TW202135816A - 以激酶抑制劑治療潰瘍性結腸炎 - Google Patents
以激酶抑制劑治療潰瘍性結腸炎 Download PDFInfo
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- TW202135816A TW202135816A TW109144272A TW109144272A TW202135816A TW 202135816 A TW202135816 A TW 202135816A TW 109144272 A TW109144272 A TW 109144272A TW 109144272 A TW109144272 A TW 109144272A TW 202135816 A TW202135816 A TW 202135816A
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- Prior art keywords
- pyrazol
- cyclobutane
- cyanomethyl
- pyrazolo
- pyridine
- Prior art date
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Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/4985—Pyrazines or piperazines ortho- or peri-condensed with heterocyclic ring systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
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- Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Chemical & Material Sciences (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201962949995P | 2019-12-18 | 2019-12-18 | |
| US62/949,995 | 2019-12-18 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| TW202135816A true TW202135816A (zh) | 2021-10-01 |
Family
ID=73856215
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| TW109144272A TW202135816A (zh) | 2019-12-18 | 2020-12-15 | 以激酶抑制劑治療潰瘍性結腸炎 |
Country Status (4)
| Country | Link |
|---|---|
| JP (1) | JP2021095402A (es) |
| AR (1) | AR120809A1 (es) |
| TW (1) | TW202135816A (es) |
| WO (1) | WO2021124095A1 (es) |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CR20180372A (es) * | 2016-02-24 | 2018-09-19 | Pfizer | Derivados de pirazolo [1,5-a] pirazin-4-ilo |
| US11254668B2 (en) * | 2017-08-14 | 2022-02-22 | Pfizer Inc. | Pyrazolo[1,5-A]pyrazin-4-yl and related derivatives |
-
2020
- 2020-12-15 TW TW109144272A patent/TW202135816A/zh unknown
- 2020-12-15 WO PCT/IB2020/061956 patent/WO2021124095A1/en not_active Ceased
- 2020-12-16 JP JP2020208048A patent/JP2021095402A/ja not_active Withdrawn
- 2020-12-17 AR ARP200103540A patent/AR120809A1/es not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| WO2021124095A1 (en) | 2021-06-24 |
| AR120809A1 (es) | 2022-03-23 |
| JP2021095402A (ja) | 2021-06-24 |
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