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SV2002000287A - Uso de inhibidor de la quinasa dependiente de la ciclina para preparar una composicion farmaceutica util para tratar enfermedades neurodegenerativas - Google Patents

Uso de inhibidor de la quinasa dependiente de la ciclina para preparar una composicion farmaceutica util para tratar enfermedades neurodegenerativas

Info

Publication number
SV2002000287A
SV2002000287A SV2001000287A SV2001000287A SV2002000287A SV 2002000287 A SV2002000287 A SV 2002000287A SV 2001000287 A SV2001000287 A SV 2001000287A SV 2001000287 A SV2001000287 A SV 2001000287A SV 2002000287 A SV2002000287 A SV 2002000287A
Authority
SV
El Salvador
Prior art keywords
neurodegenerative diseases
dependent kinase
prepare
pharmaceutical composition
kinase inhibitor
Prior art date
Application number
SV2001000287A
Other languages
English (en)
Inventor
Thomas Charles Malone
Richard John Booth
Arindam Chatterjee
Chatterjee Arindam
Original Assignee
Warner Lambert Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Warner Lambert Co filed Critical Warner Lambert Co
Publication of SV2002000287A publication Critical patent/SV2002000287A/es

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P21/00—Drugs for disorders of the muscular or neuromuscular system
    • A61P21/02—Muscle relaxants, e.g. for tetanus or cramps
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A61P25/16—Anti-Parkinson drugs
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Neurology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Psychology (AREA)
  • Psychiatry (AREA)
  • Hospice & Palliative Care (AREA)
  • Pain & Pain Management (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

Abstract

ESTA INVENCION PROPORCIONA UN METODO PARA TRATAR ENFERMEDADES NEURODEGENERATIVAS EN MAMIFEROS, QUE COMPRENDE ADMINISTRAR UNA CANTIDAD EFECTIVA DE UN INHIBIDOR DE LA QUINASA DEPENDIENTE DE CICLINA. UN METODO PREFERIDO USA INHIBIDORES DE LA CDK DE FORMULA I:VER FORMULA; Y DE LA FORMULA II: VER FORMULA; EN DONDE:W ES NH; S; SO O SO2,R1 INCLUYE FENILO Y FENILO SUSTITUIDO,R2 INCLUYE ALQUILO Y CICLOALQUILO,R3 INCLUYE ALQUILO E HIDROGENO,R8 Y R9 INCLUYEN HIDROGENO Y ALQUILO, YZ ES CARBOXI.
SV2001000287A 2000-01-27 2001-01-22 Uso de inhibidor de la quinasa dependiente de la ciclina para preparar una composicion farmaceutica util para tratar enfermedades neurodegenerativas SV2002000287A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US17840000P 2000-01-27 2000-01-27

Publications (1)

Publication Number Publication Date
SV2002000287A true SV2002000287A (es) 2002-01-08

Family

ID=22652409

Family Applications (1)

Application Number Title Priority Date Filing Date
SV2001000287A SV2002000287A (es) 2000-01-27 2001-01-22 Uso de inhibidor de la quinasa dependiente de la ciclina para preparar una composicion farmaceutica util para tratar enfermedades neurodegenerativas

Country Status (22)

Country Link
US (1) US20040224958A1 (es)
EP (1) EP1255755A1 (es)
JP (1) JP2003523358A (es)
KR (1) KR20020070520A (es)
CN (1) CN1433417A (es)
AR (1) AR029437A1 (es)
AU (1) AU1808601A (es)
BR (1) BR0017075A (es)
CA (1) CA2394525A1 (es)
CO (1) CO5280216A1 (es)
CZ (1) CZ20022521A3 (es)
GT (1) GT200100005A (es)
HN (1) HN2001000012A (es)
HU (1) HUP0203803A3 (es)
IL (1) IL150742A0 (es)
PA (1) PA8510801A1 (es)
PE (1) PE20011228A1 (es)
PL (1) PL357634A1 (es)
SK (1) SK10772002A3 (es)
SV (1) SV2002000287A (es)
TN (1) TNSN01018A1 (es)
WO (1) WO2001055148A1 (es)

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Also Published As

Publication number Publication date
KR20020070520A (ko) 2002-09-09
WO2001055148A1 (en) 2001-08-02
TNSN01018A1 (en) 2005-11-10
PA8510801A1 (es) 2002-12-11
CN1433417A (zh) 2003-07-30
CO5280216A1 (es) 2003-05-30
HN2001000012A (es) 2001-07-09
SK10772002A3 (sk) 2004-01-08
AU1808601A (en) 2001-08-07
AR029437A1 (es) 2003-06-25
BR0017075A (pt) 2002-11-05
HUP0203803A2 (hu) 2003-02-28
JP2003523358A (ja) 2003-08-05
HUP0203803A3 (en) 2004-09-28
CA2394525A1 (en) 2001-08-02
CZ20022521A3 (cs) 2003-02-12
PL357634A1 (en) 2004-07-26
GT200100005A (es) 2002-02-05
IL150742A0 (en) 2003-02-12
EP1255755A1 (en) 2002-11-13
US20040224958A1 (en) 2004-11-11
PE20011228A1 (es) 2002-01-18

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