SV2004001418A - Formulaciones farmaceuticas de 5,7,14-triazaciclo 10.3.1.0.2,11.04,9) -hexadeca-2(11),3,5,7,9-pentaeno" ref.pc 23248 - Google Patents
Formulaciones farmaceuticas de 5,7,14-triazaciclo 10.3.1.0.2,11.04,9) -hexadeca-2(11),3,5,7,9-pentaeno" ref.pc 23248Info
- Publication number
- SV2004001418A SV2004001418A SV2002001418A SV2002001418A SV2004001418A SV 2004001418 A SV2004001418 A SV 2004001418A SV 2002001418 A SV2002001418 A SV 2002001418A SV 2002001418 A SV2002001418 A SV 2002001418A SV 2004001418 A SV2004001418 A SV 2004001418A
- Authority
- SV
- El Salvador
- Prior art keywords
- pentaeno
- hexadeca
- triazaciclo
- ref
- pharmaceutical formulations
- Prior art date
Links
- 239000008194 pharmaceutical composition Substances 0.000 title 1
- 239000000203 mixture Substances 0.000 abstract 2
- SNICXCGAKADSCV-JTQLQIEISA-N (-)-Nicotine Chemical compound CN1CCC[C@H]1C1=CC=CN=C1 SNICXCGAKADSCV-JTQLQIEISA-N 0.000 abstract 1
- 206010012335 Dependence Diseases 0.000 abstract 1
- 230000002411 adverse Effects 0.000 abstract 1
- 239000002552 dosage form Substances 0.000 abstract 1
- 238000009472 formulation Methods 0.000 abstract 1
- 238000000034 method Methods 0.000 abstract 1
- 229960002715 nicotine Drugs 0.000 abstract 1
- SNICXCGAKADSCV-UHFFFAOYSA-N nicotine Natural products CN1CCCC1C1=CC=CN=C1 SNICXCGAKADSCV-UHFFFAOYSA-N 0.000 abstract 1
- 238000009827 uniform distribution Methods 0.000 abstract 1
Classifications
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-
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
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- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/498—Pyrazines or piperazines ortho- and peri-condensed with carbocyclic ring systems, e.g. quinoxaline, phenazine
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- A61K47/30—Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
- A61K47/36—Polysaccharides; Derivatives thereof, e.g. gums, starch, alginate, dextrin, hyaluronic acid, chitosan, inulin, agar or pectin
- A61K47/38—Cellulose; Derivatives thereof
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- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
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Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
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- Inorganic Chemistry (AREA)
- Psychology (AREA)
- Immunology (AREA)
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- Vascular Medicine (AREA)
- Urology & Nephrology (AREA)
- Hospice & Palliative Care (AREA)
- Diabetes (AREA)
- Rheumatology (AREA)
- Anesthesiology (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Abstract
LA PRESENTE INVENCION SE REFIERE A FORMAS DE DOSIFICACION FARMACEUTICAS ORALES DE LIBERACION CONTROLADA (ABREVIADAMENTE LC) DE 5,8,14-TRAZATETRACICLO[10.3.1.02,11.04,9]-HEXADECA-2(11)3,5,7,9-PENTAENO-VEASE 1, Y A LAS SALES FARMACEUTICAMENTE ACEPTABLES DEL MISMO, Y A PROCEDIMIENTOS EN LOS QUE SE USAN PARA REDUCIR LA ADICCION A LA NICOTINA O AYUDAR EN EL CESE O REDUCCION DEL USO DEL TABACO EN TANTO QUE REDUCEN LAS NAUSEAS COMO EFECTO ADVERSO. LA PRESENTE INVENCION SE REFIERE TAMBIEN A UNA COMPOSICION DE DOSIFICACION BAJA DE LIBERACION INMEDIATA ABREVIADAMENTE LI) QUE POSEEN UNA FORMULACION ESTABLE CON UNA DISTRIBUCION Y POTENCIA DEL FARMACO UNIFORMES, VER FORMULA.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US33465201P | 2001-11-30 | 2001-11-30 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| SV2004001418A true SV2004001418A (es) | 2004-05-07 |
Family
ID=23308160
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| SV2002001418A SV2004001418A (es) | 2001-11-30 | 2002-11-29 | Formulaciones farmaceuticas de 5,7,14-triazaciclo 10.3.1.0.2,11.04,9) -hexadeca-2(11),3,5,7,9-pentaeno" ref.pc 23248 |
