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PE20121585A1 - ANTIBODIES AGAINST THE ERbB3 RECEPTOR ECTODOMINIUM AND ITS USES - Google Patents

ANTIBODIES AGAINST THE ERbB3 RECEPTOR ECTODOMINIUM AND ITS USES

Info

Publication number
PE20121585A1
PE20121585A1 PE2012000234A PE2012000234A PE20121585A1 PE 20121585 A1 PE20121585 A1 PE 20121585A1 PE 2012000234 A PE2012000234 A PE 2012000234A PE 2012000234 A PE2012000234 A PE 2012000234A PE 20121585 A1 PE20121585 A1 PE 20121585A1
Authority
PE
Peru
Prior art keywords
seq
amino acid
acid sequence
antibody
ectodominium
Prior art date
Application number
PE2012000234A
Other languages
Spanish (es)
Inventor
Birgit Schoeberl
Ulrik Nielsen
Michael Feldhaus
Original Assignee
Merrimack Pharmaceuticals Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=43607614&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=PE20121585(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Merrimack Pharmaceuticals Inc filed Critical Merrimack Pharmaceuticals Inc
Publication of PE20121585A1 publication Critical patent/PE20121585A1/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K16/00Immunoglobulins [IGs], e.g. monoclonal or polyclonal antibodies
    • C07K16/18Immunoglobulins [IGs], e.g. monoclonal or polyclonal antibodies against material from animals or humans
    • C07K16/32Immunoglobulins [IGs], e.g. monoclonal or polyclonal antibodies against material from animals or humans against translation products of oncogenes
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K39/00Medicinal preparations containing antigens or antibodies
    • A61K2039/505Medicinal preparations containing antigens or antibodies comprising antibodies
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K2317/00Immunoglobulins specific features
    • C07K2317/20Immunoglobulins specific features characterized by taxonomic origin
    • C07K2317/21Immunoglobulins specific features characterized by taxonomic origin from primates, e.g. man
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K2317/00Immunoglobulins specific features
    • C07K2317/30Immunoglobulins specific features characterized by aspects of specificity or valency
    • C07K2317/34Identification of a linear epitope shorter than 20 amino acid residues or of a conformational epitope defined by amino acid residues
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K2317/00Immunoglobulins specific features
    • C07K2317/50Immunoglobulins specific features characterized by immunoglobulin fragments
    • C07K2317/55Fab or Fab'
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K2317/00Immunoglobulins specific features
    • C07K2317/60Immunoglobulins specific features characterized by non-natural combinations of immunoglobulin fragments
    • C07K2317/62Immunoglobulins specific features characterized by non-natural combinations of immunoglobulin fragments comprising only variable region components
    • C07K2317/622Single chain antibody (scFv)
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K2317/00Immunoglobulins specific features
    • C07K2317/70Immunoglobulins specific features characterized by effect upon binding to a cell or to an antigen
    • C07K2317/73Inducing cell death, e.g. apoptosis, necrosis or inhibition of cell proliferation
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K2317/00Immunoglobulins specific features
    • C07K2317/90Immunoglobulins specific features characterized by (pharmaco)kinetic aspects or by stability of the immunoglobulin
    • C07K2317/92Affinity (KD), association rate (Ka), dissociation rate (Kd) or EC50 value

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Oncology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Molecular Biology (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Immunology (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • Genetics & Genomics (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

