KR900007816A - 사이클로프로필-치환된 아졸릴메틸카비놀, 이의 제조방법 및 약제로서의 이의 용도 - Google Patents

사이클로프로필-치환된 아졸릴메틸카비놀, 이의 제조방법 및 약제로서의 이의 용도

Info

Publication number: KR900007816A
Authority: KR; South Korea
Prior art keywords: azolylmethylcarbinol; cyclopropyl; preparation; medicament; substituted
Prior art date: 1988-11-19
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.): Granted

Application number

KR1019890016675A

Other languages

English (en)

Other versions

KR0128662B1 (ko

Inventor

푸그만 부르크하트

프렘펠 만프레드

스트로에흐 크라우스

하인즈 뷔헬 칼

Original Assignee

바이엘 아크티엔게젤샤프트

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1988-11-19

Filing date

1989-11-17

Publication date

1990-06-02

1989-11-17 Application filed by 바이엘 아크티엔게젤샤프트 filed Critical 바이엘 아크티엔게젤샤프트

1990-06-02 Publication of KR900007816A publication Critical patent/KR900007816A/ko

1998-04-04 Application granted granted Critical

1998-04-04 Publication of KR0128662B1 publication Critical patent/KR0128662B1/ko

2009-11-17 Anticipated expiration legal-status Critical

Status Expired - Fee Related legal-status Critical Current

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
- C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
- C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C255/00—Carboxylic acid nitriles
- C07C255/45—Carboxylic acid nitriles having cyano groups bound to carbon atoms of rings other than six-membered aromatic rings
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/56—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/56—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
- C07D233/60—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms with hydrocarbon radicals, substituted by oxygen or sulfur atoms, attached to ring nitrogen atoms

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Veterinary Medicine (AREA)
Public Health (AREA)
General Health & Medical Sciences (AREA)
Medicinal Chemistry (AREA)
Animal Behavior & Ethology (AREA)
Pharmacology & Pharmacy (AREA)
General Chemical & Material Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Chemical Kinetics & Catalysis (AREA)
Oncology (AREA)
Communicable Diseases (AREA)
Epidemiology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Plural Heterocyclic Compounds (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

KR1019890016675A 1988-11-19 1989-11-17 사이클로프로필-치환된 아졸릴메틸카비놀, 이의 제조방법 및 약제로서의 이의 용도 Expired - Fee Related KR0128662B1 (ko)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
DEP3839170.8		1988-11-19
DE3839170A DE3839170A1 (de)	1988-11-19	1988-11-19	Cyclopropyl-substituierte azolylmethylcarbinole, verfahren zu ihrer herstellung und ihre verwendung als arzneimittel

Publications (2)

Publication Number	Publication Date
KR900007816A true KR900007816A (ko)	1990-06-02
KR0128662B1 KR0128662B1 (ko)	1998-04-04

Family

ID=6367500

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
KR1019890016675A Expired - Fee Related KR0128662B1 (ko)	1988-11-19	1989-11-17	사이클로프로필-치환된 아졸릴메틸카비놀, 이의 제조방법 및 약제로서의 이의 용도

Country Status (9)

