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PE20061220A1 - Bifenilsulfonamidas y proceso para su preparacion - Google Patents

Bifenilsulfonamidas y proceso para su preparacion

Info

Publication number
PE20061220A1
PE20061220A1 PE2006000293A PE2006000293A PE20061220A1 PE 20061220 A1 PE20061220 A1 PE 20061220A1 PE 2006000293 A PE2006000293 A PE 2006000293A PE 2006000293 A PE2006000293 A PE 2006000293A PE 20061220 A1 PE20061220 A1 PE 20061220A1
Authority
PE
Peru
Prior art keywords
alkyl
formula
alcoxy
halogen
amino
Prior art date
Application number
PE2006000293A
Other languages
English (en)
Inventor
Wassilios Grammenos
Joachim Rheinheimer
Thomas Grote
Christopher Koradin
Deyn Wolfgang Von
Norbert Gotz
Douglas D Anspaugh
Henry Van Tuyl Cotter
David G Kuhn
Hassan Oloumi-Sadeghi
Deborah L Culbertson
Jurgen Langewald
Ernst Baumann
Michael Puhl
Jan Klaas Lohmann
Original Assignee
Basf Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Basf Ag filed Critical Basf Ag
Publication of PE20061220A1 publication Critical patent/PE20061220A1/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D213/00Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/24Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D213/54Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/34Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom
    • A01N43/40Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom six-membered rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/14Ectoparasiticides, e.g. scabicides
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D213/00Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/24Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D213/36Radicals substituted by singly-bound nitrogen atoms
    • C07D213/42Radicals substituted by singly-bound nitrogen atoms having hetero atoms attached to the substituent nitrogen atom

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Environmental Sciences (AREA)
  • Agronomy & Crop Science (AREA)
  • Zoology (AREA)
  • Wood Science & Technology (AREA)
  • Dentistry (AREA)
  • Engineering & Computer Science (AREA)
  • Plant Pathology (AREA)
  • Pest Control & Pesticides (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Pyridine Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

DE FORMULA (I) DONDE: R1 ES H, ALQUILO C1-C4, ALQUENILO C2-C4, ALQUINILO C2-C4 o BENCILO; R2, R3, R4 Y R5 SON, EN FORMA INDEPENDIENTE, H, HALOGENO, ALQUILO C1-C4, HALOMETILO, ALCOXI C1-C4, HALOMETOXI, ALQUILTIO C1-C4, ALQUILAMINO C1-C4 o DI (ALQUIL C1-C4)AMINO; R6, R7 SON, EN FORMA INDEPENDIENTE, H, HIDROXI, CIANO, NITRO, AMINO, HALOGENO, ALQUILO C1-C8, HALOALQUILO C1-C6, ALCOXI C1-C8, HALOLCOXI C1-C8, ALQUILTIO C1-C6, (ALQUIL C1-C4)CARBONILO, (ALCOXI C1-C4)CARBONILO, -C(R8)=NOR9, (ALQUIL C1-C4)AMINO, DI(ALQUIL C1-C4) AMINO, (ALQUIL C1-C4)AMINOCARBONILO, DI(ALQUIL C1-C4)AMINOCARBONILO, FENILO O FENOXI, EN DONDE EL ANILLO FENILO PUEDE LLEVAR 1, 2 o 3 GRUPOS R10; m ES 0, 1, 2, 3 o 4; n ES 0, 1, 2, 3, 4 o 5; R8 ES ALQUILO C1-C4; R9 ES ALQUILO C1-C8, HALOALQUILO C1-C4, ALQUENILO C2-C4, HALOALQUENILO C2-C4, ALQUINILO C2-C4, HALOALQUINILO C2-C4 o BENCILO; R10 ES CIANO, NITRO, HALOGENO, ALQUILO C1-C4, HALOMETILO, ALCOXI C1-C4 o HALOMETOXI. m Y n SON 0 CUANDO R2 A R5 SON TODOS H. EL PROCESO INCLUYE: i) REACCION DE DERIVADOS DE PIRIDINA DE FORMULA (II), BAJO CONDICIONES BASICAS CON CLORURO DE SULFONILO DE FORMULA (III); o, ii) REACCION DE DERIVADOS DE PIRIDINA DE FORMULA (III) CON HALOGENUROS DE 4-HALOGENFENILSULFONILO DE FORMULA (IV), SIENDO L HIDROXI o HALOGENO, PARA CEDER DERIVADOS DE PIRIDINA DE FORMULA (V) QUE REACCIONAN CON DERIVADOS DEL ACIDO BORONICO DE FORMULA (VI) EN PRESENCIA DE UN CATALIZADOR DE PLATINO. SE USA PARA COMBATIR PLAGAS DE ARTROPODOS
PE2006000293A 2005-03-16 2006-03-16 Bifenilsulfonamidas y proceso para su preparacion PE20061220A1 (es)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US66241105P 2005-03-16 2005-03-16
DE102005018464 2005-04-20
EP05011598 2005-05-30
US77655106P 2006-02-24 2006-02-24