SE REFIERE A UN ANTICUERPO CONTRA ErbB3 QUE COMPRENDE: A) UNA REGION VARIABLE DE CADENA PESADA QUE TIENE UNA SECUENCIA DE AMINOACIDOS DE SEQ ID Nº 1 Y COMPRENDE UNA CDRH1 QUE TIENE LA SECUENCIA DE AMINOACIDOS DE SEQ ID Nº 7, UNA CDRH2 QUE TIENE LA SECUENCIA DE AMINOACIDOS DE SEQ ID Nº 8, Y UNA CDRH3 QUE TIENE LA SECUENCIA DE AMINOACIDOS DE SEQ ID Nº 9; Y B) UNA REGION VARIABLE DE CADENA LIGERA QUE TIENE UNA SECUENCIA DE AMINOACIDOS DE SEQ ID Nº 2 Y COMPRENDE UNA CDRL1 QUE TIENE LA SECUENCIA DE AMINOACIDOS DE SEQ ID Nº 10, UNA CDRL2 QUE TIENE LA SECUENCIA DE AMINOACIDOS DE SEQ ID Nº 11, Y UNA CDRL3 QUE TIENE LA SECUENCIA DE AMINOACIDOS DE SEQ ID Nº 12. TAMBIEN SE REFIERE A UN METODO DE TRATAMIENTO DE CARCINOMA RENAL, CANCER DE PROSTATA, CANCER DE OVARIO Y CANCER PULMONAR QUE COMPRENDE ADMINISTRAR EL ANTICUERPO CONTRA ErbB3 Y OTRO COMPUESTO TAL COMO ERLOTINIB, TAXOL O CISPLATINO PARA OBTENER UN EFECTO SINERGICO EN LA SUPRESION DEL CRECIMIENTO DEL TUMORIT REFERS TO AN ANTIBODY AGAINST ErbB3 WHICH INCLUDES: A) A HEAVY CHAIN VARIABLE REGION THAT HAS AN AMINO ACID SEQUENCE OF SEQ ID NO 1 AND INCLUDES A CDRH1 THAT HAS THE AMINO ACID SEQUENCE OF SEQ ID NO 7, A CDRH2 THAT HAS AMINO ACID SEQUENCE OF SEQ ID No. 8, AND A CDRH3 HAVING THE AMINO ACID SEQUENCE OF SEQ ID No. 9; AND B) A LIGHT CHAIN VARIABLE REGION THAT HAS AN AMINO ACID SEQUENCE OF SEQ ID NO. 2 AND INCLUDES A CDRL1 HAVING THE AMINO ACID SEQUENCE OF SEQ ID NO. 10, A CDRL2 HAVING THE AMINO ACID SEQUENCE OF SEQ ID NO. 11, AND A CDRL3 THAT HAS THE SEQ ID NO. 12 AMINO ACID SEQUENCE ALSO REFERS TO A TREATMENT METHOD FOR RENAL CARCINOMA, PROSTATE CANCER, OVARIAN CANCER AND LUNG CANCER THAT INCLUDES ADMINISTERING THE ANTIBODY, AS ANOTHER COMPUTER, AS ANTIBODY ERL3 TAXOL OR CISPLATINE TO OBTAIN A SYNERGIC EFFECT IN THE SUPPRESSION OF TUMOR GROWTH

PE2012000234A 2009-08-21 2010-08-23 ANTIBODIES AGAINST THE ERbB3 RECEPTOR ECTODOMINIUM AND ITS USES PE20121585A1 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US23579909P 2009-08-21 2009-08-21

Publications (1)

Publication Number Publication Date
PE20121585A1 true PE20121585A1 (en) 2012-11-29

Family

ID=43607614

Family Applications (1)

Application Number Title Priority Date Filing Date
PE2012000234A PE20121585A1 (en) 2009-08-21 2010-08-23 ANTIBODIES AGAINST THE ERbB3 RECEPTOR ECTODOMINIUM AND ITS USES

Country Status (21)

Country Link
EP (1) EP2467164A2 (en)
JP (1) JP5752687B2 (en)
KR (1) KR20120059568A (en)
CN (1) CN103002912A (en)
AU (1) AU2010284018C1 (en)
BR (1) BR112012003809A2 (en)
CA (1) CA2771744A1 (en)
CR (1) CR20120108A (en)
DO (1) DOP2012000044A (en)
EA (1) EA201200195A1 (en)
EC (1) ECSP12011740A (en)
IL (1) IL218097A0 (en)
IN (1) IN2012DN01518A (en)
MA (1) MA33582B1 (en)
MX (1) MX336091B (en)
NI (1) NI201200027A (en)
PE (1) PE20121585A1 (en)
SG (1) SG178509A1 (en)
TN (1) TN2012000057A1 (en)
WO (1) WO2011022727A2 (en)
ZA (1) ZA201201195B (en)

