LU90712I2 - Mal-ate de 5-(4-(n-m-thyl-n-(2-pyriddyl)amino)-thoxy)benzyl)) thiazolidinedione-2,4 dione ou ses sels pharmaceutiquement acceptables - Google Patents

Mal-ate de 5-(4-(n-m-thyl-n-(2-pyriddyl)amino)-thoxy)benzyl)) thiazolidinedione-2,4 dione ou ses sels pharmaceutiquement acceptables

Info

Publication number: LU90712I2
Authority: LU; Luxembourg
Prior art keywords: pyriddyl; thoxy; thiazolidinedione; thyl; dione
Prior art date: 1992-09-05

Application number

LU90712C

Other languages

English (en)

Original Assignee

Smithkline Beecham Plc

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1992-09-05

Filing date

2001-01-10

Publication date

2001-03-12

Family has litigation

First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=10721461&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=LU90712(I2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.

2001-01-10 Application filed by Smithkline Beecham Plc filed Critical Smithkline Beecham Plc

2001-03-12 Publication of LU90712I2 publication Critical patent/LU90712I2/fr

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/425—Thiazoles
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/14—Prodigestives, e.g. acids, enzymes, appetite stimulants, antidyspeptics, tonics, antiflatulents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/06—Antihyperlipidemics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Life Sciences & Earth Sciences (AREA)
General Health & Medical Sciences (AREA)
Veterinary Medicine (AREA)
Public Health (AREA)
Animal Behavior & Ethology (AREA)
Engineering & Computer Science (AREA)
Pharmacology & Pharmacy (AREA)
Medicinal Chemistry (AREA)
Bioinformatics & Cheminformatics (AREA)
General Chemical & Material Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Diabetes (AREA)
Hematology (AREA)
Obesity (AREA)
Heart & Thoracic Surgery (AREA)
Cardiology (AREA)
Emergency Medicine (AREA)
Endocrinology (AREA)
Vascular Medicine (AREA)
Urology & Nephrology (AREA)
Child & Adolescent Psychology (AREA)
Nutrition Science (AREA)
Epidemiology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)
Thiazole And Isothizaole Compounds (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)

LU90712C 1992-09-05 2001-01-10 Mal-ate de 5-(4-(n-m-thyl-n-(2-pyriddyl)amino)-thoxy)benzyl)) thiazolidinedione-2,4 dione ou ses sels pharmaceutiquement acceptables LU90712I2 (fr)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
GB929218830A GB9218830D0 (en)	1992-09-05	1992-09-05	Novel compounds
PCT/GB1993/001853 WO1994005659A1 (fr)	1992-09-05	1993-09-01	Derives substitues de la thiazolidenedione

Publications (1)

Publication Number	Publication Date
LU90712I2 true LU90712I2 (fr)	2001-03-12

Family

ID=10721461

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
LU90712C LU90712I2 (fr)	1992-09-05	2001-01-10	Mal-ate de 5-(4-(n-m-thyl-n-(2-pyriddyl)amino)-thoxy)benzyl)) thiazolidinedione-2,4 dione ou ses sels pharmaceutiquement acceptables

Country Status (37)

Country	Link
US (1)	US5910592A (fr)
EP (2)	EP0960883A1 (fr)
JP (5)	JP2828777B2 (fr)
KR (3)	KR20030097596A (fr)
CN (4)	CN1040323C (fr)
AP (1)	AP513A (fr)
AT (1)	ATE182147T1 (fr)
AU (1)	AU674880B2 (fr)
BR (1)	BR1100916A (fr)
CA (2)	CA2143849C (fr)
CY (1)	CY2138B1 (fr)
CZ (2)	CZ287473B6 (fr)
DE (2)	DE10199002I2 (fr)
DK (1)	DK0658161T3 (fr)
ES (1)	ES2133410T3 (fr)
FI (2)	FI982413A0 (fr)
GB (1)	GB9218830D0 (fr)
GR (1)	GR3030794T3 (fr)
HU (2)	HU224212B1 (fr)
IL (1)	IL106904A (fr)
LU (1)	LU90712I2 (fr)
MA (1)	MA22970A1 (fr)
MX (1)	MX9305397A (fr)
MY (1)	MY111190A (fr)
NL (1)	NL300035I2 (fr)
NO (4)	NO303016B1 (fr)
NZ (1)	NZ255505A (fr)
PL (1)	PL173725B1 (fr)
RU (3)	RU2128179C1 (fr)
SA (1)	SA93140245B1 (fr)
SG (2)	SG83747A1 (fr)
SI (1)	SI9300452B (fr)
SK (1)	SK280777B6 (fr)
TW (1)	TW385309B (fr)
UA (1)	UA41901C2 (fr)
WO (1)	WO1994005659A1 (fr)
ZA (1)	ZA936509B (fr)

