JP2008150386A

JP2008150386A - トロンボポエチン受容体アゴニスト作用を有する化合物

Info

Publication number: JP2008150386A
Application number: JP2008022275A
Authority: JP
Inventors: Hiroshi Takemoto; 浩武本; Takeshi Shioda; 武司塩田; Masami Takayama; 正己高山
Original assignee: Shionogi and Co Ltd
Current assignee: Shionogi and Co Ltd
Priority date: 2000-01-24
Filing date: 2008-02-01
Publication date: 2008-07-03
Also published as: TWI284639B; CA2397018A1; EP1253142A1; US7582665B2; US20030195231A1; KR20030016219A; EP1253142A4; AU2708901A; US20100022542A1; KR20050085991A; CN100491356C; CN1419547A; AU777777B2; WO2001053267A1; CA2397018C; JP4136371B2; KR100563795B1

Abstract

【課題】トロンボポエチンアゴニスト作用を有する化合物を提供する。
【解決手段】一般式（Ｉ）：
【化１】

［式中、Ｘ^１は置換されていてもよいアリール、置換されていてもよいヘテロアリール等；Ｙ^１は−ＮＲ^ＡＣＯ−（ＣＨ_２）_０−２−等（式中、Ｒ^Ａは水素原子等）；Ｚ^１は置換されていてもよいフェニレン等；Ｗ^１は式：
【化２】

（式中、Ｒ^１、Ｒ^２、Ｒ^３、およびＲ^４はそれぞれ独立して、水素原子、置換されていてもよい低級アルキル等、破線は結合の存在または不存在を表わす）で表わされる基等］で示される化合物、そのプロドラッグ、もしくはそれらの製薬上許容される塩、またはそれらの溶媒和物を有効成分として含有するトロンボポエチン受容体アゴニスト作用を有する医薬組成物。
【選択図】なし

Description

本発明は、トロンボポエチン受容体アゴニスト作用を有する化合物に関する。

トロンボポエチンは、３３２個のアミノ酸からなるポリペプチドサイトカインであり、受容体を介して巨核球細胞の分化、増殖を刺激することにより血小板産生を亢進することから、血小板減少症等の血小板数の異常を伴う血液疾患の病態に対する薬剤として期待されている。トロンボポエチン受容体をコードする遺伝子の塩基配列は、非特許文献１に記載されている。特許文献１および２にトロンボポエチン受容体に親和性を有する低分子ペプチドも知られているが、これらのペプチド誘導体の経口投与は一般的に実用的でない。
トロンボポエチン受容体に親和性を有する低分子化合物としては、１，４−ベンゾチアゼピン誘導体が特許文献３および４に記載されている。
本発明化合物と類似の構造を有する化合物が特許文献５等に記載されているが、トロンボポエチン受容体親和性に関する記載はない。
特開平１０−７２４９２号公報国際公開第９６／４０７５０号パンフレット特開平１１−１４７７号公報特開平１１−１５２２７６号公報特開平１０−２８７６３４号公報プロシーディングオブザナショナルアカデミーオブサイエンスオブザユナイテッドステイトオブアメリカ（Proc. Natl. Acad. Sci.）１９９２年、第８９巻、５６４０−５６４４

トロンボポエチン受容体アゴニスト作用を有する医薬組成物を創製し、経口投与可能な血小板産生調節剤を提供する。

本発明者らは以上の点に鑑み、鋭意検討を重ねた結果、以下に示す化合物が強いトロンボポエチン受容体アゴニスト活性を示すことを見出した。
すなわち、本発明は、１）一般式（Ｉ）：

［式中、Ｘ^１は置換されていてもよいアリール、置換されていてもよいアラルキル、置換されていてもよいヘテロアリール、または置換されていてもよいヘテロアリールアルキル；
Ｙ^１は−ＮＲ^ＡＣＯ−（ＣＲ^ＣＲ^Ｄ）_０−２−、−ＮＲ^ＡＣＯ−（ＣＨ_２）_０−２−Ｖ−、−ＮＲ^ＡＣＯ−ＣＲ^Ｃ＝ＣＲ^Ｄ−、−Ｖ−（ＣＨ_２）_１−５−ＮＲ^ＡＣＯ−（ＣＨ_２）_０−２−、−Ｖ−（ＣＨ_２）_１−５−ＣＯＮＲ^Ａ−（ＣＨ_２）_０−２−、−ＣＯＮＲ^Ａ−（ＣＨ_２）_０−２−、−（ＣＨ_２）_０−２−ＮＲ^Ａ−ＳＯ_２−（ＣＨ_２）_０−２−、−（ＣＨ_２）_０−２−ＳＯ_２−ＮＲ^Ａ−（ＣＨ_２）_０−２−、−ＮＲ^Ａ−（ＣＨ_２）_０−２−、−ＮＲ^Ａ−ＣＯ−ＮＲ^Ａ−、−ＮＲ^Ａ−ＣＳ−ＮＲ^Ａ−、−Ｎ＝Ｃ（−ＳＲ^Ａ）−ＮＲ^Ａ−、−ＮＲ^ＡＣＳＮＲ^ＡＣＯ−、−Ｎ＝Ｃ（−ＳＲ^Ａ）−ＮＲ^ＡＣＯ−、−ＮＲ^Ａ−（ＣＨ_２）_１−２−ＮＲ^Ａ−ＣＯ−、−ＮＲ^ＡＣＯＮＲ^ＡＮＲ^ＢＣＯ−、または−Ｎ＝Ｃ（−ＮＲ^ＡＲ^Ａ）−ＮＲ^ＡＣＯ−（式中、Ｒ^Ａはそれぞれ独立して水素原子または低級アルキル；Ｒ^Ｂは水素原子またはフェニル；Ｒ^ＣおよびＲ^Ｄはそれぞれ独立して、水素原子、ハロゲン、置換されていてもよい低級アルキル、置換されていてもよい低級アルキルオキシ、置換されていてもよい低級アルキルチオ、置換されていてもよい低級アルケニル、置換されていてもよい低級アルキニル、置換されていてもよいアリール、置換されていてもよいヘテロアリール、置換されていてもよいシクロアルキル、置換されていてもよいアラルキル、置換されていてもよいヘテロアリールアルキル、置換されていてもよい非芳香族複素環基、または置換されていてもよいアミノ；Ｖは酸素原子または硫黄原子）；
Ｚ^１は置換されていてもよいフェニレン、置換されていてもよい単環ヘテロアリレン、置換されていてもよい単環非芳香族複素環ジイル、または置換されていてもよい単環シクロアルカンジイル；
Ｗ^１は式：

（式中、Ｒ^１、Ｒ^２、Ｒ^３、Ｒ^４、Ｒ^７、およびＲ^８はそれぞれ独立して、水素原子、ハロゲン、置換されていてもよい低級アルキル、置換されていてもよい低級アルキルオキシ、置換されていてもよい低級アルキルチオ、置換されていてもよい低級アルケニル、置換されていてもよい低級アルキニル、置換されていてもよいアリール、置換されていてもよいヘテロアリール、置換されていてもよいシクロアルキル、置換されていてもよいアラルキル、置換されていてもよいヘテロアリールアルキル、置換されていてもよい非芳香族複素環基、または置換されていてもよいアミノ；
Ｒ^５、Ｒ^６、およびＲ^９はそれぞれ独立して、水素原子、置換されていてもよい低級アルキル、置換されていてもよい低級アルケニル、置換されていてもよい低級アルキニル、置換されていてもよいアリール、置換されていてもよいヘテロアリール、置換されていてもよいシクロアルキル、置換されていてもよいアラルキル、置換されていてもよいヘテロアリールアルキル、または置換されていてもよい非芳香族複素環基；
Ａ^１は置換されていてもよいアリールまたは置換されていてもよいヘテロアリール；
破線（−−−）は結合の存在または不存在を表わす）で表わされる基］で示される化合物、そのプロドラッグ、もしくはそれらの製薬上許容される塩、またはそれらの溶媒和物を有効成分として含有するトロンボポエチン受容体アゴニスト作用を有する医薬組成物、に関する。
さらに詳しくは、以下に示す２）〜２９）に関する。
２）Ｘ^１が置換されていてもよいヘテロアリールである１）記載のトロンボポエチン受容体アゴニスト作用を有する医薬組成物。
３）Ｘ^１が式：