Families Citing this family (36)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2008100624A2 (en) 2007-02-16 2008-08-21 Merrimack Pharmaceuticals, Inc. Antibodies against erbb3 and uses thereof
PT2719708T (en) * 2009-11-13 2018-01-16 Daiichi Sankyo Europe Gmbh Material and methods for treating or preventing her-3 associated diseases
HRP20160737T1 (en) 2009-12-22 2016-07-15 Roche Glycart Ag ANTI-HER3-ANTIBODIES AND THEIR USES
EP2859893A1 (en) 2010-03-11 2015-04-15 Merrimack Pharmaceuticals, Inc. Use of ERBB3 inhibitors in the treatment of triple negative and basal-like breast cancers
CN105968206B (en) 2010-04-09 2020-01-17 Aveo制药公司 Anti-ERBB3 antibody
SI2606070T1 (en) 2010-08-20 2017-04-26 Novartis Ag Antibodies for epidermal growth factor receptor 3 (her3)
TW201302793A (en) 2010-09-03 2013-01-16 Glaxo Group Ltd Novel antigen binding protein
IT1402149B1 (en) * 2010-10-04 2013-08-28 Ist Fisioterap Ospitalroma USE OF A PHOSPHOPEPTIDE WHICH IS ABLE TO BLOCK THE HER3 / P85 INTERACTION FOR THE TREATMENT OF HER2 EXPRESSION TUMORS.
DK2635604T3 (en) 2010-11-01 2017-02-27 Symphogen As PAN-HER-ANTIBODY COMPOSITION
ES2625818T3 (en) 2011-04-19 2017-07-20 Merrimack Pharmaceuticals, Inc. Bispecific anti-IGF-1R and anti-ErbB3 antibodies
WO2012176779A1 (en) * 2011-06-20 2012-12-27 協和発酵キリン株式会社 Anti-erbb3 antibody
BR112014007382A2 (en) 2011-09-30 2017-04-04 Regeneron Pharma anti-erbb3 antibodies and their uses
US9273143B2 (en) 2011-09-30 2016-03-01 Regeneron Pharmaceuticals, Inc. Methods and compositions comprising a combination of an anti-ErbB3 antibody and an anti-EGFR antibody
EP3974832A1 (en) 2011-10-06 2022-03-30 Aveo Pharmaceuticals, Inc. Predicting tumor response to anti-erbb3 antibodies
JP6149042B2 (en) * 2011-11-09 2017-06-14 ザ ユーエービー リサーチ ファンデーション HER3 antibody and use thereof
WO2013084147A2 (en) 2011-12-05 2013-06-13 Novartis Ag Antibodies for epidermal growth factor receptor 3 (her3)
US20150037336A1 (en) * 2012-02-22 2015-02-05 U3 Pharma Gmbh Combination of hb-egf binding protein and egfr inhibitor
AR094403A1 (en) 2013-01-11 2015-07-29 Hoffmann La Roche ANTI-HER3 ANTIBODY COMBINATION THERAPY
WO2015058108A1 (en) * 2013-10-17 2015-04-23 Sanford-Burnham Medical Research Institute Drug sensitivity biomarkers and methods of identifying and using drug sensitivity biomarkers
WO2015100459A2 (en) 2013-12-27 2015-07-02 Merrimack Pharmaceuticals, Inc. Biomarker profiles for predicting outcomes of cancer therapy with erbb3 inhibitors and/or chemotherapies
US10844127B2 (en) * 2014-02-28 2020-11-24 Merus N.V. Antibodies that bind EGFR and ErbB3
CN110642952B (en) * 2014-08-14 2021-05-25 上海生物制品研究所有限责任公司 anti-HER 3 antibody, preparation method and application thereof
CA2959716A1 (en) * 2014-09-08 2016-03-17 Yeda Research And Development Co. Ltd. Anti-her3 antibodies and uses of same
WO2016038610A1 (en) 2014-09-08 2016-03-17 Yeda Research And Development Co. Ltd. Compositions and methods for treating cancer resistant to a tyrosine kinase inhibitor (tki)
US10184006B2 (en) 2015-06-04 2019-01-22 Merrimack Pharmaceuticals, Inc. Biomarkers for predicting outcomes of cancer therapy with ErbB3 inhibitors
WO2017069628A2 (en) 2015-10-23 2017-04-27 Merus N.V. Binding molecules that inhibit cancer growth
WO2018182422A1 (en) 2017-03-31 2018-10-04 Merus N.V. Erbb-2 and erbb3 binding bispecific antibodies for use in the treatment f cells that have an nrg1 fusion gene
CN111148764B (en) 2017-05-17 2025-08-12 美勒斯公司 Combination of ErbB-2/ErbB-3 bispecific antibodies and endocrine treatment for breast cancer
AU2018312816B2 (en) 2017-08-09 2021-05-27 Merus N.V. Antibodies that bind EGFR and cMET
EP3665200B1 (en) 2017-08-09 2025-04-16 University of Saskatchewan Her3 binding agents and uses thereof
GB201804094D0 (en) * 2018-03-14 2018-04-25 Ultrahuman Thirteen Ltd ERBB3 Binding agents
WO2019241893A2 (en) * 2018-06-22 2019-12-26 Crd Pharmaceuticals Inc Anti-her3 antibody and uses thereof
AU2021360625A1 (en) * 2020-10-14 2023-06-01 Jiangsu Hengrui Pharmaceuticals Co., Ltd. Anti-her3 antibody and anti-her3 antibody-drug conjugate and medical use thereof
WO2022109404A1 (en) * 2020-11-20 2022-05-27 Actinium Pharmaceuticals, Inc. Her3 radioimmunotherapy for the treatment of solid cancers
IL309337A (en) * 2021-06-15 2024-02-01 Beijing Sinotau Bio Pharmaceuticals Tech Co Ltd Anti-her3 antibody, antibody drug conjugate containing the same, and use thereof
CN119013307A (en) * 2022-04-13 2024-11-22 上海翰森生物医药科技有限公司 Antibodies or antigen binding fragments thereof and medical uses thereof

