KR970702045A - 고혈압 치료, 심장 보호, 허혈증 치료 및 항지방 분해 특성을 갖는 화합물(Compounds having antihypertensive, cardioprotective, anti-ischemic and antilipolytic properties) - Google Patents
고혈압 치료, 심장 보호, 허혈증 치료 및 항지방 분해 특성을 갖는 화합물(Compounds having antihypertensive, cardioprotective, anti-ischemic and antilipolytic properties)Info
- Publication number
- KR970702045A KR970702045A KR1019960705840A KR19960705840A KR970702045A KR 970702045 A KR970702045 A KR 970702045A KR 1019960705840 A KR1019960705840 A KR 1019960705840A KR 19960705840 A KR19960705840 A KR 19960705840A KR 970702045 A KR970702045 A KR 970702045A
- Authority
- KR
- South Korea
- Prior art keywords
- cardioprotective
- antihypertensive
- ischemic
- compounds
- antilipolytic
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Ceased
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D473/00—Heterocyclic compounds containing purine ring systems
- C07D473/26—Heterocyclic compounds containing purine ring systems with an oxygen, sulphur, or nitrogen atom directly attached in position 2 or 6, but not in both
- C07D473/32—Nitrogen atom
- C07D473/34—Nitrogen atom attached in position 6, e.g. adenine
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D473/00—Heterocyclic compounds containing purine ring systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/06—Antihyperlipidemics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/08—Vasodilators for multiple indications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
- C07H19/02—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
- C07H19/04—Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
- C07H19/052—Imidazole radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
- C07H19/02—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
- C07H19/04—Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
- C07H19/16—Purine radicals
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Molecular Biology (AREA)
- Genetics & Genomics (AREA)
- Biotechnology (AREA)
- Biochemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Medicinal Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Heart & Thoracic Surgery (AREA)
- Cardiology (AREA)
- Obesity (AREA)
- Hematology (AREA)
- Diabetes (AREA)
- Urology & Nephrology (AREA)
- Vascular Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Saccharide Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US22988294A | 1994-04-19 | 1994-04-19 | |
| US08/316,761 US5561134A (en) | 1990-09-25 | 1994-10-03 | Compounds having antihypertensive, cardioprotective, anti-ischemic and antilipolytic properties |
| PCT/US1995/004800 WO1995028160A1 (en) | 1994-04-19 | 1995-04-19 | Compounds having antihypertensive, cardioprotective, anti-ischemic and antilipolytic properties |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| KR970702045A true KR970702045A (ko) | 1997-05-13 |
Family
ID=26923699
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| KR1019960705840A Ceased KR970702045A (ko) | 1994-04-19 | 1996-10-18 | 고혈압 치료, 심장 보호, 허혈증 치료 및 항지방 분해 특성을 갖는 화합물(Compounds having antihypertensive, cardioprotective, anti-ischemic and antilipolytic properties) |
Country Status (28)
| Country | Link |
|---|---|
| US (2) | US5561134A (ko) |
| EP (2) | EP1006115A3 (ko) |
| JP (1) | JPH09512020A (ko) |
| KR (1) | KR970702045A (ko) |
| CN (1) | CN1086704C (ko) |
| AP (1) | AP699A (ko) |
| AT (1) | ATE260106T1 (ko) |
| AU (1) | AU684635B2 (ko) |
| BG (1) | BG63799B1 (ko) |
| BR (1) | BR9507327A (ko) |
| CA (1) | CA2188147C (ko) |
| CZ (1) | CZ289528B6 (ko) |
| DE (1) | DE69532608T2 (ko) |
| DK (1) | DK0758897T3 (ko) |
| EE (1) | EE9600156A (ko) |
| ES (1) | ES2217279T3 (ko) |
| FI (1) | FI964218L (ko) |
| HU (1) | HUT75331A (ko) |
| NO (1) | NO317727B1 (ko) |
| NZ (1) | NZ284357A (ko) |
| OA (1) | OA10464A (ko) |
| PL (1) | PL182942B1 (ko) |
| PT (1) | PT758897E (ko) |
