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PT761218E - Processo para preparar comprimidos revestidos com polimeros compreendendo amoxicilina e clavunalato - Google Patents

Processo para preparar comprimidos revestidos com polimeros compreendendo amoxicilina e clavunalato Download PDF

Info

Publication number
PT761218E
PT761218E PT96202848T PT96202848T PT761218E PT 761218 E PT761218 E PT 761218E PT 96202848 T PT96202848 T PT 96202848T PT 96202848 T PT96202848 T PT 96202848T PT 761218 E PT761218 E PT 761218E
Authority
PT
Portugal
Prior art keywords
tablet
weight
film coating
clavulanate
amoxycillin
Prior art date
Application number
PT96202848T
Other languages
English (en)
Portuguese (pt)
Inventor
Nigel Philip Davidson
Creighton Pierce Conley
Original Assignee
Smithkline Beecham Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=10754044&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=PT761218(E) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Smithkline Beecham Corp filed Critical Smithkline Beecham Corp
Publication of PT761218E publication Critical patent/PT761218E/pt

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/42Oxazoles
    • A61K31/424Oxazoles condensed with heterocyclic ring systems, e.g. clavulanic acid
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425Thiazoles
    • A61K31/429Thiazoles condensed with heterocyclic ring systems
    • A61K31/43Compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula, e.g. penicillins, penems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/28Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806Coating materials
    • A61K9/2833Organic macromolecular compounds
    • A61K9/2853Organic macromolecular compounds obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyethylene glycol, polyethylene oxide, poloxamers, poly(lactide-co-glycolide)
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/28Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806Coating materials
    • A61K9/2833Organic macromolecular compounds
    • A61K9/286Polysaccharides, e.g. gums; Cyclodextrin
    • A61K9/2866Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/28Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2893Tablet coating processes
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Communicable Diseases (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oncology (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
PT96202848T 1994-04-23 1995-04-19 Processo para preparar comprimidos revestidos com polimeros compreendendo amoxicilina e clavunalato PT761218E (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB9408117A GB9408117D0 (en) 1994-04-23 1994-04-23 Pharmaceutical formulations

Publications (1)

Publication Number Publication Date
PT761218E true PT761218E (pt) 2001-03-30

Family

ID=10754044

Family Applications (4)

Application Number Title Priority Date Filing Date
PT00204182T PT1093813E (pt) 1994-04-23 1995-04-19 Processo para preparacao de comprimidos revestidos de polimero compreendendo amoxicilina e clavulanato revestidos com uma pelicula polimerica aquosa
PT96202848T PT761218E (pt) 1994-04-23 1995-04-19 Processo para preparar comprimidos revestidos com polimeros compreendendo amoxicilina e clavunalato
PT95917937T PT758235E (pt) 1994-04-23 1995-04-19 Comprimido revestido com polimero compreendendo amoxicilina e clavulanato
PT99200891T PT978276E (pt) 1994-04-23 1995-04-19 Comprimidos com revestimento de polimero que compreendem amoxicilina e clavulanato

Family Applications Before (1)

Application Number Title Priority Date Filing Date
PT00204182T PT1093813E (pt) 1994-04-23 1995-04-19 Processo para preparacao de comprimidos revestidos de polimero compreendendo amoxicilina e clavulanato revestidos com uma pelicula polimerica aquosa

Family Applications After (2)

Application Number Title Priority Date Filing Date
PT95917937T PT758235E (pt) 1994-04-23 1995-04-19 Comprimido revestido com polimero compreendendo amoxicilina e clavulanato
PT99200891T PT978276E (pt) 1994-04-23 1995-04-19 Comprimidos com revestimento de polimero que compreendem amoxicilina e clavulanato

Country Status (35)

Country Link
US (1) US6051255A (fr)
EP (5) EP1243267A3 (fr)
JP (1) JP3622975B2 (fr)
CN (1) CN1134258C (fr)
AP (2) AP564A (fr)
AT (6) ATE223706T1 (fr)
AU (1) AU684949B2 (fr)
BG (1) BG62842B1 (fr)
BR (1) BR9507502A (fr)
CA (1) CA2188496A1 (fr)
CZ (2) CZ294168B6 (fr)
DE (5) DE69519093T2 (fr)
DK (4) DK0761218T3 (fr)
DZ (1) DZ1876A1 (fr)
ES (4) ES2182754T3 (fr)
FI (1) FI964249A7 (fr)
GB (1) GB9408117D0 (fr)
GR (2) GR3035031T3 (fr)
HK (1) HK1050992A1 (fr)
HU (1) HU228399B1 (fr)
IL (1) IL113433A (fr)
MA (1) MA23528A1 (fr)
MY (1) MY115351A (fr)
NO (1) NO310703B1 (fr)
NZ (1) NZ285080A (fr)
OA (1) OA10377A (fr)
PL (1) PL316966A1 (fr)
PT (4) PT1093813E (fr)
RO (1) RO116997B1 (fr)
RU (1) RU2152213C1 (fr)
SA (1) SA95160343B1 (fr)
SI (1) SI0758235T1 (fr)
SK (1) SK282594B6 (fr)
WO (1) WO1995028927A1 (fr)
ZA (1) ZA953236B (fr)