Publications (1)

Publication Number Publication Date
PE20061220A1 true PE20061220A1 (es) 2006-12-21

Family

ID=36218770

Family Applications (1)

Application Number Title Priority Date Filing Date
PE2006000293A PE20061220A1 (es) 2005-03-16 2006-03-16 Bifenilsulfonamidas y proceso para su preparacion

Country Status (29)

Country Link
US (1) US20080161187A1 (es)
EP (1) EP1860941B1 (es)
JP (1) JP4637950B2 (es)
KR (1) KR20070112191A (es)
CN (1) CN101141878A (es)
AP (1) AP2108A (es)
AR (1) AR054746A1 (es)
AT (1) ATE413808T1 (es)
AU (1) AU2006224568A1 (es)
CA (1) CA2599555A1 (es)
CR (1) CR9337A (es)
CY (1) CY1108705T1 (es)
DE (1) DE602006003641D1 (es)
DK (1) DK1860941T3 (es)
EA (1) EA012526B1 (es)
EG (1) EG25264A (es)
ES (1) ES2316060T3 (es)
GT (1) GT200600118A (es)
HR (1) HRP20090037T3 (es)
IL (1) IL185447A0 (es)
MA (1) MA29383B1 (es)
MX (1) MX2007011287A (es)
PE (1) PE20061220A1 (es)
PL (1) PL1860941T3 (es)
PT (1) PT1860941E (es)
SI (1) SI1860941T1 (es)
TW (1) TW200714204A (es)
UY (1) UY29423A1 (es)
WO (1) WO2006097489A1 (es)

Families Citing this family (27)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
RU2383536C2 (ru) 2004-08-04 2010-03-10 Тайсо Фармасьютикал Ко., Лтд. Производное триазола
TW200806290A (en) * 2006-01-25 2008-02-01 Synta Pharmaceuticals Corp Substituted biaryl compounds for inflammation and immune-related uses
CN101415691B (zh) 2006-02-03 2011-12-14 大正制药株式会社 三唑衍生物
CN101415687B (zh) 2006-02-06 2012-02-08 大正制药株式会社 鞘氨醇-1-磷酸结合抑制物质
CA2645069A1 (en) * 2006-03-15 2007-09-20 Basf Se Quinoline derivatives and their use as pesticides
US20100077512A1 (en) * 2006-11-22 2010-03-25 Basf Se Pyridazin-4-ylmethyl-sulfonamides used as Fungicides and Against Arthropods
EA200900640A1 (ru) 2006-11-22 2009-12-30 Басф Се Пиримидилметилсульфонамидные соединения
HRP20120363T1 (hr) * 2007-08-01 2012-05-31 Taisho Pharmaceutical Co. Inhibitor vezivanja s1p1
CN101828111B (zh) * 2007-08-21 2014-07-23 塞诺米克斯公司 人t2r苦味受体及其用途
WO2009059603A1 (en) 2007-11-05 2009-05-14 Vestergaard Frandsen Sa Room with two counter-resistant insecticidal objects
EP2231605A1 (en) 2007-12-05 2010-09-29 Basf Se Pyridylmethyl-sulfonamide compounds
EP2252590A1 (en) * 2008-02-15 2010-11-24 Basf Se Substituted sulfonic acid amide compounds
BRPI0908840A2 (pt) * 2008-03-14 2015-07-21 Basf Se Compostos, processo para preparar os mesmos, composições agroquímicas, uso dos compostos, método para combater fungos fitopatogênicos, e, semente
EP2276746A1 (en) * 2008-04-10 2011-01-26 Basf Se Substituted pyridazinylmethyl sulfonamides
BRPI0912891A2 (pt) * 2008-05-20 2015-07-28 Basf Se Compostos, processo para preparar compostos, composições agroquímicas, método para combater fungos fitopatogênicos, e, semente
US20110077153A1 (en) * 2008-05-20 2011-03-31 Basf Se Substituted Heteroarylmethyl Sulfonamides
WO2009141290A2 (en) 2008-05-21 2009-11-26 Basf Se Substituted pyridin-4-ylmethyl sulfonamides
WO2009141274A1 (en) * 2008-05-21 2009-11-26 Basf Se Substituted pyridin-4 -yl-methyl sulfonamides as fungicides
EP2300471A1 (en) * 2008-05-28 2011-03-30 Basf Se Substituted pyridin-4-yl-methyl sulfonamidesas fungicides
IN2012DN05081A (es) * 2009-12-08 2015-10-09 Boehringer Ingelheim Int
BR112014020773A2 (pt) * 2012-02-22 2020-10-27 Sanford-Burnham Medical Research Institute compostos de sulfonamida e seus usos como inibidores tnap
WO2014099837A1 (en) * 2012-12-18 2014-06-26 E. I. Du Pont De Nemours And Company Sulfonamide anthelmintics
BR102013031043B1 (pt) * 2013-12-02 2018-03-13 Fundação Butantan Uso de compostos químicos capazes de inibir a ação tóxica das esfingomielinases d do veneno de aranhas loxosceles e composição farmacêutica compreendendo os referidos compostos
CN103755601B (zh) * 2014-01-13 2015-08-12 河北星宇化工有限公司 4,4-双(2-磺酸基苯乙烯基)-1,1-联苯的制备方法
RU2615155C2 (ru) * 2015-06-04 2017-04-04 Федеральное государственное бюджетное учреждение науки Институт нефтехимии и катализа Российской академии наук Способ получения 3-[(фенилсульфанил)метил]пентан-2,4-диона, проявляющего фунгицидную активность
RU2735251C1 (ru) * 2020-04-03 2020-10-29 Федеральное государственное бюджетное учреждение науки Сибирский федеральный научный центр агробиотехнологий Российской академии наук (СФНЦА РАН) Способ разведения капустной моли Plutella xylostella L.
CN113527152B (zh) * 2021-08-09 2023-07-28 西北农林科技大学 一种联苯磺酰胺类化合物及其防治农作物害虫的方法

