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RU2018132775A - Композиции, полезные для предупреждения и/или лечения расстройств ротовой полости, верхних дыхательных путей и пищевода - Google Patents

Композиции, полезные для предупреждения и/или лечения расстройств ротовой полости, верхних дыхательных путей и пищевода Download PDF

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Publication number
RU2018132775A
RU2018132775A RU2018132775A RU2018132775A RU2018132775A RU 2018132775 A RU2018132775 A RU 2018132775A RU 2018132775 A RU2018132775 A RU 2018132775A RU 2018132775 A RU2018132775 A RU 2018132775A RU 2018132775 A RU2018132775 A RU 2018132775A
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mass
extract
oral cavity
alginic acid
composition
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RU2018132775A
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RU2018132775A3 (ru
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Эцио БОМБАРДЕЛЛИ
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Индена С.П.А.
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Publication of RU2018132775A3 publication Critical patent/RU2018132775A3/ru

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    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0053Mouth and digestive tract, i.e. intraoral and peroral administration
    • A61K9/0056Mouth soluble or dispersible forms; Suckable, eatable, chewable coherent forms; Forms rapidly disintegrating in the mouth; Lozenges; Lollipops; Bite capsules; Baked products; Baits or other oral forms for animals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K36/00Medicinal preparations of undetermined constitution containing material from algae, lichens, fungi or plants, or derivatives thereof, e.g. traditional herbal medicines
    • A61K36/18Magnoliophyta (angiosperms)
    • A61K36/88Liliopsida (monocotyledons)
    • A61K36/906Zingiberaceae (Ginger family)
    • A61K36/9068Zingiber, e.g. garden ginger
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/22Heterocyclic compounds, e.g. ascorbic acid, tocopherol or pyrrolidones
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/30Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
    • A61K47/36Polysaccharides; Derivatives thereof, e.g. gums, starch, alginate, dextrin, hyaluronic acid, chitosan, inulin, agar or pectin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0053Mouth and digestive tract, i.e. intraoral and peroral administration
    • A61K9/006Oral mucosa, e.g. mucoadhesive forms, sublingual droplets; Buccal patches or films; Buccal sprays
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/06Ointments; Bases therefor; Other semi-solid forms, e.g. creams, sticks, gels
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/19Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles lyophilised, i.e. freeze-dried, solutions or dispersions
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2013Organic compounds, e.g. phospholipids, fats
    • A61K9/2018Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/70Web, sheet or filament bases ; Films; Fibres of the matrix type containing drug
    • A61K9/7015Drug-containing film-forming compositions, e.g. spray-on
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/02Stomatological preparations, e.g. drugs for caries, aphtae, periodontitis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/02Nasal agents, e.g. decongestants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/04Drugs for disorders of the respiratory system for throat disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • A61P31/16Antivirals for RNA viruses for influenza or rhinoviruses
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P39/00General protective or antinoxious agents

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  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Natural Medicines & Medicinal Plants (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nutrition Science (AREA)
  • Physiology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Pulmonology (AREA)
  • Virology (AREA)
  • Microbiology (AREA)
  • Mycology (AREA)
  • Inorganic Chemistry (AREA)
  • Medical Informatics (AREA)
  • Botany (AREA)
  • Biotechnology (AREA)
  • Alternative & Traditional Medicine (AREA)
  • Molecular Biology (AREA)
  • Biophysics (AREA)
  • Zoology (AREA)
  • Otolaryngology (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Toxicology (AREA)
  • Medicines Containing Plant Substances (AREA)
  • Medicinal Preparation (AREA)

Claims (11)

