RU2008148542A - Усилитель выработки тестостерона - Google Patents
Усилитель выработки тестостерона Download PDFInfo
- Publication number
- RU2008148542A RU2008148542A RU2008148542/15A RU2008148542A RU2008148542A RU 2008148542 A RU2008148542 A RU 2008148542A RU 2008148542/15 A RU2008148542/15 A RU 2008148542/15A RU 2008148542 A RU2008148542 A RU 2008148542A RU 2008148542 A RU2008148542 A RU 2008148542A
- Authority
- RU
- Russia
- Prior art keywords
- vitamin
- testosterone
- enhancer
- testosterone production
- menaquinone
- Prior art date
Links
- MUMGGOZAMZWBJJ-DYKIIFRCSA-N Testostosterone Chemical compound O=C1CC[C@]2(C)[C@H]3CC[C@](C)([C@H](CC4)O)[C@@H]4[C@@H]3CCC2=C1 MUMGGOZAMZWBJJ-DYKIIFRCSA-N 0.000 title claims abstract 26
- 229960003604 testosterone Drugs 0.000 title claims abstract 13
- 229930003448 Vitamin K Natural products 0.000 claims abstract 10
- 239000003623 enhancer Substances 0.000 claims abstract 10
- SHUZOJHMOBOZST-UHFFFAOYSA-N phylloquinone Natural products CC(C)CCCCC(C)CCC(C)CCCC(=CCC1=C(C)C(=O)c2ccccc2C1=O)C SHUZOJHMOBOZST-UHFFFAOYSA-N 0.000 claims abstract 10
- 235000019168 vitamin K Nutrition 0.000 claims abstract 10
- 239000011712 vitamin K Substances 0.000 claims abstract 10
- 150000003721 vitamin K derivatives Chemical class 0.000 claims abstract 10
- 229940046010 vitamin k Drugs 0.000 claims abstract 10
- PFRQBZFETXBLTP-UHFFFAOYSA-N Vitamin K2 Natural products C1=CC=C2C(=O)C(CC=C(C)CCC=C(C)CCC=C(C)CCC=C(C)CCC=C(C)CCC=C(C)C)=C(C)C(=O)C2=C1 PFRQBZFETXBLTP-UHFFFAOYSA-N 0.000 claims abstract 4
- 239000004480 active ingredient Substances 0.000 claims abstract 4
- 235000013305 food Nutrition 0.000 claims abstract 4
- 239000013589 supplement Substances 0.000 claims abstract 4
- 230000037213 diet Effects 0.000 claims abstract 2
- 235000005911 diet Nutrition 0.000 claims abstract 2
- 201000010099 disease Diseases 0.000 claims abstract 2
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 claims abstract 2
- 229940079593 drug Drugs 0.000 claims abstract 2
- 239000003814 drug Substances 0.000 claims abstract 2
- 235000009491 menaquinone-4 Nutrition 0.000 claims abstract 2
- 239000011676 menaquinone-4 Substances 0.000 claims abstract 2
- DKHGMERMDICWDU-GHDNBGIDSA-N menaquinone-4 Chemical group C1=CC=C2C(=O)C(C/C=C(C)/CC/C=C(C)/CC/C=C(C)/CCC=C(C)C)=C(C)C(=O)C2=C1 DKHGMERMDICWDU-GHDNBGIDSA-N 0.000 claims abstract 2
- 125000003063 menaquinone-4 group Chemical group 0.000 claims abstract 2
- 235000009464 menaquinone-7 Nutrition 0.000 claims abstract 2
- 239000011700 menaquinone-7 Substances 0.000 claims abstract 2
- RAKQPZMEYJZGPI-LJWNYQGCSA-N menaquinone-7 Chemical compound C1=CC=C2C(=O)C(C/C=C(C)/CC/C=C(C)/CC/C=C(C)/CC/C=C(C)/CC/C=C(C)/CC/C=C(C)/CCC=C(C)C)=C(C)C(=O)C2=C1 RAKQPZMEYJZGPI-LJWNYQGCSA-N 0.000 claims abstract 2
- 229960005481 menatetrenone Drugs 0.000 claims abstract 2
- 208000024891 symptom Diseases 0.000 claims abstract 2
- 235000019143 vitamin K2 Nutrition 0.000 claims abstract 2
- 239000011728 vitamin K2 Substances 0.000 claims abstract 2
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/12—Ketones