Families Citing this family (110)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB9308487D0 (en) *	1993-04-23	1993-06-09	Smithkline Beecham Plc	Novel compounds
US5919782A (en) *	1996-05-06	1999-07-06	Dr. Reddy's Research Foundation	Heterocyclic compounds having antidiabetic, hypolipidaemic, antihypertensive properties, process for their preparation and pharmaceutical compositions containing them
ZA973848B (en) *	1996-05-06	1997-12-02	Reddy Research Foundation	Novel heterocyclic compounds having antidiabetic, hypolipidaemic, antihypertensive properties, process for their preparation and pharmaceutical compositions containing them.
ZA973850B (en) *	1996-05-06	1997-12-02	Reddy Research Foundation	Novel antidiabetic compounds having hypolipidaemic, anti-hypertensive properties, process for their preparation and pharmaceutical compositions containing them.
US5801173A (en) *	1996-05-06	1998-09-01	Dr. Reddy's Research Foundation	Heterocyclic compounds having antidiabetic, hypolipidaemic, antihypertensive properties, process for their preparation and pharmaceutical compositions containing them
US6372750B2 (en)	1996-07-01	2002-04-16	Dr. Reddy's Research Foundation	Heterocyclic compounds, process for their preparation and pharmaceutical compounds containing them and their use in the treatment of diabetes and related diseases
USRE39266E1 (en) *	1996-07-01	2006-09-05	Dr. Reddy's Laboratories, Limited	Heterocyclic compounds, process for their preparation and pharmaceutical compositions containing them and their use in the treatment of diabetes and related diseases
KR100579765B1 (ko) *	1996-07-01	2006-12-28	닥터 레디스 레보러터리즈 리미티드	신규헤테로고리형화합물의제조방법,이를함유하는약제조성물및당뇨병및이와관련된질병의치료에있어서그의용도
US6114526A (en) *	1996-07-01	2000-09-05	Dr. Reddy's Research Foundation	Heterocyclic compounds, process for their preparation and pharmaceutical compositions containing them and their use in the treatment of diabetes and related diseases
US5885997A (en) *	1996-07-01	1999-03-23	Dr. Reddy's Research Foundation	Heterocyclic compounds, process for their preparation and pharmaceutical compositions containing them and their use in the treatment of diabetes and related diseases
EP0921798A1 (fr) *	1996-07-12	1999-06-16	Smithkline Beecham Plc	Nouveau traitement contre la resistance a la leptine
GB9711683D0 (en) *	1997-06-05	1997-08-06	Smithkline Beecham Plc	Composition
CZ298469B6 (cs) *	1997-06-18	2007-10-10	Smithkline Beecham Plc	Farmaceutický prostredek obsahující 5-[4-/2-(N-methyl-N-(2-pyridyl)amino)ethoxy/benzyl]thiazolidin-2,4-dion a metformin, a lécivo pro lécení diabetesmellitus
ATE353654T1 (de)	1997-06-18	2007-03-15	Smithkline Beecham Plc	Behandlung der diabetes mit thiazolidindione und sulphonylurea
GB9715306D0 (en) *	1997-07-18	1997-09-24	Smithkline Beecham Plc	Novel method of treatment
GB9721692D0 (en) *	1997-10-13	1997-12-10	Smithkline Beecham Plc	Novel treatment
GB9721693D0 (en) *	1997-10-13	1997-12-10	Smithkline Beecham Plc	Novel treatment
US20020006939A1 (en) *	1997-10-13	2002-01-17	Smithkline Beecham P.L.C.	Use of thiazolidinediones for the treatment of hyperglycaemia
US20010031776A1 (en) *	1997-10-13	2001-10-18	Smithkline Beecham P.L.C.	Use of thiazolidinediones for the treatment of hyperglycaemia