Country Status (30)
| Country | Link |
|---|---|
| US (1) | US7771748B2 (es) |
| EP (1) | EP1448235B1 (es) |
| JP (2) | JP2005528330A (es) |
| KR (2) | KR100892517B1 (es) |
| CN (2) | CN1864663A (es) |
| AR (1) | AR037592A1 (es) |
| AT (1) | ATE356625T1 (es) |
| AU (1) | AU2002351008B2 (es) |
| BR (1) | BR0214806A (es) |
| CA (1) | CA2467490C (es) |
| DE (1) | DE60218885T2 (es) |
| DK (1) | DK1448235T3 (es) |
| ES (1) | ES2282492T3 (es) |
| GT (1) | GT200200247A (es) |
| IL (1) | IL161857A0 (es) |
| MX (1) | MXPA04003807A (es) |
| MY (1) | MY130619A (es) |
| NO (1) | NO20042739L (es) |
| NZ (1) | NZ532435A (es) |
| PA (1) | PA8559501A1 (es) |
| PE (1) | PE20040121A1 (es) |
| PL (1) | PL208080B1 (es) |
| PT (1) | PT1448235E (es) |
| RU (2) | RU2272629C2 (es) |
| SI (1) | SI1448235T1 (es) |
| SV (1) | SV2004001418A (es) |
| TW (1) | TWI327471B (es) |
| UY (1) | UY27553A1 (es) |
| WO (1) | WO2003045437A1 (es) |
| ZA (1) | ZA200403068B (es) |
Families Citing this family (35)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| BR9814592B1 (pt) * | 1997-12-31 | 2010-06-01 | composto azapolicìclico condensado com arila, composição farmacêutica contendo o mesmo e seu uso na fabricação de um medicamento. | |
| SE521512C2 (sv) * | 2001-06-25 | 2003-11-11 | Niconovum Ab | Anordning för administrering av en substans till främre delen av en individs munhåla |
| EP1448235B1 (en) | 2001-11-30 | 2007-03-14 | Pfizer Products Inc. | Oral controlled release pharmaceutical compositions of 5,8,14-triazatetracyclo 10.3.1.0(2,11).0(4,9)]-hexadeca-2(11)3,5,7,9-pentaene |
| DK3473251T3 (da) * | 2002-12-20 | 2024-01-22 | Niconovum Ab | Nikotin-cellulose-kombination |
| JP2006528237A (ja) * | 2003-05-20 | 2006-12-14 | ファイザー・プロダクツ・インク | バレニクリンの医薬組成物 |
| US7051606B2 (en) * | 2004-01-30 | 2006-05-30 | Andrx Labs Llc | Dosage form holder device and methods for immersion testing |
| JP2008516942A (ja) * | 2004-10-15 | 2008-05-22 | ファイザー・プロダクツ・インク | バレニクリンの鼻腔内、バッカル、舌下および肺送達のための組成物および方法 |
| CA2593432A1 (en) * | 2005-01-07 | 2006-07-13 | Prizer Products Inc. | Fast-disintegrating dosage forms of 5,8,14-triazatetracyclo[10.3.1.02,11.04,9]-hexadeca-2(11),3,5,7,9-pentaene |
| US20110086086A1 (en) * | 2005-07-26 | 2011-04-14 | Pfizer Inc | Transdermal system for varenicline |
| US20080248107A1 (en) * | 2005-08-24 | 2008-10-09 | Rubicon Research Pvt. Ltd. | Controlled Release Formulation |
| CA2646942C (en) | 2006-03-16 | 2014-07-29 | Niconovum Ab | Improved snuff composition |
| BRPI0710914A2 (pt) * | 2006-04-24 | 2011-09-27 | Pfizer Prod Inc | forma de dosagem e método para o tratamento de dependência, adição e supressão de nicotina, em particular para uso na terapia para parar de fumar |
| WO2007132344A2 (en) * | 2006-05-09 | 2007-11-22 | Aurobindo Pharma Limited | Controlled release compositions of an antidepressant agent |
| US20080145423A1 (en) * | 2006-12-14 | 2008-06-19 | Ajmal Ali Khan | Chewable tablet and method of formulating |
| WO2009027786A2 (en) * | 2007-08-29 | 2009-03-05 | Pfizer Inc. | Matrix dosage forms of varenicline |
| WO2009034431A2 (en) | 2007-09-10 | 2009-03-19 | Pfizer Inc. | Controlled-release dosage forms for varenicline |
| WO2009123580A1 (en) * | 2008-04-01 | 2009-10-08 | Schering-Plough Healthcare Products, Inc. | Chewable tablet and method of formulating |
| EP2268639A2 (en) | 2008-05-22 | 2011-01-05 | Teva Pharmaceutical Industries Ltd. | Varenicline tosylate, an intermediate in the preparation process of varenicline l-tartrate |
| US20090318695A1 (en) * | 2008-06-19 | 2009-12-24 | Vinod Kumar Kansal | Processes for the preparation of varenicline and intermediates thereof |
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