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PE20221462A1 - Composiciones y metodos para la activacion de integrinas - Google Patents

Composiciones y metodos para la activacion de integrinas

Info

Publication number
PE20221462A1
PE20221462A1 PE2022000784A PE2022000784A PE20221462A1 PE 20221462 A1 PE20221462 A1 PE 20221462A1 PE 2022000784 A PE2022000784 A PE 2022000784A PE 2022000784 A PE2022000784 A PE 2022000784A PE 20221462 A1 PE20221462 A1 PE 20221462A1
Authority
PE
Peru
Prior art keywords
protein
alpha6
alpha7
alpha3
integrin
Prior art date
Application number
PE2022000784A
Other languages
English (en)
Inventor
Patrick Andre
Chun Chen
Scott Turner
Original Assignee
Pliant Therapeutics Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pliant Therapeutics Inc filed Critical Pliant Therapeutics Inc
Publication of PE20221462A1 publication Critical patent/PE20221462A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K39/00Medicinal preparations containing antigens or antibodies
    • A61K39/395Antibodies; Immunoglobulins; Immune serum, e.g. antilymphocytic serum
    • A61K39/39533Antibodies; Immunoglobulins; Immune serum, e.g. antilymphocytic serum against materials from animals
    • A61K39/39541Antibodies; Immunoglobulins; Immune serum, e.g. antilymphocytic serum against materials from animals against normal tissues, cells
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K16/00Immunoglobulins [IGs], e.g. monoclonal or polyclonal antibodies
    • C07K16/18Immunoglobulins [IGs], e.g. monoclonal or polyclonal antibodies against material from animals or humans
    • C07K16/28Immunoglobulins [IGs], e.g. monoclonal or polyclonal antibodies against material from animals or humans against receptors, cell surface antigens or cell surface determinants
    • C07K16/2839Immunoglobulins [IGs], e.g. monoclonal or polyclonal antibodies against material from animals or humans against receptors, cell surface antigens or cell surface determinants against the integrin superfamily
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P21/00Drugs for disorders of the muscular or neuromuscular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K16/00Immunoglobulins [IGs], e.g. monoclonal or polyclonal antibodies
    • C07K16/18Immunoglobulins [IGs], e.g. monoclonal or polyclonal antibodies against material from animals or humans
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K39/00Medicinal preparations containing antigens or antibodies
    • A61K2039/505Medicinal preparations containing antigens or antibodies comprising antibodies
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K2317/00Immunoglobulins specific features
    • C07K2317/20Immunoglobulins specific features characterized by taxonomic origin
    • C07K2317/24Immunoglobulins specific features characterized by taxonomic origin containing regions, domains or residues from different species, e.g. chimeric, humanized or veneered
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K2317/00Immunoglobulins specific features
    • C07K2317/30Immunoglobulins specific features characterized by aspects of specificity or valency
    • C07K2317/31Immunoglobulins specific features characterized by aspects of specificity or valency multispecific
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K2317/00Immunoglobulins specific features
    • C07K2317/70Immunoglobulins specific features characterized by effect upon binding to a cell or to an antigen
    • C07K2317/75Agonist effect on antigen
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02ATECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
    • Y02A50/00TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
    • Y02A50/30Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Immunology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Biochemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Biophysics (AREA)
  • Neurosurgery (AREA)
  • Epidemiology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychiatry (AREA)
  • Mycology (AREA)
  • Microbiology (AREA)
  • Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Micro-Organisms Or Cultivation Processes Thereof (AREA)

Abstract

La invencion proporciona un agente farmaceutico que es un agonista de al menos una de la integrina alfa7beta1, integrina alfa6beta1 e integrina alfa3beta1 y que se une a al menos uno de: el dominio de union a laminina de al menos una de la proteina alfa7, proteina alfa6 y proteina alfa3; el dominio CALF-1 de al menos una de la proteina alfa7, proteina alfa6 y proteina alfa3; y el dominio CALF-2 de al menos una de la proteina alfa7, proteina alfa6 y proteina alfa3. Dicho agente es un anticuerpo monoclonal, multiespecifico o biespecifico. Tambien proporcionan una composicion farmaceutica que lo comprende; siendo utiles para tratar enfermedades relacionadas con el mal funcionamiento muscular, que incluyen distrofias musculares.
PE2022000784A 2019-11-15 2020-11-13 Composiciones y metodos para la activacion de integrinas PE20221462A1 (es)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US201962935732P 2019-11-15 2019-11-15
US202063009020P 2020-04-13 2020-04-13
US202063029070P 2020-05-22 2020-05-22
PCT/US2020/060574 WO2021097338A1 (en) 2019-11-15 2020-11-13 Compositions and methods for activation of integrins