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2008100624A2 (en) * 2007-02-16 2008-08-21 Merrimack Pharmaceuticals, Inc. Antibodies against erbb3 and uses thereof

Also Published As

Publication number Publication date
JP2013506622A (en) 2013-02-28
AU2010284018B2 (en) 2014-06-05
MA33582B1 (en) 2012-09-01
ECSP12011740A (en) 2013-02-28
CA2771744A1 (en) 2011-02-24
WO2011022727A3 (en) 2013-06-27
IL218097A0 (en) 2012-04-30
TN2012000057A1 (en) 2013-09-19
AU2010284018C1 (en) 2015-10-15
IN2012DN01518A (en) 2015-06-05
EA201200195A1 (en) 2012-12-28
JP5752687B2 (en) 2015-07-22
ZA201201195B (en) 2015-07-29
CR20120108A (en) 2012-06-05
KR20120059568A (en) 2012-06-08
BR112012003809A2 (en) 2019-09-24
CN103002912A (en) 2013-03-27
MX336091B (en) 2016-01-08
SG178509A1 (en) 2012-04-27
EP2467164A2 (en) 2012-06-27
MX2012002172A (en) 2012-05-29
DOP2012000044A (en) 2012-06-30
AU2010284018A1 (en) 2012-03-22
WO2011022727A2 (en) 2011-02-24
NI201200027A (en) 2013-01-29

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