（式中、Ｒ^１０およびＲ^１１はそれぞれ独立して水素原子、置換されていてもよい低級アルキル、カルボキシ、低級アルキルオキシカルボニル、ハロゲン、置換されていてもよいアミノカルボニル、置換されていてもよいヘテロアリール、または置換されていてもよいアリール；Ｒ^１２は水素原子または低級アルキル）で示される基である１）記載のトロンボポエチン受容体アゴニスト作用を有する医薬組成物。
４）Ｘ^１が式：

（式中、Ｒ^１０およびＲ^１１は３）と同意義）で示される基である１）記載のトロンボポエチン受容体アゴニスト作用を有する医薬組成物。
５）Ｙ^１が−ＮＨＣＯ−、−ＣＯＮＨ−、−ＮＨＣＨ_２−、−ＮＨＣＯ−ＣＨ＝ＣＨ−、または−ＮＨＳＯ_２−である１）〜４）のいずれかに記載のトロンボポエチン受容体アゴニスト作用を有する医薬組成物。
６）Ｙ^１が−ＮＨＣＯ−である１）〜４）のいずれかに記載のトロンボポエチン受容体アゴニスト作用を有する医薬組成物。
７）Ｚ^１がハロゲンまたは低級アルキルで置換されていてもよい１，４−フェニレンである１）〜６）のいずれかに記載のトロンボポエチン受容体アゴニスト作用を有する医薬組成物。
８）Ｒ^１が水素原子または低級アルキルである１）〜７）のいずれかに記載のトロンボポエチン受容体アゴニスト作用を有する医薬組成物。
９）Ｒ^２が水素原子、低級アルキル、ハロゲン、低級アルキルオキシ、低級アルキルチオ、または置換されていてもよいアミノである１）〜８）のいずれかに記載のトロンボポエチン受容体アゴニスト作用を有する医薬組成物。
１０）Ｗ^１が式：

（式中、Ｒ^１３は水素原子、低級アルキル、低級アルキルオキシ、低級アルキルチオ、またはハロゲン；Ｒ^１４およびＲ^１５はそれぞれ独立して水素原子、またはそれぞれ以下の置換基群Ａから選択される１以上の置換基によって置換されていてもよい低級アルキル、低級アルケニル、低級アルキニル、シクロアルキル、アリール、アラルキル、ヘテロアリール、もしくはヘテロアリールアルキル；破線は１）と同意義；
置換基群Ａ：ハロゲン、ハロ低級アルキル、置換されていてもよいアミノ、カルボキシ、低級アルキルチオ、低級アルキルシリル、または低級アルキルオキシ）で表わされる基である、１）〜９）のいずれかに記載のトロンボポエチン受容体アゴニスト作用を有する医薬組成物。
１１）Ｗ^１が式：

（式中、Ｒ^１３は水素原子、低級アルキル、低級アルキルオキシ、低級アルキルチオ、またはハロゲン；Ｒ^２６は水素原子または低級アルキル；破線は１）と同意義）で表わされる基である、１）〜９）のいずれかに記載のトロンボポエチン受容体アゴニスト作用を有する医薬組成物。
１２）血小板産生調節剤である１）〜１１）のいずれかに記載のトロンボポエチン受容体アゴニスト作用を有する医薬組成物。
１３）血小板産生を調節するための医薬を製造するための１）〜１１）のいずれかに記載の化合物の使用。
１４）１）〜１１）のいずれかに記載の化合物の治療上効果を示す量を人を含む哺乳動物に投与することからなる、哺乳動物の血小板産生を調節する方法。
１５）一般式（ＩＩ）：

［式中、Ｘ^２は置換されていてもよい５員ヘテロアリールまたは置換されていてもよいピリジル；
Ｙ^２は−ＮＲ^ＡＣＯ−（ＣＲ^ＣＲ^Ｄ）_０−２−、−ＮＲ^ＡＣＯ−（ＣＨ_２）_０−２−Ｖ−、−ＮＲ^ＡＣＯ−ＣＲ^Ｃ＝ＣＲ^Ｄ−、−Ｖ−（ＣＨ_２）_１−５−ＮＲ^ＡＣＯ−（ＣＨ_２）_０−２−、−Ｖ−（ＣＨ_２）_１−５−ＣＯＮＲ^Ａ−（ＣＨ_２）_０−２−、−ＣＯＮＲ^Ａ−（ＣＨ_２）_０−２−、−（ＣＨ_２）_０−２−ＮＲ^Ａ−ＳＯ_２−（ＣＨ_２）_０−２−、−（ＣＨ_２）_０−２−ＳＯ_２−ＮＲ^Ａ−（ＣＨ_２）_０−２−、−ＮＲ^Ａ−（ＣＨ_２）_０−２−、−ＮＲ^Ａ−ＣＯ−ＮＲ^Ａ−、−ＮＲ^Ａ−ＣＳ−ＮＲ^Ａ−、−Ｎ＝Ｃ（−ＳＲ^Ａ）−ＮＲ^Ａ−、−ＮＲ^ＡＣＳＮＲ^ＡＣＯ−、−Ｎ＝Ｃ（−ＳＲ^Ａ）−ＮＲ^ＡＣＯ−、−ＮＲ^Ａ−（ＣＨ_２）_１−２−ＮＲ^Ａ−ＣＯ−、−ＮＲ^ＡＣＯＮＲ^ＡＮＲ^ＢＣＯ−、または−Ｎ＝Ｃ（−ＮＲ^ＡＲ^Ａ）−ＮＲ^ＡＣＯ−（式中、Ｒ^Ａはそれぞれ独立して水素原子または低級アルキル；Ｒ^Ｂは水素原子またはフェニル；Ｒ^ＣおよびＲ^Ｄはそれぞれ独立して、水素原子、ハロゲン、置換されていてもよい低級アルキル、置換されていてもよい低級アルキルオキシ、置換されていてもよい低級アルキルチオ、置換されていてもよい低級アルケニル、置換されていてもよい低級アルキニル、置換されていてもよいアリール、置換されていてもよいヘテロアリール、置換されていてもよいシクロアルキル、置換されていてもよいアラルキル、置換されていてもよいヘテロアリールアルキル、置換されていてもよい非芳香族複素環基、または置換されていてもよいアミノ；Ｖは酸素原子または硫黄原子）；
Ｚ^２は置換されていてもよいフェニレン、置換されていてもよい２，５−ピリジンジイル、置換されていてもよい２，５−チオフェンジイル、または置換されていてもよい２，５−フランジイル；
Ｗ^２は式：

（式中、Ｒ^１、Ｒ^２、Ｒ^３、Ｒ^４、Ｒ^７、およびＲ^８はそれぞれ独立して、水素原子、ハロゲン、置換されていてもよい低級アルキル、置換されていてもよい低級アルキルオキシ、置換されていてもよい低級アルキルチオ、置換されていてもよい低級アルケニル、置換されていてもよい低級アルキニル、置換されていてもよいアリール、置換されていてもよいヘテロアリール、置換されていてもよいシクロアルキル、置換されていてもよいアラルキル、置換されていてもよいヘテロアリールアルキル、置換されていてもよい非芳香族複素環基、または置換されていてもよいアミノ；
Ｒ^５、Ｒ^６、およびＲ^９はそれぞれ独立して、水素原子、置換されていてもよい低級アルキル、置換されていてもよい低級アルケニル、置換されていてもよい低級アルキニル、置換されていてもよいアリール、置換されていてもよいヘテロアリール、置換されていてもよいシクロアルキル、置換されていてもよいアラルキル、置換されていてもよいヘテロアリールアルキル、または置換されていてもよい非芳香族複素環基；
Ａ^２は置換されていてもよいアリールまたは置換されていてもよいヘテロアリール；
破線（−−−）は結合の存在または不存在を表わす）で表わされる基；
ただし、Ｒ^２はイミダゾリル、トリアゾリル、またはテトラゾリルではない］で示される化合物、そのプロドラッグ、もしくはそれらの製薬上許容される塩、またはそれらの溶媒和物。
１６）Ｘ^２が式：

（式中、Ｒ^１０およびＲ^１１はそれぞれ独立して水素原子、置換されていてもよい低級アルキル、カルボキシ、低級アルキルオキシカルボニル、ハロゲン、置換されていてもよいアミノカルボニル、置換されていてもよいヘテロアリール、または置換されていてもよいアリール）で示される基である１５）記載の化合物、そのプロドラッグ、もしくはそれらの製薬上許容される塩、またはそれらの溶媒和物。
１７）Ｘ^２が式：

