RU2007122284A - Предотвращениеи вертикальных инфекций, вызываемых эндопаразитами - Google Patents
Предотвращениеи вертикальных инфекций, вызываемых эндопаразитами Download PDFInfo
- Publication number
- RU2007122284A RU2007122284A RU2007122284/15A RU2007122284A RU2007122284A RU 2007122284 A RU2007122284 A RU 2007122284A RU 2007122284/15 A RU2007122284/15 A RU 2007122284/15A RU 2007122284 A RU2007122284 A RU 2007122284A RU 2007122284 A RU2007122284 A RU 2007122284A
- Authority
- RU
- Russia
- Prior art keywords
- endoparasites
- endoparasitis
- prevention
- infections caused
- acting against
- Prior art date
Links
- 208000015181 infectious disease Diseases 0.000 title claims abstract 5
- 230000002265 prevention Effects 0.000 title 1
- 244000079386 endoparasite Species 0.000 claims abstract 8
- 108010002156 Depsipeptides Proteins 0.000 claims abstract 4
- 241000282472 Canis lupus familiaris Species 0.000 claims abstract 2
- 239000003814 drug Substances 0.000 claims abstract 2
- 229940079593 drug Drugs 0.000 claims abstract 2
- 108010056417 emodepside Proteins 0.000 claims abstract 2
- ZMQMTKVVAMWKNY-YSXLEBCMSA-N emodepside Chemical compound C([C@@H]1C(=O)N(C)[C@@H](CC(C)C)C(=O)O[C@H](C)C(=O)N(C)[C@H](C(O[C@H](CC=2C=CC(=CC=2)N2CCOCC2)C(=O)N(C)[C@@H](CC(C)C)C(=O)O[C@H](C)C(=O)N(C)[C@@H](CC(C)C)C(=O)O1)=O)CC(C)C)C(C=C1)=CC=C1N1CCOCC1 ZMQMTKVVAMWKNY-YSXLEBCMSA-N 0.000 claims abstract 2
- 229960001575 emodepside Drugs 0.000 claims abstract 2
- OHRURASPPZQGQM-GCCNXGTGSA-N romidepsin Chemical compound O1C(=O)[C@H](C(C)C)NC(=O)C(=C/C)/NC(=O)[C@H]2CSSCC\C=C\[C@@H]1CC(=O)N[C@H](C(C)C)C(=O)N2 OHRURASPPZQGQM-GCCNXGTGSA-N 0.000 claims abstract 2
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
- A61K38/04—Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
- A61K38/15—Depsipeptides; Derivatives thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/10—Anthelmintics
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
- Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
- Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- General Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical & Material Sciences (AREA)
- Immunology (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Epidemiology (AREA)
- Gastroenterology & Hepatology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Tropical Medicine & Parasitology (AREA)
- Communicable Diseases (AREA)
- Oncology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Peptides Or Proteins (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Medicinal Preparation (AREA)
Abstract
1. Применение депсипептидов, действующих против эндопаразитов, для получения лекарственных средств для предотвращения вертикальной инфекции, вызываемой эндопаразитами.2. Применение по п.1, причем в качестве депсипептида, действующего против эндопаразитов, используют эмодепсид.3. Применение по п.1 или 2 для предотвращения вертикальной инфекции, вызываемой эндопаразитами, у собак.
Claims (3)
1. Применение депсипептидов, действующих против эндопаразитов, для получения лекарственных средств для предотвращения вертикальной инфекции, вызываемой эндопаразитами.
2. Применение по п.1, причем в качестве депсипептида, действующего против эндопаразитов, используют эмодепсид.
