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CR8695A - Preparado polifasico para la contracepcion a base de un estrogeno natural - Google Patents

Preparado polifasico para la contracepcion a base de un estrogeno natural

Info

Publication number
CR8695A
CR8695A CR8695A CR8695A CR8695A CR 8695 A CR8695 A CR 8695A CR 8695 A CR8695 A CR 8695A CR 8695 A CR8695 A CR 8695A CR 8695 A CR8695 A CR 8695A
Authority
CR
Costa Rica
Prior art keywords
natural
strogen
polyphasic
preparation
contraception based
Prior art date
Application number
CR8695A
Other languages
English (en)
Inventor
Jan Endrikat
Bernd Dusterberg
Original Assignee
Bayer Schering Pharma Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=34979546&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CR8695(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Bayer Schering Pharma Ag filed Critical Bayer Schering Pharma Ag
Publication of CR8695A publication Critical patent/CR8695A/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/56Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/565Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/56Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/57Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/56Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • A61P15/18Feminine contraceptives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • A61P5/24Drugs for disorders of the endocrine system of the sex hormones

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Endocrinology (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Reproductive Health (AREA)
  • Gynecology & Obstetrics (AREA)
  • Diabetes (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Orthopedics, Nursing, And Contraception (AREA)
  • Steroid Compounds (AREA)
  • Compositions Of Macromolecular Compounds (AREA)

Abstract

La invencion se refiere a un preparado polifasico para la contracepcion a base de un estrogeno natural en combinacion con un gestageno sintetico que asegura mayor seguridad contraceptiva durante todo el ciclo, que mejora el comportamiento ciclico de la hemorragia y minimiza o elimina los efectos secundarios tales como tension en los pechos, dolores de cabeza, estados de animo depresivos y modificaciones de la libido, etc. en comparacion con los contraceptivos anovulatorios tradicionales del mismo tipo.
CR8695A 2004-04-20 2006-10-19 Preparado polifasico para la contracepcion a base de un estrogeno natural CR8695A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE102004019743A DE102004019743B4 (de) 2004-04-20 2004-04-20 Mehrphasenpräparat zur Kontrazeption auf der Basis eines natürlichen Estrogens

Publications (1)

Publication Number Publication Date
CR8695A true CR8695A (es) 2008-07-29

Family

ID=34979546

Family Applications (1)

Application Number Title Priority Date Filing Date
CR8695A CR8695A (es) 2004-04-20 2006-10-19 Preparado polifasico para la contracepcion a base de un estrogeno natural

Country Status (37)

Country Link
US (3) US8071577B2 (es)
EP (1) EP1740163B2 (es)
JP (1) JP4908399B2 (es)
KR (1) KR20060134168A (es)
CN (1) CN1946383B (es)
AR (2) AR048830A1 (es)
AT (1) ATE473734T1 (es)
AU (1) AU2005235418C1 (es)
BR (1) BRPI0510005A (es)
CA (1) CA2561839C (es)
CR (1) CR8695A (es)
CY (1) CY1111292T1 (es)
DE (2) DE102004019743B4 (es)
DK (1) DK1740163T4 (es)
EA (1) EA010313B1 (es)
EC (1) ECSP067000A (es)
ES (1) ES2348038T5 (es)
GT (1) GT200500093A (es)
HR (1) HRP20100513T4 (es)
IL (2) IL178510A (es)
ME (1) ME01183B (es)
MX (1) MXPA06012213A (es)
MY (1) MY143669A (es)
NO (1) NO344098B1 (es)
NZ (1) NZ550417A (es)
PA (1) PA8630901A1 (es)
PE (1) PE20060308A1 (es)
PL (1) PL1740163T5 (es)
PT (1) PT1740163E (es)
RS (1) RS51434B2 (es)
SI (1) SI1740163T2 (es)
SV (1) SV2006002090A (es)
TW (1) TWI351960B (es)
UA (1) UA83915C2 (es)
UY (1) UY28863A1 (es)
WO (1) WO2005102247A2 (es)
ZA (1) ZA200609594B (es)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE102004019743B4 (de) 2004-04-20 2008-11-27 Bayer Schering Pharma Aktiengesellschaft Mehrphasenpräparat zur Kontrazeption auf der Basis eines natürlichen Estrogens
DE502005006837D1 (de) * 2005-10-13 2009-04-23 Bayer Schering Pharma Ag Verwendung von Estradiolvalerat in Kombination mit Dienogest zur oralen Therapie der dysfunktionellen uterinen Blutung in Einheit mit einer oralen Kontrazeption
DK1937274T3 (da) * 2005-10-13 2012-06-18 Bayer Pharma AG Anvendelse af estradiolvalerat i kombination med dienogest til oral behandling af dysfunktionel uterin blødning i enhed med en oral kontraception
US8153616B2 (en) * 2005-10-17 2012-04-10 Bayer Pharma Aktiengesellschaft Combination preparation for oral contraception and oral therapy of dysfunctional uterine bleeding containing estradiol valerate and dienogest and method of using same
EP1993531B1 (en) * 2006-03-02 2015-10-14 Warner Chilcott Company, LLC Extended cycle multiphasic oral contraceptive method
DE102006010329A1 (de) * 2006-03-06 2007-09-13 Höltge, Michael, Dipl.-Med. Hormonelles Kontrazeptivum auf der Basis eines Estrogens, eines Gestagens oder einer Kombination von Estrogenen und Gestagenen unter der Zugabe von Testosteron
EP1930010A1 (de) * 2006-10-20 2008-06-11 Bayer Schering Pharma Aktiengesellschaft Verwendung von Estradiolvalerat oder 17ß-Estradiol in Kombination mit Dienogest zur oralen Therapie für den Erhalt und/oder die Steigerung der weiblichen Libido
US20090117184A1 (en) * 2007-11-05 2009-05-07 Sabine Fricke Use of a gestagen in combination with an estrogen and one or more pharmaceutically acceptable auxiliary agents/excipients for lactose-free oral contraception
AR086395A1 (es) * 2011-05-11 2013-12-11 Kirax Corp Envase para el tratamiento de patologias