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* Cited by examiner, † Cited by third party
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US20030109503A1 (en) * 1995-06-06 2003-06-12 Smithkline Beecham P.L.C. Pharmaceutical formulations comprising clavulanic acid alone or in combination with other beta-lactam antibiotics
ATE208618T1 (de) 1995-09-07 2001-11-15 Smithkline Beecham Corp Verwendung einer amoxicillin und clavulanat enthaltenden paediatrischen pharmazeutischen formulierung
AT403375B (de) * 1995-11-15 1998-01-26 Biochemie Gmbh Verfahren zur fällung von alkalisalzen der clavulansäure
TWI225402B (en) * 1996-03-13 2004-12-21 Biochemie Gmbh Auxiliary-free agglomerates
AT407701B (de) * 1996-08-12 2001-05-25 Biochemie Gmbh Zur direkttablettierung geeignete mischung, die als wesentliche komponenten amoxicillin-trihydrat und das kaliumsalz der clavulansäure enthält und verfahren zur herstellung dieser mischung
GB9613470D0 (en) 1996-06-27 1996-08-28 Ciba Geigy Ag Small solid oral dosage form
GB9616536D0 (en) * 1996-08-06 1996-09-25 Quadrant Holdings Cambridge Co-amoxiclav dosage form
GB9617780D0 (en) 1996-08-24 1996-10-02 Smithkline Beecham Plc Method of treatment
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US20030124187A1 (en) * 1997-02-14 2003-07-03 Smithkline Beecham Laboratoires Pharmaceutiques, Pharmaceutical formulations comprising amoxycillin and clavulanate
SK110299A3 (en) * 1997-02-14 2000-08-14 Smithkline Beecham Lab Pharmaceutical formulations comprising amoxocyllin and clavulanate, preparation method and use thereof
TR200000529T2 (tr) * 1997-08-29 2000-08-21 Dsm N.V. İçinde eksipiyan olmayan granüller
EP1032425A1 (fr) 1997-10-31 2000-09-06 Monsanto Company Enrobage de comprimes a l'aide de gomme gellane
WO2000041478A2 (fr) 1999-04-01 2000-07-20 Dsm N.V. Agglomerats obtenus par cristallisation
US6294199B1 (en) * 1999-04-13 2001-09-25 Beecham Pharmaceuticals (Pte) Limited Method of treating a bacterial infection comprising administering amoxycillin
US7250176B1 (en) * 1999-04-13 2007-07-31 Beecham Pharmaceuticals (Pte) Limited Method of treating a bacterial infection
US6878386B1 (en) 1999-04-13 2005-04-12 Beecham Pharmaceuticals (Pte) Limited Method of treating a bacterial infection comprising amoxycillin and potassium clavulanate
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US20060083759A1 (en) * 2002-07-17 2006-04-20 Aleksander Resman Stabilization of the profile of release of active substances from a formulation
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CL2008003230A1 (es) * 2007-11-01 2009-11-27 Sanofi Aventis Healthcare Pty Ltd Composicion de recubrimiento de tableta que comprende polimero celulosico, plastificante, edulcorante y composicion de sabor en polvo la que comprende saborizante asociado con portador solido; fluido de recubrimiento de tableta que comprende dicha composicion; tableta farmaceutica; proceso de preparacion de dicha tableta.
CN102596184B (zh) * 2009-09-18 2015-03-11 赛诺菲 稳定性提高的(z)-2-氰基-3-羟基-丁-2-烯酸-(4’-三氟甲基苯基)-酰胺片剂制剂
TR200909787A2 (tr) 2009-12-25 2011-07-21 Bi̇lgi̇ç Mahmut Üçüncü kuşak bir sefalosporin ve klavulanik asit içeren farmasötik formülasyonlar.
TR201000686A1 (tr) 2010-01-29 2011-08-22 B�Lg�� Mahmut Bakteriyel enfeksiyonların tedavisinde suda çözünebilir sefdinir ve klavulanik asit formülasyonları.@
TR201000687A1 (tr) 2010-01-29 2011-08-22 Bi̇lgi̇ç Mahmut Aktif madde olarak sefiksim ve klavulanik asit içeren efervesan formülasyonlar
TR201000688A2 (tr) 2010-01-29 2011-08-22 B�Lg�� Mahmut Aktif madde olarak sefaklor ve klavulanik asit içeren efervesan formülasyonlar.
JP6041591B2 (ja) * 2011-09-13 2016-12-14 大日本住友製薬株式会社 イルベサルタンとアムロジピンまたはその塩を含有する安定化された医薬組成物
US9387250B2 (en) 2013-03-15 2016-07-12 Rutgers, The State University Of New Jersey Therapeutic compositions for bone repair