GB9723295D0 (en)	1997-11-04	1998-01-07	Smithkline Beecham Plc	Novel process
US7091359B2 (en)	1997-11-04	2006-08-15	Smithkline Beecham Plc	Process for the preparation of thiazolidinedione derivatives
GB9726563D0 (en)	1997-12-16	1998-02-11	Smithkline Beecham Plc	Novel pharmaceutical
GB9726568D0 (en) *	1997-12-16	1998-02-11	Smithkline Beecham Plc	Novel pharmaceutical
US6664278B2 (en)	1997-12-16	2003-12-16	Smithkline Beecham P.L.C.	Hydrate of 5-[4-[2-(N-methyl-N-(2-pyridil)amino)ethoxy]benzyl]thiazolidine-2,4-dione maleic acid salt
AU774613B2 (en) *	1997-12-16	2004-07-01	Smithkline Beecham Plc	Hydrate of 5-(4-(2- (N-methyl-N- (2-pyridil)amino) ethoxy)benzyl) thiazolidine-2,4-dione maleic acid salt
GB9726566D0 (en) *	1997-12-16	1998-02-11	Smithkline Beecham Plc	Novel pharmaceutical
US20020137940A1 (en)	1997-12-16	2002-09-26	Smithkline Beecham P.L.C.	5-[4-[2-(N-methyl-N-(2-pyridyl)amino)ethoxy]benzyl]thiazolidine-2, 4-dione, maleic acid salt, hydrate as pharmaceutical
AU770817B2 (en) *	1997-12-16	2004-03-04	Smithkline Beecham Plc	5-(4-(2-(N-methyl-N-(2-pyridyl)amino)ethoxy)benzyl) thiazolidine-2,dione,maleic acid salt, hydrate as pharmaceutical
US7045519B2 (en)	1998-06-19	2006-05-16	Chiron Corporation	Inhibitors of glycogen synthase kinase 3
MA26662A1 (fr) *	1998-07-21	2004-12-20	Smithkline Beecham Plc	Derives de thiazolidinedione, compositions pharmaceutiques les contenant et leur utilisation
US6613785B2 (en)	1998-07-21	2003-09-02	Smithkline Beecham Plc	Use of glucose uptake enhancer for reducing post-ischemic injury of the heart
AP2001002036A0 (en) *	1998-07-21	2001-03-31	Smithkline Beecham Plc	Use of glucose uptake enhancer for reducing apoptosis.
US20030153607A1 (en) *	1998-11-12	2003-08-14	Smithkline Beecham P.L.C.	Novel composition and use
SK287038B6 (sk)	1998-11-12	2009-10-07	Smithkline Beecham Plc	Farmaceutický prostriedok na postupné uvoľňovanie 5-[4-[2-(N- metyl-N-(2-pyridyl)amino)etoxy]benzyl]tiazolidín-2,4-diónu a metformínu a spôsob jeho výroby
DZ2937A1 (fr) *	1998-11-12	2004-03-15	Smithkline Beecham Plc	Compositions nouvelles de sensibilidants à l'insuline.
GB9824893D0 (en) *	1998-11-12	1999-01-06	Smithkline Beckman Corp	Novel method of treatment
US20040102486A1 (en) *	1998-11-12	2004-05-27	Smithkline Beecham Corporation	Novel method of treatment
GB9909041D0 (en) *	1999-04-20	1999-06-16	Smithkline Beecham Plc	Novel pharmaceutical
GB9909075D0 (en) *	1999-04-20	1999-06-16	Smithkline Beecham Plc	Novel pharmaceutical
ATE246191T1 (de) *	1999-04-23	2003-08-15	Smithkline Beecham Plc	Polymorph von 5-(4-(2-(n-methyl-n-(2- pyrdyl)amino)äthoxy)benzyl)thiazolidin-2,4-dion maleinsäuresalz
US20040248945A1 (en)	1999-04-23	2004-12-09	Smithkline Beecham P.L.C.	Thiazolidinedione derivative and its use as antidiabetic
JP2002543076A (ja) *	1999-04-23	2002-12-17	スミスクラインビーチャムパブリックリミテッドカンパニー	チアゾリジンジオン誘導体および抗糖尿病薬としてのその使用
BR0009934A (pt) *	1999-04-23	2002-06-04	Smithkline Beecham Plc	Produto farmacêutico
JP2003507379A (ja) *	1999-08-17	2003-02-25	スミスクラインビーチャムパブリックリミテッドカンパニー	チアゾリジンジオン誘導体を含有する医薬組成物およびその調製法
AR030920A1 (es) *	1999-11-16	2003-09-03	Smithkline Beecham Plc	Composiciones farmaceuticas para el tratamiento de la diabetes mellitus y condiciones asociadas con la diabetes mellitus, y procedimientos para preparar dichas composiciones
