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RU2008148461A - Комбинации вазоактивных веществ и их применение в лечении сексуальных дисфункций - Google Patents

Комбинации вазоактивных веществ и их применение в лечении сексуальных дисфункций Download PDF

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Publication number
RU2008148461A
RU2008148461A RU2008148461/15A RU2008148461A RU2008148461A RU 2008148461 A RU2008148461 A RU 2008148461A RU 2008148461/15 A RU2008148461/15 A RU 2008148461/15A RU 2008148461 A RU2008148461 A RU 2008148461A RU 2008148461 A RU2008148461 A RU 2008148461A
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RU
Russia
Prior art keywords
icarin
derivatives
amentoflavone
gingko biloba
composition
Prior art date
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RU2008148461/15A
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English (en)
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RU2480229C2 (ru
Inventor
Эцио БОМБАРДЕЛЛИ (IT)
Эцио БОМБАРДЕЛЛИ
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Индена С.П.А. (It)
Индена С.П.А.
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Publication of RU2008148461A publication Critical patent/RU2008148461A/ru
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Publication of RU2480229C2 publication Critical patent/RU2480229C2/ru

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    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/335Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/35Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom
    • A61K31/352Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom condensed with carbocyclic rings, e.g. methantheline 
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K36/00Medicinal preparations of undetermined constitution containing material from algae, lichens, fungi or plants, or derivatives thereof, e.g. traditional herbal medicines
    • A61K36/16Ginkgophyta, e.g. Ginkgoaceae (Ginkgo family)
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K36/00Medicinal preparations of undetermined constitution containing material from algae, lichens, fungi or plants, or derivatives thereof, e.g. traditional herbal medicines
    • A61K36/18Magnoliophyta (angiosperms)
    • A61K36/185Magnoliopsida (dicotyledons)
    • A61K36/39Convolvulaceae (Morning-glory family), e.g. bindweed
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K36/00Medicinal preparations of undetermined constitution containing material from algae, lichens, fungi or plants, or derivatives thereof, e.g. traditional herbal medicines
    • A61K36/18Magnoliophyta (angiosperms)
    • A61K36/185Magnoliopsida (dicotyledons)
    • A61K36/53Lamiaceae or Labiatae (Mint family), e.g. thyme, rosemary or lavender
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • A61P15/10Drugs for genital or sexual disorders; Contraceptives for impotence
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K2300/00Mixtures or combinations of active ingredients, wherein at least one active ingredient is fully defined in groups A61K31/00 - A61K41/00

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  • Health & Medical Sciences (AREA)
  • Natural Medicines & Medicinal Plants (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Medical Informatics (AREA)
  • Microbiology (AREA)
  • Mycology (AREA)
  • Botany (AREA)
  • Biotechnology (AREA)
  • Alternative & Traditional Medicine (AREA)
  • Organic Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Endocrinology (AREA)
  • Reproductive Health (AREA)
  • Gynecology & Obstetrics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines Containing Plant Substances (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Saccharide Compounds (AREA)
  • Pyrane Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)

Abstract

1. Композиция для местного применения, содержащая: ! виснадин; ! очищенный экстракт Coleus forskolii; ! этиловый эфир ксимениновой кислоты; ! и, необязательно, ! одно соединение, выбранное из икарина или его производных, или содержащих его экстрактов, аментофлавона и димерных флавонов Gingko biloba. ! 2. Композиция по п.1, где производные икарина включают 7-гидроксиэтил-7-десглюкоикарин, 7-гидроксиэтиликарин, 7-аминоэтиликарин, 7-гидроксиэтил-3-0-рамнозиликарин, 7-аминоэтил-3-рамнозиликарин, 8-дигидроикарин или его гликозиды по 7 и 3 положениям. ! 3. Композиция по п.1, где димерные флавоны Gingko biloba включают аментофлавон. ! 4. Применение комбинации, содержащей: ! виснадин; ! очищенный экстракт Coleus forskolii; ! этиловый эфир ксимениновой кислоты; ! и, необязательно, ! одно соединение, выбранное из икарина или его производных, или содержащих его экстрактов, аментофлавона и димерных флавонов Gingko biloba; ! для получения композиции для местного лечения сексуальных дисфункций.

