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UA111147C2 - Способи та композиції для лікування або профілактики зовнішнього отиту - Google Patents

Способи та композиції для лікування або профілактики зовнішнього отиту

Info

Publication number
UA111147C2
UA111147C2 UAA201207023A UAA201207023A UA111147C2 UA 111147 C2 UA111147 C2 UA 111147C2 UA A201207023 A UAA201207023 A UA A201207023A UA A201207023 A UAA201207023 A UA A201207023A UA 111147 C2 UA111147 C2 UA 111147C2
Authority
UA
Ukraine
Prior art keywords
agents
composition
enhancing
auditory canal
viscosity
Prior art date
Application number
UAA201207023A
Other languages
English (en)
Inventor
Вільям Р. Кемпбелл
Ніл Е. Паулсен
Роналд Х. ДЖОНСОН
Дуглас І. Хеплер
Original Assignee
Байєр Б.В.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=43992011&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=UA111147(C2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Байєр Б.В. filed Critical Байєр Б.В.
Publication of UA111147C2 publication Critical patent/UA111147C2/uk

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/496Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/56Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/57Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone
    • A61K31/573Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone substituted in position 21, e.g. cortisone, dexamethasone, prednisone or aldosterone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K36/00Medicinal preparations of undetermined constitution containing material from algae, lichens, fungi or plants, or derivatives thereof, e.g. traditional herbal medicines
    • A61K36/18Magnoliophyta (angiosperms)
    • A61K36/185Magnoliopsida (dicotyledons)
    • A61K36/75Rutaceae (Rue family)
    • A61K36/752Citrus, e.g. lime, orange or lemon
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/08Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
    • A61K47/14Esters of carboxylic acids, e.g. fatty acid monoglycerides, medium-chain triglycerides, parabens or PEG fatty acid esters
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0019Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0046Ear
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/10Dispersions; Emulsions
    • A61K9/107Emulsions ; Emulsion preconcentrates; Micelles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/10Dispersions; Emulsions
    • A61K9/127Synthetic bilayered vehicles, e.g. liposomes or liposomes with cholesterol as the only non-phosphatidyl surfactant
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P23/00Anaesthetics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • A61P27/16Otologicals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10Antimycotics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Natural Medicines & Medicinal Plants (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Dispersion Chemistry (AREA)
  • Biotechnology (AREA)
  • Microbiology (AREA)
  • Mycology (AREA)
  • Medical Informatics (AREA)
  • Botany (AREA)
  • Alternative & Traditional Medicine (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Dermatology (AREA)
  • Rheumatology (AREA)
  • Anesthesiology (AREA)
  • Virology (AREA)
  • Pain & Pain Management (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

Abstract

Винахід належать до способу лікування або профілактики інфікування зовнішнього отиту та його наслідків шляхом місцевого введення фармацевтично прийнятної композиції в зовнішній слуховий прохід, де зазначена композиція не містить целюлоз, що підвищують в’язкість, або засобів, що підвищують в’язкість, вибраних з альгінової кислоти, желатину, карбомеру акації та цетостеарилового спирту, або адгезивних компонентів, і не є у формі гелю, і де зазначена композиція містить ліпідний носій, і принаймні два активні засоби, вибрані із групи, що складається з антибіотиків, протигрибкових засобів, антипаразитарних засобів, противірусних засобів, нестероїдних протизапальних засобів, знеболювальних засобів, анестетичних засобів і стероїдів, де ліпідний носій є ліпідною емульсією типу «масло у воді», ліпідною мікроемульсією або ліпідною везикулою, та де ліпіди вибирають з фосфоліпідів, які вибирають зі сполук фосфатидилу, що вибираються з фосфатидилгліцерину, фосфатидилінозитолу, фосфатидилхоліну, фосфоліпону 90Н, фосфатидилсерину, фосфатидилетаноламіну, сфінголіпідів, цереброзидів, гангліозидів, кардіоліпінів, трилінолеїнів, лецетину та церамідів, при цьому зазначений спосіб включає введення зазначеної композиції в зовнішній слуховий прохід однією дозою, достатньою для клінічного покращення або повного виліковування даного хворого стану.Також винахід належить до застосування заявленої композиції.
UAA201207023A 2009-11-11 2010-10-11 Способи та композиції для лікування або профілактики зовнішнього отиту UA111147C2 (uk)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US26030909P 2009-11-11 2009-11-11
PCT/US2010/056255 WO2011060083A1 (en) 2009-11-11 2010-11-10 Methods and compositions for rapid treatment of otitis externa

Publications (1)

Publication Number Publication Date
UA111147C2 true UA111147C2 (uk) 2016-04-11

Family

ID=43992011

Family Applications (1)

Application Number Title Priority Date Filing Date
UAA201207023A UA111147C2 (uk) 2009-11-11 2010-10-11 Способи та композиції для лікування або профілактики зовнішнього отиту

Country Status (29)