GB0006133D0 (en) *	2000-03-14	2000-05-03	Smithkline Beecham Plc	Novel pharmaceutical
GB0014006D0 (en) *	2000-06-08	2000-08-02	Smithkline Beecham Plc	Novel pharmaceutical
GB0014005D0 (en) *	2000-06-08	2000-08-02	Smithkline Beecham Plc	Novel pharmaceutical
AP2002002688A0 (en) *	2000-06-16	2002-12-31	Smithkline Beecham Plc	Treatment and prevention of cardiac insulin resistance associated associated conditions.
GB0014969D0 (en)	2000-06-19	2000-08-09	Smithkline Beecham Plc	Novel method of treatment
GB0019228D0 (en) *	2000-08-04	2000-09-27	Smithkline Beecham Plc	Novel pharmaceutical
AU2005229687B2 (en) *	2000-08-04	2008-03-13	Smithkline Beecham P.L.C.	Tartrate salts of thiazolidinedione derivative
GB0019223D0 (en) *	2000-08-04	2000-09-27	Smithkline Beecham Plc	Novel pharmaceutical
GB0019226D0 (en) *	2000-08-04	2000-09-27	Smithkline Beecham Plc	Novel pharmaceutical
AU2005229688B2 (en) *	2000-08-04	2008-04-03	Smithkline Beecham P.L.C.	Tartrate salts of thiazolidinedione derivative
GB0019224D0 (en) *	2000-08-04	2000-09-27	Smithkline Beecham Plc	Novel pharmaceutical
GB0021784D0 (en) *	2000-09-05	2000-10-18	Smithkline Beecham Plc	Novel pharmaceutical
GB0021785D0 (en) *	2000-09-05	2000-10-18	Smithkline Beecham Plc	Novel Pharmaceutical
GB0021865D0 (en) *	2000-09-06	2000-10-18	Smithkline Beecham Plc	Novel pharmaceutical
GB0021978D0 (en) *	2000-09-07	2000-10-25	Smithkline Beecham Plc	Novel pharmaceutical
PL360661A1 (en) *	2000-09-26	2004-09-20	Dr.Reddy's Research Foundation	Novel polymorphic forms of 5-[4-[2-[n-methyl-n-(2-pyridyl)amino]ethoxy]benzyl] thiazolidine-2,4-dione maleate and process for their preparation
US7241895B2 (en)	2000-09-26	2007-07-10	Dr. Reddy's Laboratories Limited	Polymorphic forms of 5-[4-[2-[n-methyl-n-(2-pyridyl)amino[ethoxy]benzyl] thiazolidine-2,4-dione maleate and process for their preparation
UA75370C2 (en) *	2000-09-26	2006-04-17	Reddys Lab Ltd Dr	Polymorphic forms of 5-[4-[2(n-methyl-n-(2-pyridyl)amino]ethoxy]benzyl] thiazolidine-2.4-dione maleate
GB0023971D0 (en) *	2000-09-29	2000-11-15	Smithkline Beecham Plc	Novel pharmaceutical
WO2002051839A1 (fr) *	2000-12-22	2002-07-04	Smithkline Beecham P.L.C.	Mesylate de 5-[4-[2-(n-methyl-n-(2-pyridyl)amino)ethoxy]benzyl]thiazolidine-2,4-dione
WO2002051823A1 (fr)	2000-12-26	2002-07-04	Torrent Pharmaceuticals Ltd	Procede de preparation de maleate de rosiglitazone
GB0127805D0 (en)	2001-11-20	2002-01-09	Smithkline Beecham Plc	Pharmaceutical composition
EP1446404B1 (fr) *	2001-11-21	2006-06-14	Smithkline Beecham Plc	Edisylates de rosiglitazone et leur utilisation en tant qu'antidiabetiques
SI1448559T1 (sl) *	2001-11-21	2007-06-30	Smithkline Beecham Plc	5-(4-(2-(n-metil-n-(2-piridil)amino)etoksi)benzil-tiazolidin-2,4-dion- benzensulfonat; postopek za njegovo pripravo; njegovi polimorfi i, ii, iii; in njegova uporaba kot farmacevtska uäśinkovina
GB0129872D0 (en) *	2001-12-13	2002-02-06	Smithkline Beecham Plc	Novel pharmaceutical
GB0129871D0 (en) *	2001-12-13	2002-02-06	Smithkline Beecham Plc	Novel pharmaceutical
GB0129851D0 (en) *	2001-12-13	2002-01-30	Smithkline Beecham Plc	Novel compounds