Claims (4)

1. Композиция для местного применения, содержащая:
виснадин;
очищенный экстракт Coleus forskolii;
этиловый эфир ксимениновой кислоты;
и, необязательно,
одно соединение, выбранное из икарина или его производных, или содержащих его экстрактов, аментофлавона и димерных флавонов Gingko biloba.
2. Композиция по п.1, где производные икарина включают 7-гидроксиэтил-7-десглюкоикарин, 7-гидроксиэтиликарин, 7-аминоэтиликарин, 7-гидроксиэтил-3-0-рамнозиликарин, 7-аминоэтил-3-рамнозиликарин, 8-дигидроикарин или его гликозиды по 7 и 3 положениям.
3. Композиция по п.1, где димерные флавоны Gingko biloba включают аментофлавон.
4. Применение комбинации, содержащей:
виснадин;
очищенный экстракт Coleus forskolii;
этиловый эфир ксимениновой кислоты;
и, необязательно,
одно соединение, выбранное из икарина или его производных, или содержащих его экстрактов, аментофлавона и димерных флавонов Gingko biloba;
для получения композиции для местного лечения сексуальных дисфункций.
RU2008148461/15A 2003-07-11 2008-12-08 Комбинации вазоактивных веществ и их применение в лечении сексуальных дисфункций RU2480229C2 (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
IT001428A ITMI20031428A1 (it) 2003-07-11 2003-07-11 Combinazioni di agenti vasoattivi e loro uso per il trattamento di disfunzioni sessuali
ITMI2003A001428 2003-07-11

Related Parent Applications (1)

Application Number Title Priority Date Filing Date
RU2006100305/15A Division RU2356568C2 (ru) 2003-07-11 2004-07-06 Комбинации вазоактивных веществ и их применение в лечении сексуальных дисфункций

Publications (2)

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RU2008148461A true RU2008148461A (ru) 2010-06-20
RU2480229C2 RU2480229C2 (ru) 2013-04-27

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RU2006100305/15A RU2356568C2 (ru) 2003-07-11 2004-07-06 Комбинации вазоактивных веществ и их применение в лечении сексуальных дисфункций
RU2008148461/15A RU2480229C2 (ru) 2003-07-11 2008-12-08 Комбинации вазоактивных веществ и их применение в лечении сексуальных дисфункций

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Country Status (18)

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US (3) US20060193927A1 (ru)
EP (2) EP1797876B1 (ru)
JP (1) JP4892342B2 (ru)
KR (1) KR101146867B1 (ru)
CN (1) CN1822848B (ru)
AT (2) ATE361087T1 (ru)
AU (1) AU2004255441B2 (ru)
CA (1) CA2532825C (ru)
DE (2) DE602004006271T2 (ru)
DK (2) DK1644014T3 (ru)
ES (2) ES2330795T3 (ru)
IT (1) ITMI20031428A1 (ru)
NO (2) NO335002B1 (ru)
PL (2) PL1644014T3 (ru)
PT (2) PT1644014E (ru)
RU (2) RU2356568C2 (ru)
SI (2) SI1797876T1 (ru)
WO (1) WO2005004890A1 (ru)

