PE20010744A1 - Uso de (2s,3s,5r)-2-(3,5-difluorofenil)-3,5-dimetil-2-morfolinol para el tratamiento de la obesidad - Google Patents
Uso de (2s,3s,5r)-2-(3,5-difluorofenil)-3,5-dimetil-2-morfolinol para el tratamiento de la obesidadInfo
- Publication number
- PE20010744A1 PE20010744A1 PE2000001089A PE0010892000A PE20010744A1 PE 20010744 A1 PE20010744 A1 PE 20010744A1 PE 2000001089 A PE2000001089 A PE 2000001089A PE 0010892000 A PE0010892000 A PE 0010892000A PE 20010744 A1 PE20010744 A1 PE 20010744A1
- Authority
- PE
- Peru
- Prior art keywords
- morpholinol
- dimethyl
- obesity
- difluorophenyl
- treatment
- Prior art date
Links
- 208000008589 Obesity Diseases 0.000 title abstract 2
- 235000020824 obesity Nutrition 0.000 title abstract 2
- OZGPVYJHWWPEFT-RGNHYFCHSA-N manifaxine Chemical compound C[C@@H]1N[C@H](C)CO[C@@]1(O)C1=CC(F)=CC(F)=C1 OZGPVYJHWWPEFT-RGNHYFCHSA-N 0.000 title 1
- 230000036528 appetite Effects 0.000 abstract 1
- 235000019789 appetite Nutrition 0.000 abstract 1
- 230000004584 weight gain Effects 0.000 abstract 1
- 235000019786 weight gain Nutrition 0.000 abstract 1
- 230000004580 weight loss Effects 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
- A61K31/5375—1,4-Oxazines, e.g. morpholine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
Landscapes
- Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Organic Chemistry (AREA)
- Diabetes (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Engineering & Computer Science (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Child & Adolescent Psychology (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Coloring Foods And Improving Nutritive Qualities (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
Abstract
SE REFIERE AL USO DE (2S,3S,5R)-2-(3,5-DIFLUOROFENIL)-3,5-DIMETIL-2-MORFOLINOL DE FORMULA I, PARA TRATAR LA OBESIDAD, SUPRIMIR EL APETITO, CAUSAR LA PERDIDA DE PESO, PREVENIR EL AUMENTO DE PESO
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GBGB9924275.2A GB9924275D0 (en) | 1999-10-13 | 1999-10-13 | Method for the treatment of obesity |
| GB0001861A GB0001861D0 (en) | 2000-01-28 | 2000-01-28 | Method for the treatment of obesity |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| PE20010744A1 true PE20010744A1 (es) | 2001-07-23 |
Family
ID=26243494
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| PE2000001089A PE20010744A1 (es) | 1999-10-13 | 2000-10-11 | Uso de (2s,3s,5r)-2-(3,5-difluorofenil)-3,5-dimetil-2-morfolinol para el tratamiento de la obesidad |
Country Status (6)
| Country | Link |
|---|---|
| EP (1) | EP1220673A2 (es) |
| JP (1) | JP2003511410A (es) |
| AR (1) | AR026022A1 (es) |
| AU (1) | AU7750100A (es) |
| PE (1) | PE20010744A1 (es) |
| WO (1) | WO2001026641A2 (es) |
Families Citing this family (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| MXPA04001165A (es) | 2001-08-08 | 2004-05-20 | R Orton Kevin | Aparato y metodo para una reduccion de peso electricamente conductiva. |
| KR20110043664A (ko) * | 2002-05-17 | 2011-04-27 | 듀크 유니버시티 | 비만치료방법 |
| CA2522708C (en) | 2003-04-29 | 2013-05-28 | Orexigen Therapeutics, Inc. | Compositions for affecting weight loss |
| ES2761812T3 (es) | 2005-11-22 | 2020-05-21 | Nalpropion Pharmaceuticals Inc | Composición y métodos de aumento de la sensibilidad a la insulina |
| US8916195B2 (en) | 2006-06-05 | 2014-12-23 | Orexigen Therapeutics, Inc. | Sustained release formulation of naltrexone |
| AU2007319472B2 (en) | 2006-11-09 | 2013-01-17 | Nalpropion Pharmaceuticals Llc | Methods Of Administering Weight Loss Medications |
| US20090203695A1 (en) * | 2007-12-05 | 2009-08-13 | Biovitrum Ab | Compounds IV |
| WO2009158114A1 (en) | 2008-05-30 | 2009-12-30 | Orexigen Therapeutics, Inc. | Methods for treating visceral fat conditions |
| MX2010013353A (es) * | 2008-06-04 | 2010-12-21 | Astrazeneca Ab | Nuevos compuestos vii. |
| EP2523557B1 (en) | 2010-01-11 | 2019-09-25 | Nalpropion Pharmaceuticals, Inc. | Methods of providing weight loss therapy in patients with major depression |
| PT2858640T (pt) | 2012-06-06 | 2020-06-30 | Nalpropion Pharmaceuticals Llc | Composição para utilização num método de tratamento de excesso de peso e obesidade em doentes com alto risco cardiovascular |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB8924528D0 (en) * | 1989-10-31 | 1989-12-20 | Wellcome Found | Heterocyclic pharmaceutical compounds,preparation and use |
| JP2001524960A (ja) * | 1997-04-24 | 2001-12-04 | メルク シヤープ エンド ドーム リミテツド | 摂食障害を治療するためのnk−1受容体拮抗薬の使用 |
| WO1999025355A1 (en) * | 1997-11-14 | 1999-05-27 | Glaxo Group Ltd. | Method of treating addiction to nicotine products |
| AP1229A (en) * | 1998-01-21 | 2003-12-04 | Glaxo Group Ltd | Pharmaceutically active morpholinol. |
| MA26693A1 (fr) * | 1998-09-28 | 2004-12-20 | Glaxo Group Ltd | Compositions pour administration par voie buccale |
-
2000
- 2000-10-03 AU AU77501/00A patent/AU7750100A/en not_active Abandoned
- 2000-10-03 JP JP2001529431A patent/JP2003511410A/ja active Pending
- 2000-10-03 WO PCT/US2000/027252 patent/WO2001026641A2/en not_active Ceased
- 2000-10-03 EP EP00967281A patent/EP1220673A2/en not_active Withdrawn
- 2000-10-11 PE PE2000001089A patent/PE20010744A1/es not_active Application Discontinuation
- 2000-10-12 AR ARP000105369A patent/AR026022A1/es unknown
Also Published As
| Publication number | Publication date |
|---|---|
| WO2001026641A3 (en) | 2002-01-10 |
| AU7750100A (en) | 2001-04-23 |
| WO2001026641A2 (en) | 2001-04-19 |
| EP1220673A2 (en) | 2002-07-10 |
| JP2003511410A (ja) | 2003-03-25 |
| AR026022A1 (es) | 2002-12-26 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FA | Abandonment or withdrawal |