[go: up one dir, main page]

TN2010000011A1 - Improved pharmaceutical composition containing dihydropyridine calcium channel antagonist and method for the preparation thereof - Google Patents

Improved pharmaceutical composition containing dihydropyridine calcium channel antagonist and method for the preparation thereof

Info

Publication number
TN2010000011A1
TN2010000011A1 TNP2010000011A TN2010000011A TN2010000011A1 TN 2010000011 A1 TN2010000011 A1 TN 2010000011A1 TN P2010000011 A TNP2010000011 A TN P2010000011A TN 2010000011 A TN2010000011 A TN 2010000011A TN 2010000011 A1 TN2010000011 A1 TN 2010000011A1
Authority
TN
Tunisia
Prior art keywords
preparation
calcium channel
channel antagonist
pharmaceutical composition
composition containing
Prior art date
Application number
TNP2010000011A
Other languages
English (en)
Inventor
Evangelos Karavas
Makis Koutris
Vicky Samara
Christina Matsingou
Athina Iliopoulou
Original Assignee
Pharmathen Sa
Recordati Ireland Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=39223083&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=TN2010000011(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Pharmathen Sa, Recordati Ireland Ltd filed Critical Pharmathen Sa
Publication of TN2010000011A1 publication Critical patent/TN2010000011A1/fr

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2009Inorganic compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/44221,4-Dihydropyridines, e.g. nifedipine, nicardipine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2072Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
    • A61K9/2077Tablets comprising drug-containing microparticles in a substantial amount of supporting matrix; Multiparticulate tablets

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Epidemiology (AREA)
  • Vascular Medicine (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Urology & Nephrology (AREA)
  • Inorganic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Hydrogenated Pyridines (AREA)
TNP2010000011A 2007-07-23 2010-01-08 Improved pharmaceutical composition containing dihydropyridine calcium channel antagonist and method for the preparation thereof TN2010000011A1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
PCT/EP2007/006517 WO2009012791A1 (fr) 2007-07-23 2007-07-23 Composition pharmaceutique contenant un antagoniste des canaux calciques de type dihydropyridine et son procédé de préparation
PCT/EP2008/059645 WO2009013306A1 (fr) 2007-07-23 2008-07-23 Composition pharmaceutique améliorée contenant un antagoniste de canal calcique de dihydropyridine et son procédé de préparation

Publications (1)

Publication Number Publication Date
TN2010000011A1 true TN2010000011A1 (en) 2011-09-26

Family

ID=39223083

Family Applications (2)

Application Number Title Priority Date Filing Date
TNP2010000011A TN2010000011A1 (en) 2007-07-23 2010-01-08 Improved pharmaceutical composition containing dihydropyridine calcium channel antagonist and method for the preparation thereof
TNP2010000022A TN2010000022A1 (en) 2007-07-23 2010-01-13 Pharmaceutical composition containing dihydropyridine calcium channel antagonist and method for the preparation thereof

Family Applications After (1)

Application Number Title Priority Date Filing Date
TNP2010000022A TN2010000022A1 (en) 2007-07-23 2010-01-13 Pharmaceutical composition containing dihydropyridine calcium channel antagonist and method for the preparation thereof

Country Status (20)

