SV2006002201A - Polimorfo ii de rapamicina y sus utilizaciones ref. am- 101733salvo - Google Patents
Polimorfo ii de rapamicina y sus utilizaciones ref. am- 101733salvoInfo
- Publication number
- SV2006002201A SV2006002201A SV2005002201A SV2005002201A SV2006002201A SV 2006002201 A SV2006002201 A SV 2006002201A SV 2005002201 A SV2005002201 A SV 2005002201A SV 2005002201 A SV2005002201 A SV 2005002201A SV 2006002201 A SV2006002201 A SV 2006002201A
- Authority
- SV
- El Salvador
- Prior art keywords
- rapamycin
- rapamycin polymorph
- ref
- uses ref
- poliform
- Prior art date
Links
- ZAHRKKWIAAJSAO-UHFFFAOYSA-N rapamycin Natural products COCC(O)C(=C/C(C)C(=O)CC(OC(=O)C1CCCCN1C(=O)C(=O)C2(O)OC(CC(OC)C(=CC=CC=CC(C)CC(C)C(=O)C)C)CCC2C)C(C)CC3CCC(O)C(C3)OC)C ZAHRKKWIAAJSAO-UHFFFAOYSA-N 0.000 title abstract 3
- QFJCIRLUMZQUOT-HPLJOQBZSA-N sirolimus Chemical compound C1C[C@@H](O)[C@H](OC)C[C@@H]1C[C@@H](C)[C@H]1OC(=O)[C@@H]2CCCCN2C(=O)C(=O)[C@](O)(O2)[C@H](C)CC[C@H]2C[C@H](OC)/C(C)=C/C=C/C=C/[C@@H](C)C[C@@H](C)C(=O)[C@H](OC)[C@H](O)/C(C)=C/[C@@H](C)C(=O)C1 QFJCIRLUMZQUOT-HPLJOQBZSA-N 0.000 title abstract 3
- 229960002930 sirolimus Drugs 0.000 title abstract 3
- 239000008194 pharmaceutical composition Substances 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D498/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
- C07D498/18—Bridged systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Public Health (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Oncology (AREA)
- Communicable Diseases (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Abstract
PROVEE FORMA POLIFORMA II DE RAPAMICINA. ESTA INVENCION TAMBIEN PROVEE PROCESOS PARA PREPARAR FORMA POLIFORMA II DE RAPAMICINA Y COMPOSICIONES FARMACEUTICAS QUE INCLUYEN FORMA POLIFORMA II DE RAPAMICINA.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US60309604P | 2004-08-20 | 2004-08-20 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| SV2006002201A true SV2006002201A (es) | 2006-05-09 |
Family
ID=35431373
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| SV2005002201A SV2006002201A (es) | 2004-08-20 | 2005-08-18 | Polimorfo ii de rapamicina y sus utilizaciones ref. am- 101733salvo |
Country Status (22)
| Country | Link |
|---|---|
| US (1) | US7282505B2 (es) |
| EP (1) | EP1781671A1 (es) |
| JP (1) | JP2008510710A (es) |
| KR (1) | KR20070051863A (es) |
| CN (1) | CN101039948A (es) |
| AR (1) | AR050374A1 (es) |
| AU (1) | AU2005277407A1 (es) |
| BR (1) | BRPI0514407A (es) |
| CA (1) | CA2575887A1 (es) |
| CR (1) | CR8929A (es) |
| EC (1) | ECSP077268A (es) |
| GT (1) | GT200500223A (es) |
| IL (1) | IL181170A0 (es) |
| MX (1) | MX2007002044A (es) |
| NO (1) | NO20071050L (es) |
| PA (1) | PA8642501A1 (es) |
| PE (1) | PE20060649A1 (es) |
| RU (1) | RU2007104518A (es) |
| SV (1) | SV2006002201A (es) |
| TW (1) | TW200608973A (es) |
| WO (1) | WO2006023627A1 (es) |
| ZA (1) | ZA200701453B (es) |
Families Citing this family (46)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| KR101131794B1 (ko) | 2002-07-30 | 2012-03-30 | 와이어쓰 엘엘씨 | Cci-779 공용매 농축액, 비경구 cci-779 제형 및 비경구 cci-779 제형의 제조방법 |
