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UA83915C2 - Многофазный препарат для контрацепции на основе натурального эстрогена - Google Patents

Многофазный препарат для контрацепции на основе натурального эстрогена

Info

Publication number
UA83915C2
UA83915C2 UAA200611799A UAA200611799A UA83915C2 UA 83915 C2 UA83915 C2 UA 83915C2 UA A200611799 A UAA200611799 A UA A200611799A UA A200611799 A UAA200611799 A UA A200611799A UA 83915 C2 UA83915 C2 UA 83915C2
Authority
UA
Ukraine
Prior art keywords
natural estrogen
preparation based
preparation
contraceptive preparation
phase
Prior art date
Application number
UAA200611799A
Other languages
English (en)
Ukrainian (uk)
Inventor
Ян Эндрикат
Бернд Дюстерберг
Original Assignee
Байер Шеринг Фарма Акциенгезелльшафт
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=34979546&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=UA83915(C2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Байер Шеринг Фарма Акциенгезелльшафт filed Critical Байер Шеринг Фарма Акциенгезелльшафт
Publication of UA83915C2 publication Critical patent/UA83915C2/ru

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/565—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/57—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/18—Feminine contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/24—Drugs for disorders of the endocrine system of the sex hormones

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Endocrinology (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Reproductive Health (AREA)
  • Gynecology & Obstetrics (AREA)
  • Diabetes (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Orthopedics, Nursing, And Contraception (AREA)
  • Steroid Compounds (AREA)
  • Compositions Of Macromolecular Compounds (AREA)

Abstract

Изобретение касается многофазного препарата для контрацепции на основе натурального эстрогена в комбинации с синтетическим гестагеном, который по сравнению с обычными известными препаратами, угнетающими овуляцию, обеспечивает более высокую контрацептивную надежность.
UAA200611799A 2004-04-20 2005-04-15 Многофазный препарат для контрацепции на основе натурального эстрогена UA83915C2 (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE102004019743A DE102004019743B4 (de) 2004-04-20 2004-04-20 Mehrphasenpräparat zur Kontrazeption auf der Basis eines natürlichen Estrogens
PCT/EP2005/004022 WO2005102247A2 (de) 2004-04-20 2005-04-15 Mehrphasenpräparat zur kontrazeption auf der basis eines natürlichen estrogens

Publications (1)

Publication Number Publication Date
UA83915C2 true UA83915C2 (ru) 2008-08-26

Family

ID=34979546

Family Applications (1)

Application Number Title Priority Date Filing Date
UAA200611799A UA83915C2 (ru) 2004-04-20 2005-04-15 Многофазный препарат для контрацепции на основе натурального эстрогена

Country Status (37)

Country Link
US (3) US8071577B2 (ru)
EP (1) EP1740163B2 (ru)
JP (1) JP4908399B2 (ru)
KR (1) KR20060134168A (ru)
CN (1) CN1946383B (ru)
AR (2) AR048830A1 (ru)
AT (1) ATE473734T1 (ru)
AU (1) AU2005235418C1 (ru)
BR (1) BRPI0510005A (ru)
CA (1) CA2561839C (ru)
CR (1) CR8695A (ru)
CY (1) CY1111292T1 (ru)
DE (2) DE102004019743B4 (ru)
DK (1) DK1740163T4 (ru)
EA (1) EA010313B1 (ru)
EC (1) ECSP067000A (ru)
ES (1) ES2348038T5 (ru)
GT (1) GT200500093A (ru)
HR (1) HRP20100513T4 (ru)
IL (2) IL178510A (ru)
ME (1) ME01183B (ru)
MX (1) MXPA06012213A (ru)
MY (1) MY143669A (ru)
NO (1) NO344098B1 (ru)
NZ (1) NZ550417A (ru)
PA (1) PA8630901A1 (ru)
PE (1) PE20060308A1 (ru)
PL (1) PL1740163T5 (ru)
PT (1) PT1740163E (ru)
RS (1) RS51434B2 (ru)
SI (1) SI1740163T2 (ru)
SV (1) SV2006002090A (ru)
TW (1) TWI351960B (ru)
UA (1) UA83915C2 (ru)
UY (1) UY28863A1 (ru)
WO (1) WO2005102247A2 (ru)
ZA (1) ZA200609594B (ru)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE102004019743B4 (de) 2004-04-20 2008-11-27 Bayer Schering Pharma Aktiengesellschaft Mehrphasenpräparat zur Kontrazeption auf der Basis eines natürlichen Estrogens
DE502005006837D1 (de) * 2005-10-13 2009-04-23 Bayer Schering Pharma Ag Verwendung von Estradiolvalerat in Kombination mit Dienogest zur oralen Therapie der dysfunktionellen uterinen Blutung in Einheit mit einer oralen Kontrazeption
DK1937274T3 (da) * 2005-10-13 2012-06-18 Bayer Pharma AG Anvendelse af estradiolvalerat i kombination med dienogest til oral behandling af dysfunktionel uterin blødning i enhed med en oral kontraception
US8153616B2 (en) * 2005-10-17 2012-04-10 Bayer Pharma Aktiengesellschaft Combination preparation for oral contraception and oral therapy of dysfunctional uterine bleeding containing estradiol valerate and dienogest and method of using same
EP1993531B1 (en) * 2006-03-02 2015-10-14 Warner Chilcott Company, LLC Extended cycle multiphasic oral contraceptive method
DE102006010329A1 (de) * 2006-03-06 2007-09-13 Höltge, Michael, Dipl.-Med. Hormonelles Kontrazeptivum auf der Basis eines Estrogens, eines Gestagens oder einer Kombination von Estrogenen und Gestagenen unter der Zugabe von Testosteron
EP1930010A1 (de) * 2006-10-20 2008-06-11 Bayer Schering Pharma Aktiengesellschaft Verwendung von Estradiolvalerat oder 17ß-Estradiol in Kombination mit Dienogest zur oralen Therapie für den Erhalt und/oder die Steigerung der weiblichen Libido
US20090117184A1 (en) * 2007-11-05 2009-05-07 Sabine Fricke Use of a gestagen in combination with an estrogen and one or more pharmaceutically acceptable auxiliary agents/excipients for lactose-free oral contraception
AR086395A1 (es) * 2011-05-11 2013-12-11 Kirax Corp Envase para el tratamiento de patologias