| RO (1) | RO119225B1 (ko) |
| RU (1) | RU2166319C2 (ko) |
| SI (1) | SI9520055A (ko) |
| SK (1) | SK284039B6 (ko) |
| WO (1) | WO1995028160A1 (ko) |
Families Citing this family (83)
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| US5721263A (en) * | 1993-06-07 | 1998-02-24 | Takeda Chemical Industries, Ltd. | Pharmaceutical composition for angiotensin II-mediated diseases |
| US5792776A (en) * | 1994-06-27 | 1998-08-11 | Cytomed, Inc., | Compounds and methods for the treatment of cardiovascular, inflammatory and immune disorders |
| SI0828740T1 (en) * | 1995-05-30 | 2001-12-31 | Aventis Pharma Sa | 2-azabicyclo(2.2.1)heptane derivatives, preparation and application thereof |
| US6992188B1 (en) | 1995-12-08 | 2006-01-31 | Pfizer, Inc. | Substituted heterocyclic derivatives |
| US6376472B1 (en) | 1996-07-08 | 2002-04-23 | Aventis Pharmaceuticals, Inc. | Compounds having antihypertensive, cardioprotective, anti-ischemic and antilipolytic properties |
| UA51716C2 (uk) * | 1996-07-08 | 2002-12-16 | Авентіс Фармасьютікалз Продактс Інк. | Сполуки, що мають гіпотензивну, кардіопротекторну, анти-ішемічну та антиліполітичну властивості, фармацевтична композиція та способи лікування |
| US5747474A (en) * | 1996-07-29 | 1998-05-05 | Immune Modulation, Inc. | Immunosuppression by administration of N6,N6 -disubstituted cAMP's, analogues thereof, and related nucleosides |
| WO1998016539A1 (en) * | 1996-10-14 | 1998-04-23 | Novo Nordisk A/S | Novel therapeutically active adenosine derivatives |
| GB9723590D0 (en) * | 1997-11-08 | 1998-01-07 | Glaxo Group Ltd | Chemical compounds |
| GB9723566D0 (en) * | 1997-11-08 | 1998-01-07 | Glaxo Group Ltd | Chemical compounds |
| AU774155B2 (en) * | 1998-12-21 | 2004-06-17 | Aventis Pharmaceuticals Inc. | Process for preparing N6-substituted deaza-adenosine derivatives |
| AU2187100A (en) | 1998-12-31 | 2000-07-24 | Aventis Pharmaceuticals Products Inc. | Process for preparing n6-substituted deaza-adenosine derivatives |
| US7378400B2 (en) * | 1999-02-01 | 2008-05-27 | University Of Virginia Patent Foundation | Method to reduce an inflammatory response from arthritis |
| US7018365B2 (en) | 1999-05-21 | 2006-03-28 | Micro Therapeutics, Inc. | Threaded syringe with quick stop |
| US6576619B2 (en) * | 1999-05-24 | 2003-06-10 | Cv Therapeutics, Inc. | Orally active A1 adenosine receptor agonists |
| DE19951701A1 (de) * | 1999-10-27 | 2001-05-03 | Aventis Pharma Gmbh | Verwendung von 2-Imidazolyl-substituierten Carbinolen zur Herstellung eines Medikaments zur Behandlung oder Prophylaxe von durch ischämischen Zuständen bewirkten Krankheiten |
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1994
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1995
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- 1995-04-19 AT AT95916451T patent/ATE260106T1/de active
- 1995-04-19 RU RU96121567/14A patent/RU2166319C2/ru not_active IP Right Cessation
- 1995-04-19 SK SK1340-96A patent/SK284039B6/sk unknown
- 1995-04-19 CZ CZ19963032A patent/CZ289528B6/cs not_active IP Right Cessation
- 1995-04-19 RO RO96-01991A patent/RO119225B1/ro unknown
- 1995-04-19 CA CA002188147A patent/CA2188147C/en not_active Expired - Fee Related
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- 1995-04-19 WO PCT/US1995/004800 patent/WO1995028160A1/en not_active Ceased
- 1995-04-19 HU HU9602829A patent/HUT75331A/hu unknown
- 1995-04-19 SI SI9520055A patent/SI9520055A/sl not_active IP Right Cessation
- 1995-04-19 JP JP7527171A patent/JPH09512020A/ja not_active Ceased
- 1995-04-19 AP APAP/P/1996/000904A patent/AP699A/en active
- 1995-05-31 US US08/455,361 patent/US5736554A/en not_active Expired - Fee Related
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- 1996-10-18 KR KR1019960705840A patent/KR970702045A/ko not_active Ceased
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