Country Link
US (1) US8927006B2 (uk)
EP (1) EP2498792B1 (uk)
JP (2) JP2013510861A (uk)
KR (2) KR101901083B1 (uk)
CN (1) CN102612372B (uk)
AU (1) AU2010319538B2 (uk)
BR (1) BR112012011017A2 (uk)
CA (1) CA2780160C (uk)
CL (1) CL2012001227A1 (uk)
CO (1) CO6540004A2 (uk)
DK (1) DK2498792T3 (uk)
EC (1) ECSP12011967A (uk)
ES (1) ES2645200T3 (uk)
HR (1) HRP20171520T1 (uk)
HU (1) HUE034617T2 (uk)
IL (1) IL219483A (uk)
LT (1) LT2498792T (uk)
MX (1) MX2012005521A (uk)
MY (1) MY162687A (uk)
NO (1) NO2498792T3 (uk)
NZ (1) NZ599559A (uk)
PH (1) PH12012500913A1 (uk)
PL (1) PL2498792T3 (uk)
PT (1) PT2498792T (uk)
RU (1) RU2680137C2 (uk)
SI (1) SI2498792T1 (uk)
UA (1) UA111147C2 (uk)
WO (1) WO2011060083A1 (uk)
ZA (1) ZA201203239B (uk)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2014036165A1 (en) * 2012-08-29 2014-03-06 Bayer Healthcare, Llc Aqueous based compositions for treating otitis externa
CN104337952A (zh) * 2013-08-10 2015-02-11 李谊 一种中西医结合治疗爆震性耳聋的组合药物
CN104739768A (zh) * 2013-12-27 2015-07-01 河南惠通天下生物工程有限公司 一种甲砜霉素纳米脂质体及其制备方法
EP3482744A1 (de) * 2017-11-14 2019-05-15 ProFem GmbH Emulsionen zur topischen behandlung urogenitaler und dermaler infektionen
IL274630B2 (en) * 2017-11-14 2025-05-01 Profem Gmbh Emulsions for treating mucosal infections
WO2021056106A1 (en) 2019-09-23 2021-04-01 Dds Research Inc. Lipid vesicle compositions with penetration enhancing agents
US11986483B2 (en) * 2019-10-11 2024-05-21 Dechra Veterinary Products, Llc Otic formulations, methods and devices
WO2022204305A2 (en) 2021-03-24 2022-09-29 Glo Pharma, Inc. Peptides and methods for reducing skin pigmentation
CN113876658B (zh) * 2021-11-01 2023-10-20 仙乐健康科技股份有限公司 水包油型乳液组合物及其制备方法

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EP0744939B1 (en) 1994-02-04 2002-09-25 Lipocore Holding AB Bilayer preparations made from digalactosyldiacylglycerol containing galactolipid
CA2201134A1 (en) * 1994-10-10 1996-04-18 Alfred Sallmann Ophthalmic and aural compositions containing diclofenac potassium
ZA964653B (en) * 1995-06-06 1996-12-12 Bayer Ag Non-irritation non-sensitizing non-ototoxic otic anti-bacterial compositions
IT1295369B1 (it) 1997-10-21 1999-05-12 Fatro Spa Composizione a base di tiamfenicolo e diclofenac
US6433024B1 (en) * 2000-05-08 2002-08-13 Karl F. Popp Topical anti-acne composition
AUPR798901A0 (en) * 2001-09-28 2001-10-25 Medvet Science Pty. Ltd. Spheroidal hdl particles with a defined phospholipid composition
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WO2004091578A2 (en) * 2003-04-09 2004-10-28 Biodelivery Sciences International, Inc. Novel encochleation methods, cochleates and methods of use
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US20090082337A1 (en) * 2007-09-21 2009-03-26 Srini Venkastesh Compositions Comprising Quinolone and Methods for Treating or Controlling Infections
US20090111780A1 (en) * 2007-10-31 2009-04-30 Everett Laboratories, Inc. Compositions and methods for treatment of ear canal infection and inflammation

Also Published As

Publication number Publication date
ECSP12011967A (es) 2012-08-31
ES2645200T3 (es) 2017-12-04
HRP20171520T1 (hr) 2017-11-17
CN102612372B (zh) 2016-01-20
JP6138891B2 (ja) 2017-05-31
RU2680137C2 (ru) 2019-02-18
ZA201203239B (en) 2013-07-31
IL219483A0 (en) 2012-06-28
NO2498792T3 (uk) 2017-12-30
IL219483A (en) 2017-12-31
MY162687A (en) 2017-07-14
US8927006B2 (en) 2015-01-06
CL2012001227A1 (es) 2012-08-24
EP2498792B1 (en) 2017-08-02
KR20120116398A (ko) 2012-10-22
DK2498792T3 (da) 2017-11-06
NZ599559A (en) 2014-08-29
AU2010319538B2 (en) 2015-04-09
CA2780160C (en) 2018-03-06
US20110281809A1 (en) 2011-11-17
MX2012005521A (es) 2012-06-19
CA2780160A1 (en) 2011-05-19
JP2016102112A (ja) 2016-06-02
HUE034617T2 (en) 2018-02-28
PH12012500913A1 (en) 2012-11-26
PL2498792T3 (pl) 2018-01-31
CO6540004A2 (es) 2012-10-16
WO2011060083A1 (en) 2011-05-19
PT2498792T (pt) 2017-10-18
EP2498792A1 (en) 2012-09-19
EP2498792A4 (en) 2013-06-12
AU2010319538A1 (en) 2012-05-17
BR112012011017A2 (pt) 2015-09-15
CN102612372A (zh) 2012-07-25
LT2498792T (lt) 2017-10-25
KR101901083B1 (ko) 2018-09-20
KR20170100680A (ko) 2017-09-04
SI2498792T1 (sl) 2017-11-30
JP2013510861A (ja) 2013-03-28
RU2012124067A (ru) 2013-12-20

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