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TR200001530T2 - Gastrik asit salgılamasının önlenmesi için heterosiklik bileşimler - Google Patents

Gastrik asit salgılamasının önlenmesi için heterosiklik bileşimler

Info

Publication number
TR200001530T2
TR200001530T2 TR2000/01530T TR200001530T TR200001530T2 TR 200001530 T2 TR200001530 T2 TR 200001530T2 TR 2000/01530 T TR2000/01530 T TR 2000/01530T TR 200001530 T TR200001530 T TR 200001530T TR 200001530 T2 TR200001530 T2 TR 200001530T2
Authority
TR
Turkey
Prior art keywords
gastric acid
acid secretion
prevent gastric
heterocyclic compositions
heterocyclic
Prior art date
Application number
TR2000/01530T
Other languages
English (en)
Inventor
Amin Kostrat
Dahlstr�m Mikael
Nordberg Peter
Starke Ingemar
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Publication of TR200001530T2 publication Critical patent/TR200001530T2/tr

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

Mevcut bulus, egzojen ve endojen olarak stimüle edilmis gastrik asit salgilanmasini önleyen ve böylece gastrointestinal iltihapli hastaliklarin önlenmesi ve tedavisinde kullanilabilen formül (I)'in heteosiklik bilesimleri ile ilgilidir, burada fenil parçaci 2- e 6- pozisyonunda düsük alkil ile ikame edilir.
TR2000/01530T 1997-11-28 1998-11-18 Gastrik asit salgılamasının önlenmesi için heterosiklik bileşimler TR200001530T2 (tr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
SE9704404A SE9704404D0 (sv) 1997-11-28 1997-11-28 New compounds

Publications (1)

Publication Number Publication Date
TR200001530T2 true TR200001530T2 (tr) 2000-11-21

Family

ID=20409181

Family Applications (1)

Application Number Title Priority Date Filing Date
TR2000/01530T TR200001530T2 (tr) 1997-11-28 1998-11-18 Gastrik asit salgılamasının önlenmesi için heterosiklik bileşimler

Country Status (32)

Country Link
US (1) US6518270B1 (tr)
EP (1) EP1042324B1 (tr)
JP (1) JP2001525322A (tr)
KR (1) KR20010032559A (tr)
CN (1) CN1142933C (tr)
AR (1) AR016972A1 (tr)
AT (1) ATE233263T1 (tr)
AU (1) AU752187C (tr)
BR (1) BR9814755A (tr)
CA (1) CA2311798A1 (tr)
CZ (1) CZ292349B6 (tr)
DE (1) DE69811735T2 (tr)
DK (1) DK1042324T3 (tr)
EE (1) EE04060B1 (tr)
ES (1) ES2191356T3 (tr)
HU (1) HUP0100601A3 (tr)
ID (1) ID24730A (tr)
IL (1) IL136145A0 (tr)
IS (1) IS5486A (tr)
MY (1) MY121032A (tr)
NO (1) NO315704B1 (tr)
NZ (1) NZ504355A (tr)
PL (1) PL340920A1 (tr)
PT (1) PT1042324E (tr)
RU (1) RU2241000C2 (tr)
SE (1) SE9704404D0 (tr)
SK (1) SK283904B6 (tr)
TR (1) TR200001530T2 (tr)
TW (1) TW515798B (tr)
UA (1) UA70932C2 (tr)
WO (1) WO1999028322A1 (tr)
ZA (1) ZA9810468B (tr)

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EP1805177B9 (en) * 2004-09-03 2010-09-15 Yuhan Corporation Pyrrolo[3,2-c]pyridine derivatives and process for the preparation thereof
US7642269B2 (en) 2004-09-03 2010-01-05 Yuhan Corporation Pyrrolo[3,2-B]pyridine derivatives and processes for the preparation thereof
ES2367312T3 (es) * 2004-09-03 2011-11-02 Yuhan Corporation DERIVADOS DE PIRROLO [3,2-c] PIRIDINA Y PROCESOS PARA LA PREPARACIÓN DE LOS MISMOS.
US7777040B2 (en) 2005-05-03 2010-08-17 Cgi Pharmaceuticals, Inc. Certain substituted ureas, as modulators of kinase activity
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US20090156578A1 (en) * 2005-12-05 2009-06-18 PAULS Henry 3-Heterocyclylacrylamide Compounds as Fab I Inhibitors and Antibacterial Agents
JP2009539840A (ja) 2006-06-06 2009-11-19 シェーリング コーポレイション プロテインキナーゼ阻害剤としてのイミダゾピラジン
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Also Published As

Publication number Publication date
PT1042324E (pt) 2003-06-30
AR016972A1 (es) 2001-08-01
AU1356599A (en) 1999-06-16
AU752187C (en) 2003-09-18
KR20010032559A (ko) 2001-04-25
ZA9810468B (en) 1999-05-21
DK1042324T3 (da) 2003-05-05
ID24730A (id) 2000-08-03
EP1042324A1 (en) 2000-10-11
HUP0100601A3 (en) 2002-10-28
RU2241000C2 (ru) 2004-11-27
AU752187B2 (en) 2002-09-12
IL136145A0 (en) 2001-05-20
NZ504355A (en) 2001-12-21
HK1030216A1 (en) 2001-04-27
US6518270B1 (en) 2003-02-11
MY121032A (en) 2005-12-30
EE04060B1 (et) 2003-06-16
EP1042324B1 (en) 2003-02-26
ATE233263T1 (de) 2003-03-15
WO1999028322A1 (en) 1999-06-10
CA2311798A1 (en) 1999-06-10
CZ292349B6 (cs) 2003-09-17
DE69811735T2 (de) 2003-12-18
SK283904B6 (sk) 2004-04-06
NO20002721L (no) 2000-07-28
TW515798B (en) 2003-01-01
HUP0100601A2 (hu) 2001-09-28
UA70932C2 (uk) 2004-11-15
CN1142933C (zh) 2004-03-24
EE200000315A (et) 2001-10-15
SE9704404D0 (sv) 1997-11-28
SK6742000A3 (en) 2001-03-12
CN1284078A (zh) 2001-02-14
NO20002721D0 (no) 2000-05-26
CZ20001947A3 (cs) 2000-11-15
ES2191356T3 (es) 2003-09-01
PL340920A1 (en) 2001-03-12
DE69811735D1 (de) 2003-04-03
BR9814755A (pt) 2000-10-03
NO315704B1 (no) 2003-10-13
IS5486A (is) 2000-05-10
JP2001525322A (ja) 2001-12-11

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