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PT900793E - Derivados de cicloalquilaminometilpirrolidina - Google Patents

Derivados de cicloalquilaminometilpirrolidina

Info

Publication number
PT900793E
PT900793E PT97919690T PT97919690T PT900793E PT 900793 E PT900793 E PT 900793E PT 97919690 T PT97919690 T PT 97919690T PT 97919690 T PT97919690 T PT 97919690T PT 900793 E PT900793 E PT 900793E
Authority
PT
Portugal
Prior art keywords
group
carbon atoms
alkyl
hydrogen atom
halogenomethyl
Prior art date
Application number
PT97919690T
Other languages
English (en)
Inventor
Katsuhiro Kawakami
Makoto Takemura
Youichi Kimura
Hitoshi Ohki
Original Assignee
Daiichi Seiyaku Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Daiichi Seiyaku Co filed Critical Daiichi Seiyaku Co
Publication of PT900793E publication Critical patent/PT900793E/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pyrrole Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
  • Cosmetics (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Silicon Compounds (AREA)
  • Liquid Crystal (AREA)
  • Pyridine Compounds (AREA)
PT97919690T 1996-04-24 1997-04-24 Derivados de cicloalquilaminometilpirrolidina PT900793E (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP10233496 1996-04-24

Publications (1)

Publication Number Publication Date
PT900793E true PT900793E (pt) 2002-11-29

Family

ID=14324624

Family Applications (1)

Application Number Title Priority Date Filing Date
PT97919690T PT900793E (pt) 1996-04-24 1997-04-24 Derivados de cicloalquilaminometilpirrolidina

Country Status (17)

Country Link
US (1) US6194434B1 (pt)
EP (1) EP0900793B1 (pt)
JP (1) JP4127322B2 (pt)
KR (1) KR100458146B1 (pt)
CN (1) CN1116295C (pt)
AT (1) ATE221063T1 (pt)
AU (1) AU726378B2 (pt)
BR (1) BR9708824A (pt)
CA (1) CA2251927C (pt)
DE (1) DE69714249T2 (pt)
DK (1) DK0900793T3 (pt)
EA (1) EA000878B1 (pt)
ES (1) ES2180975T3 (pt)
ID (1) ID16655A (pt)
PT (1) PT900793E (pt)
TW (1) TW425394B (pt)
WO (1) WO1997040037A1 (pt)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR100768034B1 (ko) 1999-03-17 2007-10-17 다이이찌 세이야꾸 가부시기가이샤 의약 조성물
MXPA04009026A (es) * 2002-03-18 2005-01-25 Kyorin Seiyaku Kk Derivados de acido 10- (3- ciclopropilaminometil -1-pirrolidinil) piridobenzoxazin- carboxilico efectivos contra bacterias resistentes a farmacos.
CA2536429C (en) 2003-09-10 2012-02-14 Kyorin Pharmaceutical Co., Ltd. 7-(4-substituted-3-cyclopropylaminomethyl-1-pyrrolidinyl) quinolonecarboxylic acid derivative
GB0428250D0 (en) * 2004-12-23 2005-01-26 Novartis Ag Organic compounds
US8222407B2 (en) 2007-05-24 2012-07-17 Kyorin Pharmaceutical Co., Ltd. Mutilin derivative having heterocyclic aromatic ring carboxylic acid structure in substituent at 14-position
AU2016234411C1 (en) * 2015-03-13 2020-04-30 Kyorin Pharmaceutical Co., Ltd. Respiratory infection treating agent

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IE55898B1 (en) 1982-09-09 1991-02-14 Warner Lambert Co Antibacterial agents
US4657913A (en) * 1985-04-18 1987-04-14 Warner-Lambert Company Trifluoro- quinoline -3- carboxylic acids and their use as anti-bacterial agents
JPH0696572B2 (ja) * 1985-07-17 1994-11-30 大日本製薬株式会社 ピリドンカルボン酸誘導体、そのエステルおよびその塩
US4771055A (en) * 1986-07-28 1988-09-13 Warner-Lambert Company 7-[[3-(aminomethyl)-3-alkyl]-1-pyrrolidinyl]-quinoline-carboxylic acids
US4965273A (en) * 1986-10-08 1990-10-23 Bristol-Myers Company Certain 1-tertiary-butyl-naphthyridone carboxylic acid derivatives anti-bacterial agents
ZA877471B (en) * 1986-10-08 1988-04-05 Bristol-Myers Company 1-tertiary-alkyl-substituted naphthyridine-and quinoline-carboxylic acid antibacterial agents
US4954507A (en) * 1986-10-08 1990-09-04 Bristol-Myers Company 1-tertiary-alkyl-substituted naphthyridine carboxylic acid antibacterial agents
US4780468A (en) * 1987-08-07 1988-10-25 Warner-Lambert Company 8-trifluoromethyl quinolones as antibacterial agents
US5173484A (en) * 1988-02-05 1992-12-22 Bayer Aktiengesellschaft Quinolone- and naphthyridone carboxylic acid derivatives, process for their production, antibacterial compositions and feed additives containing them
DE3814517A1 (de) * 1988-02-05 1989-08-17 Bayer Ag Chinolon- und naphthyridoncarbonsaeurederivate, verfahren zu ihrer herstellung und sie enthaltende antibakterielle mittel und futterzusatzstoffe
IL90062A (en) * 1988-04-27 1994-10-07 Daiichi Seiyaku Co Pyridonecarboxylic acid derivatives, their preparation and pharmaceutical compositions containing them

Also Published As

Publication number Publication date
JP4127322B2 (ja) 2008-07-30
ID16655A (id) 1997-10-30
KR20000010578A (ko) 2000-02-15
AU726378B2 (en) 2000-11-02
EP0900793A1 (en) 1999-03-10
DE69714249D1 (en) 2002-08-29
TW425394B (en) 2001-03-11
AU2407297A (en) 1997-11-12
ES2180975T3 (es) 2003-02-16
KR100458146B1 (ko) 2005-06-13
CN1222151A (zh) 1999-07-07
CA2251927A1 (en) 1997-10-30
EA199800952A1 (ru) 1999-04-29
ATE221063T1 (de) 2002-08-15
WO1997040037A1 (en) 1997-10-30
EP0900793B1 (en) 2002-07-24
HK1018786A1 (en) 2000-01-07
DE69714249T2 (de) 2003-03-27
EA000878B1 (ru) 2000-06-26
BR9708824A (pt) 1999-08-03
DK0900793T3 (da) 2002-10-14
CN1116295C (zh) 2003-07-30
CA2251927C (en) 2005-02-15
US6194434B1 (en) 2001-02-27
EP0900793A4 (en) 1999-07-07

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