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EP2011496A1 (en) * 2007-07-03 2009-01-07 Indena S.P.A. Combinations of vasoactive substances with estrogens and their use in the treatment of female sexual dysfunctions
US20090054497A1 (en) * 2007-08-21 2009-02-26 Nawaz Ahmad Methods for attaining enhanced sexual wellness using anhydrous compositions
US20090197892A1 (en) * 2007-08-21 2009-08-06 Nawaz Ahmad Anhydrous compositions useful for attaining enhanced sexual wellness
US20090054498A1 (en) * 2007-08-21 2009-02-26 Nawaz Ahmad Anhydrous Compositions Useful for Attaining Enhanced Sexual Wellness
CN101606928B (zh) * 2008-06-18 2011-12-07 河南大学 化合物穗花衫双黄酮在制备降血脂药物方面的应用
WO2015099521A2 (en) 2013-12-24 2015-07-02 Biotropics Malaysia Bhd Fruit extracts and extract formulations of canarium odontophyllum as actives and related invention embodiments
US10226418B2 (en) 2014-05-12 2019-03-12 Susie Q, Ltd. Arginine-containing topical composition
US9927614B2 (en) 2015-12-29 2018-03-27 Microsoft Technology Licensing, Llc Augmented reality display system with variable focus
WO2018031216A1 (en) * 2016-08-12 2018-02-15 Steven Rothman Treatment of disorders of sexual arousal with local application of agents that increase membrane excitability
WO2018094377A1 (en) * 2016-11-21 2018-05-24 REV Pharmaceuticals LLC Sexual health enhancement composition
IN201941006993A (ru) * 2019-02-22 2019-03-01
CN112546453B (zh) * 2020-10-15 2022-11-29 西安蓝极医疗电子科技有限公司 基于激光照射治疗男性勃起功能障碍的发光体组件及装置
KR102820913B1 (ko) * 2021-09-08 2025-06-17 주식회사 바이오의생명공학연구소 뮤슬리, 푸나르나바 및 칼라다나의 혼합 발효 추출물을 이용한 자양강장 및 전립선질환 또는 발기부전 개선용 조성물
EP4646204A1 (en) * 2023-01-03 2025-11-12 Initiator Pharma A/S Compound for treatment of erectile dysfunction

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Also Published As

Publication number Publication date
ATE442138T1 (de) 2009-09-15
US8287926B2 (en) 2012-10-16
EP1797876B1 (en) 2009-09-09
PL1644014T3 (pl) 2007-09-28
CA2532825C (en) 2013-12-10
RU2006100305A (ru) 2006-06-10
JP4892342B2 (ja) 2012-03-07
ES2330795T3 (es) 2009-12-15
EP1797876A1 (en) 2007-06-20
NO20140193L (no) 2006-02-10
CN1822848A (zh) 2006-08-23
DE602004023137D1 (de) 2009-10-22
PT1797876E (pt) 2009-11-02
DE602004006271D1 (de) 2007-06-14
RU2356568C2 (ru) 2009-05-27
US20120009283A1 (en) 2012-01-12
ES2286658T3 (es) 2007-12-01
AU2004255441A1 (en) 2005-01-20
WO2005004890A1 (en) 2005-01-20
KR101146867B1 (ko) 2012-05-16
HK1091123A1 (en) 2007-01-12
JP2009513518A (ja) 2009-04-02
ATE361087T1 (de) 2007-05-15
DK1644014T3 (da) 2007-09-10
DK1797876T3 (da) 2009-12-21
EP1644014B1 (en) 2007-05-02
SI1644014T1 (sl) 2007-08-31
US8092844B2 (en) 2012-01-10
ITMI20031428A1 (it) 2005-01-12
AU2004255441B2 (en) 2010-02-25
NO20060679L (no) 2006-02-10
PL1797876T3 (pl) 2009-12-31
NO335002B1 (no) 2014-08-18
NO340484B1 (no) 2017-05-02
CA2532825A1 (en) 2005-01-20
EP1644014A1 (en) 2006-04-12
SI1797876T1 (sl) 2009-12-31
US20060193927A1 (en) 2006-08-31
PT1644014E (pt) 2007-07-31
CN1822848B (zh) 2010-05-26
DE602004006271T2 (de) 2008-01-10
RU2480229C2 (ru) 2013-04-27
US20090269426A1 (en) 2009-10-29
KR20060028746A (ko) 2006-03-31

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Effective date: 20170707