TW200626559A - Anilino-pyrimidine analogs - Google Patents
Anilino-pyrimidine analogsInfo
- Publication number
- TW200626559A TW200626559A TW094135620A TW94135620A TW200626559A TW 200626559 A TW200626559 A TW 200626559A TW 094135620 A TW094135620 A TW 094135620A TW 94135620 A TW94135620 A TW 94135620A TW 200626559 A TW200626559 A TW 200626559A
- Authority
- TW
- Taiwan
- Prior art keywords
- anilino
- pyrimidine analogs
- pyrimidine
- analogs
- compounds
- Prior art date
Links
- 150000008059 anilinopyrimidines Chemical class 0.000 title 1
- 150000001875 compounds Chemical class 0.000 abstract 1
Classifications
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- C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
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- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
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| US7122544B2 (en) | 2000-12-06 | 2006-10-17 | Signal Pharmaceuticals, Llc | Anilinopyrimidine derivatives as IKK inhibitors and compositions and methods related thereto |
| CN1307173C (zh) * | 2000-12-21 | 2007-03-28 | 葛兰素集团有限公司 | 作为血管生成调节剂的嘧啶胺 |
| US20020132823A1 (en) * | 2001-01-17 | 2002-09-19 | Jiahuai Han | Assay method |
| GB0103926D0 (en) * | 2001-02-17 | 2001-04-04 | Astrazeneca Ab | Chemical compounds |
| JP4309657B2 (ja) * | 2001-02-20 | 2009-08-05 | アストラゼネカ・アクチエボラーグ | Gsk−3関連障害の治療のための2−アリルアミノ−ピリミジン |
| WO2002079197A1 (en) * | 2001-03-29 | 2002-10-10 | Vertex Pharmaceuticals Incorporated | Inhibitors of c-jun n-terminal kinases (jnk) and other protein kinases |
| CA2443234A1 (en) * | 2001-04-10 | 2002-10-24 | Vertex Pharmaceuticals Incorporated | Isoxaxole derivatives as inhibitors of src and other protein kinases |
| MXPA03009378A (es) * | 2001-04-13 | 2004-01-29 | Vertex Pharma | Inhibidores de cinasas c-jun n-terminales (jnk) y otras proteinas cinasas. |
| JP4316893B2 (ja) * | 2001-05-16 | 2009-08-19 | バーテックス ファーマシューティカルズ インコーポレイテッド | Srcおよび他のプロテインキナーゼのインヒビター |
| DE50213202D1 (de) * | 2001-05-29 | 2009-02-26 | Bayer Schering Pharma Ag | Cdk inhibitorische pyrimidine, deren herstellung und verwendung als arzneimittel |
| WO2002096905A1 (en) | 2001-06-01 | 2002-12-05 | Vertex Pharmaceuticals Incorporated | Thiazole compounds useful as inhibitors of protein kinases |
| EP1399440B1 (en) * | 2001-06-15 | 2009-06-03 | Vertex Pharmaceuticals Incorporated | 5-(2-aminopyrimidin-4-yl)benzisoxazoles as protein kinase inhibitors |
| US6939874B2 (en) * | 2001-08-22 | 2005-09-06 | Amgen Inc. | Substituted pyrimidinyl derivatives and methods of use |
| US6703414B2 (en) | 2001-09-14 | 2004-03-09 | Arizona Board Of Regents On Behalf Of The University Of Arizona | Device and method for treating restenosis |
| CA2476281A1 (en) * | 2002-02-08 | 2003-08-14 | Smithkline Beecham Corporation | Pyrimidine compounds |
| ATE365165T1 (de) * | 2002-03-01 | 2007-07-15 | Smithkline Beecham Corp | Diaminopyrimidine und deren verwendung als angiogenesehemmer |