（式中、Ｒ^１６は水素原子、置換されていてもよい低級アルキル、カルボキシ、低級アルキルオキシカルボニル、ハロゲン、または置換されていてもよいアミノカルボニル；
Ｒ^１７、Ｒ^１８、Ｒ^１９、Ｒ^２０、Ｒ^２１、Ｒ^２２、およびＲ^２３はそれぞれ独立して水素原子、置換基群Ｂから選択される１以上の置換基によって置換されていてもよいアルキル、シクロアルキル、置換基群Ｂから選択される１以上の置換基によって置換されていてもよいアルキルオキシ、アルキルチオ、ハロゲン、置換基群Ｃから選択される１以上の置換基によって置換されていてもよいフェニル、置換基群Ｃから選択される１以上の置換基によって置換されていてもよいヘテロアリール、または置換基群Ｃから選択される１以上の置換基によって置換されていてもよい非芳香族複素環基、
置換基群Ｂ：ヒドロキシ、アルキルオキシ、ハロゲン、カルボキシ、低級アルキルオキシカルボニル、アリールオキシカルボニル、置換されていてもよいアミノ、置換基群Ｃから選択される１以上の置換基によって置換されていてもよいフェニル、非芳香族複素環基、およびヘテロアリール、
置換基群Ｃ：ヒドロキシ、アルキル、ハロゲン、ハロ低級アルキル、カルボキシ、低級アルキルオキシカルボニル、アルキルオキシ、置換されていてもよいアミノ、非芳香族複素環、およびヘテロアリール；
Ｒ^１６およびＲ^１７は一緒になって−ＣＨ_２−、−ＣＨ_２ＣＨ_２−、−ＣＨ_２ＣＨ_２ＣＨ_２−、−ＯＣＨ_２−、または−ＳＣＨ_２−を形成してもよい）で示される基である１５）または１６）記載の化合物、そのプロドラッグ、もしくはそれらの製薬上許容される塩、またはそれらの溶媒和物。
１８）Ｙ^２が−ＮＨＣＯ−である１５）〜１７）のいずれかに記載の化合物、そのプロドラッグ、もしくはそれらの製薬上許容される塩、またはそれらの溶媒和物。
１９）Ｚ^２がハロゲンまたは低級アルキルで置換されていてもよい１，４−フェニレンである１５）〜１８）のいずれかに記載の化合物、そのプロドラッグ、もしくはそれらの製薬上許容される塩、またはそれらの溶媒和物。
２０）Ｒ^１が水素原子または低級アルキルである１５）〜１９）のいずれかに記載の化合物、そのプロドラッグ、もしくはそれらの製薬上許容される塩、またはそれらの溶媒和物。
２１）Ｒ^２が水素原子、低級アルキル、ハロゲン、低級アルキルオキシ、低級アルキルチオ、または置換されていてもよいアミノである１５）〜２０）のいずれかに記載の化合物、そのプロドラッグ、もしくはそれらの製薬上許容される塩、またはそれらの溶媒和物。
２２）Ｗ^２が式：

（式中、Ｒ^１、Ｒ^２、Ｒ^３、Ｒ^４、Ｒ^５、Ｒ^６、Ｒ^７、Ｒ^８、およびＡ^２は１５）と同意義、ただし、Ｒ^２はイミダゾリル、トリアゾリル、またはテトラゾリルではない）である１５）〜２１）のいずれかに記載の化合物、そのプロドラッグ、もしくはそれらの製薬上許容される塩、またはそれらの溶媒和物。
２３）Ｗ^２が式：

（式中、Ｒ^１３は水素原子、低級アルキル、低級アルキルオキシ、低級アルキルチオ、またはハロゲン、Ｒ^１４およびＲ^１５はそれぞれ独立して水素原子、またはそれぞれ以下の置換基群Ａから選択される１以上の置換基によって置換されていてもよい低級アルキル、低級アルケニル、低級アルキニル、シクロアルキル、アリール、アラルキル、ヘテロアリール、ヘテロアリールアルキル、もしくは非芳香族複素環基；
置換基群Ａ：ハロゲン、ハロ低級アルキル、置換されていてもよいアミノ、カルボキシ、低級アルキルチオ、低級アルキルシリル、または低級アルキルオキシ）である１５）〜２２）のいずれかに記載の化合物、そのプロドラッグ、もしくはそれらの製薬上許容される塩、またはそれらの溶媒和物。
２４）Ｗ^２が式：

（式中、Ｒ^１３は水素原子、低級アルキル、低級アルキルオキシ、低級アルキルチオ、またはハロゲン；Ｒ^２６は水素原子または低級アルキル；破線は１５）と同意義）で表わされる基である、１５）〜２２）のいずれかに記載の化合物、そのプロドラッグ、もしくはそれらの製薬上許容される塩、またはそれらの溶媒和物。
２５）一般式（ＩＩＩ）：

［式中、Ｒ^１６は水素原子、置換されていてもよい低級アルキル、カルボキシ、低級アルキルオキシカルボニル、ハロゲン、または置換されていてもよいアミノカルボニル；
Ｒ^１７、Ｒ^１８、Ｒ^１９、Ｒ^２０、およびＲ^２１はそれぞれ独立して水素原子、置換基群Ｂから選択される１以上の置換基によって置換されていてもよいアルキル、シクロアルキル、置換基群Ｂから選択される１以上の置換基によって置換されていてもよいアルキルオキシ、アルキルチオ、ハロゲン、置換基群Ｃから選択される１以上の置換基によって置換されていてもよいフェニル、置換基群Ｃから選択される１以上の置換基によって置換されていてもよいヘテロアリール、または置換基群Ｃから選択される１以上の置換基によって置換されていてもよい非芳香族複素環基、
置換基群Ｂ：ヒドロキシ、アルキルオキシ、ハロゲン、カルボキシ、低級アルキルオキシカルボニル、アリールオキシカルボニル、置換されていてもよいアミノ、置換基群Ｃから選択される１以上の置換基によって置換されていてもよいフェニル、非芳香族複素環基、およびヘテロアリール、
置換基群Ｃ：ヒドロキシ、アルキル、ハロゲン、ハロ低級アルキル、カルボキシ、低級アルキルオキシカルボニル、アルキルオキシ、置換されていてもよいアミノ、非芳香族複素環、およびヘテロアリール；
Ｒ^１６およびＲ^１７は一緒になって−ＣＨ_２−、−ＣＨ_２ＣＨ_２−、−ＣＨ_２ＣＨ_２ＣＨ_２−、−ＯＣＨ_２−、または−ＳＣＨ_２−を形成してもよい；
Ｒ^３１およびＲ^３２はそれぞれ独立して、水素原子、低級アルキル、ハロゲン、ハロ低級アルキル、低級アルキルオキシ、ハロ低級アルキルオキシ、またはヒドロキシ；
Ｗ^３は式：

（式中、Ｒ^１３は水素原子、低級アルキル、低級アルキルオキシ、低級アルキルチオ、またはハロゲン；
Ｒ^１４およびＲ^１５はそれぞれ独立して水素原子、またはそれぞれ以下の置換基群Ａにより置換されていてもよい低級アルキル、低級アルケニル、低級アルキニル、シクロアルキル、アリール、アラルキル、ヘテロアリール、ヘテロアリールアルキル、もしくは非芳香族複素環基；
置換基群Ａ：ハロゲン、ハロ低級アルキル、置換されていてもよいアミノ、カルボキシ、低級アルキルチオ、低級アルキルシリル、または低級アルキルオキシ；
Ｒ^２４は水素原子または低級アルキル；
Ｒ^２５は低級アルキル、置換されていてもよいアリール、または置換されていてもよい非芳香族複素環；
Ａ^３はヘテロアリール）で表わされる基］で示される化合物、そのプロドラッグ、もしくはそれらの製薬上許容される塩、またはそれらの溶媒和物。
２６）一般式（ＩＶ−Ａ）：

