TW200407123A - Combinations of atorvastatin and α1 adrenergic receptor antagonists - Google Patents

Combinations of atorvastatin and α1 adrenergic receptor antagonists Download PDF

Info

Publication number: TW200407123A
Authority: TW; Taiwan
Prior art keywords: pharmaceutically acceptable; acceptable derivative; bph; atovastatin; patent application
Prior art date: 2002-09-17

Application number

TW092125472A

Other languages

English (en)

Chinese (zh)

Inventor

Nicholas Pullen

Richard James Thurlow

Original Assignee

Pfizer

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2002-09-17

Filing date

2003-09-16

Publication date

2004-05-16

2003-09-16 Application filed by Pfizer filed Critical Pfizer

2004-05-16 Publication of TW200407123A publication Critical patent/TW200407123A/zh

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XUKUURHRXDUEBC-KAYWLYCHSA-N Atorvastatin Chemical compound C=1C=CC=CC=1C1=C(C=2C=CC(F)=CC=2)N(CC[C@@H](O)C[C@@H](O)CC(O)=O)C(C(C)C)=C1C(=O)NC1=CC=CC=C1 XUKUURHRXDUEBC-KAYWLYCHSA-N 0.000 title abstract description 4
XUKUURHRXDUEBC-UHFFFAOYSA-N Atorvastatin Natural products C=1C=CC=CC=1C1=C(C=2C=CC(F)=CC=2)N(CCC(O)CC(O)CC(O)=O)C(C(C)C)=C1C(=O)NC1=CC=CC=C1 XUKUURHRXDUEBC-UHFFFAOYSA-N 0.000 title abstract description 4
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Classifications

- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/517—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with carbocyclic ring systems, e.g. quinazoline, perimidine
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system

Landscapes

Health & Medical Sciences (AREA)
Veterinary Medicine (AREA)
Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Epidemiology (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Urology & Nephrology (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Organic Chemistry (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Pyrrole Compounds (AREA)

TW092125472A 2002-09-17 2003-09-16 Combinations of atorvastatin and α1 adrenergic receptor antagonists TW200407123A (en)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
GBGB0221579.6A GB0221579D0 (en)	2002-09-17	2002-09-17	Combinations of atorvastatin and, adrenergic receptor antagonists

Publications (1)

Publication Number	Publication Date
TW200407123A true TW200407123A (en)	2004-05-16

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EP (1)	EP1542677A1 (fr)
CN (1)	CN1681492A (fr)
AU (1)	AU2003263420A1 (fr)
BR (1)	BR0314388A (fr)
CA (1)	CA2498894A1 (fr)
GB (1)	GB0221579D0 (fr)
PL (1)	PL374656A1 (fr)
TW (1)	TW200407123A (fr)
WO (1)	WO2004026300A1 (fr)
ZA (1)	ZA200502225B (fr)

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* Cited by examiner, † Cited by third party
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CN100418529C (zh) *	2006-06-30	2008-09-17	南京美瑞制药有限公司	萘哌地尔在制备促进泌尿系统结石排出的药物中的应用

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IT1238011B (it) *	1989-12-13	1993-06-21	Pulitzer Italiana	Composizioni farmaceutiche a base di inibitori della riduttasi del hmg-coa per il trattamento della ipertrofia prostatica benigna.
GB9700504D0 (en) *	1997-01-11	1997-02-26	Pfizer Ltd	Pharmaceutical compounds
GT199800126A (es) *	1997-08-29	2000-01-29		Terapia de combinacion.
US6534537B2 (en) *	2000-01-07	2003-03-18	Kenneth Weisman	Use of HMG-COA reductase inhibitors to prevent and treat BPH
GB0206033D0 (en) *	2002-03-14	2002-04-24	Pfizer Ltd	Compounds useful in therapy

2002
- 2002-09-17 GB GBGB0221579.6A patent/GB0221579D0/en not_active Ceased
2003
- 2003-09-05 CA CA002498894A patent/CA2498894A1/fr not_active Abandoned
- 2003-09-05 PL PL03374656A patent/PL374656A1/xx not_active Application Discontinuation
- 2003-09-05 EP EP03797447A patent/EP1542677A1/fr not_active Withdrawn
- 2003-09-05 WO PCT/IB2003/003940 patent/WO2004026300A1/fr not_active Ceased
- 2003-09-05 CN CNA038217864A patent/CN1681492A/zh active Pending
- 2003-09-05 AU AU2003263420A patent/AU2003263420A1/en not_active Abandoned
- 2003-09-05 BR BR0314388-0A patent/BR0314388A/pt not_active Application Discontinuation
- 2003-09-16 TW TW092125472A patent/TW200407123A/zh unknown
2005
- 2005-03-16 ZA ZA200502225A patent/ZA200502225B/en unknown

Also Published As

Publication number	Publication date
WO2004026300A1 (fr)	2004-04-01
AU2003263420A1 (en)	2004-04-08
CA2498894A1 (fr)	2004-04-01
EP1542677A1 (fr)	2005-06-22
GB0221579D0 (en)	2002-10-23
ZA200502225B (en)	2006-02-22
CN1681492A (zh)	2005-10-12
PL374656A1 (en)	2005-10-31
BR0314388A (pt)	2005-07-19

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