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GB9408117D0 (en) * 1994-04-23 1994-06-15 Smithkline Beecham Corp Pharmaceutical formulations
ES2202004T3 (es) * 1999-04-13 2004-04-01 Beecham Pharmaceuticals (Pte) Limited Novedoso procedimiento de tratamiento usando un fuerte regimen de dosificacion de amoxicilina y clavulanato potasico.
WO2002030392A2 (fr) * 2000-10-12 2002-04-18 Beecham Pharmaceuticals (Pte) Limited Nouvelle formulation

Also Published As

Publication number Publication date
EP1093813A3 (fr) 2001-05-30
EP0978276B1 (fr) 2002-09-11
GR3035031T3 (en) 2001-03-30
DZ1876A1 (fr) 2002-02-17
ZA953236B (en) 1995-12-27
PT978276E (pt) 2003-01-31
CZ294168B6 (cs) 2004-10-13
ATE223706T1 (de) 2002-09-15
OA10377A (en) 2001-11-21
EP0978276A3 (fr) 2000-04-12
WO1995028927A1 (fr) 1995-11-02
AT5349U1 (de) 2002-06-25
HK1009936A1 (en) 1999-06-11
RO116997B1 (ro) 2001-09-28
HU9602922D0 (en) 1996-12-30
HK1021860A1 (en) 2000-07-07
ES2182754T3 (es) 2003-03-16
EP1093813A2 (fr) 2001-04-25
PT1093813E (pt) 2003-02-28
HK1050992A1 (en) 2003-07-18
FI964249L (fi) 1996-10-22
AP9500733A0 (en) 1995-04-30
IL113433A (en) 2003-06-24
RU2152213C1 (ru) 2000-07-10
ES2161288T3 (es) 2001-12-01
CN1134258C (zh) 2004-01-14
EP0758235A1 (fr) 1997-02-19
SI0758235T1 (en) 2001-10-31
AU2406895A (en) 1995-11-16
DE69528204D1 (de) 2002-10-17
DE69521799D1 (de) 2001-08-23
CZ11376U1 (cs) 2001-07-12
MA23528A1 (fr) 1995-12-31
CZ309096A3 (en) 1997-04-16
FI964249A0 (fi) 1996-10-22
NO964488L (no) 1996-12-17
AU684949B2 (en) 1998-01-08
AT5350U1 (de) 2002-06-25
DE69519093T2 (de) 2001-07-19
NO964488D0 (no) 1996-10-22
DE69528204T2 (de) 2003-08-07
EP0761218B1 (fr) 2000-10-11
GB9408117D0 (en) 1994-06-15
HUT76335A (en) 1997-08-28
US6051255A (en) 2000-04-18
EP0758235B1 (fr) 2001-07-18
DK0978276T3 (da) 2003-01-20
HK1027024A1 (en) 2001-01-05
MY115351A (en) 2003-05-31
HK1036404A1 (en) 2002-01-04
DK0761218T3 (da) 2000-12-18
EP0761218A1 (fr) 1997-03-12
DE69519093D1 (de) 2000-11-16
AP564A (en) 1996-11-21
DK1093813T3 (da) 2003-02-17
DE69528608D1 (de) 2002-11-21
SA95160343B1 (ar) 2005-05-04
SK282594B6 (sk) 2002-10-08
AP9600868A0 (en) 1996-10-31
FI964249A7 (fi) 1996-10-22
ATE196845T1 (de) 2000-10-15
EP1243267A2 (fr) 2002-09-25
NZ285080A (en) 1998-05-27
ATE226074T1 (de) 2002-11-15
PT758235E (pt) 2001-10-31
DE29522153U1 (de) 2000-04-06
PL316966A1 (en) 1997-03-03
CN1149829A (zh) 1997-05-14
ES2152485T3 (es) 2001-02-01
NO310703B1 (no) 2001-08-20
SK135496A3 (en) 1997-05-07
BG62842B1 (bg) 2000-09-29
EP0978276A2 (fr) 2000-02-09
ES2180251T3 (es) 2003-02-01
ATE203161T1 (de) 2001-08-15
CA2188496A1 (fr) 1995-11-02
IL113433A0 (en) 1995-07-31
BG100933A (en) 1997-07-31
EP1093813B1 (fr) 2002-10-16
DK0758235T3 (da) 2001-10-29
JP3622975B2 (ja) 2005-02-23
JPH09512027A (ja) 1997-12-02
EP1243267A3 (fr) 2002-10-30
GR3036844T3 (en) 2002-01-31
DE69521799T2 (de) 2002-06-13
DE69528608T2 (de) 2003-06-26
HU228399B1 (en) 2013-03-28
BR9507502A (pt) 1997-09-02

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