WO2003050116A1 (fr) *	2001-12-13	2003-06-19	Smithkline Beecham Plc	Sel d'acide 10-camphorsulphonique de 5(-4-(2-(n-methyl-n-(2-pyridil)amino)ethoxy)benzyl)thiazolidine-2,4-dione et son utilisation contre le diabete sucre
WO2003050112A1 (fr) *	2001-12-13	2003-06-19	Smithkline Beecham Plc	Hydrates de toluenesulfonate d'un derive de thiazolidinedione
GB0129876D0 (en) *	2001-12-13	2002-02-06	Smithkline Beecham Plc	Novel pharmaceutical
GB0130510D0 (en) *	2001-12-20	2002-02-06	Smithkline Beecham Plc	Novel pharmaceutical
GB0130509D0 (en) *	2001-12-20	2002-02-06	Smithkline Beecham Plc	Novel pharmaceutical
GB0130511D0 (en) *	2001-12-20	2002-02-06	Smithkline Beecham Plc	Novel pharmaceutical
AU2002352479A1 (en) *	2001-12-20	2003-07-09	Smithkline Beecham Plc	5- (4- (2- (n-methyl-n- (2-pyridyl) amino) ethoxy) benzyl) thiazolidine-2, 4-dione malic acid salt and use against diabetes mellitus
US8268352B2 (en)	2002-08-05	2012-09-18	Torrent Pharmaceuticals Limited	Modified release composition for highly soluble drugs
US8216609B2 (en)	2002-08-05	2012-07-10	Torrent Pharmaceuticals Limited	Modified release composition of highly soluble drugs
US7232828B2 (en) *	2002-08-10	2007-06-19	Bethesda Pharmaceuticals, Inc.	PPAR Ligands that do not cause fluid retention, edema or congestive heart failure
WO2004062667A1 (fr) *	2003-01-08	2004-07-29	Dr. Reddy's Laboratories Limited	Forme amorphe du maleate de rosiglitazone et procede de preparation
GB0307259D0 (en) *	2003-03-28	2003-05-07	Glaxo Group Ltd	Process
GB2405403A (en) *	2003-08-29	2005-03-02	Cipla Ltd	Rosiglitazone maleate of particular polymorphic forms and methods of preparing rosiglitazone free base
WO2005058813A2 (fr) *	2003-12-17	2005-06-30	Ranbaxy Laboratories Limited	Agents antidiabetiques
EP1732513A2 (fr) *	2003-12-31	2006-12-20	Alpharma, Inc.	Preparations de rosiglitazone
WO2005073227A2 (fr) *	2004-01-28	2005-08-11	Usv Limited	Procede de preparation de maleate de 5-[4-[2-[n-methyl-n-(2-pyridyl) amino] ethoxy] phenyl methyl] thiazolidine-2, 4-dione
GB2410948A (en) *	2004-02-13	2005-08-17	Sandoz Ag	Novel phosphoric acid salt of rosiglitazone
AR047541A1 (es) *	2004-02-13	2006-01-25	Sandoz Ag	Fosfato de 5-[[4-[2-metil-2-piridinil-amino-etoxi]fenil]metil]-2,4 tiazolidinadiona (rosiglitazona) y sus formas polimorficas
GB2421240A (en) *	2004-12-14	2006-06-21	Sandoz Ag	Phosphoric acid salt of rosiglitazone
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1992
- 1992-09-05 GB GB929218830A patent/GB9218830D0/en active Pending
1993
- 1993-09-01 DE DE2001199002 patent/DE10199002I2/de active Active
- 1993-09-01 EP EP99108192A patent/EP0960883A1/fr not_active Ceased
- 1993-09-01 FI FI982413A patent/FI982413A0/fi unknown
- 1993-09-01 HU HU9500659A patent/HU224212B1/hu active Protection Beyond IP Right Term
- 1993-09-01 EP EP93919489A patent/EP0658161B1/fr not_active Expired - Lifetime
- 1993-09-01 NZ NZ255505A patent/NZ255505A/xx not_active IP Right Cessation
- 1993-09-01 KR KR1020027006870A patent/KR20030097596A/ko not_active Ceased
- 1993-09-01 AT AT93919489T patent/ATE182147T1/de active
- 1993-09-01 ES ES93919489T patent/ES2133410T3/es not_active Expired - Lifetime