| CA2539324A1 (en) | 2003-09-18 | 2005-03-31 | Macusight, Inc. | Transscleral delivery |
| US7349971B2 (en) * | 2004-02-05 | 2008-03-25 | Scenera Technologies, Llc | System for transmitting data utilizing multiple communication applications simultaneously in response to user request without specifying recipient's communication information |
| US8551512B2 (en) | 2004-03-22 | 2013-10-08 | Advanced Cardiovascular Systems, Inc. | Polyethylene glycol/poly(butylene terephthalate) copolymer coated devices including EVEROLIMUS |
| GB2438544A (en) | 2005-02-09 | 2007-11-28 | Cooper Internat Corp | Liquid formulations for treatment of diseases or conditions |
| US8663639B2 (en) | 2005-02-09 | 2014-03-04 | Santen Pharmaceutical Co., Ltd. | Formulations for treating ocular diseases and conditions |
| JP5528708B2 (ja) | 2006-02-09 | 2014-06-25 | 参天製薬株式会社 | 安定な製剤ならびにそれらを調製および使用する方法 |
| AU2007230964B2 (en) | 2006-03-23 | 2012-07-19 | Santen Pharmaceutical Co., Ltd. | Formulations and methods for vascular permeability-related diseases or conditions |
| NZ574654A (en) * | 2006-07-25 | 2012-03-30 | Abbott Lab | Crystalline forms of rapamycin analogs |
| US7812032B2 (en) | 2006-07-25 | 2010-10-12 | Abbott Laboratories | Crystalline forms of rapamycin analogs |
| US7820812B2 (en) | 2006-07-25 | 2010-10-26 | Abbott Laboratories | Methods of manufacturing crystalline forms of rapamycin analogs |
| US8486926B2 (en) * | 2006-11-17 | 2013-07-16 | Harbor Therapeutics, Inc. | Steroid tetrol solid state forms |
| US8414526B2 (en) * | 2006-11-20 | 2013-04-09 | Lutonix, Inc. | Medical device rapid drug releasing coatings comprising oils, fatty acids, and/or lipids |
| US8414910B2 (en) | 2006-11-20 | 2013-04-09 | Lutonix, Inc. | Drug releasing coatings for medical devices |
| US8998846B2 (en) | 2006-11-20 | 2015-04-07 | Lutonix, Inc. | Drug releasing coatings for balloon catheters |
| US9700704B2 (en) | 2006-11-20 | 2017-07-11 | Lutonix, Inc. | Drug releasing coatings for balloon catheters |
| US8425459B2 (en) | 2006-11-20 | 2013-04-23 | Lutonix, Inc. | Medical device rapid drug releasing coatings comprising a therapeutic agent and a contrast agent |
| US8414525B2 (en) | 2006-11-20 | 2013-04-09 | Lutonix, Inc. | Drug releasing coatings for medical devices |
| US9737640B2 (en) | 2006-11-20 | 2017-08-22 | Lutonix, Inc. | Drug releasing coatings for medical devices |
| US8430055B2 (en) | 2008-08-29 | 2013-04-30 | Lutonix, Inc. | Methods and apparatuses for coating balloon catheters |
| US20080276935A1 (en) * | 2006-11-20 | 2008-11-13 | Lixiao Wang | Treatment of asthma and chronic obstructive pulmonary disease with anti-proliferate and anti-inflammatory drugs |
| US20080175887A1 (en) * | 2006-11-20 | 2008-07-24 | Lixiao Wang | Treatment of Asthma and Chronic Obstructive Pulmonary Disease With Anti-proliferate and Anti-inflammatory Drugs |
| JP2008305262A (ja) * | 2007-06-08 | 2008-12-18 | Konica Minolta Business Technologies Inc | サーバ及びシンクライアント環境でのプリンタ紹介方法 |
| ES2645692T3 (es) | 2008-11-11 | 2017-12-07 | The Board Of Regents,The University Of Texas System | Microcápsulas de rapamicina y su uso para el tratamiento del cáncer |
