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TNSN97010A1 - Cyclopentanopyridyl-oxazolidinones contenant des heteroatomes. - Google Patents

Cyclopentanopyridyl-oxazolidinones contenant des heteroatomes.

Info

Publication number
TNSN97010A1
TNSN97010A1 TNTNSN97010A TNSN97010A TNSN97010A1 TN SN97010 A1 TNSN97010 A1 TN SN97010A1 TN TNSN97010 A TNTNSN97010 A TN TNSN97010A TN SN97010 A TNSN97010 A TN SN97010A TN SN97010 A1 TNSN97010 A1 TN SN97010A1
Authority
TN
Tunisia
Prior art keywords
cyclopentanopyridyl
heteroatomes
oxazolidinones containing
oxazolidinones
drugs
Prior art date
Application number
TNTNSN97010A
Other languages
English (en)
Inventor
Bernd Riedl Dr
Dieter Habich Dr
Andreas Stolle Dr
Martin Ruppelt Dr
Stephan Bartel Dr
Walter Guarnieri Dr
Rainer Endermann Dr
Hein Peter Kroll Dr
Hanno Wild Dr
Original Assignee
Bayer Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Ag filed Critical Bayer Ag
Publication of TNSN97010A1 publication Critical patent/TNSN97010A1/fr

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/6561—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing systems of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring or ring system, with or without other non-condensed hetero rings
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Biochemistry (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Molecular Biology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)

Abstract

LA PRESENTE INVENTION CONCERNE DES CYCLOPENTANOPYRIDYL- OXAZOLIDINONES CONTENANT DES HETEROATOMES, DES PROCEDES POUR LEUR PREPARATION ET LEUR UTILISATION COMME MEDICAMENTS, EN PARTICULIER COMME MEDICAMENTS ANTIBACTERIENS.
TNTNSN97010A 1996-01-18 1997-01-15 Cyclopentanopyridyl-oxazolidinones contenant des heteroatomes. TNSN97010A1 (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19601627A DE19601627A1 (de) 1996-01-18 1996-01-18 Heteroatomhaltige Cyclopentanopyridyl-Oxazolidinone

Publications (1)

Publication Number Publication Date
TNSN97010A1 true TNSN97010A1 (fr) 2005-03-15

Family

ID=7783042

Family Applications (1)

Application Number Title Priority Date Filing Date
TNTNSN97010A TNSN97010A1 (fr) 1996-01-18 1997-01-15 Cyclopentanopyridyl-oxazolidinones contenant des heteroatomes.

Country Status (21)

Country Link
US (1) US5869659A (fr)
EP (1) EP0785201A1 (fr)
JP (1) JPH09202787A (fr)
KR (1) KR970059170A (fr)
AU (1) AU1012397A (fr)
BG (1) BG101139A (fr)
BR (1) BR9700716A (fr)
CA (1) CA2195177A1 (fr)
CZ (1) CZ15897A3 (fr)
DE (1) DE19601627A1 (fr)
EE (1) EE9700020A (fr)
HU (1) HU9700152D0 (fr)
IL (1) IL120016A0 (fr)
MA (1) MA24062A1 (fr)
NO (1) NO970210L (fr)
PL (1) PL317985A1 (fr)
SG (1) SG50001A1 (fr)
SK (1) SK6997A3 (fr)
TN (1) TNSN97010A1 (fr)
TR (1) TR199700039A2 (fr)
ZA (1) ZA97393B (fr)

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US8110578B2 (en) 2008-10-27 2012-02-07 Signal Pharmaceuticals, Llc Pyrazino[2,3-b]pyrazine mTOR kinase inhibitors for oncology indications and diseases associated with the mTOR/PI3K/Akt pathway
EP2493472B1 (fr) 2009-10-26 2016-12-07 Signal Pharmaceuticals, LLC Procédés de synthèse et de purification de composés hétéroaryles
EA034512B1 (ru) 2011-10-19 2020-02-14 СИГНАЛ ФАРМАСЬЮТИКАЛЗ, ЭлЭлСи Лечение злокачественной опухоли ингибиторами tor-киназы
SG10201604558SA (en) 2011-12-02 2016-07-28 Signal Pharm Llc Pharmaceutical compositions of 7-(6-(2-hydroxypropan-2-yl)pyridin-3-yl)-1-((trans)-4 methoxycyclohexyl)-3,4-dihydropyrazino [2,3-b]pyrazin-2(1h)-one, a solid form thereof and methods of their use
MY174308A (en) 2012-02-24 2020-04-06 Signal Pharm Llc Methods for treating non-small cell lung using tor kinase inhibitor combination therapy
AU2013203714B2 (en) 2012-10-18 2015-12-03 Signal Pharmaceuticals, Llc Inhibition of phosphorylation of PRAS40, GSK3-beta or P70S6K1 as a marker for TOR kinase inhibitory activity
EP3202403A1 (fr) 2013-01-16 2017-08-09 Signal Pharmaceuticals, LLC Composés de pyrrolopyrimidine substitués, leurs compositions et procédés de traitement
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WO2015160882A1 (fr) 2014-04-16 2015-10-22 Signal Pharmaceuticals, Llc Formes solides comprenant de la 7-(6- (2-hydroxypropan-2-yl) pyridin-3-yl)-1-(trans)-4-méthoxycyclohexyl)-3, 4-dihydropyrazino[2,3-b] pyrazin-2(1h)-one, et un co-formeur, leurs compositions et leurs procédés d'utilisation
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Also Published As

Publication number Publication date
DE19601627A1 (de) 1997-07-24
TR199700039A2 (tr) 1997-08-21
BR9700716A (pt) 1998-10-06
MA24062A1 (fr) 1997-10-01
ZA97393B (en) 1997-07-17
JPH09202787A (ja) 1997-08-05
HU9700152D0 (en) 1997-03-28
KR970059170A (ko) 1997-08-12
IL120016A0 (en) 1997-04-15
CA2195177A1 (fr) 1997-07-19
CZ15897A3 (en) 1997-08-13
MX9700388A (es) 1997-07-31
PL317985A1 (en) 1997-07-21
US5869659A (en) 1999-02-09
SG50001A1 (en) 1998-06-15
EE9700020A (et) 1997-08-15
BG101139A (en) 1998-04-30
AU1012397A (en) 1997-07-24
NO970210L (no) 1997-07-21
NO970210D0 (no) 1997-01-17
EP0785201A1 (fr) 1997-07-23
SK6997A3 (en) 1997-09-10

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