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PE20110945A1 - Nuevo procedimiento de preparacion de granulados de principios activos y granulados tal como se lo ha obtenido - Google Patents

Nuevo procedimiento de preparacion de granulados de principios activos y granulados tal como se lo ha obtenido

Info

Publication number
PE20110945A1
PE20110945A1 PE2011001032A PE2011001032A PE20110945A1 PE 20110945 A1 PE20110945 A1 PE 20110945A1 PE 2011001032 A PE2011001032 A PE 2011001032A PE 2011001032 A PE2011001032 A PE 2011001032A PE 20110945 A1 PE20110945 A1 PE 20110945A1
Authority
PE
Peru
Prior art keywords
active principles
granulates
preparation
alcoholic
new procedure
Prior art date
Application number
PE2011001032A
Other languages
English (en)
Inventor
Christophe Lebon
Pascal Suplie
Original Assignee
Debregeas Et Associes Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=40348849&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=PE20110945(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Debregeas Et Associes Pharma filed Critical Debregeas Et Associes Pharma
Publication of PE20110945A1 publication Critical patent/PE20110945A1/es

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A61K9/5073—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings
    • A61K9/5078—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings with drug-free core
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/08—Antiepileptics; Anticonvulsants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/06—Antihyperlipidemics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/141—Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers
    • A61K9/145—Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers with organic compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A61K9/5005—Wall or coating material
    • A61K9/5021—Organic macromolecular compounds
    • A61K9/5036—Polysaccharides, e.g. gums, alginate; Cyclodextrin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A61K9/5005—Wall or coating material
    • A61K9/5021—Organic macromolecular compounds
    • A61K9/5036—Polysaccharides, e.g. gums, alginate; Cyclodextrin
    • A61K9/5042—Cellulose; Cellulose derivatives, e.g. phthalate or acetate succinate esters of hydroxypropyl methylcellulose
    • A61K9/5047—Cellulose ethers containing no ester groups, e.g. hydroxypropyl methylcellulose

Landscapes

  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Epidemiology (AREA)
  • Diabetes (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Emergency Medicine (AREA)
  • Neurology (AREA)
  • Endocrinology (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Pain & Pain Management (AREA)
  • Medicinal Preparation (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Glanulating (AREA)
  • Fertilizers (AREA)
  • Seasonings (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Fodder In General (AREA)
  • Medicines Containing Plant Substances (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

REFERIDA A UN PROCEDIMIENTO DE PREPARACION DE UN GRANULADO DE AL MENOS DOS PRINCIPIOS ACTIVOS QUE CONSITE EN POLVIFICAR DICHOS PRINCIPIOS ACTIVOS SOBRE UN SOPORTE SOLIDO, DONDE LA ETAPA DE POLVIFICADO COMPRENDE PULVERIZAR UNA SOLUCION ACUOSA, ALCOHOLICA O HIDROALCOHOLICA DE UN AGLUTINANTE Y LUEGO RECUBRIR EL GRANULADO RESULTANTE SEGUIDA DE UNA ETAPA DE MEZCLADO CON UN LUBRICANTE Y/O UN AROMATIZANTE Y/O UN EDULCOLRANTE Y/O UN COLORANTE. EL SOPORTE ES UN POLIOL TAL COMO MANITOL, SORBITOL, MALTITOL, ENTRE OTROS, UN CARBONATO TAL COMO CARBONATO DE CALCIO, MAGNESIO, POTASIO O SODIO, ENTRE OTROS; EL AGLUTINANTE ES ALMIDON, SACAROSA, CELULOSA, GOMA ARABIGA, ENTRE OTROS; EL AGENTE DE RECUBRIMIENTO ES GOMA LACA, POLIVINILPIRROLIDONA, POLIETILENGLICOL, ENTRE OTROS; Y LOS PRINCIPIOS ACTIVOS NO SON EXTRACTOS DE PLANTAS
PE2011001032A 2008-11-14 2009-11-13 Nuevo procedimiento de preparacion de granulados de principios activos y granulados tal como se lo ha obtenido PE20110945A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR0857764A FR2938432B1 (fr) 2008-11-14 2008-11-14 Nouveau procede de preparation de granules de principes actifs, et granules tels qu'obtenus

Publications (1)

Publication Number Publication Date
PE20110945A1 true PE20110945A1 (es) 2012-02-01

Family

ID=40348849

Family Applications (1)

Application Number Title Priority Date Filing Date
PE2011001032A PE20110945A1 (es) 2008-11-14 2009-11-13 Nuevo procedimiento de preparacion de granulados de principios activos y granulados tal como se lo ha obtenido

Country Status (25)