- 1993-09-01 JP JP6506983A patent/JP2828777B2/ja not_active Expired - Lifetime
- 1993-09-01 DE DE69325658T patent/DE69325658T2/de not_active Expired - Lifetime
- 1993-09-01 PL PL93307812A patent/PL173725B1/pl unknown
- 1993-09-01 AU AU49730/93A patent/AU674880B2/en not_active Expired
- 1993-09-01 WO PCT/GB1993/001853 patent/WO1994005659A1/fr not_active Ceased
- 1993-09-01 DK DK93919489T patent/DK0658161T3/da active
- 1993-09-01 CZ CZ1995565A patent/CZ287473B6/cs not_active IP Right Cessation
- 1993-09-01 RU RU95108329A patent/RU2128179C1/ru active
- 1993-09-01 KR KR1020087020116A patent/KR20080081099A/ko not_active Ceased
- 1993-09-01 SG SG9904980A patent/SG83747A1/en unknown
- 1993-09-01 CA CA002143849A patent/CA2143849C/fr not_active Expired - Lifetime
- 1993-09-01 HU HU0500355A patent/HU0500355D0/hu not_active Application Discontinuation
- 1993-09-01 UA UA95038295A patent/UA41901C2/uk unknown
- 1993-09-01 SG SG1996008773A patent/SG48302A1/en unknown
- 1993-09-01 SK SK277-95A patent/SK280777B6/sk not_active IP Right Cessation
- 1993-09-01 KR KR1019950700873A patent/KR100371297B1/ko not_active Expired - Lifetime
- 1993-09-01 CA CA002273147A patent/CA2273147A1/fr not_active Abandoned
- 1993-09-02 AP APAP/P/1993/000562A patent/AP513A/en active
- 1993-09-02 SI SI9300452A patent/SI9300452B/sl unknown
- 1993-09-03 MA MA23279A patent/MA22970A1/fr unknown
- 1993-09-03 ZA ZA936509A patent/ZA936509B/xx unknown
- 1993-09-03 IL IL106904A patent/IL106904A/xx not_active IP Right Cessation
- 1993-09-03 MX MX9305397A patent/MX9305397A/es unknown
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- 1993-09-04 CN CN93119067A patent/CN1040323C/zh not_active Expired - Lifetime
- 1993-10-07 TW TW082108297A patent/TW385309B/zh not_active IP Right Cessation
- 1993-10-10 SA SA93140245A patent/SA93140245B1/ar unknown
1995
- 1995-03-03 NO NO950852A patent/NO303016B1/no not_active IP Right Cessation
- 1995-03-03 FI FI951004A patent/FI106263B/fi not_active IP Right Cessation
1997
- 1997-05-14 BR BR1100916-0A patent/BR1100916A/pt active IP Right Grant
- 1997-07-14 US US08/892,045 patent/US5910592A/en not_active Ceased
- 1997-10-08 NO NO974646A patent/NO305802B1/no not_active IP Right Cessation
- 1997-10-30 CN CN97122519A patent/CN1051312C/zh not_active Expired - Lifetime
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- 1997-12-08 CZ CZ19973958A patent/CZ290591B6/cs not_active IP Right Cessation
1998
- 1998-06-02 JP JP10152828A patent/JPH11147885A/ja active Pending
- 1998-09-24 RU RU98117673/14A patent/RU98117673A/ru not_active Application Discontinuation
- 1998-09-24 RU RU98117628/04A patent/RU98117628A/ru not_active Application Discontinuation
1999
- 1999-07-15 GR GR990401864T patent/GR3030794T3/el unknown
- 1999-10-05 CY CY9900033A patent/CY2138B1/xx unknown
2001
- 2001-01-05 NL NL300035C patent/NL300035I2/nl unknown
- 2001-01-10 LU LU90712C patent/LU90712I2/fr unknown
- 2001-04-10 NO NO2001005C patent/NO2001005I2/no unknown
- 2001-04-10 NO NO2001006C patent/NO2001006I1/no unknown
- 2001-08-06 JP JP2001238154A patent/JP2002047288A/ja active Pending
2004
- 2004-05-12 JP JP2004142553A patent/JP2004359676A/ja active Pending
2008
- 2008-05-13 JP JP2008125985A patent/JP2008208142A/ja active Pending