- A61K31/122—Ketones having the oxygen directly attached to a ring, e.g. quinones, vitamin K1, anthralin
-
- A—HUMAN NECESSITIES
- A23—FOODS OR FOODSTUFFS; TREATMENT THEREOF, NOT COVERED BY OTHER CLASSES
- A23L—FOODS, FOODSTUFFS OR NON-ALCOHOLIC BEVERAGES, NOT OTHERWISE PROVIDED FOR; PREPARATION OR TREATMENT THEREOF
- A23L33/00—Modifying nutritive qualities of foods; Dietetic products; Preparation or treatment thereof
- A23L33/10—Modifying nutritive qualities of foods; Dietetic products; Preparation or treatment thereof using additives
- A23L33/15—Vitamins
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/10—Drugs for genital or sexual disorders; Contraceptives for impotence
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P21/00—Drugs for disorders of the muscular or neuromuscular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/02—Nutrients, e.g. vitamins, minerals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/06—Antihyperlipidemics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
- A61P5/26—Androgens
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Endocrinology (AREA)
- Diabetes (AREA)
- Neurology (AREA)
- Epidemiology (AREA)
- Biomedical Technology (AREA)
- Neurosurgery (AREA)
- Nutrition Science (AREA)
- Obesity (AREA)
- Reproductive Health (AREA)
- Hematology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Urology & Nephrology (AREA)
- Cardiology (AREA)
- Gynecology & Obstetrics (AREA)
- Heart & Thoracic Surgery (AREA)
- Hospice & Palliative Care (AREA)
- Physical Education & Sports Medicine (AREA)
- Psychiatry (AREA)
- Mycology (AREA)
- Food Science & Technology (AREA)
- Polymers & Plastics (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Coloring Foods And Improving Nutritive Qualities (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Abstract
1. Усилитель выработки тестостерона, включающий витамин К в качестве активного ингредиента. ! 2. Усилитель выработки тестостерона по п.1, отличающийся тем, что витамин К является витамином К2. ! 3. Усилитель выработки тестостерона по п.1, отличающийся тем, что описанный выше витамин К является менахиноном-4 и/или менахиноном-7. ! 4. Лекарство, которое предотвращает появление и/или лечит симптомы или заболевания, вызванные снижением тестостерона, созданные на основе усилителя выработки тестостерона, который включает витамин К в качестве активного компонента. ! 5. Добавка, диетическая пища, пищевые продукты, содержащие добавки, которые содержат усилитель тестостерона, включая витамин К в качестве активного компонента.
Claims (5)
1. Усилитель выработки тестостерона, включающий витамин К в качестве активного ингредиента.
2. Усилитель выработки тестостерона по п.1, отличающийся тем, что витамин К является витамином К2.
3. Усилитель выработки тестостерона по п.1, отличающийся тем, что описанный выше витамин К является менахиноном-4 и/или менахиноном-7.
4. Лекарство, которое предотвращает появление и/или лечит симптомы или заболевания, вызванные снижением тестостерона, созданные на основе усилителя выработки тестостерона, который включает витамин К в качестве активного компонента.