Publications (1)

Publication Number Publication Date
PE20221462A1 true PE20221462A1 (es) 2022-09-21

Family

ID=73740612

Family Applications (1)

Application Number Title Priority Date Filing Date
PE2022000784A PE20221462A1 (es) 2019-11-15 2020-11-13 Composiciones y metodos para la activacion de integrinas

Country Status (17)

Country Link
US (2) US12134642B2 (es)
EP (1) EP4058481A1 (es)
JP (1) JP2023503851A (es)
KR (1) KR20220113386A (es)
CN (1) CN115151566A (es)
AU (1) AU2020381534A1 (es)
BR (1) BR112022009430A2 (es)
CA (1) CA3163339A1 (es)
CL (1) CL2022001261A1 (es)
CO (1) CO2022006653A2 (es)
EC (1) ECSP22043116A (es)
IL (1) IL292773A (es)
MX (1) MX2022005904A (es)
PE (1) PE20221462A1 (es)
PH (1) PH12022551166A1 (es)
TW (1) TW202128764A (es)
WO (1) WO2021097338A1 (es)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US10696672B2 (en) 2016-12-23 2020-06-30 Pliant Therapeutics, Inc. Amino acid compounds and methods of use
TWI841573B (zh) 2018-06-27 2024-05-11 美商普萊恩醫療公司 具有未分支連接子之胺基酸化合物及使用方法
JP7579805B2 (ja) 2019-04-08 2024-11-08 プライアント・セラピューティクス・インコーポレイテッド アミノ酸化合物の剤形およびレジメン
CN115151566A (zh) 2019-11-15 2022-10-04 普利安特治疗公司 用于活化整合素的组合物和方法
PE20240114A1 (es) 2020-11-19 2024-01-22 Pliant Therapeutics Inc Inhibidor de integrina y usos de este
WO2025194093A2 (en) * 2024-03-15 2025-09-18 Morphic Therapeutic, Inc. INTEGRIN α7β1 ANTIBODIES AND USES THEREOF

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4522811A (en) 1982-07-08 1985-06-11 Syntex (U.S.A.) Inc. Serial injection of muramyldipeptides and liposomes enhances the anti-infective activity of muramyldipeptides
GB8308235D0 (en) 1983-03-25 1983-05-05 Celltech Ltd Polypeptides
US4816567A (en) 1983-04-08 1989-03-28 Genentech, Inc. Recombinant immunoglobin preparations
JPS61122292A (ja) 1984-11-16 1986-06-10 Teijin Ltd 新規カルバサイクリン中間体の製法
US5225539A (en) 1986-03-27 1993-07-06 Medical Research Council Recombinant altered antibodies and methods of making altered antibodies
US4975369A (en) 1988-04-21 1990-12-04 Eli Lilly And Company Recombinant and chimeric KS1/4 antibodies directed against a human adenocarcinoma antigen
WO1990005144A1 (en) 1988-11-11 1990-05-17 Medical Research Council Single domain ligands, receptors comprising said ligands, methods for their production, and use of said ligands and receptors
US5530101A (en) 1988-12-28 1996-06-25 Protein Design Labs, Inc. Humanized immunoglobulins
IL162181A (en) 1988-12-28 2006-04-10 Pdl Biopharma Inc A method of producing humanized immunoglubulin, and polynucleotides encoding the same
DE69531187T2 (de) 1994-12-20 2004-04-22 Merck Patent Gmbh Monoklonaler Antikörper gegen das Alpha-V-Integrin
WO2002066989A2 (en) 2001-02-20 2002-08-29 The Board Of Trustees Of The University Of Illinois Diagnostics, assay methods and amelioration of muscular dystrophy symptoms
CN115151566A (zh) 2019-11-15 2022-10-04 普利安特治疗公司 用于活化整合素的组合物和方法

Also Published As

Publication number Publication date
IL292773A (en) 2022-07-01
CN115151566A (zh) 2022-10-04
BR112022009430A2 (pt) 2022-10-25
CA3163339A1 (en) 2021-05-20
CL2022001261A1 (es) 2023-03-17
KR20220113386A (ko) 2022-08-12
WO2021097338A1 (en) 2021-05-20
JP2023503851A (ja) 2023-02-01
PH12022551166A1 (en) 2023-10-02
AU2020381534A1 (en) 2022-06-23
MX2022005904A (es) 2022-09-07
CO2022006653A2 (es) 2022-08-09
ECSP22043116A (es) 2022-08-31
TW202128764A (zh) 2021-08-01
US20250026819A1 (en) 2025-01-23
US12134642B2 (en) 2024-11-05
US20210147526A1 (en) 2021-05-20
EP4058481A1 (en) 2022-09-21

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