［式中、Ｒ^２７は水素原子、Ｃ１−３アルキル、トリフルオロメチル、またはハロゲン；
Ｒ^２８、Ｒ^２９、およびＲ^３０はそれぞれ独立して水素原子、置換基群Ｂから選択される１以上の置換基によって置換されていてもよいアルキル、シクロアルキル、置換基群Ｂから選択される１以上の置換基によって置換されていてもよいアルキルオキシ、アルキルチオ、ハロゲン、置換基群Ｃから選択される１以上の置換基によって置換されていてもよいフェニル、置換基群Ｃから選択される１以上の置換基によって置換されていてもよいヘテロアリール、または置換基群Ｃから選択される１以上の置換基によって置換されていてもよい非芳香族複素環基、
置換基群Ｂ：ヒドロキシ、アルキルオキシ、ハロゲン、カルボキシ、低級アルキルオキシカルボニル、アリールオキシカルボニル、置換されていてもよいアミノ、置換基群Ｃから選択される１以上の置換基によって置換されていてもよいフェニル、非芳香族複素環基、およびヘテロアリール、
置換基群Ｃ：ヒドロキシ、アルキル、ハロゲン、ハロ低級アルキル、カルボキシ、低級アルキルオキシカルボニル、アルキルオキシ、置換されていてもよいアミノ、非芳香族複素環、およびヘテロアリール；
Ｒ^３１およびＲ^３２はそれぞれ独立して、水素原子、低級アルキル、ハロゲン、ハロ低級アルキル、低級アルキルオキシ、ハロ低級アルキルオキシ、またはヒドロキシ；
Ｗ^４は式：

（式中、Ｒ^１３は水素原子、低級アルキル、低級アルキルオキシ、低級アルキルチオ、またはハロゲン；
Ｒ^１４およびＲ^１５はそれぞれ独立して水素原子、またはそれぞれ以下の置換基群Ａにより置換されていてもよい低級アルキル、低級アルケニル、低級アルキニル、シクロアルキル、アリール、アラルキル、ヘテロアリール、ヘテロアリールアルキル、もしくは非芳香族複素環基；
置換基群Ａ：ハロゲン、ハロ低級アルキル、置換されていてもよいアミノ、カルボキシ、低級アルキルチオ、低級アルキルシリル、または低級アルキルオキシ；
Ｒ^２４は水素原子または低級アルキル）で表わされる基］で示される化合物、そのプロドラッグ、もしくはそれらの製薬上許容される塩、またはそれらの溶媒和物。
２７）一般式（ＩＶ−Ｂ）：

［式中、Ｒ^２８、Ｒ^２９、およびＲ^３０はそれぞれ独立して水素原子、置換基群Ｂから選択される１以上の置換基によって置換されていてもよいアルキル、シクロアルキル、置換基群Ｂから選択される１以上の置換基によって置換されていてもよいアルキルオキシ、アルキルチオ、ハロゲン、置換基群Ｃから選択される１以上の置換基によって置換されていてもよいフェニル、置換基群Ｃから選択される１以上の置換基によって置換されていてもよいヘテロアリール、または置換基群Ｃから選択される１以上の置換基によって置換されていてもよい非芳香族複素環基、
置換基群Ｂ：ヒドロキシ、アルキルオキシ、ハロゲン、カルボキシ、低級アルキルオキシカルボニル、アリールオキシカルボニル、置換されていてもよいアミノ、置換基群Ｃから選択される１以上の置換基によって置換されていてもよいフェニル、非芳香族複素環基、およびヘテロアリール、
置換基群Ｃ：ヒドロキシ、アルキル、ハロゲン、ハロ低級アルキル、カルボキシ、低級アルキルオキシカルボニル、アルキルオキシ、置換されていてもよいアミノ、非芳香族複素環、およびヘテロアリール；
Ｒ^３１およびＲ^３２はそれぞれ独立して、水素原子、低級アルキル、ハロゲン、ハロ低級アルキル、低級アルキルオキシ、ハロ低級アルキルオキシ、またはヒドロキシ；
Ｗ^４は式：

（式中、Ｒ^１３は水素原子、低級アルキル、低級アルキルオキシ、低級アルキルチオ、またはハロゲン；
Ｒ^１４およびＲ^１５はそれぞれ独立して水素原子、またはそれぞれ以下の置換基群Ａにより置換されていてもよい低級アルキル、低級アルケニル、低級アルキニル、シクロアルキル、アリール、アラルキル、ヘテロアリール、ヘテロアリールアルキル、もしくは非芳香族複素環基；
置換基群Ａ：ハロゲン、ハロ低級アルキル、置換されていてもよいアミノ、カルボキシ、低級アルキルチオ、低級アルキルシリル、または低級アルキルオキシ；
Ｒ^２４は水素原子または低級アルキル）で表わされる基；
Ｔは−ＣＨ_２−、−ＣＨ_２ＣＨ_２−、−ＣＨ_２ＣＨ_２ＣＨ_２−、−ＯＣＨ_２−、または−ＳＣＨ_２−］で示される化合物、そのプロドラッグ、もしくはそれらの製薬上許容される塩、またはそれらの溶媒和物。
２８）１５）〜２７）のいずれかに記載の化合物を有効成分として含有する医薬組成物。
２９）１５）〜２７）のいずれかに記載の化合物を有効成分として含有するトロンボポエチン受容体アゴニスト作用を有する医薬組成物。
３０）１５）〜２７）のいずれかに記載の化合物を有効成分として含有する血小板産生調節剤。
３１）血小板産生を調節するための医薬を製造するための１５）〜２７）のいずれかに記載の化合物の使用。
３２）１５）〜２７）のいずれかに記載の化合物の治療上効果を示す量を人を含む哺乳動物に投与することからなる、哺乳動物の血小板産生を調節する方法。

本明細書中、「ハロゲン」とは、フッ素、塩素、臭素、ヨウ素を意味する。フッ素、塩素、および臭素が好ましい。
本明細書中、単独でもしくは他の用語と組み合わせて用いられる「アルキル」とは、炭素原子数１〜１５の直鎖または分枝鎖の１価の炭化水素基を包含する。例えば、メチル、エチル、ｎ−プロピル、イソプロピル、ｎ−ブチル、イソブチル、ｓｅｃ−ブチル、ｔｅｒｔ−ブチル、ｎ−ペンチル、イソペンチル、ｎｅｏ−ペンチル、ｎ−ヘキシル、イソヘキシル、ｎ−ヘプチル、ｎ−オクチル、ｎ−ノナニル、ｎ−デカニル、ｎ−ウンデカニル、ｎ−ドデカニル、ｎ−トリデカニル、ｎ−テトラデカニル、ｎ−ペンタデカニル等が挙げられる。好ましくは、Ｃ１〜Ｃ１０アルキルが挙げられる。さらに好ましくは、Ｃ１〜Ｃ６アルキルが挙げられる。
本明細書中、単独でもしくは他の用語と組み合わせて用いられる「低級アルキル」とは、炭素原子数１〜８の直鎖または分枝鎖の１価の炭化水素基を包含する。例えば、メチル、エチル、ｎ−プロピル、イソプロピル、ｎ−ブチル、イソブチル、ｓｅｃ−ブチル、ｔｅｒｔ−ブチル、ｎ−ペンチル、イソペンチル、ｎｅｏ−ペンチル、ｎ−ヘキシル、イソヘキシル、ｎ−ヘプチル、ｎ−オクチル等が挙げられる。好ましくは、Ｃ１〜Ｃ６アルキルが挙げられる。さらに好ましくは、Ｃ１〜Ｃ３アルキルが挙げられる。
本明細書中、単独でもしくは他の用語と組み合わせて用いられる「Ｃ１−３アルキレン」としては、メチレン、エチレン、およびプロピレンが挙げられる。
本明細書中、単独でもしくは他の用語と組み合わせて用いられる「シクロアルカン」とは、炭素原子数が３〜８個である単環のシクロアルカンを包含する。例えば、シクロプロパン、シクロブタン、シクロペンタン、シクロヘキサン、シクロヘプタン、シクロオクタンが挙げられる。好ましくはＣ３〜Ｃ６シクロアルカンが挙げられる。
本明細書中、単独でもしくは他の用語と組み合わせて用いられる「シクロアルキル」とは、炭素原子数が３〜８個である単環のシクロアルキルを包含する。例えば、シクロプロピル、シクロブチル、シクロペンチル、シクロヘキシル、シクロヘプチル、シクロオクチルが挙げられる。好ましくはＣ３〜Ｃ６シクロアルキルが挙げられる。
本明細書中、「低級アルケニル」とは、炭素原子数が２〜８個であり、１個もしくは２個以上の二重結合を有する、直鎖または分枝鎖の１価の炭化水素基を包含する。例えば、ビニル、アリル、１−プロペニル、２−プロペニル、種々のブチニル異性体等が挙げられる。好ましくは、Ｃ２〜Ｃ６アルキニルが挙げられる。さらに好ましくは、Ｃ２〜Ｃ４アルキニルが挙げられる。
本明細書中、「低級アルキニル」とは、炭素原子数が２〜８個であり、１個もしくは２個以上の三重結合を有する、直鎖または分枝鎖の１価の炭化水素基を包含する。例えば、エチニル、１−プロピニル、２−プロピニル、１−プロペニル、２−プロペニル、クロトニル、イソペンテニル、種々のブテニル異性体等が挙げられる。好ましくは、Ｃ２〜Ｃ６アルケニルが挙げられる。さらに好ましくは、Ｃ２〜Ｃ４アルケニルが挙げられる。

