UA88444C2 - Aza spiro alkane derivatives as inhibitors of metallproteases - Google Patents
Aza spiro alkane derivatives as inhibitors of metallproteasesInfo
- Publication number
- UA88444C2 UA88444C2 UAA200511110A UAA200511110A UA88444C2 UA 88444 C2 UA88444 C2 UA 88444C2 UA A200511110 A UAA200511110 A UA A200511110A UA A200511110 A UAA200511110 A UA A200511110A UA 88444 C2 UA88444 C2 UA 88444C2
- Authority
- UA
- Ukraine
- Prior art keywords
- metallproteases
- inhibitors
- formula
- alkane derivatives
- aza spiro
- Prior art date
Links
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
Даний винахід описує сполуку формули І або формули II:, I, IIїї енантіомери, діастереомери, проліки, сольвати, метаболіти або фармацевтично прийнятні солі, де складові змінні визначені в описі даної заявки.Сполуки формули І і II є модуляторами металопротеаз і корисні для лікування захворювань, пов'язаних з активністю металопротеаз, таких як артрит, рак, серцево-судинні розлади, шкірні захворювання, запальні та алергійні стани.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US46615903P | 2003-04-24 | 2003-04-24 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| UA88444C2 true UA88444C2 (en) | 2009-10-26 |
Family
ID=37390761
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| UAA200511110A UA88444C2 (en) | 2003-04-24 | 2004-04-23 | Aza spiro alkane derivatives as inhibitors of metallproteases |
Country Status (4)
| Country | Link |
|---|---|
| CN (1) | CN1863532A (uk) |
| CR (1) | CR8045A (uk) |
| UA (1) | UA88444C2 (uk) |
| ZA (1) | ZA200509496B (uk) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US11851475B2 (en) | 2018-01-03 | 2023-12-26 | Xi'an Jiaotong-Liverpool University | Membrane-type metalloprotease inhibitory protein and pharmaceutical and pharmaceutical composition containing same, and respective uses thereof |
| CN109394786A (zh) * | 2018-10-26 | 2019-03-01 | 西交利物浦大学 | 一种抗肿瘤的药物组合物 |
-
2004
- 2004-04-23 CN CN 200480017350 patent/CN1863532A/zh active Pending
- 2004-04-23 UA UAA200511110A patent/UA88444C2/ru unknown
-
2005
- 2005-10-14 CR CR8045A patent/CR8045A/es not_active Application Discontinuation
- 2005-11-23 ZA ZA200509496A patent/ZA200509496B/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| CN1863532A (zh) | 2006-11-15 |
| ZA200509496B (en) | 2006-10-25 |
| CR8045A (es) | 2006-05-29 |
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