1. Композиции, содержащие по меньшей мере один пленкообразующий агент, способный прикрепляться стабильным образом к слизистой оболочке ротовой полости, пищевода и верхних дыхательных путей, где пленкообразующий агент выбран из группы, состоящей из солей гиалуроновой кислоты, протеогликанов или альгиновой кислоты с антоцианидинами или проантоцианидинами в свободной или гликозилированной форме, или из танинов, полученных из процианидинов или эллаговой кислоты, включенных в поперечно-сшитую гиалуроновую кислоту или альгиновую кислоту.
2. Композиции по п. 1, где пленкообразующий агент получен путем приведения во взаимодействие гиалуроновой кислоты или альгиновой кислоты с экстрактами, полученными из лекарственных растений.
3. Композиции по п. 1 или 2, где гиалуроновая кислота или альгиновая кислота имеет молекулярную массу в диапазоне от 100000 до 10000000 Дальтон, предпочтительно 1000000 Дальтон.
4. Композиции по п. 2, где экстракты выбраны из экстракта Vaccinium myrtillus, Vaccinium uliginosum, Punica grcmatum, Vitis vinifera uAesculus ippocastanum.
5. Композиции по n. 4, где экстракт представляет собой экстракт Vaccinium myrtillus или экстракт Vaccinium uliginosum.
6. Композиции по любому из пп. 1-5, где гиалуроновая или альгиновая кислота поперечно сшиты сшивающими агентами, выбранными из дивинилсульфона (DVS), диглицидилового эфира 1,4-бутандиола, водорастворимых карбодиимидов, таких как 1-этил-3-(3-диметиламинопропил)карбодиимид, и сшивающими агентами с аминогруппами или мочевиной.
7. Композиции по любому из пп. 1-6, дополнительно содержащие по меньшей мере одно соединение или экстракт, полученные из лекарственного растения, обладающего противомикробной или противовирусной активностью.
8. Композиции по п. 7, где экстракт, полученный из лекарственного растения, обладающего противомикробной или противовирусной активностью, представляет собой липофильный экстракт Zingiber officinale.
9. Композиции по п. 8, где количество липофильного экстракта Zingiber officinale находится в диапазоне от 0,01% масс/масс, до 1% масс/масс, предпочтительно от 0,1% масс/масс, до 0,8% масс/масс, и еще более предпочтительно составляет 0,5% масс/масс.
10. Композиции по любому из пп. 1-9 для применения в предупреждении и/или лечении расстройств ротовой полости, пищевода и верхних дыхательных путей, вызванных химическими и/или бактериальными и/или вирусными агентами.
11. Композиции для применения по п. 10, где расстройства, вызванные химическими и/или бактериальными и/или вирусными агентами, представляют собой простуды, грипп, воспаление слизистой оболочки ротовой полости и пищевода различного происхождения и повреждения слизистой оболочки пищевода, вызванные повышенной кислотностью или гастроэзофагеальным рефлюксом.
RU2018132775A 2016-03-18 2017-03-15 Композиции, полезные для предупреждения и/или лечения расстройств ротовой полости, верхних дыхательных путей и пищевода RU2018132775A (ru)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
IT102016000028801 2016-03-18
ITUA2016A001822A ITUA20161822A1 (it) 2016-03-18 2016-03-18 Composizioni utili nella prevenzione e/o nel trattamento di patologie del cavo orale, delle prime vie aeree e dell’esofago
PCT/EP2017/056148 WO2017158041A1 (en) 2016-03-18 2017-03-15 Compositions useful in the prevention and/or treatment of disorders of the oral cavity, upper airways and esophagus

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RU2018132775A true RU2018132775A (ru) 2020-04-20
RU2018132775A3 RU2018132775A3 (ru) 2020-04-20

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US (2) US20190083392A1 (ru)
EP (1) EP3429607B1 (ru)
JP (1) JP2019508470A (ru)
KR (1) KR20180123042A (ru)
CN (1) CN108778304A (ru)
AU (1) AU2017234987A1 (ru)
BR (1) BR112018068642A2 (ru)
CA (1) CA3017791A1 (ru)
DK (1) DK3429607T3 (ru)
ES (1) ES2906803T3 (ru)
HU (1) HUE058136T2 (ru)
IL (1) IL261737A (ru)
IT (1) ITUA20161822A1 (ru)
MX (1) MX2018011205A (ru)
PL (1) PL3429607T3 (ru)
PT (1) PT3429607T (ru)
RU (1) RU2018132775A (ru)
SG (1) SG11201807963WA (ru)
SI (1) SI3429607T1 (ru)
WO (1) WO2017158041A1 (ru)

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SG11201807963WA (en) 2018-10-30
ITUA20161822A1 (it) 2017-09-18
KR20180123042A (ko) 2018-11-14
DK3429607T3 (da) 2022-01-10
IL261737A (en) 2018-10-31
SI3429607T1 (sl) 2022-04-29
CN108778304A (zh) 2018-11-09
PL3429607T3 (pl) 2022-04-04
EP3429607A1 (en) 2019-01-23
MX2018011205A (es) 2018-11-22
US20190083392A1 (en) 2019-03-21
ES2906803T3 (es) 2022-04-20
PT3429607T (pt) 2022-02-22
JP2019508470A (ja) 2019-03-28
AU2017234987A1 (en) 2018-10-04
US20200289413A1 (en) 2020-09-17
RU2018132775A3 (ru) 2020-04-20
WO2017158041A1 (en) 2017-09-21
CA3017791A1 (en) 2017-09-21
BR112018068642A2 (pt) 2019-02-05
EP3429607B1 (en) 2021-12-15
HUE058136T2 (hu) 2022-07-28

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