本明細書中、単独でもしくは他の用語と組み合わせて用いられる「アリール」とは、単環状もしくは縮合環状芳香族炭化水素を包含する。例えば、フェニル、１−ナフチル、２−ナフチル、アントリル等が挙げられる。
本明細書中、「アラルキル」とは、前記「低級アルキル」に前記「アリ−ル」が１または２以上置換したものを包含し、これらは可能な全ての位置で置換しうる。例えば、ベンジル、フェニルエチル（例えば、２−フェニルエチル等）、フェニルプロピル（例えば、３−フェニルプロピル等）、ナフチルメチル（例えば、１−ナフチルメチル、２−ナフチルメチル等）、アントリルメチル（例えば、９−アントリルメチル等）等が挙げられる。好ましくは、ベンジル、フェニルエチルが挙げられる。
本明細書中、単独でもしくは他の用語と組み合わせて用いられる「非芳香族複素環基」なる用語は、任意に選ばれる、酸素原子、硫黄原子又は窒素原子を環内に１個以上含む非芳香族の５〜７員環またはそれらが２個以上縮合した環を包含する。例えば、ピロリジニル（例えば、１−ピロリジニル、２−ピロリジニル）、ピロリニル（例えば、３−ピロリニル）、イミダゾリジニル（例えば、２−イミダゾリジニル）、イミダゾリニル（例えば、イミダゾリニル）、ピラゾリジニル（例えば、１−ピラゾリジニル、２−ピラゾリジニル）、ピラゾリニル（例えば、ピラゾリニル）、ピペリジル（例えば、ピペリジノ、２−ピペリジル）、ピペラジニル（例えば、１−ピペラジニル）、インドリニル（例えば、１−インドリニル）、イソインドリニル（例えば、イソインドリニル）、モルホリニル（例えば、モルホリノ、３−モルホリニル）、テトラヒドロフラニル、テトラヒドロピラニル等が挙げられる。
Ｒ^１７、Ｒ^１８、Ｒ^１９、Ｒ^２０、Ｒ^２１、Ｒ^２２、Ｒ^２３、Ｒ^２８、Ｒ^２９、およびＲ^３０における「非芳香族複素環基」としては、モルホリノ、ピペラジノ、ピロリジノ、テトラヒドロフラニル、テトラヒドロピラニル等が好ましい。
置換基群Ｂにおける「非芳香族複素環基」としては、モルホリノ、ピペラジノ、ピペリジノ、テトラヒドロフラニル、テトラヒドロピラニル等が好ましい。
置換基群Ｃにおける「非芳香族複素環基」としては、モルホリノ、ピペラジノ、ピペリジノ、ピロリジノ、テトラヒドロフラニル、テトラヒドロピラニル等が好ましい。
本明細書中、単独でもしくは他の用語と組み合わせて用いられる「ヘテロアリール」とは、任意に選ばれる、酸素原子、硫黄原子又は窒素原子を環内に１個以上含む５〜６員の芳香環を包含する。これは前記「シクロアルキル」、前記「アリール」、前記「非芳香族複素環基」、もしくは他のヘテロアリールと可能な全ての位置で縮合していてもよい。ヘテロアリールが単環および縮合環のいずれである場合も、すべての可能な位置で結合しうる。例えば、ピロリル（例えば、１−ピロリル、２−ピロリル、３−ピロリル）、フリル（例えば、２−フリル、３−フリル）、チエニル（例えば、２−チエニル、３−チエニル）、イミダゾリル（例えば、２−イミダゾリル、４−イミダゾリル）、ピラゾリル（例えば、１−ピラゾリル、３−ピラゾリル）、イソチアゾリル（例えば、３−イソチアゾリル）、イソキサゾリル（例えば、３−イソキサゾリル）、オキサゾリル（例えば、２−オキサゾリル）、チアゾリル（例えば、２−チアゾリル）、ピリジル（例えば、２−ピリジル、３−ピリジル、４−ピリジル）、ピラジニル（例えば、２−ピラジニル）、ピリミジニル（例えば、２−ピリミジニル、４−ピリミジニル）、ピリダジニル（例えば、３−ピリダジニル）、テトラゾリル（例えば、１Ｈ−テトラゾリル）、オキサジアゾリル（例えば、１，３，４−オキサジアゾリル）、チアジアゾリル（例えば、１，３，４−チアジアゾリル）、インドリジニル（例えば、２−インドリジニル、６−インドリジニル）、イソインドリル（例えば、２−イソインドリル）、インドリル（例えば、１−インドリル、２−インドリル、３−インドリル）、インダゾリル（例えば、３−インダゾリル）、プリニル（例えば、８−プリニル）、キノリジニル（例えば、２−キノリジニル）、イソキノリル（例えば、３−イソキノリル）、キノリル（例えば、２−キノリル、５−キノリル）、フタラジニル（例えば、１−フタラジニル）、ナフチリジニル（例えば、２−ナフチリジニル）、キノラニル（例えば、２−キノラニル）、キナゾリニル（例えば、２−キナゾリニル）、シンノリニル（例えば、３−シンノリニル）、プテリジニル（例えば、２−プテリジニル）、カルバゾリル（例えば、２−カルバゾリル、４−カルバゾリル）、フェナントリジニル（例えば、２−フェナントリジニル、３−フェナントリジニル）、アクリジニル（例えば、１−アクリニジル、２−アクリニジル）、ジベンゾフラニル（例えば、１−ジベンゾフラニル、２−ジベンゾフラニル）、ベンゾイミダゾリル（例えば、２−ベンゾイミダゾリル）、ベンゾイソキサゾリル（例えば、３−ベンゾイソキサゾリル）、ベンゾオキサゾリル（例えば、２−ベンゾオキサゾリル）、ベンゾオキサジアゾリル（例えば、４−ベンゾオキサジアゾリル）、ベンゾイソチアゾリル（例えば、３−ベンゾイソチアゾリル）、ベンゾチアゾリル（例えば、２−ベンゾチアゾリル）、ベンゾフリル（例えば、３−ベンゾフリル）、ベンゾチエニル（例えば、２−ベンゾチエニル）、４，５−ジヒドロナフト［１，２−ｄ］チアゾリル、４Ｈ−クロメノ［４，３−ｄ］チアゾリル、４Ｈ−チオクロメノ［４，３−ｄ］チアゾリル、４，５−ジヒドロチアゾロ［５，４−ｃ］キノリル、８Ｈ−インデノ［１，２−ｄ］チアゾリル、５，６−ジヒドロ−４Ｈ−３−チア−１−アザ−ベンゾ［ｅ］アズレニル等が挙げられる。
Ｘ^１における「ヘテロアリール」としては、チアゾリル、イソキサゾリル、チエニル、カルバゾリル、ベンゾチアゾリル、ピリジル、ピラゾリル等が好ましい。さらに好ましくは、チアゾリル、ピリジル等が挙げられる。
Ｒ^１、Ｒ^２、Ｒ^３、Ｒ^４、Ｒ^７、およびＲ^８における「ヘテロアリール」としては、ピリジル、チアゾリル、ベンゾチアゾリル等が好ましい。
Ｒ^１０およびＲ^１１における「ヘテロアリール」としては、ピリジル、チエニル、フリル、ピリミジニル、イミダゾリル、チアゾリル、オキサゾリル、トリアゾリル等が好ましい。
Ａ^１、Ａ^２、およびＡ^３における「ヘテロアリール」としては、イミダゾリル、トリアゾリル、テトラゾリル、ピリジル、ピリミジニル等が好ましい。
Ｒ^１７、Ｒ^１８、Ｒ^１９、Ｒ^２０、Ｒ^２１、Ｒ^２２、Ｒ^２３、Ｒ^２８、Ｒ^２９、およびＲ^３０における「ヘテロアリール」としては、ピリジル、チエニル、フリル、ピリミジニル、イミダゾリル、チアゾリル、オキサゾリル、トリアゾリル等が好ましい。
置換基群Ｂにおける「ヘテロアリール」としては、ピリジル、ピラゾリル、ピリミジル、イミダゾリル、オキサゾリル、チアゾリル、フリル、チエニル等が好ましい。
置換基群Ｃにおける「ヘテロアリール」としては、ピリジル、ピラゾリル、イミダゾリル等が好ましい。
本明細書中、「５員ヘテロアリール」とは、任意に選ばれる、酸素原子、硫黄原子又は窒素原子を環内に１個以上含む５員の芳香環を包含する。例えば、チエニル、フリル、ピロリル、イミダゾリル、ピラゾリル、イソチアゾリル、イソキサゾリル、チアゾリル、オキサゾリル、１，２，３−トリアゾリル、１，２，４−トリアゾリル、１，２，４−チアジアゾリル、１，３，４−チアジアゾリル、１，２，４−オキサジアゾリル、１，３，４−オキサジアゾリル等が挙げられる。チアゾリルが好ましい。
本明細書中、「ヘテロアリールアルキル」とは、前記「低級アルキル」の任意の位置に前記「ヘテロアリ−ル」が１または２以上置換したものを包含し、これらは可能な全ての位置で置換しうる。例えば、チエニルメチル（例えば、２−チエニルメチル）、チエニルエチル（例えば、２−（チオフェン−２−イル）エチル）、フリルメチル（例えば、２−フリルメチル）、フリルエチル（例えば２−（フラン−２−イル）エチル）、ピロリルメチル（例えば、２−ピロリルメチル）、ピロリルエチル（例えば、２−（ピロール−２−イル）エチル）、イミダゾリルメチル（例えば、２−イミダゾリルメチル、４−イミダゾリルメチル）、イミダゾリルエチル（例えば、２−（イミダゾール−２−イル）エチル）、ピラゾリルメチル（例えば、３−ピラゾリルメチル）、ピラゾリルエチル（例えば、２−（ピラゾール−３−イル）エチル）、チアゾリルメチル（例えば、２−チアゾリルメチル）、チアゾリルエチル（例えば、２−（チアゾール−２−イル）エチル）、イソチアゾリルメチル（例えば、３−イソチアゾリルメチル）、イソキサゾリルメチル（例えば、３−イソキサゾリルメチル）、オキサゾリルメチル（例えば、２−オキサゾリルメチル）、オキサゾリルエチル（例えば、２−（オキサゾール−２−イル）エチル）、ピリジルメチル（例えば、２−ピリジルメチル、３−ピリジルメチル、４−ピリジルメチル）、ピリジルエチル（例えば、２−ピリジルエチル）等が挙げられる。
Ｒ^１、Ｒ^２、Ｒ^３、Ｒ^４、Ｒ^７、およびＲ^８における「ヘテロアリールアルキル」としては、２−チエニルメチル、２−フリルメチル等が挙げられる。
本明細書中、「フェニレン」とは、フェニルの２価基を意味する。例えば、１，２−フェニレン、１，３−フェニレン、１，４−フェニレンが挙げられる。好ましくは１，４−フェニレンが挙げられる。
本明細書中、「単環ヘテロアリレン」とは、前記「ヘテロアリール」のうち単環のヘテロアリールの２価基を意味する。例えば、チオフェンジイル、フランジイル、ピリジンジイル等が挙げられる。さらに詳しくは、２，５−チオフェンジイル、２，５−フランジイル、２，５−ピリジンジイル、２，５−チアゾールジイル、２，５−（１，３，４−チアジアゾール）ジイル、２，５−ピリジンジイル、２，５−ピラジンジイル、３，６−ピリダジンジイル、２，５−（４Ｈ−ピラン）ジイル等が挙げられる。２，５−チオフェンジイル、２，５−フランジイル、２，５−ピリジンジイルが好ましい。
本明細書中、「単環非芳香族複素環ジイル」とは、前記「非芳香族複素環基」のうち単環の非芳香族複素環基の２価基を意味する。例えば、ピロリジンジイル、ピペリジンジイル、ピラジンジイル等が挙げられる。
本明細書中、「単環シクロアルカンジイル」とは、前記「シクロアルカン」のうち単環のシクロアルカンの２価基を意味する。例えば、１，４−シクロペンタンジイル、１，４−シクロヘキサンジイル等が挙げられる。