Country	Link
US (1)	US5059615A (ko)
EP (1)	EP0370300B1 (ko)
JP (1)	JP2839161B2 (ko)
KR (1)	KR0128662B1 (ko)
AT (1)	ATE103907T1 (ko)
CA (1)	CA2003213C (ko)
DE (2)	DE3839170A1 (ko)
ES (1)	ES2052863T3 (ko)
ZA (1)	ZA898775B (ko)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
DE4206529A1 (de) *	1992-03-02	1993-09-09	Bayer Ag	Azolylmethyl-cyclopropyl-derivate
EP3173406A1 (en) *	2012-12-19	2017-05-31	Basf Se	Substituted [1,2,4]triazole compounds and their use as fungicides
AR100743A1 (es) *	2014-06-06	2016-10-26	Basf Se	Compuestos de [1,2,4]triazol sustituido
BR112017000694A2 (pt) *	2014-07-18	2018-07-03	Bayer Cropscience Ag	vinil e alquinil cianocicloalcanóis e vinil e alquinil cianoheterocicloalcanóis substituídos como agentes ativos contra estresse abiótico em plantas
AR101214A1 (es)	2014-07-22	2016-11-30	Bayer Cropscience Ag	Ciano-cicloalquilpenta-2,4-dienos, ciano-cicloalquilpent-2-en-4-inas, ciano-heterociclilpenta-2,4-dienos y ciano-heterociclilpent-2-en-4-inas sustituidos como principios activos contra el estrés abiótico de plantas
RS58961B1 (sr)	2015-01-22	2019-08-30	Sanofi Aventis Deutschland	Proces proizvodnje 2-[4-(ciklopropankarbonil)fenil]-2-metil-propannitrila
US20180354928A1 (en) *	2015-11-17	2018-12-13	Dow Agrosciences Llc	4-((6-(2-(2,4-difluorophenyl)-1,1-difluoro-2-hydroxy-3-(1h-1,2,4-triazol-1-yl)propyl)pyridin-3-yl)oxy)benzonitrile and processes of preparation
US20180370946A1 (en) *	2015-11-17	2018-12-27	Dow Agrosciences Llc	4-((6-(2-(2,4-difluorophenyl)-1,1-difluoro-2-hydroxy-3-(1h-1,2,4-triazol-1-yl)propyl)pyridin-3-yl)oxy)benzonitrile and processes of preparation

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
EP0106515B1 (en) *	1982-09-30	1988-12-28	Pfizer Limited	Triazole anti-fungal agents
EP0180850A3 (de) *	1984-11-02	1987-05-27	Bayer Ag	Antimykotische Azolylmethyl-cyclopropyl-carbinol Derivate
US4859232A (en) *	1986-12-05	1989-08-22	Monsanto Company	Substituted-aryl cyclopropanecarbonitriles and derivatives thereof as herbicide antidotes
DE3732385A1 (de) *	1987-09-25	1989-04-06	Bayer Ag	Hydroxyalkylcyclopropyl1-1,2,4-triazolyl- oder -imidazolyl-derivate und ihre verwendung als antimykotische mittel

1988
- 1988-11-19 DE DE3839170A patent/DE3839170A1/de not_active Withdrawn
1989
- 1989-11-01 US US07/430,204 patent/US5059615A/en not_active Expired - Fee Related
- 1989-11-07 AT AT89120575T patent/ATE103907T1/de not_active IP Right Cessation
- 1989-11-07 ES ES89120575T patent/ES2052863T3/es not_active Expired - Lifetime
- 1989-11-07 DE DE89120575T patent/DE58907399D1/de not_active Expired - Fee Related
- 1989-11-07 EP EP89120575A patent/EP0370300B1/de not_active Expired - Lifetime
- 1989-11-17 CA CA002003213A patent/CA2003213C/en not_active Expired - Fee Related
- 1989-11-17 JP JP1297767A patent/JP2839161B2/ja not_active Expired - Lifetime
- 1989-11-17 KR KR1019890016675A patent/KR0128662B1/ko not_active Expired - Fee Related
- 1989-11-17 ZA ZA898775A patent/ZA898775B/xx unknown

Also Published As

Publication number	Publication date
JP2839161B2 (ja)	1998-12-16
CA2003213A1 (en)	1990-05-19
DE3839170A1 (de)	1990-05-31
CA2003213C (en)	1999-08-03
EP0370300B1 (de)	1994-04-06
EP0370300A2 (de)	1990-05-30
US5059615A (en)	1991-10-22
ATE103907T1 (de)	1994-04-15
ES2052863T3 (es)	1994-07-16
DE58907399D1 (de)	1994-05-11
KR0128662B1 (ko)	1998-04-04
ZA898775B (en)	1990-08-29
EP0370300A3 (de)	1991-07-03
JPH02243673A (ja)	1990-09-27