Country Link
EP (2) EP2180883B1 (fr)
JP (2) JP5769963B2 (fr)
KR (2) KR101632079B1 (fr)
CN (3) CN101784260A (fr)
AU (2) AU2007356942B2 (fr)
BR (2) BRPI0721883A2 (fr)
CA (2) CA2691752C (fr)
CO (1) CO6290639A2 (fr)
CR (1) CR11285A (fr)
EA (2) EA021645B1 (fr)
EC (1) ECSP109984A (fr)
ES (2) ES2622495T3 (fr)
MA (1) MA31684B1 (fr)
MX (2) MX2010000856A (fr)
MY (1) MY153857A (fr)
NZ (2) NZ582648A (fr)
TN (2) TN2010000011A1 (fr)
UA (2) UA97161C2 (fr)
WO (2) WO2009012791A1 (fr)
ZA (2) ZA201000586B (fr)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2008063888A2 (fr) 2006-11-22 2008-05-29 Plexxikon, Inc. Composés modulant l'activité de c-fms et/ou de c-kit et utilisations associées
MX2010000617A (es) 2007-07-17 2010-05-17 Plexxikon Inc Compuestos y metodos para modulacion de cinasa, e indicaciones de estos.
UA97161C2 (ru) * 2007-07-23 2012-01-10 Фарматен С.А. Фармацевтическая композиция, которая содержит дигидропиридиновый антагонист кальциевого канала лерканидипин и коллоидный диоксид кремния, способ ее приготовления
AU2010232670B2 (en) 2009-04-03 2015-07-09 F. Hoffmann-La Roche Ag Propane- I-sulfonic acid {3- [5- (4 -chloro-phenyl) -1H-pyrrolo [2, 3-b] pyridine-3-carbonyl] -2, 4-difluoro-pheny l } -amide compositions and uses thereof
US8329724B2 (en) 2009-08-03 2012-12-11 Hoffmann-La Roche Inc. Process for the manufacture of pharmaceutically active compounds
MA33975B1 (fr) 2009-11-06 2013-02-01 Plexxikon Inc Composés et méthodes de modulation des kinases et leurs indications d'emploi
HUE040136T2 (hu) 2011-02-07 2019-02-28 Plexxikon Inc Vegyületek és eljárások kináz modulációra és azok indikációi
TWI558702B (zh) 2011-02-21 2016-11-21 普雷辛肯公司 醫藥活性物質的固態形式
US9150570B2 (en) 2012-05-31 2015-10-06 Plexxikon Inc. Synthesis of heterocyclic compounds
JP2015537029A (ja) 2012-11-14 2015-12-24 ダブリュー・アール・グレース・アンド・カンパニー−コーンW R Grace & Co−Conn 生物学的に活性な物質及び不規則性無機酸化物を含有する組成物
GR1008554B (el) * 2014-06-12 2015-09-03 ΦΑΡΜΑΤΕΝ ΑΝΩΝΥΜΟΣ ΒΙΟΜΗΧΑΝΙΚΗ ΚΑΙ ΕΜΠΟΡΙΚΗ ΕΤΑΙΡΕΙΑ ΦΑΡΜΑΚΕΥΤΙΚΩΝ ΙΑΤΡΙΚΩΝ ΚΑΙ ΚΑΛΛΥΝΤΙΚΩΝ ΠΡΟΪΟΝΤΩΝ με δ.τ. ΦΑΡΜΑΤΕΝ, Φαρμακευτικο σκευασμα περιεχον εναν αντιμυκητιασικο παραγοντα τριaζολης και μεθοδος για την παρασκευη αυτου
CN104069500A (zh) * 2014-06-20 2014-10-01 湖南天地恒一制药有限公司 一种包含乐卡地平的药物组合物
CN105168165B (zh) * 2015-08-28 2018-06-26 江苏福邦药业有限公司 一种盐酸乐卡地平片及其制备方法
WO2018004379A1 (fr) * 2016-07-01 2018-01-04 Общество С Ограниченной Ответственностью "Гиостин" Produit sous forme de capsule pour traiter des maladies d'articulations
AU2019225236B2 (en) 2018-02-26 2025-01-30 R.P. Scherer Technologies, Llc Pharmaceutical dosage form for an emulsion of simethicone and loperamide
EA202092186A1 (ru) 2018-03-22 2020-12-16 Комифарм Интернэшнл Австралия Пти Лтд Фармацевтическая композиция, содержащая метаарсенит, и способ изготовления
CN114533686B (zh) * 2022-02-15 2023-10-20 湖南普道医药技术有限公司 一种二氢吡啶类药物的口服固体制剂及其制备方法
KR20240040407A (ko) * 2022-09-21 2024-03-28 주식회사 종근당 사쿠비트릴ㆍ발사르탄 칼슘염을 포함하는 약제학적 조성물

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3720757A1 (de) * 1987-06-24 1989-01-05 Bayer Ag Dhp-manteltablette
US5209933A (en) * 1990-01-10 1993-05-11 Syntex (U.S.A.) Inc. Long acting calcium channel blocker composition
GB9025251D0 (en) * 1990-11-20 1991-01-02 Solomon Montague C Nifedipine dosage forms
BR9903490A (pt) * 1998-12-15 2000-09-26 Oscar Gold Processo para a preparação de composições farmacêuticas de liberação programada contendo nimodipine, que permitem a liberação gradual e a manuntenção da ação terapeutica
DE19944803A1 (de) * 1999-09-20 2001-03-29 Bayer Ag Kombination von Dihydropyridinverbindungen und HMG-CoA-Reduktase-Inhibitoren und ihre Verwendung in Arzneimitteln
US20040185097A1 (en) * 2003-01-31 2004-09-23 Glenmark Pharmaceuticals Ltd. Controlled release modifying complex and pharmaceutical compositions thereof
WO2005053689A2 (fr) * 2003-12-01 2005-06-16 Lifecycle Pharma A/S Compositions pharmaceutiques comprenant de la lercanidipine
CN1901888A (zh) * 2003-12-01 2007-01-24 生命周斯药物公司 包含乐卡地平的药物组合物
EP2063872B2 (fr) * 2006-08-30 2019-12-04 Jagotec AG Formulations posologiques à libération contrôlée administrées par voie orale comprenant un noyau et une ou plusieurs couches barrières
EP2101771A2 (fr) * 2006-12-06 2009-09-23 Torrent Pharmaceuticals Ltd Formulation stable de lercanidipine
UA97161C2 (ru) * 2007-07-23 2012-01-10 Фарматен С.А. Фармацевтическая композиция, которая содержит дигидропиридиновый антагонист кальциевого канала лерканидипин и коллоидный диоксид кремния, способ ее приготовления