本明細書中、「アルキルオキシ」としては、メチルオキシ、エチルオキシ、ｎ−プロピルオキシ、イソプロピルオキシ、ｎ−ブチルオキシ、イソブチルオキシ、ｓｅｃ−ブチルオキシ、ｔｅｒｔ−ブチルオキシ、ｎ−ペンチルオキシ、ｎ−ヘキシルオキシ、ｎ−ヘプチルオキシ、ｎ−オクチルオキシ、ｎ−ノナニルオキシ、ｎ−デカニルオキシ等が挙げられる。好ましくは、メチルオキシ、エチルオキシ、ｎ−プロピルオキシ、イソプロピルオキシ、ｎ−ブチルオキシが挙げられる。
本明細書中、「低級アルキルオキシ」としては、メチルオキシ、エチルオキシ、ｎ−プロピルオキシ、イソプロピルオキシ、ｎ−ブチルオキシ、イソブチルオキシ、ｓｅｃ−ブチルオキシ、ｔｅｒｔ−ブチルオキシ等が挙げられる。好ましくは、メチルオキシ、エチルオキシ、ｎ−プロピルオキシ、イソプロピルオキシ、ｎ−ブチルオキシが挙げられる。
本明細書中、「低級アルキルチオ」としては、メチルチオ、エチルチオ等が挙げられる。
本明細書中、「低級アルキルオキシカルボニル」としては、メチルオキシカルボニル、エチルオキシカルボニル、ｎ−プロピルオキシカルボニル、イソプロピルオキシカルボニル、ｎ−ブチルオキシカルボニル、ｔ−ブチルオキシカルボニル、ｎ−ペンチルオキシカルボニル等が挙げられる。
本明細書中、「アリールオキシカルボニル」としては、フェニルオキシカルボニル、１−ナフチルオキシカルボニル、２−ナフチルオキシカルボニル等が挙げられる。
本明細書中、単独でもしくは他の用語と組み合わせて用いられる「アシル」なる用語は、アルキル部分が前記「低級アルキル」であるアルキルカルボニルまたはアリール部分が前記「アリール」であるアリールカルボニルを包含する。例えば、アセチル、プロピオニル、ブチロイル、ベンゾイル等が挙げられる。「低級アルキル」および「アリール」は後述のそれぞれの置換基によって置換されていてもよい。
本明細書中、単独でもしくは他の用語と組み合わせて用いられる「ハロ低級アルキル」なる用語は、前記ハロゲンによって１〜８個所、好ましくは１〜５個所置換された前記「低級アルキル」を包含する。例えば、トリフルオロメチル、トリクロロメチル、ジフルオロエチル、トリフルオロエチル、ジクロロエチル、トリクロロエチル等が挙げられる。好ましくは、トリフルオロメチルが挙げられる。
本明細書中、「ハロ低級アルキルオキシ」としては、トリフルオロメチルオキシ、トリクロロメチルオキシ、ジフルオロエチルオキシ、トリフルオロエチルオキシ、ジクロロエチルオキシ、トリクロロエチルオキシ等が挙げられる。好ましくは、トリフルオロメチルオキシが挙げられる。
本明細書中、「アシルオキシ」としては、アセチルオキシ、プロピオニルオキシ、ベンゾイルオキシ等が挙げられる。
本明細書中、「低級アルキルシリル」としては、トリエチルシリル、ｔ−ブチルジメチルシリル等が挙げられる。
本明細書中、単独でもしくは他の用語と組み合わせて用いられる「置換されていてもよいアミノ」なる用語は、前記「低級アルキル」、前記「アリール」、前記「アラルキル」、前記「ヘテロアリール」、前記「ヘテロアリールアルキル」、または前記「アシル」で１または２個所置換されいてもよいアミノを包含する。例えば、アミノ、メチルアミノ、ジメチルアミノ、エチルメチルアミノ、ジエチルアミノ、エチルメチルアミノ、ベンジルアミノ、アセチルアミノ、ベンゾイルアミノ等が挙げられる。好ましくはアミノ、メチルアミノ、ジメチルアミノ、エチルメチルアミノ、ジエチルアミノ、アセチルアミノが挙げられる。
本明細書中、「置換されていてもよいアミノカルボニル」としては、アミノカルボニル、メチルアミノカルボニル、ジメチルアミノカルボニル、エチルメチルアミノカルボニル、ジエチルアミノカルボニル等が挙げられる。好ましくは、アミノカルボニル、メチルアミノカルボニル、ジメチルアミノカルボニルが挙げられる。
本明細書中、「置換されていてもよいウレイド」なる用語は、前記「低級アルキル」、前記「アリール」、前記「アラルキル」、前記「ヘテロアリール」、前記「ヘテロアリールアルキル」、または前記「アシル」で１または２個所以上置換されいてもよいウレイドを包含する。
本明細書中、「置換されていてもよい低級アルキル」における置換基としては、シクロアルキル、低級アルケニル、低級アルキリデン、ヒドロキシ、低級アルキルオキシ、メルカプト、低級アルキルチオ、ハロゲン、ニトロ、シアノ、カルボキシ、低級アルキルオキシカルボニル、ハロ低級アルキル、ハロ低級アルキルオキシ、置換されていてもよいアミノ、置換されていてもよいアミノカルボニル、アシル、アシルオキシ、置換されていてもよい非芳香族複素環基、アリールオキシ（例えば、フェニルオキシ）、アラルキルオキシ（例えば、ベンジルオキシ）、低級アルキルスルホニル、グアニジノ、アゾ基、置換されていてもよいウレイド、＝Ｎ−Ｏ−（アシル）等が挙げられる。これらは、全ての可能な位置で１個以上置換しうる。
Ｒ^ＣおよびＲ^Ｄにおける「置換されていてもよい低級アルキル」の置換基としては、ハロゲン、ハロ低級アルキル等が好ましい。
Ｒ^１、Ｒ^２、Ｒ^３、Ｒ^４、Ｒ^５、Ｒ^６、Ｒ^７、Ｒ^８、およびＲ^９における「置換されていてもよい低級アルキル」の置換基としては、ヒドロキシ、カルボキシ、ハロゲン、アルキルオキシ、アルキルチオ、アルキルシリル、置換されていてもよいアミノ、シアノ、アシル等が好ましい。
Ｒ^１０、Ｒ^１１、およびＲ^１６における「置換されていてもよい低級アルキル」の置換基としては、低級アルキルオキシカルボニル、ハロゲンが好ましい。
Ｒ^１２における「置換されていてもよい低級アルキル」の置換基としては、シクロアルキル、低級アルケニル、低級アルキリデン等が好ましい。
本明細書中、「置換されていてもよい低級アルキルオキシ」および「置換されていてもよい低級アルキルチオ」における置換基としては、シクロアルキル、低級アルケニル、低級アルキリデン、ヒドロキシ、低級アルキルオキシ、メルカプト、低級アルキルチオ、ハロゲン、ニトロ、シアノ、カルボキシ、低級アルキルオキシカルボニル、ハロ低級アルキル、ハロ低級アルキルオキシ、置換されていてもよいアミノ、置換されていてもよいアミノカルボニル、アシル、アシルオキシ、置換されていてもよい非芳香族複素環基、アリールオキシ（例えば、フェニルオキシ）、アラルキルオキシ（例えば、ベンジルオキシ）、低級アルキルスルホニル、グアニジノ、アゾ基、置換されていてもよいウレイド、＝Ｎ−Ｏ−（アシル）等が挙げられる。これらは、全ての可能な位置で１個以上置換しうる。好ましくは、ハロゲン等が挙げられる。
本明細書中、「置換されていてもよい低級アルケニル」および「置換されていてもよい低級アルキニル」における置換基としては、シクロアルキル、低級アルキリデン、ヒドロキシ、低級アルキルオキシ、メルカプト、低級アルキルチオ、ハロゲン、ニトロ、シアノ、カルボキシ、低級アルキルオキシカルボニル、ハロ低級アルキル、ハロ低級アルキルオキシ、置換されていてもよいアミノ、置換されていてもよいアミノカルボニル、アシル、アシルオキシ、置換されていてもよい非芳香族複素環基、アリール、アリールオキシ（例えば、フェニルオキシ）、アラルキル、アラルキルオキシ（例えば、ベンジルオキシ）、低級アルキルスルホニル、グアニジノ、アゾ基、置換されていてもよいウレイド等が挙げられる。これらは、全ての可能な位置で１個以上置換しうる。