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US4154744A (en) * 1976-10-12 1979-05-15 Sumitomo Chemical Company, Limited Process for producing a furan derivative
US4874775A (en) * 1985-06-11 1989-10-17 Eli Lilly And Company Agriculturally useful sulfonamides
WO1997000857A1 (fr) * 1995-06-21 1997-01-09 Otsuka Kagaku Kabushiki Kaisha Derives de sulfonamides et insecticide, miticide et nematicide les contenant
JP4477006B2 (ja) * 2003-09-18 2010-06-09 ビーエーエスエフ ソシエタス・ヨーロピア 殺真菌植物保護剤としての4−ピリジニルメチルスルホンアミド誘導体

Also Published As

Publication number Publication date
IL185447A0 (en) 2008-01-06
EG25264A (en) 2011-11-30
CA2599555A1 (en) 2006-09-21
WO2006097489A8 (en) 2007-03-08
JP4637950B2 (ja) 2011-02-23
ES2316060T3 (es) 2009-04-01
EP1860941B1 (en) 2008-11-12
AU2006224568A1 (en) 2006-09-21
CR9337A (es) 2008-01-21
AP2007004152A0 (en) 2007-10-31
SI1860941T1 (sl) 2009-04-30
MA29383B1 (fr) 2008-04-01
AR054746A1 (es) 2007-07-11
US20080161187A1 (en) 2008-07-03
PL1860941T3 (pl) 2009-04-30
GT200600118A (es) 2006-11-13
CN101141878A (zh) 2008-03-12
JP2008533096A (ja) 2008-08-21
EA200701839A1 (ru) 2008-02-28
KR20070112191A (ko) 2007-11-22
UY29423A1 (es) 2006-10-31
MX2007011287A (es) 2007-11-08
DE602006003641D1 (de) 2008-12-24
HRP20090037T3 (en) 2009-03-31
EP1860941A1 (en) 2007-12-05
CY1108705T1 (el) 2014-04-09
PT1860941E (pt) 2008-12-22
WO2006097489A1 (en) 2006-09-21
EA012526B1 (ru) 2009-10-30
AP2108A (en) 2010-02-25
DK1860941T3 (da) 2009-03-02
ATE413808T1 (de) 2008-11-15
TW200714204A (en) 2007-04-16

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