| DE102008060549A1 (de) | 2008-12-04 | 2010-06-10 | MAX-PLANCK-Gesellschaft zur Förderung der Wissenschaften e.V. | Wirkstoff-Peptid-Konstrukt zur extrazellulären Anreicherung |
| US20110275798A1 (en) * | 2009-01-21 | 2011-11-10 | Rakesh Bhaiyyaram Mendhe | Method for Determination of Sirolimus Stability and Process for Preparing Its Stable Form |
| US20120231037A1 (en) | 2009-02-02 | 2012-09-13 | Yissum Research Development Companyof the Hebrew U | Crystalline drug-containing coatings |
| US20120252834A1 (en) * | 2009-08-05 | 2012-10-04 | The Government Of United States, As Represented By The Secretary Of The Army | Novel use and method of rapamycin to treat toxic shock |
| WO2015103447A1 (en) | 2013-12-31 | 2015-07-09 | Rapamycin Holdings, Llc | Oral rapamycin nanoparticle preparations and use |
| US9283211B1 (en) | 2009-11-11 | 2016-03-15 | Rapamycin Holdings, Llc | Oral rapamycin preparation and use for stomatitis |
| AU2012338869A1 (en) | 2011-11-15 | 2014-06-05 | Novartis Ag | Combination of a phosphoinositide 3-kinase inhibitor and a modulator of the Janus Kinase 2-Signal Transducer and Activator of Transcription 5 pathway |
| EP2869818A1 (en) | 2012-07-06 | 2015-05-13 | Novartis AG | Combination of a phosphoinositide 3-kinase inhibitor and an inhibitor of the il-8/cxcr interaction |
| DK2968281T3 (da) | 2013-03-13 | 2020-11-02 | Univ Texas | Mtor-hæmmere til forebyggelse af vækst af tarmpolyp |
| EP3738592B1 (en) | 2013-10-08 | 2022-01-26 | AI Therapeutics, Inc. | Rapamycin for the treatment of lymphangioleiomyomatosis |
| US9700544B2 (en) | 2013-12-31 | 2017-07-11 | Neal K Vail | Oral rapamycin nanoparticle preparations |
| JP2017505789A (ja) * | 2014-02-11 | 2017-02-23 | ラム・セラピューティクス,インコーポレーテッド | リンパ脈管筋腫症の治療のためのラパマイシン |
| US10307371B2 (en) | 2014-02-11 | 2019-06-04 | AI Therapeutics, Inc. | Rapamycin for the treatment of lymphangioleiomyomatosis |
| HUP1400075A2 (hu) | 2014-02-14 | 2015-08-28 | Druggability Technologies Ip Holdco Jersey Ltd | Sirolimus és származékainak komplexei, elõállítása és gyógyszerészeti kompozíciói |
| BR112016022598A8 (pt) | 2014-04-04 | 2021-06-29 | Ai Therapeutics Inc | composição aerossol farmacêutica na forma de um pó seco para liberação pulmonar, forma de dosagem unitária, pacote farmacêutico, kit e uso |
| CA2963085C (en) | 2014-10-07 | 2023-02-21 | Lam Therapeutics, Inc. | An inhalable rapamycin formulation for the treatment of pulmonary hypertension |
| MA40910A (fr) | 2014-11-07 | 2017-09-12 | Civitas Therapeutics Inc | Poudres de rapamycine pour administration pulmonaire |
| CN106478663A (zh) * | 2015-08-26 | 2017-03-08 | 博瑞生物医药(苏州)股份有限公司 | 一种依维莫司的干燥方法 |
| ES2871499T3 (es) | 2017-05-15 | 2021-10-29 | Bard Inc C R | Dispositivo médico con recubrimiento de elución de fármaco y capa intermedia |
| CN109020995A (zh) * | 2017-06-12 | 2018-12-18 | 鲁南制药集团股份有限公司 | 一种替西罗莫司的晶型物 |
| WO2020101675A1 (en) | 2018-11-14 | 2020-05-22 | Lutonix, Inc. | Medical device with drug-eluting coating on modified device surface |
