UA87515C2 - Фармацевтическая композиция толтеродина с пролонгированным высвобождением - Google Patents
Фармацевтическая композиция толтеродина с пролонгированным высвобождениемInfo
- Publication number
- UA87515C2 UA87515C2 UAA200703260A UAA200703260A UA87515C2 UA 87515 C2 UA87515 C2 UA 87515C2 UA A200703260 A UAA200703260 A UA A200703260A UA A200703260 A UAA200703260 A UA A200703260A UA 87515 C2 UA87515 C2 UA 87515C2
- Authority
- UA
- Ukraine
- Prior art keywords
- pharmaceutical composition
- tolterodine
- sustained release
- release pharmaceutical
- composition
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
- A61K9/5005—Wall or coating material
- A61K9/5021—Organic macromolecular compounds
- A61K9/5026—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/13—Amines
- A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
- A61K31/137—Arylalkylamines, e.g. amphetamine, epinephrine, salbutamol, ephedrine or methadone
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
- A61K9/5073—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings
- A61K9/5078—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings with drug-free core
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/10—Drugs for disorders of the urinary system of the bladder
Landscapes
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Epidemiology (AREA)
- Emergency Medicine (AREA)
- Urology & Nephrology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Medicinal Preparation (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Abstract
Данное изобретение относится к фармацевтической композиции с пролонгированным высвобождением, которая содержит толтеродин, преимущественно толтеродина тартрат, применения указанной композиции для приготовления лекарственного средства и способа получения такой фармацевтической композиции.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP04020431A EP1629834A1 (en) | 2004-08-27 | 2004-08-27 | Sustained release pharmaceutical composition of tolterodine |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| UA87515C2 true UA87515C2 (ru) | 2009-07-27 |
Family
ID=34926332
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| UAA200703260A UA87515C2 (ru) | 2004-08-27 | 2005-08-23 | Фармацевтическая композиция толтеродина с пролонгированным высвобождением |
Country Status (7)
| Country | Link |
|---|---|
| EP (3) | EP1629834A1 (ru) |
| AT (1) | ATE505187T1 (ru) |
| DE (1) | DE602005027469D1 (ru) |
| EA (1) | EA200700484A1 (ru) |
| NO (1) | NO20071299L (ru) |
| UA (1) | UA87515C2 (ru) |
| WO (1) | WO2006021425A1 (ru) |
Families Citing this family (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA2645940A1 (en) * | 2006-03-21 | 2007-09-27 | Teva Pharmaceutical Industries Ltd. | Controlled release formulation of tolterodine |
| EP1839649A1 (en) * | 2006-03-31 | 2007-10-03 | LEK Pharmaceuticals D.D. | Coated formulations for tolterodine |
| KR100851033B1 (ko) * | 2007-02-12 | 2008-08-12 | 명문제약주식회사 | 엘-주석산 톨터로딘 함유 서방성 제제의 제조방법 |
| WO2009019599A2 (en) * | 2007-08-08 | 2009-02-12 | Themis Laboratories Private Limited | Extended release compositions comprising tolterodine |
| WO2011061616A2 (en) | 2009-11-23 | 2011-05-26 | Micro Labs Limited | Extended release compositions containing tolterodine and process for preparing the same |
| WO2011095388A1 (en) | 2010-02-04 | 2011-08-11 | Synthon Bv | Tolterodine bead |
| GB2479213B (en) | 2010-04-01 | 2013-07-10 | Theravida Inc | Pharmaceutical formulations for the treatment of overactive bladder |