Country Link
US (1) US20110280945A1 (es)
EP (1) EP2349226A1 (es)
JP (1) JP5608681B2 (es)
KR (1) KR101585705B1 (es)
CN (1) CN102223879A (es)
AR (1) AR074330A1 (es)
AU (1) AU2009315449B2 (es)
BR (1) BRPI0916019A2 (es)
CA (1) CA2743753A1 (es)
CL (1) CL2011001115A1 (es)
CO (1) CO6382108A2 (es)
CU (1) CU20110107A7 (es)
EA (1) EA201100757A1 (es)
FR (1) FR2938432B1 (es)
IL (1) IL212850A0 (es)
MA (1) MA32789B1 (es)
MX (1) MX2011005072A (es)
NZ (1) NZ592857A (es)
PE (1) PE20110945A1 (es)
SG (1) SG195651A1 (es)
TN (1) TN2011000235A1 (es)
TW (1) TWI522113B (es)
UA (1) UA103781C2 (es)
WO (1) WO2010055268A1 (es)
ZA (1) ZA201103543B (es)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2971422B1 (fr) * 2011-02-11 2016-05-20 Debregeas Et Associes Pharma Granules d'acide gamma-hydroxybutyrique
US9241956B2 (en) * 2012-11-05 2016-01-26 Kenneth John Tibbs Pharmaceutical preparation and method for treatment of diabetes
US20140127296A1 (en) * 2012-11-05 2014-05-08 Kenneth John Tibbs Pharmaceutical preparation and method for treatment of diabetes
US11058635B1 (en) * 2020-10-15 2021-07-13 King Abdulaziz University Oral administration of 5-FU in a gelling nanosuspension for targeted delivery to treat colorectal cancers
KR20240157168A (ko) * 2023-04-24 2024-11-01 주식회사 케이티앤지 바인더를 사용하는 파우치 충진 물질의 제조 방법

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS6327424A (ja) * 1986-07-17 1988-02-05 Shionogi & Co Ltd 徐放性製剤およびその製造法
JP2820829B2 (ja) * 1991-03-07 1998-11-05 武田薬品工業株式会社 有核散剤およびその製造方法
JPH08310969A (ja) * 1995-05-22 1996-11-26 Lion Corp 固形薬品組成物及びその製造方法
FR2790668B1 (fr) * 1999-03-12 2002-07-26 D B F Granules contenant une substance vegetale et leur procede de preparation
MXPA01011800A (es) * 1999-05-17 2003-08-19 D B F Granulos que contienen una sustancia vegetal y procedimiento para prepararlos.
MY148805A (en) * 2002-10-16 2013-05-31 Takeda Pharmaceutical Controlled release preparation
US9247765B2 (en) * 2004-01-14 2016-02-02 Omniactive Health Technologies Limited Stable beadlets of lipophilic nutrients
FR2880541B1 (fr) * 2005-01-10 2008-02-22 Amalric Veret Une nouvelle formule de plantes sous forme de micro-granules de xilitol pour renforcer les effets des plantes et leurs proprietes par une meilleure assimilation
US20060182796A1 (en) * 2005-02-03 2006-08-17 Abrika Pharmaceuticals, Inc. Taste masked pharmaceutical compositions
WO2008027993A2 (en) * 2006-08-31 2008-03-06 Eurand, Inc. Drug delivery systems comprising solid solutions of weakly basic drugs
KR101180163B1 (ko) * 2007-02-14 2012-09-05 다이니치 세이카 고교 가부시키가이샤 유기안료의 분산제 및 그 사용
US20090004281A1 (en) * 2007-06-26 2009-01-01 Biovail Laboratories International S.R.L. Multiparticulate osmotic delivery system

Also Published As

Publication number Publication date
SG195651A1 (en) 2013-12-30
MX2011005072A (es) 2011-10-03
TN2011000235A1 (fr) 2012-12-17
TW201029667A (en) 2010-08-16
EA201100757A1 (ru) 2011-12-30
ZA201103543B (en) 2012-01-25
NZ592857A (en) 2013-07-26
WO2010055268A1 (fr) 2010-05-20
BRPI0916019A2 (pt) 2015-11-10
AU2009315449B2 (en) 2015-03-26
CO6382108A2 (es) 2012-02-15
CN102223879A (zh) 2011-10-19
US20110280945A1 (en) 2011-11-17
CL2011001115A1 (es) 2011-11-11
JP5608681B2 (ja) 2014-10-15
IL212850A0 (en) 2011-07-31
JP2012508786A (ja) 2012-04-12
FR2938432A1 (fr) 2010-05-21
EP2349226A1 (fr) 2011-08-03
UA103781C2 (uk) 2013-11-25
CA2743753A1 (fr) 2010-05-20
MA32789B1 (fr) 2011-11-01
KR20110095888A (ko) 2011-08-25
CU20110107A7 (es) 2012-01-31
TWI522113B (zh) 2016-02-21
KR101585705B1 (ko) 2016-01-15
AR074330A1 (es) 2011-01-05
FR2938432B1 (fr) 2011-05-20
AU2009315449A1 (en) 2010-05-20

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