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DE2365103C3 (de) 1973-12-21 1980-08-28 Schering Ag, 1000 Berlin Und 4619 Bergkamen V erwendung von Hormonen zur Kontrazeption
DE2431704A1 (de) 1974-07-02 1976-01-22 Asche Ag Stufenkombinationspraeparate per kontrazeption
DE2645307A1 (de) 1976-10-05 1978-04-06 Schering Ag Neue mittel und neue methoden zur behandlung klimakterischer ausfallerscheinungen
JPS6019734B2 (ja) 1977-05-12 1985-05-17 三共株式会社 安定なプロスタグランジンｅ類製剤の製法
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PT1635843E (pt) 2003-06-25 2009-04-07 Bayer Schering Pharma Ag Terapia de substituição hormonal e de depressão compreendendo dienogest
DE102004019743B4 (de) 2004-04-20 2008-11-27 Bayer Schering Pharma Aktiengesellschaft Mehrphasenpräparat zur Kontrazeption auf der Basis eines natürlichen Estrogens
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DE502005006837D1 (de) 2005-10-13 2009-04-23 Bayer Schering Pharma Ag Verwendung von Estradiolvalerat in Kombination mit Dienogest zur oralen Therapie der dysfunktionellen uterinen Blutung in Einheit mit einer oralen Kontrazeption
US8153616B2 (en) 2005-10-17 2012-04-10 Bayer Pharma Aktiengesellschaft Combination preparation for oral contraception and oral therapy of dysfunctional uterine bleeding containing estradiol valerate and dienogest and method of using same
EP1930010A1 (de) 2006-10-20 2008-06-11 Bayer Schering Pharma Aktiengesellschaft Verwendung von Estradiolvalerat oder 17ß-Estradiol in Kombination mit Dienogest zur oralen Therapie für den Erhalt und/oder die Steigerung der weiblichen Libido

Also Published As

Publication number Publication date
US20070259840A1 (en) 2007-11-08
WO2005102247A2 (de) 2005-11-03
NO344098B1 (no) 2019-09-02
PL1740163T3 (pl) 2010-12-31
TW200534860A (en) 2005-11-01
DK1740163T3 (da) 2010-10-18
DE102004019743B4 (de) 2008-11-27
NZ550417A (en) 2010-01-29
CA2561839C (en) 2009-09-29
WO2005102247A3 (de) 2006-01-12
HK1099701A1 (zh) 2007-08-24
ECSP067000A (es) 2006-12-29
MXPA06012213A (es) 2007-01-17
CY1111292T1 (el) 2015-08-05
US8071577B2 (en) 2011-12-06
PT1740163E (pt) 2010-09-28
US20100173877A1 (en) 2010-07-08
IL178510A0 (en) 2007-02-11
SI1740163T1 (sl) 2010-11-30
NO20065292L (no) 2007-01-17
HRP20100513T4 (hr) 2020-10-02
PL1740163T5 (pl) 2020-10-05
PE20060308A1 (es) 2006-05-25
AR084229A2 (es) 2013-05-02
CR8695A (es) 2008-07-29
ES2348038T5 (es) 2020-09-14
CA2561839A1 (en) 2005-11-03
IL178510A (en) 2015-08-31
CN1946383A (zh) 2007-04-11
RS51434B2 (sr) 2020-11-30
GT200500093A (es) 2006-04-17
DE102004019743A1 (de) 2005-11-24
KR20060134168A (ko) 2006-12-27
ZA200609594B (en) 2008-04-30
RS51434B (sr) 2011-04-30
AU2005235418A1 (en) 2005-11-03
MY143669A (en) 2011-06-30
UY28863A1 (es) 2005-11-30
EA200601844A1 (ru) 2007-04-27
JP2007533681A (ja) 2007-11-22
ES2348038T3 (es) 2010-11-29
EA010313B1 (ru) 2008-08-29
DK1740163T4 (da) 2020-04-06
SV2006002090A (es) 2006-02-15
DE502005009904D1 (de) 2010-08-26
IL239861A0 (en) 2015-08-31
AU2005235418B2 (en) 2009-08-06
EP1740163B2 (de) 2020-01-15
HRP20100513T1 (hr) 2010-11-30
AU2005235418C1 (en) 2015-05-21
AR048830A1 (es) 2006-05-31
TWI351960B (en) 2011-11-11
JP4908399B2 (ja) 2012-04-04
SI1740163T2 (sl) 2020-04-30
EP1740163B1 (de) 2010-07-14
ATE473734T1 (de) 2010-07-15
CN1946383B (zh) 2010-06-09
US20110124612A1 (en) 2011-05-26
ME01183B (me) 2013-03-20
EP1740163A2 (de) 2007-01-10
BRPI0510005A (pt) 2007-09-18
PA8630901A1 (es) 2006-05-16

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