PE20191502A1 - Complejo medicinal para tratar diabetes tipo 2 y dislipidemia diabetica - Google Patents
Complejo medicinal para tratar diabetes tipo 2 y dislipidemia diabeticaInfo
- Publication number
- PE20191502A1 PE20191502A1 PE2019001004A PE2019001004A PE20191502A1 PE 20191502 A1 PE20191502 A1 PE 20191502A1 PE 2019001004 A PE2019001004 A PE 2019001004A PE 2019001004 A PE2019001004 A PE 2019001004A PE 20191502 A1 PE20191502 A1 PE 20191502A1
- Authority
- PE
- Peru
- Prior art keywords
- diabetes
- treat type
- pharmaceutically acceptable
- diabetic dyslipidemia
- medical complex
- Prior art date
Links
- 208000001072 type 2 diabetes mellitus Diseases 0.000 title abstract 2
- 206010070901 Diabetic dyslipidaemia Diseases 0.000 title 1
- 150000003839 salts Chemical class 0.000 abstract 2
- 208000032928 Dyslipidaemia Diseases 0.000 abstract 1
- ZWPRRQZNBDYKLH-VIFPVBQESA-N Gemigliptin Chemical compound C([C@@H](N)CC(=O)N1CC2=C(C(=NC(=N2)C(F)(F)F)C(F)(F)F)CC1)N1CC(F)(F)CCC1=O ZWPRRQZNBDYKLH-VIFPVBQESA-N 0.000 abstract 1
- 229940121710 HMGCoA reductase inhibitor Drugs 0.000 abstract 1
- 208000017170 Lipid metabolism disease Diseases 0.000 abstract 1
- 102000035195 Peptidases Human genes 0.000 abstract 1
- 108091005804 Peptidases Proteins 0.000 abstract 1
- 239000011230 binding agent Substances 0.000 abstract 1
- 239000004067 bulking agent Substances 0.000 abstract 1
- 206010012601 diabetes mellitus Diseases 0.000 abstract 1
- 239000007884 disintegrant Substances 0.000 abstract 1
- 229960002458 gemigliptin Drugs 0.000 abstract 1
- -1 glidants Substances 0.000 abstract 1
- 239000002471 hydroxymethylglutaryl coenzyme A reductase inhibitor Substances 0.000 abstract 1
- 239000003112 inhibitor Substances 0.000 abstract 1
- 239000000546 pharmaceutical excipient Substances 0.000 abstract 1
- 235000019833 protease Nutrition 0.000 abstract 1
- BPRHUIZQVSMCRT-VEUZHWNKSA-N rosuvastatin Chemical compound CC(C)C1=NC(N(C)S(C)(=O)=O)=NC(C=2C=CC(F)=CC=2)=C1\C=C\[C@@H](O)C[C@@H](O)CC(O)=O BPRHUIZQVSMCRT-VEUZHWNKSA-N 0.000 abstract 1
- 229960000672 rosuvastatin Drugs 0.000 abstract 1
- 239000003381 stabilizer Substances 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/21—Esters, e.g. nitroglycerine, selenocyanates
- A61K31/215—Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids
- A61K31/22—Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids of acyclic acids, e.g. pravastatin
- A61K31/225—Polycarboxylic acids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
- A61P31/06—Antibacterial agents for tuberculosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K2300/00—Mixtures or combinations of active ingredients, wherein at least one active ingredient is fully defined in groups A61K31/00 - A61K41/00
Landscapes
- Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Epidemiology (AREA)
- Emergency Medicine (AREA)
- Diabetes (AREA)
- General Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Engineering & Computer Science (AREA)
- Communicable Diseases (AREA)
- Endocrinology (AREA)
- Oncology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Pulmonology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Abstract
La presente invencion se refiere a una combinacion que comprende gemigliptina, que es un inhibidor de peptidasa IV o una sal farmaceuticamente aceptable del mismo, y rosuvastatina, que es un inhibidor de la HMG-CoA reductasa o una sal farmaceuticamente aceptable del mismo. Ademas, puede comprender estabilizadores, aglutinantes, desintegrantes, deslizantes, agentes de carga y similares como excipientes farmaceuticamente aceptables. Dicha preparacion sirve para tratar eficazmente la diabetes mellitus tipo 2 y la dislipidemia en pacientes diabeticos.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| KR20160152195 | 2016-11-15 | ||