5. Добавка, диетическая пища, пищевые продукты, содержащие добавки, которые содержат усилитель тестостерона, включая витамин К в качестве активного компонента.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2006-173455 | 2006-06-23 | ||
| JP2006173455 | 2006-06-23 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| RU2008148542A true RU2008148542A (ru) | 2010-06-20 |
| RU2431475C2 RU2431475C2 (ru) | 2011-10-20 |
Family
ID=38833237
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| RU2008148542/15A RU2431475C2 (ru) | 2006-06-23 | 2007-05-21 | Усилитель выработки тестостерона |
Country Status (7)
| Country | Link |
|---|---|
| US (2) | US8686049B2 (ru) |
| EP (1) | EP2033634A4 (ru) |
| JP (1) | JP5110478B2 (ru) |
| KR (1) | KR20090023562A (ru) |
| CN (1) | CN101472574B (ru) |
| RU (1) | RU2431475C2 (ru) |
| WO (1) | WO2007148494A1 (ru) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2014093818A2 (en) * | 2012-12-14 | 2014-06-19 | Bioject, Inc. | Use of a novel subcutaneous needle-free technique to deliver testosterone in hypogonadal men |
| WO2023170591A2 (en) * | 2022-03-09 | 2023-09-14 | Synergia Life Sciences Pvt Ltd. | Novel menaquinone-n (vitamin-k2-7) supplementation for livestock and poultry |
Family Cites Families (14)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2943031B2 (ja) | 1991-11-30 | 1999-08-30 | 株式会社ホーネンコーポレーション | 天然ビタミンk濃縮物の製造方法 |
| JP2900238B2 (ja) | 1994-07-07 | 1999-06-02 | 株式会社ホーネンコーポレーション | 天然メナキノン−7高含量脂質 |
| JP3845923B2 (ja) * | 1996-12-10 | 2006-11-15 | 熊本製粉株式会社 | 食品用ビタミンk補給組成物の製造方法 |
| JPH10295393A (ja) | 1997-04-30 | 1998-11-10 | New Food Kurieeshiyon Gijutsu Kenkyu Kumiai | ビタミンkの製造法 |
| JPH1156232A (ja) | 1997-08-26 | 1999-03-02 | Snow Brand Milk Prod Co Ltd | ビタミンk及びカルシウムを強化した乳及び乳製品 |
| JP3876395B2 (ja) | 1997-09-25 | 2007-01-31 | 株式会社J−オイルミルズ | ビタミンk2濃縮物の製造法 |
| JPH11127816A (ja) | 1997-10-27 | 1999-05-18 | Sanei Gen Ffi Inc | ビタミンkを含有する食品 |
| JP3836242B2 (ja) * | 1998-01-16 | 2006-10-25 | 陽子 竹中 | ビタミンk類及び機能性食品の製造方法並びに機能性食品 |
| US6093421A (en) | 1999-08-31 | 2000-07-25 | Biotics Research Corporation | Maca and antler for augmenting testosterone levels |
| JP2001136959A (ja) | 1999-11-17 | 2001-05-22 | Hiroyuki Sumi | 枯草菌菌体および/またはその産生物を含む培養物、これに由来する水溶性ビタミンk誘導体、これらを含む医薬、食品および飼料ならびにこれらの製造方法 |
| JP4131443B2 (ja) | 2001-08-27 | 2008-08-13 | 株式会社J−オイルミルズ | 抗骨粗鬆症組成物 |
| EP1441724B8 (en) | 2001-09-27 | 2007-10-17 | Laboratoires Serono SA | Methods of increasing endogenous testosterone levels |
| JP2003226639A (ja) * | 2002-01-31 | 2003-08-12 | Hisamitsu Pharmaceut Co Inc | 神経成長因子活性増強剤としてのビタミンk類を含む医薬組成物およびその使用 |
| JP2005306754A (ja) | 2004-04-19 | 2005-11-04 | Towa Corporation 株式会社 | テストステロン増加組成物、テストステロン増加食品、テストステロン増加皮膚外用およびテストステロン増加薬 |
-
2007
- 2007-05-21 JP JP2008522346A patent/JP5110478B2/ja active Active
- 2007-05-21 KR KR1020087027209A patent/KR20090023562A/ko not_active Ceased
- 2007-05-21 WO PCT/JP2007/060341 patent/WO2007148494A1/ja not_active Ceased
- 2007-05-21 US US12/305,403 patent/US8686049B2/en not_active Expired - Fee Related
- 2007-05-21 CN CN2007800233762A patent/CN101472574B/zh not_active Expired - Fee Related
- 2007-05-21 RU RU2008148542/15A patent/RU2431475C2/ru not_active IP Right Cessation
- 2007-05-21 EP EP07743775A patent/EP2033634A4/en not_active Withdrawn
-
2014
- 2014-02-12 US US14/178,409 patent/US20140228447A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| US20140228447A1 (en) | 2014-08-14 |
| CN101472574B (zh) | 2011-06-15 |
| CN101472574A (zh) | 2009-07-01 |
| KR20090023562A (ko) | 2009-03-05 |
| JPWO2007148494A1 (ja) | 2009-11-19 |
| EP2033634A4 (en) | 2010-12-22 |
| RU2431475C2 (ru) | 2011-10-20 |
| EP2033634A1 (en) | 2009-03-11 |
| US20090209653A1 (en) | 2009-08-20 |
| JP5110478B2 (ja) | 2012-12-26 |
| US8686049B2 (en) | 2014-04-01 |
| WO2007148494A1 (ja) | 2007-12-27 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| MM4A | The patent is invalid due to non-payment of fees |
Effective date: 20160522 |