Publication	Publication Date	Title
FI903215A7 (fi)	1990-12-29	Heteroaryyliamino- ja heteroaryylioksipyridiiniamiineja ja niihin liittyviä yhdisteitä, menetelmä niiden valmistamiseksi sekä niiden käyttö lääkkeinä
IT1219811B (it)	1990-05-24	Derivati peptidici,loro preparazione e loro impiego come medicamenti
IT8219730A0 (it)	1982-02-18	Derivati 5-amminometil-ossazolidinici, procedimento per la loro preparazione, e loro applicazione in terapia.
ES511433A0 (es)	1983-02-16	"procedimiento de preparacion de productos utiles particularmente en medicamentos utilizables para el tratamiento de melanomas".
IT8821719A0 (it)	1988-08-19	Piperidine pontate, loro preparazione e loro impiego come medicamenti.
FI940810L (fi)	1994-08-24	Substituoidut bentseenisulfonyylivirtsa-aineet ja -tiovirtsa-aineet, menetelmä niiden valmistamiseksi ja niiden käyttö lääkkeinä
DE68908374D1 (de)	1993-09-16	Propenonoximether, verfahren zu dessen herstellung sowie diese enthaltende arzneinmittel.
FI902248A7 (fi)	1990-11-09	N-heteroaryyli-4-kinoliiniamiineja, menetelmä niiden valmistamiseksi ja niiden käyttö lääkkeinä
NL8601838A (nl)	1987-02-16	Distamycinederivaten, werkwijze voor de bereiding ervan, alsmede farmaceutische preparaten, die deze derivaten bevatten.
IT1219542B (it)	1990-05-18	Derivati pepticidi,loro preparazione e loro impiego come medicamenti
FI902850A7 (fi)	1990-12-10	N-heteroaryylipuriini-6-amiineja, menetelmä niiden valmistamiseksi ja niiden käyttö lääkeaineina
PT89478A (pt)	1989-10-04	Processo para a preparacao de piridinas di-substituidas
KR900007816A (ko)	1990-06-02	사이클로프로필-치환된 아졸릴메틸카비놀, 이의 제조방법 및 약제로서의 이의 용도
EP0230264A3 (en)	1988-12-14	Pharmaceutical composition for nasal application, process for its preparation and its use
FI903214A7 (fi)	1990-12-29	Naftyyliamino- ja naftyylioksi-pyrimidiinit ja niihin liittyvät yhdisteet, menetelmä niiden valmistamiseksi ja niiden käyttö dermatologisinalääkeaineina
FI896243A7 (fi)	1990-06-28	N-pyridinyyli-9H-karbatsoli-9-amiineja, menetelmä niiden valmistamiseksi sekä niiden käyttö lääkkeinä
NO890096D0 (no)	1989-01-10	Pyrazol- og indozolpyridinaminer, en fremgangsmaate for fremstilling og anvendelse derav som medikamenter.
PT87186A (pt)	1988-05-01	Imidazothiadiazine derivatives a process for preparing the same and their use as medicaments
IL89401A0 (en)	1989-09-10	Medicaments containing 1,4-dihydropyridine derivatives for the treatment of alcohol addiction
FI883692A7 (fi)	1989-02-08	Menetelmä ulkoisesti käytettävän, ihoon erääntyvän antiviraalisen farmaseuttisen koostumuksen valmistamiseksi
DE3380989D1 (de)	1990-01-25	2-aminobenzosaeurederivate, verfahren zu ihrer herstellung und pharmazeutische zubereitungen.
FI810990A7 (fi)	1981-10-03	Bifenylyyli- atsolyylietaanijohdannaiset, menetelmä niiden valmistamiseksi ja niiden käyttö lääkeaineina.
IT1211681B (it)	1989-11-03	Peptidi e derivati peptidici, loro preparazione e loro impiego come medicamenti
PT86642A (pt)	1988-02-01	Arylthiadiazolylsulfonamides and derivatives a process for thir preparation and their use as medicaments
DK256689D0 (da)	1989-05-26	1,2-dithiol-3-thion-s-oxid-forbindelser til anven delse som laegemidler

