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HK83384A - Long-acting parenteral compositions of haloperidol and bromperidol derivatives - Google Patents

Long-acting parenteral compositions of haloperidol and bromperidol derivatives

Info

Publication number
HK83384A
HK83384A HK833/84A HK83384A HK83384A HK 83384 A HK83384 A HK 83384A HK 833/84 A HK833/84 A HK 833/84A HK 83384 A HK83384 A HK 83384A HK 83384 A HK83384 A HK 83384A
Authority
HK
Hong Kong
Prior art keywords
bromperidol
haloperidol
long
derivatives
parenteral compositions
Prior art date
Application number
HK833/84A
Inventor
Niemegeers Carlos
Original Assignee
Janssen Pharmaceutica N.V.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Janssen Pharmaceutica N.V. filed Critical Janssen Pharmaceutica N.V.
Publication of HK83384A publication Critical patent/HK83384A/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/36—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D211/40—Oxygen atoms
    • C07D211/44—Oxygen atoms attached in position 4
    • C07D211/52—Oxygen atoms attached in position 4 having an aryl radical as the second substituent in position 4
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/20—Hypnotics; Sedatives

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Anesthesiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
  • Medicinal Preparation (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

Abstract

Long-acting neuraleptic compositions for parenteral, in particular intramuscular or subcutaneous, administration, comprise a decanoate ester of haloperidol or bromperidol in sesame oil as a solvent. The esters may be prepared by known methods.
HK833/84A 1979-06-28 1984-11-01 Long-acting parenteral compositions of haloperidol and bromperidol derivatives HK83384A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP8082679A JPS568318A (en) 1979-06-28 1979-06-28 Non oral long acting composition of haloperidol and bromperidol derivative

Publications (1)

Publication Number Publication Date
HK83384A true HK83384A (en) 1984-11-09

Family

ID=13729223

Family Applications (1)

Application Number Title Priority Date Filing Date
HK833/84A HK83384A (en) 1979-06-28 1984-11-01 Long-acting parenteral compositions of haloperidol and bromperidol derivatives

Country Status (9)

Country Link
JP (1) JPS568318A (en)
BE (1) BE883994A (en)
CY (1) CY1255A (en)
DE (1) DE3024305A1 (en)
FR (1) FR2460932A1 (en)
GB (1) GB2054371B (en)
HK (1) HK83384A (en)
KE (1) KE3427A (en)
NL (1) NL190775C (en)

Families Citing this family (21)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8621892D0 (en) * 1986-09-11 1986-10-15 Lundbeck & Co As H Organic compound
DK238190D0 (en) * 1990-10-03 1990-10-03 Lundbeck & Co As H DEPOT DERIVATIVES
ES2077547T3 (en) * 1992-11-17 2000-06-16 Yoshitomi Pharmaceutical SUSTAINED RELEASE MICROSPHERE CONTAINING AN ANTIPSYCHOTIC AND PRODUCTION PROCEDURE.
EP0937053A1 (en) * 1996-10-31 1999-08-25 THE UNITED STATES OF AMERICA, as represented by the Secretary of the Department of Health and Human Services Sustained-release derivatives of hydroxylated analogs of substituted 1- 2 bis(aryl)methoxy]ethyl]-piperazines and -homopiperazines and their use as noncompetitive antagonists of dopamine reuptake
RU2178297C1 (en) * 2001-02-02 2002-01-20 Открытое акционерное общество "Химико-фармацевтический комбинат "Акрихин" Pharmaceutical composition eliciting antipsychotic and antiemetic action and method of its preparing
US8003617B2 (en) 2004-11-10 2011-08-23 Genzyme Corporation Methods of treating diabetes mellitus
US8716327B2 (en) 2006-05-09 2014-05-06 Genzyme Corporation Methods of treating fatty liver disease
EP2594563B1 (en) 2007-05-31 2018-07-18 Genzyme Corporation 2-acylaminopropanol-type glucosylceramide synthase inhibitors
WO2009045503A1 (en) 2007-10-05 2009-04-09 Genzyme Corporation Method of treating polycystic kidney diseases with ceramide derivatives
JP2011529500A (en) 2008-07-28 2011-12-08 ジェンザイム コーポレーション Glucosylceramide synthase inhibition for the treatment of collapsing glomerulopathy and other glomerular diseases
CA2738768C (en) 2008-10-03 2017-10-31 Genzyme Corporation 2-acylaminopropoanol-type glucosylceramide synthase inhibitors
LT2685979T (en) 2011-03-18 2016-12-12 Alkermes Pharma Ireland Limited Injectable pharmaceutical compositions comprising a water-insoluble anti-psychotic, sorbitan laurate and polysorbate 20
CN103301461B (en) * 2012-03-08 2018-09-07 江苏豪森药业集团有限公司 A kind of long acting injection and its preparation method and application
WO2013142198A1 (en) 2012-03-19 2013-09-26 Alkermes Pharma Ireland Limited Pharmaaceutical compositions comprising fatty acid esters
CA2867137C (en) 2012-03-19 2020-12-08 Alkermes Pharma Ireland Limited Pharmaceutical compositions comprising aripiprazole prodrugs and benzyl alcohol
ES2764383T3 (en) 2012-03-19 2020-06-03 Alkermes Pharma Ireland Ltd Pharmaceutical compositions comprising glycerol esters
NZ631345A (en) 2012-09-19 2017-06-30 Alkermes Pharma Ireland Ltd Pharmaceutical compositions having improved storage stability
BR112016021535A8 (en) 2014-03-20 2021-07-20 Alkermes Pharma Ireland Ltd kit comprising aripiprazole formulations having increased injection rates useful for the treatment of a central nervous system disorder and use
CA3092335A1 (en) 2018-03-05 2019-09-12 Alkermes Pharma Ireland Limited Aripiprazole dosing strategy
CN113117092A (en) * 2020-01-14 2021-07-16 中国科学院上海药物研究所 Non-aqueous sustained-release drug delivery system
HUP2100259A1 (en) 2021-07-07 2023-01-28 Richter Gedeon Nyrt Controlled release injectable cariprazine formulation

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3408356A (en) * 1965-08-31 1968-10-29 Squibb & Sons Inc Long chain esters of 4'-fluoro-4-[4-hydroxy-4-(alpha, alpha, alpha-trifluorotolyl)piperi-dino]butyrophenone and the like
DE1695194A1 (en) * 1966-07-11 1971-03-18 Hoffmann La Roche Process for the preparation of piperidine derivatives
US3850935A (en) * 1971-10-16 1974-11-26 Sumitomo Chemical Co Process for producing piperidine derivatives by degrading quaternary piperidinium salts

Also Published As

Publication number Publication date
FR2460932B1 (en) 1984-11-16
DE3024305C2 (en) 1989-12-07
FR2460932A1 (en) 1981-01-30
DE3024305A1 (en) 1981-01-22
NL190775B (en) 1994-03-16
CY1255A (en) 1984-08-31
JPS568318A (en) 1981-01-28
KE3427A (en) 1984-08-10
NL190775C (en) 1994-08-16
BE883994A (en) 1980-12-29
GB2054371B (en) 1983-08-03
NL8003583A (en) 1980-12-30
GB2054371A (en) 1981-02-18

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Legal Events

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PE Patent expired