx) |
| UA (1) | UA92047C2 (xx) |
| ZA (1) | ZA200804667B (xx) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN113234081A (zh) * | 2021-05-27 | 2021-08-10 | 东南大学 | 一种吡咯并吡唑衍生物与dmpeda做脲的制备方法 |
| CN117185993B (zh) * | 2023-08-28 | 2025-08-12 | 南通华祥医药科技有限公司 | 一种含取代苯巯基吡啶结构单元的酰胺类化合物的制备与应用 |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| UA81790C2 (uk) * | 2002-12-19 | 2008-02-11 | Фармация Италия С.П.А. | Заміщені піролопіразольні похідні як інгібітори кінази |
-
2006
- 2006-12-12 SI SI200631657T patent/SI1979356T1/sl unknown
- 2006-12-12 CN CN2006800486846A patent/CN101346382B/zh not_active Expired - Fee Related
- 2006-12-12 UA UAA200807387A patent/UA92047C2/uk unknown
-
2008
- 2008-05-29 ZA ZA200804667A patent/ZA200804667B/xx unknown
- 2008-06-20 TN TNP2008000274A patent/TNSN08274A1/fr unknown
Also Published As
| Publication number | Publication date |
|---|---|
| ZA200804667B (en) | 2010-05-26 |
| CN101346382B (zh) | 2011-07-06 |
| TNSN08274A1 (fr) | 2009-10-30 |
| SI1979356T1 (sl) | 2013-11-29 |
| CN101346382A (zh) | 2009-01-14 |
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