本明細書中、「置換されていてもよいフェニレン」、「置換されていてもよい単環ヘテロアリレン」、「置換されていてもよい２，５−ピリジンジイル」、「置換されていてもよい２，５−チオフェンジイル」、「置換されていてもよい２，５−フランジイル」、「置換されていてもよい単環非芳香族複素環ジイル」、「置換されていてもよい単環シクロアルカンジイル」、「置換されていてもよいアリール」、「置換されていてもよいフェニル」、「置換されていてもよいヘテロアリール」、「置換されていてもよい５員ヘテロアリール」、「置換されていてもよいピリジル」「置換されていてもよい非芳香族複素環基」、「置換されていてもよいシクロアルキル」、「置換されていてもよいアラルキル」、および「置換されていてもよいヘテロアリールアルキル」における置換基としては、置換されていてもよいアルキル、シクロアルキル、低級アルケニル、低級アルキニル、ヒドロキシ、アルキルオキシ、アラルキルオキシ、メルカプト、低級アルキルチオ、ハロゲン、ニトロ、シアノ、カルボキシ、低級アルキルオキシカルボニル、アリールオキシカルボニル、ハロ低級アルキル、ハロ低級アルキルオキシ、置換されていてもよいアミノ、置換されていてもよいアミノカルボニル、アシル、アシルオキシ、置換されていてもよいアリール（置換基としては、ハロゲン、カルボキシ、アルキル、アルキルオキシ等）、置換されていてもよいヘテロアリ−ル（置換基としては、ハロゲン、カルボキシ、アルキル、アルキルオキシ等）、置換されていてもよい非芳香族複素環基、置換されていてもよいアラルキル、低級アルキルスルホニル、グアニジノ、アゾ基、−Ｎ＝Ｎ−（置換されていてもよいフェニル）、または置換されていてもよいウレイド等が挙げられる。これらは、全ての可能な位置で１個以上置換しうる。
「置換されていてもよいフェニレン」、「置換されていてもよい単環ヘテロアリレン」、「置換されていてもよい２，５−ピリジンジイル」、「置換されていてもよい２，５−チオフェンジイル」、「置換されていてもよい２，５−フランジイル」、「置換されていてもよい単環非芳香族複素環ジイル」、および「置換されていてもよい単環シクロアルカンジイル」の置換基としては、ハロゲン、ニトロ、シアノ、低級アルキル、低級アルキルオキシ等が好ましい。非置換のものが好ましい。
Ｘ^１における「置換されていてもよいアリール」および「置換されていてもよいアラルキル」の置換基としては、低級アルキル、ヒドロキシ低級アルキル、ヒドロキシ、低級アルキルオキシ、低級アルキルチオ、ハロゲン、ニトロ、シアノ、カルボキシ、ハロ低級アルキル、ハロ低級アルキルオキシ、アラルキルオキシ、置換されていてもよいアミノ、置換されていてもよいアミノカルボニル、アリール、ヘテロアリール、非芳香族複素環基、−Ｎ＝Ｎ−（フェニル）等が挙げられる。好ましい置換基としては、低級アルキル、ヒドロキシ、低級アルキルオキシ、低級アルキルチオ、ハロゲン、ハロ低級アルキル、アラルキルオキシ、−Ｎ＝Ｎ−（フェニル）、アルキレンジオキシ等が挙げられる。
Ｘ^１における「置換されていてもよいアリール」としては、フェニル、３−メチルフェニル、４−メチルフェニル、３，４−ジメチルフェニル、４−エチルフェニル、４−ｔ−ブチルフェニル、４−ｎ−ブチルフェニル、４−ｎ−ヘキシルフェニル、４−ｎ−オクチルフェニル、３，５−ジ−ｔ−ブチル−４−ヒドロキシフェニル、４−エチルオキシフェニル、４−フルオロフェニル、３，５−ジクロロフェニル、４−ヨードフェニル、４−トリフルオロメチルフェニル、４−メチルチオフェニル、４−フェニルオキシメチルフェニル、アゾベンゼン−４−イル、ベンゾジオキソリル（例えば、１，３−ベンゾジオキソリル）等が挙げられる。
Ｒ^１０およびＲ^１１における「置換されていてもよいアリール」の置換基としては、ハロゲン、置換されていてもよいアルキル、シクロアルキル、低級アルケニル、低級アルキニル、ヒドロキシ、アルキルオキシ、メルカプト、低級アルキルチオ、ニトロ、シアノ、カルボキシ、低級アルキルオキシカルボニル、ハロ低級アルキル、ハロ低級アルキルオキシ、置換されていてもよいアミノ、置換されていてもよいアミノカルボニル、アシル、ホルミル、アシルオキシ、置換されていてもよいアリール、置換されていてもよいヘテロアリ−ル（例えば、ピリジル、イミダゾリル）、非芳香族複素環基（例えば、モルホリノ、ピペラジニル）、アラルキル等が挙げられる。好ましくは、置換基群Ｂから選択される１以上の置換基によって置換されていてもよいアルキル、シクロアルキル、置換基群Ｂから選択される１以上の置換基によって置換されていてもよいアルキルオキシ、アルキルチオ、ハロゲン、置換基群Ｃから選択される１以上の置換基によって置換されていてもよいフェニル、置換基群Ｃから選択される１以上の置換基によって置換されていてもよいヘテロアリール、または置換基群Ｃから選択される１以上の置換基によって置換されていてもよい非芳香族複素環基等が挙げられる（置換基群Ｂ：ヒドロキシ、アルキルオキシ、ハロゲン、カルボキシ、低級アルキルオキシカルボニル、アリールオキシカルボニル、置換されていてもよいアミノ、置換基群Ｃから選択される１以上の置換基によって置換されていてもよいフェニル、非芳香族複素環基、およびヘテロアリール、
置換基群Ｃ：ヒドロキシ、アルキル、ハロゲン、ハロ低級アルキル、カルボキシ、低級アルキルオキシカルボニル、アルキルオキシ、置換されていてもよいアミノ、非芳香族複素環、およびヘテロアリール）。また、該アリールはＣ５−Ｃ７シクロヘキサン環（例えば、シクロペンタン、シクロヘキサン等）または非芳香族複素環基（例えば、テトラヒドロフラニル、１，３−ジオキソリル、１，４−ジオキシニル、ピロリジニル等）と縮合し、インダン、１，２，３，４−テトラヒドロナフタレン、１，２，３，４−テトラヒドロキノリン、２，３−ジヒドロベンゾ［１，４］ジオキシン、ベンゾ［１，３］ジオキソール、２，３−ジヒドロベンゾフラン、２，３−ジヒドロ−１Ｈ−インドールを形成してもよい。