| WO2003076434A1 (en) | 2002-03-09 | 2003-09-18 | Astrazeneca Ab | 4- imidazolyl substuited pyrimidine derivatives with cdk inhibitiory activity |
| GB0215844D0 (en) * | 2002-07-09 | 2002-08-14 | Novartis Ag | Organic compounds |
| CA2506772A1 (en) * | 2002-11-01 | 2004-05-21 | Vertex Pharmaceuticals Incorporated | Compositions useful as inhibitors of jak and other protein kinases |
| US7348335B2 (en) * | 2002-11-05 | 2008-03-25 | Vertex Pharmaceuticals Incorporated | Compositions useful as inhibitors of JAK and other protein kinases |
| GB0226582D0 (en) * | 2002-11-14 | 2002-12-18 | Cyclacel Ltd | Anti-viral compounds |
| GB0226583D0 (en) * | 2002-11-14 | 2002-12-18 | Cyclacel Ltd | Compounds |
-
2005
- 2005-10-13 RU RU2007114080/04A patent/RU2007114080A/ru not_active Application Discontinuation
- 2005-10-13 KR KR1020077010445A patent/KR20070084067A/ko not_active Withdrawn
- 2005-10-13 CA CA002580913A patent/CA2580913A1/en not_active Abandoned
- 2005-10-13 AR ARP050104293A patent/AR051387A1/es not_active Application Discontinuation
- 2005-10-13 PE PE2005001207A patent/PE20060582A1/es not_active Application Discontinuation
- 2005-10-13 CN CNA2005800349350A patent/CN101039919A/zh not_active Withdrawn
- 2005-10-13 MX MX2007004488A patent/MX2007004488A/es unknown
- 2005-10-13 TW TW094135620A patent/TW200626559A/zh unknown
- 2005-10-13 EP EP05812654A patent/EP1799652A1/en not_active Withdrawn
- 2005-10-13 GT GT200500286A patent/GT200500286A/es unknown
- 2005-10-13 AU AU2005295788A patent/AU2005295788A1/en not_active Abandoned
- 2005-10-13 US US11/248,495 patent/US7799915B2/en not_active Expired - Fee Related
- 2005-10-13 PA PA20058649401A patent/PA8649401A1/es unknown
- 2005-10-13 JP JP2007536838A patent/JP2008515986A/ja active Pending
- 2005-10-13 BR BRPI0516597-0A patent/BRPI0516597A/pt not_active IP Right Cessation
- 2005-10-13 WO PCT/US2005/036674 patent/WO2006044457A1/en not_active Ceased
-
2007
- 2007-03-28 NO NO20071642A patent/NO20071642L/no not_active Application Discontinuation
- 2007-03-29 IL IL182316A patent/IL182316A0/en unknown
- 2007-04-11 CR CR9048A patent/CR9048A/es unknown
- 2007-04-12 ZA ZA200703022A patent/ZA200703022B/xx unknown
Also Published As
| Publication number | Publication date |
|---|---|
| AU2005295788A1 (en) | 2006-04-27 |
| EP1799652A1 (en) | 2007-06-27 |
| IL182316A0 (en) | 2007-07-24 |
| US7799915B2 (en) | 2010-09-21 |
| WO2006044457A1 (en) | 2006-04-27 |
| PE20060582A1 (es) | 2006-08-17 |
| RU2007114080A (ru) | 2008-11-27 |
| US20060079543A1 (en) | 2006-04-13 |
| GT200500286A (es) | 2006-06-13 |
| ZA200703022B (en) | 2009-04-29 |
| AR051387A1 (es) | 2007-01-10 |
| PA8649401A1 (es) | 2006-09-22 |
| BRPI0516597A (pt) | 2008-09-16 |
| CN101039919A (zh) | 2007-09-19 |
| NO20071642L (no) | 2007-06-01 |
| MX2007004488A (es) | 2007-09-11 |
| CR9048A (es) | 2007-08-28 |
| KR20070084067A (ko) | 2007-08-24 |
| CA2580913A1 (en) | 2006-04-27 |
| JP2008515986A (ja) | 2008-05-15 |
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