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DE2431704A1 (de) 1974-07-02 1976-01-22 Asche Ag Stufenkombinationspraeparate per kontrazeption
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JPS6019734B2 (ja) 1977-05-12 1985-05-17 三共株式会社 安定なプロスタグランジンe類製剤の製法
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US8153616B2 (en) 2005-10-17 2012-04-10 Bayer Pharma Aktiengesellschaft Combination preparation for oral contraception and oral therapy of dysfunctional uterine bleeding containing estradiol valerate and dienogest and method of using same
EP1930010A1 (de) 2006-10-20 2008-06-11 Bayer Schering Pharma Aktiengesellschaft Verwendung von Estradiolvalerat oder 17ß-Estradiol in Kombination mit Dienogest zur oralen Therapie für den Erhalt und/oder die Steigerung der weiblichen Libido

Also Published As

Publication number Publication date
US20070259840A1 (en) 2007-11-08
WO2005102247A2 (de) 2005-11-03
NO344098B1 (no) 2019-09-02
PL1740163T3 (pl) 2010-12-31
TW200534860A (en) 2005-11-01
DK1740163T3 (da) 2010-10-18
DE102004019743B4 (de) 2008-11-27
NZ550417A (en) 2010-01-29
CA2561839C (en) 2009-09-29
WO2005102247A3 (de) 2006-01-12
HK1099701A1 (zh) 2007-08-24
ECSP067000A (es) 2006-12-29
MXPA06012213A (es) 2007-01-17
CY1111292T1 (el) 2015-08-05
US8071577B2 (en) 2011-12-06
PT1740163E (pt) 2010-09-28
US20100173877A1 (en) 2010-07-08
IL178510A0 (en) 2007-02-11
SI1740163T1 (sl) 2010-11-30
NO20065292L (no) 2007-01-17
HRP20100513T4 (hr) 2020-10-02
PL1740163T5 (pl) 2020-10-05
PE20060308A1 (es) 2006-05-25
AR084229A2 (es) 2013-05-02
ES2348038T5 (es) 2020-09-14
CA2561839A1 (en) 2005-11-03
IL178510A (en) 2015-08-31
CN1946383A (zh) 2007-04-11
RS51434B2 (sr) 2020-11-30
GT200500093A (es) 2006-04-17
DE102004019743A1 (de) 2005-11-24
KR20060134168A (ko) 2006-12-27
ZA200609594B (en) 2008-04-30
RS51434B (sr) 2011-04-30
AU2005235418A1 (en) 2005-11-03
MY143669A (en) 2011-06-30
UY28863A1 (es) 2005-11-30
EA200601844A1 (ru) 2007-04-27
JP2007533681A (ja) 2007-11-22
ES2348038T3 (es) 2010-11-29
EA010313B1 (ru) 2008-08-29
DK1740163T4 (da) 2020-04-06
SV2006002090A (es) 2006-02-15
DE502005009904D1 (de) 2010-08-26
IL239861A0 (en) 2015-08-31
AU2005235418B2 (en) 2009-08-06
EP1740163B2 (de) 2020-01-15
HRP20100513T1 (hr) 2010-11-30
AU2005235418C1 (en) 2015-05-21
AR048830A1 (es) 2006-05-31
TWI351960B (en) 2011-11-11
JP4908399B2 (ja) 2012-04-04
SI1740163T2 (sl) 2020-04-30
EP1740163B1 (de) 2010-07-14
ATE473734T1 (de) 2010-07-15
UA83915C2 (ru) 2008-08-26
CN1946383B (zh) 2010-06-09
US20110124612A1 (en) 2011-05-26
ME01183B (me) 2013-03-20
EP1740163A2 (de) 2007-01-10
BRPI0510005A (pt) 2007-09-18
PA8630901A1 (es) 2006-05-16

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