3. Применение по п.1 или 2 для предотвращения вертикальной инфекции, вызываемой эндопаразитами, у собак.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE102004055316A DE102004055316A1 (de) | 2004-11-16 | 2004-11-16 | Verhinderung vertikaler Endoparasiten-Infektionen |
| DE102004055316.5 | 2004-11-16 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| RU2007122284A true RU2007122284A (ru) | 2008-12-27 |
| RU2405565C2 RU2405565C2 (ru) | 2010-12-10 |
Family
ID=35767587
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| RU2007122284/15A RU2405565C2 (ru) | 2004-11-16 | 2005-11-03 | Предотвращение вертикальных инфекций, вызываемых эндопаразитами |
Country Status (29)
| Country | Link |
|---|---|
| US (1) | US20090215678A1 (ru) |
| EP (1) | EP1814572B1 (ru) |
| JP (1) | JP5078619B2 (ru) |
| KR (1) | KR101280511B1 (ru) |
| CN (1) | CN101102785B (ru) |
| AR (1) | AR052133A1 (ru) |
| AT (1) | ATE469652T1 (ru) |
| AU (1) | AU2005306070B2 (ru) |
| BR (1) | BRPI0518172A (ru) |
| CA (1) | CA2587537C (ru) |
| CR (1) | CR9108A (ru) |
| DE (2) | DE102004055316A1 (ru) |
| DK (1) | DK1814572T3 (ru) |
| ES (1) | ES2345265T3 (ru) |
| HR (1) | HRP20100471T1 (ru) |
| IL (1) | IL183200A (ru) |
| MX (1) | MX2007005766A (ru) |
| MY (1) | MY142727A (ru) |
| NO (1) | NO341472B1 (ru) |
| NZ (1) | NZ555117A (ru) |
| PE (1) | PE20061079A1 (ru) |
| PL (1) | PL1814572T3 (ru) |
| PT (1) | PT1814572E (ru) |
| RU (1) | RU2405565C2 (ru) |
| SI (1) | SI1814572T1 (ru) |
| TW (1) | TWI358293B (ru) |
| UA (1) | UA91694C2 (ru) |
| WO (1) | WO2006053641A1 (ru) |
| ZA (1) | ZA200703982B (ru) |
Families Citing this family (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE102008022520A1 (de) * | 2008-05-07 | 2009-11-12 | Bayer Animal Health Gmbh | Feste Arzneimittelformulierung mit verzögerter Freisetzung |
| KR101978620B1 (ko) * | 2011-12-21 | 2019-08-28 | 바이엘 파마 악티엔게젤샤프트 | 무정형 에모뎁시드를 함유하는 제제 |
| SG10202103403SA (en) | 2015-05-20 | 2021-05-28 | Boehringer Ingelheim Animal Health Usa Inc | Anthelmintic depsipeptide compounds |
| NZ743913A (en) | 2015-12-28 | 2019-04-26 | Boehringer Ingelheim Animal Health Usa Inc | Anthelmintic depsipeptide compounds |
| US11382949B2 (en) | 2016-11-16 | 2022-07-12 | Boehringer Ingelheim Animal Health USA Inc. | Anthelmintic depsipeptide compounds |
| EP3480195A1 (en) | 2017-11-07 | 2019-05-08 | Bayer Animal Health GmbH | Method for the synthesis of cyclic depsipeptides |
| EP3676265B1 (en) | 2017-11-07 | 2025-08-20 | Elanco Animal Health GmbH | Method for the synthesis of cyclic depsipeptides |
Family Cites Families (21)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE2362539C2 (de) * | 1973-12-17 | 1986-05-07 | Merck Patent Gmbh, 6100 Darmstadt | 2-Acyl-4-oxo-1,2,3,6,7,11b-hexahydro-4H-pyrazino[2,1-a]isochinoline, Verfahren zu ihrer Herstellung und diese Verbindungen enthaltende Arzneimittel |
| NO176766C (no) * | 1989-02-07 | 1995-05-24 | Meiji Seika Kaisha | Fremgangsmåte for fremstilling av en forbindelse med anthelmintaktivitet |
| ATE211466T1 (de) * | 1992-03-17 | 2002-01-15 | Fujisawa Pharmaceutical Co | Depsipeptide, herstellung und anwendung |
| DE4317458A1 (de) * | 1992-06-11 | 1993-12-16 | Bayer Ag | Verwendung von cyclischen Depsipeptiden mit 18 Ringatomen zur Bekämpfung von Endoparasiten, neue cyclische Depsipeptide mit 18 Ringatomen und Verfahren zu ihrer Herstellung |
| KR100309091B1 (ko) * | 1993-02-19 | 2001-12-28 | 이치로 키타사토 | 환상 데프시펩티드 pf 1022의 유도체 |
| WO1994025038A1 (en) * | 1993-05-05 | 1994-11-10 | Palo Alto Medical Foundation | Use of rifamycin derivatives for the manufacture of a medicament for the treatment of toxoplasmosis |
| DE4317457A1 (de) * | 1993-05-26 | 1994-12-01 | Bayer Ag | Octacyclodepsipeptide mit endoparasitizider Wirkung |
| DE4317432A1 (de) * | 1993-05-26 | 1994-12-01 | Bayer Ag | Octacyclodepsipeptide mit endoparasitizider Wirkung |
| EP0718293B1 (en) * | 1993-09-06 | 2002-03-13 | Fujisawa Pharmaceutical Co., Ltd. | Cyclodepsipeptide compound |
| DE4400464A1 (de) * | 1994-01-11 | 1995-07-13 | Bayer Ag | Endoparasitizide Mittel |