| RU2671575C2 (ru) | 2011-05-10 | 2018-11-02 | Теравида, Инк. | Применение солифенацина и стимуляторов слюноотделения в лечении гиперактивного мочевого пузыря |
| CN103211784B (zh) * | 2012-01-18 | 2017-07-11 | 北京天衡药物研究院有限公司 | 酒石酸托特罗定膜控缓释微丸胶囊 |
| TW201422254A (zh) | 2012-11-21 | 2014-06-16 | Ferring Bv | 用於速釋及延釋的組成物 |
| DK3405191T3 (da) | 2016-01-20 | 2025-05-19 | Theravida Inc | Sammensætninger til anvendelse ved behandling af hyperhidrose |
Family Cites Families (18)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| SE2061C1 (ru) † | 1890-01-25 | |||
| SE8800207D0 (sv) | 1988-01-22 | 1988-01-22 | Kabivitrum Ab | Nya aminer, deras anvendning och framstellning |
| SE9203318D0 (sv) | 1992-11-06 | 1992-11-06 | Kabi Pharmacia Ab | Novel 3,3-diphenylpropylamines, their use and preparation |
| US6274171B1 (en) † | 1996-03-25 | 2001-08-14 | American Home Products Corporation | Extended release formulation of venlafaxine hydrochloride |
| JP2000515525A (ja) | 1996-07-19 | 2000-11-21 | アベーグ,グンナー | 尿と胃腸の疾患の治療におけるs(―)―トルテロジン |
| KR20000057548A (ko) | 1996-12-13 | 2000-09-25 | 알프레드 엘. 미첼슨 | 광학적 전송물질 및 결합재 |
| SE9803871D0 (sv) † | 1998-11-11 | 1998-11-11 | Pharmacia & Upjohn Ab | Therapeutic method and formulation |
| SI1039882T1 (sl) * | 1998-08-27 | 2011-01-31 | Pfizer Health Ab | Terapevtska formulacija za dajanje tolterodina s kontroliranim sproščanjem |
| DE19901692C2 (de) † | 1999-01-18 | 2002-06-20 | Gruenenthal Gmbh | Verfahren zur Herstellung von Pellets mit einem Gehalt von bis zu 90 Gew.% eines pharmazeutischen Wirkstoffes |
| KR100838930B1 (ko) * | 1999-11-11 | 2008-06-16 | 화이자 헬스 에이비 | 톨테로딘을 포함하는 약학 제제 및 이의 용도 |
| SE9904850D0 (sv) | 1999-12-30 | 1999-12-30 | Pharmacia & Upjohn Ab | Novel process and intermediates |
| IN191835B (ru) | 2001-08-03 | 2004-01-10 | Ranbaxy Lab Ltd | |
| US20030185882A1 (en) * | 2001-11-06 | 2003-10-02 | Vergez Juan A. | Pharmaceutical compositions containing oxybutynin |
| WO2003053428A1 (en) * | 2001-12-20 | 2003-07-03 | Pharmacia Corporation | Controlled release dosage form having improved drug release properties |
| KR100540035B1 (ko) † | 2002-02-01 | 2005-12-29 | 주식회사 태평양 | 다단계 경구 약물 방출 제어 시스템 |
| US7005449B2 (en) | 2002-04-23 | 2006-02-28 | Pharmacia & Upjohn Company | Tolterodine salts |
| CN1150160C (zh) | 2002-04-29 | 2004-05-19 | 上海医药工业研究院 | L-酒石酸托特罗定的合成方法 |
| EP1635795A1 (en) | 2003-05-30 | 2006-03-22 | Ranbaxy Laboratories, Ltd. | Controlled release pharmaceutical compositions of tolterodine and processes for their preparation |
-
2004
- 2004-08-27 EP EP04020431A patent/EP1629834A1/en not_active Withdrawn
-
2005
- 2005-08-23 AT AT05784596T patent/ATE505187T1/de not_active IP Right Cessation
- 2005-08-23 EA EA200700484A patent/EA200700484A1/ru unknown
- 2005-08-23 EP EP08007539A patent/EP1964553A1/en not_active Withdrawn
- 2005-08-23 UA UAA200703260A patent/UA87515C2/ru unknown
- 2005-08-23 DE DE602005027469T patent/DE602005027469D1/de not_active Expired - Lifetime
- 2005-08-23 WO PCT/EP2005/009102 patent/WO2006021425A1/en not_active Ceased
- 2005-08-23 EP EP05784596.8A patent/EP1781275B2/en not_active Expired - Lifetime
-
2007
- 2007-03-09 NO NO20071299A patent/NO20071299L/no not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| NO20071299L (no) | 2007-05-29 |
| WO2006021425A1 (en) | 2006-03-02 |
| EP1629834A1 (en) | 2006-03-01 |
| DE602005027469D1 (de) | 2011-05-26 |
| ATE505187T1 (de) | 2011-04-15 |
| EA200700484A1 (ru) | 2007-10-26 |
| EP1781275A1 (en) | 2007-05-09 |
| EP1781275B1 (en) | 2011-04-13 |
| EP1781275B2 (en) | 2014-04-16 |
| EP1964553A1 (en) | 2008-09-03 |
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