Legal Events

Date	Code	Title	Description
1989-11-17	PA0109	Patent application	St.27 status event code: A-0-1-A10-A12-nap-PA0109
1989-11-17	R17-X000	Change to representative recorded	St.27 status event code: A-3-3-R10-R17-oth-X000
1989-12-05	P11-X000	Amendment of application requested	St.27 status event code: A-2-2-P10-P11-nap-X000
1989-12-05	P13-X000	Application amended	St.27 status event code: A-2-2-P10-P13-nap-X000
1990-06-02	PG1501	Laying open of application	St.27 status event code: A-1-1-Q10-Q12-nap-PG1501
1991-03-13	R17-X000	Change to representative recorded	St.27 status event code: A-3-3-R10-R17-oth-X000
1994-08-12	A201	Request for examination
1994-08-12	PA0201	Request for examination	St.27 status event code: A-1-2-D10-D11-exm-PA0201
1997-03-05	E902	Notification of reason for refusal
1997-03-05	PE0902	Notice of grounds for rejection	St.27 status event code: A-1-2-D10-D21-exm-PE0902
1997-05-03	P11-X000	Amendment of application requested	St.27 status event code: A-2-2-P10-P11-nap-X000
1997-05-03	P13-X000	Application amended	St.27 status event code: A-2-2-P10-P13-nap-X000
1997-05-03	R17-X000	Change to representative recorded	St.27 status event code: A-3-3-R10-R17-oth-X000
1997-08-25	E701	Decision to grant or registration of patent right
1997-08-25	PE0701	Decision of registration	St.27 status event code: A-1-2-D10-D22-exm-PE0701
1997-11-04	GRNT	Written decision to grant
1997-11-04	PR0701	Registration of establishment	St.27 status event code: A-2-4-F10-F11-exm-PR0701
1997-11-04	PR1002	Payment of registration fee	St.27 status event code: A-2-2-U10-U11-oth-PR1002 Fee payment year number: 1
1998-04-04	PG1601	Publication of registration	St.27 status event code: A-4-4-Q10-Q13-nap-PG1601
1999-01-06	R18-X000	Changes to party contact information recorded	St.27 status event code: A-5-5-R10-R18-oth-X000
1999-02-22	R18-X000	Changes to party contact information recorded	St.27 status event code: A-5-5-R10-R18-oth-X000
1999-02-25	R18-X000	Changes to party contact information recorded	St.27 status event code: A-5-5-R10-R18-oth-X000
1999-03-03	PN2301	Change of applicant	St.27 status event code: A-5-5-R10-R13-asn-PN2301 St.27 status event code: A-5-5-R10-R11-asn-PN2301
2000-08-11	R18-X000	Changes to party contact information recorded	St.27 status event code: A-5-5-R10-R18-oth-X000
2000-11-05	LAPS	Lapse due to unpaid annual fee
2000-11-05	PC1903	Unpaid annual fee	St.27 status event code: A-4-4-U10-U13-oth-PC1903 Not in force date: 20001105 Payment event data comment text: Termination Category : DEFAULT_OF_REGISTRATION_FEE
2000-11-09	R18-X000	Changes to party contact information recorded	St.27 status event code: A-5-5-R10-R18-oth-X000
2001-08-11	PC1903	Unpaid annual fee	St.27 status event code: N-4-6-H10-H13-oth-PC1903 Ip right cessation event data comment text: Termination Category : DEFAULT_OF_REGISTRATION_FEE Not in force date: 20001105
2004-01-06	R18-X000	Changes to party contact information recorded	St.27 status event code: A-5-5-R10-R18-oth-X000
2010-12-27	R18-X000	Changes to party contact information recorded	St.27 status event code: A-5-5-R10-R18-oth-X000
2016-10-19	R18-X000	Changes to party contact information recorded	St.27 status event code: A-5-5-R10-R18-oth-X000