| WO2020209828A1 (en) | 2019-04-08 | 2020-10-15 | Bard Peripheral Vascular, Inc. | Medical device with drug-eluting coating on modified device surface |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| ZA737247B (en) * | 1972-09-29 | 1975-04-30 | Ayerst Mckenna & Harrison | Rapamycin and process of preparation |
| US3993749A (en) | 1974-04-12 | 1976-11-23 | Ayerst Mckenna And Harrison Ltd. | Rapamycin and process of preparation |
| UA41884C2 (uk) | 1993-11-05 | 2001-10-15 | Амерікан Хоум Продактс Корпорейшн | Спосіб відокремлення рапаміцину від кислотних, основних та неполярних нейтральних домішок, присутніх в концентраті екстрактів ферментаційного бульйону або маточних розчинів |
-
2005
- 2005-08-16 AR ARP050103448A patent/AR050374A1/es unknown
- 2005-08-18 BR BRPI0514407-8A patent/BRPI0514407A/pt not_active IP Right Cessation
- 2005-08-18 GT GT200500223A patent/GT200500223A/es unknown
- 2005-08-18 KR KR1020077003941A patent/KR20070051863A/ko not_active Withdrawn
- 2005-08-18 US US11/206,472 patent/US7282505B2/en not_active Expired - Fee Related
- 2005-08-18 PA PA20058642501A patent/PA8642501A1/es unknown
- 2005-08-18 SV SV2005002201A patent/SV2006002201A/es unknown
- 2005-08-18 PE PE2005000957A patent/PE20060649A1/es not_active Application Discontinuation
- 2005-08-18 JP JP2007528004A patent/JP2008510710A/ja not_active Withdrawn
- 2005-08-18 RU RU2007104518/04A patent/RU2007104518A/ru not_active Application Discontinuation
- 2005-08-18 CN CNA2005800353638A patent/CN101039948A/zh active Pending
- 2005-08-18 EP EP05788650A patent/EP1781671A1/en not_active Withdrawn
- 2005-08-18 WO PCT/US2005/029364 patent/WO2006023627A1/en not_active Ceased
- 2005-08-18 TW TW094128147A patent/TW200608973A/zh unknown
- 2005-08-18 AU AU2005277407A patent/AU2005277407A1/en not_active Abandoned
- 2005-08-18 MX MX2007002044A patent/MX2007002044A/es unknown
- 2005-08-18 CA CA002575887A patent/CA2575887A1/en not_active Abandoned
-
2007
- 2007-02-05 IL IL181170A patent/IL181170A0/en unknown
- 2007-02-15 CR CR8929A patent/CR8929A/es not_active Application Discontinuation
- 2007-02-19 ZA ZA200701453A patent/ZA200701453B/xx unknown
- 2007-02-21 EC EC2007007268A patent/ECSP077268A/es unknown
- 2007-02-23 NO NO20071050A patent/NO20071050L/no not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| ECSP077268A (es) | 2007-03-29 |
| MX2007002044A (es) | 2007-03-29 |
| PA8642501A1 (es) | 2006-05-16 |
| US7282505B2 (en) | 2007-10-16 |
| KR20070051863A (ko) | 2007-05-18 |
| NO20071050L (no) | 2007-05-15 |
| ZA200701453B (en) | 2010-08-25 |
| GT200500223A (es) | 2006-03-09 |
| US20060040971A1 (en) | 2006-02-23 |
| EP1781671A1 (en) | 2007-05-09 |
| IL181170A0 (en) | 2007-07-04 |
| CA2575887A1 (en) | 2006-03-02 |
| AU2005277407A1 (en) | 2006-03-02 |
| AR050374A1 (es) | 2006-10-18 |
| BRPI0514407A (pt) | 2008-06-10 |
| WO2006023627A1 (en) | 2006-03-02 |
| WO2006023627A8 (en) | 2006-11-30 |
| CR8929A (es) | 2007-08-28 |
| RU2007104518A (ru) | 2008-09-27 |
| TW200608973A (en) | 2006-03-16 |
| PE20060649A1 (es) | 2006-08-10 |
| JP2008510710A (ja) | 2008-04-10 |
| CN101039948A (zh) | 2007-09-19 |
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