| DE4401389A1 (de) * | 1994-01-19 | 1995-07-20 | Bayer Ag | Verwendung von cyclischen Depsipeptiden mit 12 Ringatomen zur Bekämpfung von Endoparasiten, neue cyclische Depsipeptide mit 12 Ringatomen und Verfahren zu ihrer Herstellung |
| DE4406025A1 (de) * | 1994-02-24 | 1995-08-31 | Bayer Ag | Milchsäure-haltige cyclische Depsipeptide mit 18 Ringatomen als endoparasitizide Mittel und Verfahren zu ihrer Herstellung |
| DE4437198A1 (de) * | 1994-10-18 | 1996-04-25 | Bayer Ag | Verfahren zur Sulfonylierung, Sulfenylierung und Phosphorylierung von cyclischen Depsipeptiden |
| WO1997002256A1 (en) * | 1995-06-30 | 1997-01-23 | Fujisawa Pharmaceutical Co., Ltd. | Depsipeptide derivative, process for production thereof, and novel intermediate therefor |
| ATE299871T1 (de) * | 1995-09-22 | 2005-08-15 | Meiji Seika Kaisha | Neue zyklische depsipeptid pf1022 derivate |
| DE19545639A1 (de) * | 1995-12-07 | 1997-06-12 | Bayer Ag | Verfahren zur Herstellung von substituierten Arylmilchsäure-haltigen Cyclodepsipeptiden mit 24 Ringatomen |
| DE19962147A1 (de) * | 1999-12-22 | 2001-06-28 | Bayer Ag | Schädlingsbekämpfungsmittel / PF 1022-221 |
| US20010036922A1 (en) * | 2000-04-03 | 2001-11-01 | Benchaoui Hafid Abdelaali | Method of treating a parasitic infection |
| GB0008353D0 (en) * | 2000-04-03 | 2000-05-24 | Pfizer Ltd | Method of treating a parasitic infection |
| DE10358525A1 (de) * | 2003-12-13 | 2005-07-07 | Bayer Healthcare Ag | Endoparasitizide Mittel zur topischen Applikation |
| DE102005011779A1 (de) * | 2005-03-11 | 2006-09-14 | Bayer Healthcare Ag | Endoparasitizide Mittel |
-
2004
- 2004-11-16 DE DE102004055316A patent/DE102004055316A1/de not_active Withdrawn
-
2005
- 2005-11-03 ES ES05800013T patent/ES2345265T3/es not_active Expired - Lifetime
- 2005-11-03 WO PCT/EP2005/011748 patent/WO2006053641A1/de not_active Ceased
- 2005-11-03 HR HR20100471T patent/HRP20100471T1/hr unknown
- 2005-11-03 BR BRPI0518172-0A patent/BRPI0518172A/pt not_active Application Discontinuation
- 2005-11-03 CA CA2587537A patent/CA2587537C/en not_active Expired - Lifetime
- 2005-11-03 PT PT05800013T patent/PT1814572E/pt unknown
- 2005-11-03 EP EP05800013A patent/EP1814572B1/de not_active Expired - Lifetime
- 2005-11-03 DK DK05800013.4T patent/DK1814572T3/da active
- 2005-11-03 US US11/719,379 patent/US20090215678A1/en not_active Abandoned
- 2005-11-03 DE DE502005009697T patent/DE502005009697D1/de not_active Expired - Lifetime
- 2005-11-03 JP JP2007541733A patent/JP5078619B2/ja not_active Expired - Lifetime
- 2005-11-03 KR KR1020077011479A patent/KR101280511B1/ko not_active Expired - Lifetime
- 2005-11-03 MX MX2007005766A patent/MX2007005766A/es active IP Right Grant
- 2005-11-03 UA UAA200706853A patent/UA91694C2/ru unknown
- 2005-11-03 NZ NZ555117A patent/NZ555117A/en not_active IP Right Cessation
- 2005-11-03 RU RU2007122284/15A patent/RU2405565C2/ru active
- 2005-11-03 AU AU2005306070A patent/AU2005306070B2/en not_active Expired
- 2005-11-03 CN CN2005800466551A patent/CN101102785B/zh not_active Expired - Lifetime
- 2005-11-03 AT AT05800013T patent/ATE469652T1/de active
- 2005-11-03 SI SI200531078T patent/SI1814572T1/sl unknown
- 2005-11-03 PL PL05800013T patent/PL1814572T3/pl unknown
- 2005-11-15 AR ARP050104792A patent/AR052133A1/es not_active Application Discontinuation
- 2005-11-15 MY MYPI20055348A patent/MY142727A/en unknown
- 2005-11-15 TW TW094140003A patent/TWI358293B/zh not_active IP Right Cessation
- 2005-11-15 PE PE2005001335A patent/PE20061079A1/es not_active Application Discontinuation
-
2007
- 2007-05-09 CR CR9108A patent/CR9108A/es unknown
- 2007-05-15 IL IL183200A patent/IL183200A/en active IP Right Grant
- 2007-05-16 ZA ZA200703982A patent/ZA200703982B/xx unknown
- 2007-06-13 NO NO20073023A patent/NO341472B1/no unknown
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| TK4A | Correction to the publication in the bulletin (patent) |
Free format text: AMENDMENT TO CHAPTER -FG4A- IN JOURNAL: 34-2010 |
|
| PC41 | Official registration of the transfer of exclusive right |
Effective date: 20130207 |