Also Published As

Publication number Publication date
KR20100047848A (ko) 2010-05-10
CA2691752A1 (fr) 2009-01-29
AU2008280106B2 (en) 2014-03-20
ES2622495T3 (es) 2017-07-06
EA019614B1 (ru) 2014-05-30
NZ582690A (en) 2011-12-22
WO2009012791A1 (fr) 2009-01-29
AU2008280106A1 (en) 2009-01-29
NZ582648A (en) 2012-06-29
JP5769963B2 (ja) 2015-08-26
MX2010000801A (es) 2010-07-05
CN103976968A (zh) 2014-08-13
TN2010000022A1 (en) 2011-09-26
EA201000220A1 (ru) 2010-08-30
BRPI0721883A2 (pt) 2014-02-18
UA97161C2 (ru) 2012-01-10
EP2170295A1 (fr) 2010-04-07
JP2010534211A (ja) 2010-11-04
KR101512404B1 (ko) 2015-04-21
UA99136C2 (ru) 2012-07-25
KR101632079B1 (ko) 2016-06-20
CA2693233A1 (fr) 2009-01-29
AU2007356942B2 (en) 2011-12-15
CA2691752C (fr) 2016-01-26
MA31684B1 (fr) 2010-09-01
MY153857A (en) 2015-03-31
EP2180883A1 (fr) 2010-05-05
EA201070160A1 (ru) 2010-06-30
CR11285A (es) 2010-04-27
AU2008280106B9 (en) 2014-08-07
AU2007356942A1 (en) 2009-01-29
CN101801347A (zh) 2010-08-11
BRPI0814666A2 (pt) 2017-05-09
MX2010000856A (es) 2010-04-30
ECSP109984A (es) 2010-04-30
ES2537063T3 (es) 2015-06-02
JP2010534220A (ja) 2010-11-04
ZA201000586B (en) 2011-03-30
CN101784260A (zh) 2010-07-21
EP2180883B1 (fr) 2017-01-11
EP2170295B1 (fr) 2015-04-22
KR20100045456A (ko) 2010-05-03
EA021645B1 (ru) 2015-08-31
CO6290639A2 (es) 2011-06-20
WO2009013306A1 (fr) 2009-01-29
AU2008280106A2 (en) 2010-02-25
ZA201001176B (en) 2010-11-24

Similar Documents

Publication Publication Date Title
TN2010000011A1 (en) Improved pharmaceutical composition containing dihydropyridine calcium channel antagonist and method for the preparation thereof
WO2010065709A3 (fr) Dérivés d'acide hydroxamique, préparation et utilisations thérapeutiques de ceux-ci
MY149731A (en) Compounds
JO2973B1 (en) Fumarate salt for (alpha-beta-R) -6-bromo-alpha-[2- (methylamino) ethyl-2-methoxy-alpha-1-naphthalenyl-beta-phenyl-3-quinoline ethanol
EA201170753A1 (ru) Налмефена гидрохлорид дигидрат
WO2014016754A3 (fr) Compositions pharmaceutiques d'inhibiteur de la pompe à protons
WO2010049449A3 (fr) Nouveaux sels de sunitinib
ZA201003380B (en) Improved pharmaceutical composition containing a pyrrolidone anticonvulsant agent and methhod for the preparation thereof
WO2008001201A3 (fr) Compositions pharmaceutiques de clopidogrel
WO2010070677A3 (fr) Procédé de préparation de prasugrel et de ses sels pharmaceutiquement acceptables
NZ591204A (en) Pharmaceutical compositions and methods for stabilizing the same
EA200900463A1 (ru) Арипипразола гемифумарат и способ его получения
WO2010044097A3 (fr) Nouvelle forme pharmaceutique de palipéridone et procédé de préparation de celle-ci
WO2007110765A3 (fr) Procedes de preparation d'octreotide
GR1008821B (el) Φαρμακευτικο σκευασμα που περιλαμβανει υδροχλωρικη ιβαμπραδινη και μεθοδος παρασκευης αυτου
WO2010061220A3 (fr) Nouveaux procédés et polymorphes purs
GR20070100405A (el) Βελτιωμενες φαρμακοτεχνικες μορφες που περιεχουν αναστολεις της ακετυλοχοληνεστερασης και μεθοδοι παρασκευης αυτων
MY150480A (en) Pharmaceutical composition containing dihydropyridine calcium channel antagonist and method for the preparation thereof
CY1108846T1 (el) Βελτιωμενη φαρμακευτικη συνθεση που περιεχει αναστολεα ace και μεθοδος για την παρασκευη της
WO2011086577A3 (fr) Composition pharmaceutique de moxifloxacine et ses sels pharmaceutiquement acceptables
WO2010061219A3 (fr) Formes polymorphiques
WO2010046912A3 (fr) Analogues de fluconazole contenant du tiophène utilisés en tant qu'agents et procédé d'utilisation associé
CO6260055A2 (es) Composicion farmaceutica que contiene un antagonista del canal de calcio de tipo dihidropiridina y metodo para la preparacion de la misma
GR1007741B (el) Φαρμακευτικο σκευασμα περιεχον εναν ατυπικο αντιψυχωτικο παραγοντα και μεθοδος για την παρασκευη αυτου
GR1008082B (el) Φαρμακευτικο σκευασμα περιεχον εναν ατυπο αντιψυχωσικο παραγοντα και μεθοδος για την παρασκευη αυτου