| PCT/KR2017/012941 WO2018093144A1 (ko) | 2016-11-15 | 2017-11-15 | 제2형 당뇨병 및 당뇨성 이상지질혈증 치료용 복합제제 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| PE20191502A1 true PE20191502A1 (es) | 2019-10-22 |
Family
ID=62146049
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| PE2019001004A PE20191502A1 (es) | 2016-11-15 | 2017-11-15 | Complejo medicinal para tratar diabetes tipo 2 y dislipidemia diabetica |
Country Status (10)
| Country | Link |
|---|---|
| KR (1) | KR102055894B1 (es) |
| CN (1) | CN109996545A (es) |
| BR (1) | BR112019009709A2 (es) |
| CO (1) | CO2019005207A2 (es) |
| MX (1) | MX2019005572A (es) |
| PE (1) | PE20191502A1 (es) |
| PH (1) | PH12019501028A1 (es) |
| RU (1) | RU2721406C1 (es) |
| UA (1) | UA122847C2 (es) |
| WO (1) | WO2018093144A1 (es) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN119874701A (zh) * | 2025-01-14 | 2025-04-25 | 深圳格莱恩生物医药科技有限公司 | 一种吉格列汀马来酸盐晶体及其制备方法与应用 |
| CN120004890B (zh) * | 2025-02-17 | 2025-10-21 | 安徽峆一药业股份有限公司 | 一种吉格列汀盐酸盐微晶及其制备方法与应用 |
Family Cites Families (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB0322552D0 (en) * | 2003-09-26 | 2003-10-29 | Astrazeneca Uk Ltd | Therapeutic treatment |
| AP2007004234A0 (en) * | 2005-04-22 | 2007-12-31 | Alantos Pharm Holding | Dipeptidyl peptidase-IV inhibitors |
| EP2464344A2 (en) * | 2009-08-13 | 2012-06-20 | Synthon B.V. | Pharmaceutical tablet comprising rosuvastatin calcium |
| CN107115530A (zh) * | 2009-11-27 | 2017-09-01 | 勃林格殷格翰国际有限公司 | 基因型糖尿病患者利用dpp‑iv抑制剂例如利拉利汀的治疗 |
| WO2011139256A2 (en) * | 2010-05-04 | 2011-11-10 | Bilgic Mahmut | Stable rosuvastatin formulations |
| KR20140013436A (ko) * | 2012-07-24 | 2014-02-05 | 한미약품 주식회사 | 메트포르민 및 로수바스타틴을 포함하는 경구용 복합 제제 |
| TWI606848B (zh) * | 2012-10-08 | 2017-12-01 | Lg生命科學股份有限公司 | 包含格米列汀與美氟明的組合藥物及其製備方法 |
| WO2014080383A1 (en) * | 2012-11-26 | 2014-05-30 | Ranbaxy Laboratories Limited | Pharmaceutical composition of dipeptidyl peptidase-iv (dpp-iv) inhibitors in combination with other antidiabetics |
| TW201636015A (zh) * | 2013-07-05 | 2016-10-16 | 卡地拉保健有限公司 | 協同性組成物 |
| CN103494788B (zh) * | 2013-10-10 | 2015-08-05 | 齐晓彤 | 瑞舒伐他汀钙片的药物组合物及其制备方法 |
| CN104473929B (zh) * | 2014-12-17 | 2018-05-29 | 深圳翰宇药业股份有限公司 | 一种西格列汀辛伐他汀缓释组合物 |
-
2017
- 2017-11-15 KR KR1020170152253A patent/KR102055894B1/ko active Active
- 2017-11-15 UA UAA201906759A patent/UA122847C2/uk unknown
- 2017-11-15 WO PCT/KR2017/012941 patent/WO2018093144A1/ko not_active Ceased
- 2017-11-15 RU RU2019118301A patent/RU2721406C1/ru active
- 2017-11-15 CN CN201780070583.7A patent/CN109996545A/zh active Pending
- 2017-11-15 MX MX2019005572A patent/MX2019005572A/es unknown
- 2017-11-15 PE PE2019001004A patent/PE20191502A1/es unknown
- 2017-11-15 BR BR112019009709A patent/BR112019009709A2/pt not_active IP Right Cessation
-
2019
- 2019-05-09 PH PH12019501028A patent/PH12019501028A1/en unknown
- 2019-05-22 CO CONC2019/0005207A patent/CO2019005207A2/es unknown
Also Published As
| Publication number | Publication date |
|---|---|
| CN109996545A (zh) | 2019-07-09 |
| CO2019005207A2 (es) | 2019-08-20 |
| UA122847C2 (uk) | 2021-01-06 |
| MX2019005572A (es) | 2019-08-14 |
| KR102055894B1 (ko) | 2019-12-13 |
| RU2721406C1 (ru) | 2020-05-19 |
| BR112019009709A2 (pt) | 2019-08-13 |
| WO2018093144A1 (ko) | 2018-05-24 |
| KR20180054500A (ko) | 2018-05-24 |
| PH12019501028A1 (en) | 2020-01-20 |
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