Also Published As

Publication number	Publication date
PL173725B1 (pl)	1998-04-30
BR1100916A (pt)	2000-07-04
DE69325658T2 (de)	1999-12-30
NL300035I1 (nl)	2001-03-01
NO974646L (no)	1995-03-03
HK1012363A1 (en)	1999-07-30
NZ255505A (en)	1997-08-22
FI982413L (fi)	1998-11-06
FI951004A0 (fi)	1995-03-03
IL106904A (en)	1997-09-30
HU224212B1 (hu)	2005-06-28
RU98117628A (ru)	2000-08-20
CN1101911A (zh)	1995-04-26
NO305802B1 (no)	1999-07-26
JP2828777B2 (ja)	1998-11-25
CN1183413A (zh)	1998-06-03
CN1183275A (zh)	1998-06-03
RU98117673A (ru)	2000-07-20
DE69325658D1 (de)	1999-08-19
EP0658161B1 (fr)	1999-07-14
KR950702982A (ko)	1995-08-23
CZ56595A3 (en)	1995-11-15
SG48302A1 (en)	1998-04-17
CZ290591B6 (cs)	2002-08-14
ES2133410T3 (es)	1999-09-16
NO950852D0 (no)	1995-03-03
IL106904A0 (en)	1993-12-28
SI9300452B (sl)	2003-02-28
MY111190A (en)	1999-09-30
CA2143849A1 (fr)	1994-03-17
NO303016B1 (no)	1998-05-18
UA41901C2 (uk)	2001-10-15
CA2273147A1 (fr)	1994-03-17
EP0960883A1 (fr)	1999-12-01
CN1051312C (zh)	2000-04-12
NO950852L (no)	1995-03-03
SI9300452A (en)	1994-06-30
CN1066939C (zh)	2001-06-13
EP0658161A1 (fr)	1995-06-21
TW385309B (en)	2000-03-21
HUT72639A (en)	1996-05-28
MA22970A1 (fr)	1994-04-01
KR20030097596A (ko)	2003-12-31
KR100371297B1 (ko)	2003-05-09
HU0500355D0 (en)	2005-05-30
JPH08501095A (ja)	1996-02-06
DE10199002I2 (de)	2001-12-13
RU2128179C1 (ru)	1999-03-27
DK0658161T3 (da)	1999-11-29
NL300035I2 (nl)	2001-07-02
CN1040323C (zh)	1998-10-21
NO2001005I2 (no)	2004-06-01
AU4973093A (en)	1994-03-29
ATE182147T1 (de)	1999-07-15
SK27795A3 (en)	1995-08-09
JP2002047288A (ja)	2002-02-12
US5910592A (en)	1999-06-08
CZ287473B6 (en)	2000-12-13
GR3030794T3 (en)	1999-11-30
KR20080081099A (ko)	2008-09-05
CN1063942C (zh)	2001-04-04
JP2004359676A (ja)	2004-12-24
HU9500659D0 (en)	1995-04-28
SK280777B6 (sk)	2000-07-11
AU674880B2 (en)	1997-01-16
CY2138B1 (en)	2002-06-21
JPH11147885A (ja)	1999-06-02
JP2008208142A (ja)	2008-09-11
NO2001006I1 (no)	2001-04-30
CA2143849C (fr)	2000-04-25
ZA936509B (en)	1994-06-16
FI951004L (fi)	1995-03-03
SG83747A1 (en)	2001-10-16
RU95108329A (ru)	1996-12-20
FI982413A7 (fi)	1998-11-06
AP9300562A0 (en)	1993-10-31
MX9305397A (es)	1995-01-31
WO1994005659A1 (fr)	1994-03-17
NO974646D0 (no)	1997-10-08
CN1183276A (zh)	1998-06-03
GB9218830D0 (en)	1992-10-21
FI106263B (fi)	2000-12-29
PL307812A1 (en)	1995-06-26
SA93140245B1 (ar)	2005-10-15
FI982413A0 (fi)	1998-11-06
AP513A (en)	1996-07-30

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ITGE940099A0 (it)	1994-09-07	Dispositivo per l'agugliatura di una falda di ovatta.
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