Ｘ^１における「置換されていてもよいヘテロアリール」および「置換されていてもよいヘテロアリールアルキル」の置換基としては、置換されていてもよい低級アルキル、低級アルケニル（例えば、＝ＣＨ−ＣＨ_３）、低級アルキニル、ヒドロキシ、低級アルキルオキシ、メルカプト、低級アルキルチオ、ハロゲン、ニトロ、シアノ、カルボキシ、低級アルキルオキシカルボニル、ハロ低級アルキル、ハロ低級アルキルオキシ、置換されていてもよいアミノ、置換されていてもよいアミノカルボニル、アシル（例えば、ハロゲン、ニトロ、シアノ等で置換されていてもよいアリールオキシカルボニル等）、アシルオキシ、置換されていてもよいアリール、置換されていてもよいヘテロアリ−ル（例えば、２−ピリジル、３−ピリジル、４−ピリジル、３−チエニル、５−メチルピリジン−２−イル、３−キノリル、５−クロロチオフェン−２−イル、５−ブロモチオフェン−２−イル）、非芳香族複素環基、アラルキル、＝Ｎ−Ｏ−（アシル）等が挙げられる。好ましくは、置換されていてもよい低級アルキル、低級アルケニル、低級アルキルオキシカルボニル、置換されていてもよいフェニル、ヘテロアリール、＝Ｎ−Ｏ−（アシル）等が挙げられる。
ヘテロ原子が窒素原子である場合は、該窒素原子がアルキル、オキソ等で置換されていてもよい。
Ｘ^２における「置換されていてもよい５員ヘテロアリール」の置換基としては、置換されていてもよい低級アルキル、低級アルケニル（例えば、＝ＣＨ−ＣＨ_３）、低級アルキニル、ヒドロキシ、低級アルキルオキシ、メルカプト、低級アルキルチオ、ハロゲン、ニトロ、シアノ、カルボキシ、低級アルキルオキシカルボニル、ハロ低級アルキル、ハロ低級アルキルオキシ、置換されていてもよいアミノ、置換されていてもよいアミノカルボニル、アシル（例えば、ハロゲン、ニトロ、シアノ等で置換されていてもよいアリールオキシカルボニル等）、アシルオキシ、置換されていてもよいアリール、置換されていてもよいヘテロアリ−ル（例えば、２−ピリジル、３−ピリジル、４−ピリジル、２−フリル、３−フリル、２−チエニル、３−チエニル、５−メチルピリジン−２−イル、インドール−３−イル、３−キノリル、５−クロロチオフェン−２−イル、５−ブロモチオフェン−２−イル）、非芳香族複素環基、アラルキル、＝Ｎ−Ｏ−（アシル）等が挙げられる。好ましくは、置換基群Ｂから選択される１以上の置換基によって置換されていてもよいアルキル、シクロアルキル、置換基群Ｂから選択される１以上の置換基によって置換されていてもよいアルキルオキシ、アルキルチオ、ハロゲン、置換基群Ｃから選択される１以上の置換基によって置換されていてもよいフェニル、置換基群Ｃから選択される１以上の置換基によって置換されていてもよいヘテロアリール、または置換基群Ｃから選択される１以上の置換基によって置換されていてもよい非芳香族複素環基等が挙げられる（置換基群Ｂ：ヒドロキシ、アルキルオキシ、ハロゲン、カルボキシ、低級アルキルオキシカルボニル、アリールオキシカルボニル、置換されていてもよいアミノ、置換基群Ｃから選択される１以上の置換基によって置換されていてもよいフェニル、非芳香族複素環基、およびヘテロアリール、
置換基群Ｃ：ヒドロキシ、アルキル、ハロゲン、ハロ低級アルキル、カルボキシ、低級アルキルオキシカルボニル、アルキルオキシ、置換されていてもよいアミノ、非芳香族複素環、およびヘテロアリール）。
Ｒ^１０およびＲ^１１における「置換されていてもよいヘテロアリール」の置換基としては、ハロゲン、置換されていてもよいアルキル、シクロアルキル、低級アルケニル、低級アルキニル、ヒドロキシ、アルキルオキシ、メルカプト、低級アルキルチオ、ニトロ、シアノ、カルボキシ、低級アルキルオキシカルボニル、ハロ低級アルキル、ハロ低級アルキルオキシ、置換されていてもよいアミノ、置換されていてもよいアミノカルボニル、アシル、ホルミル、アシルオキシ、置換されていてもよいアリール、置換されていてもよいヘテロアリ−ル（例えば、ピリジル、イミダゾリル）、非芳香族複素環基（例えば、モルホリノ、ピペラジニル）、アラルキル等が挙げられる。好ましくは、置換基群Ｂから選択される１以上の置換基によって置換されていてもよいアルキル、シクロアルキル、置換基群Ｂから選択される１以上の置換基によって置換されていてもよいアルキルオキシ、アルキルチオ、ハロゲン、置換基群Ｃから選択される１以上の置換基によって置換されていてもよいフェニル、置換基群Ｃから選択される１以上の置換基によって置換されていてもよいヘテロアリール、または置換基群Ｃから選択される１以上の置換基によって置換されていてもよい非芳香族複素環基等が挙げられる（置換基群Ｂ：ヒドロキシ、アルキルオキシ、ハロゲン、カルボキシ、低級アルキルオキシカルボニル、アリールオキシカルボニル、置換されていてもよいアミノ、置換基群Ｃから選択される１以上の置換基によって置換されていてもよいフェニル、非芳香族複素環基、およびヘテロアリール、
置換基群Ｃ：ヒドロキシ、アルキル、ハロゲン、ハロ低級アルキル、カルボキシ、低級アルキルオキシカルボニル、アルキルオキシ、置換されていてもよいアミノ、非芳香族複素環、およびヘテロアリール）。

本明細書中、（α）_β−γはαがβ〜γ個存在することを意味する。例えば、（ＣＲ^ＣＲ^Ｄ）_０−２は（ＣＲ^ＣＲ^Ｄ）が０〜２個存在することを、（ＣＨ_２）_０−２は（ＣＨ_２）が０〜２個存在することを、（ＣＨ_２）_１−５は（ＣＨ_２）が１〜５個存在することを意味する。
本明細書中、「血小板産生調節剤」とは、血小板減少症（骨髄移植後の血小板減少、化学療法後の血小板減少、再生不良性貧血、骨髄異形成症候群、難治性突発性血小板減少性紫斑病等の後天性血小板減少症、トロンボポエチン欠損症等の先天性血小板減少症）等の血小板数の異常を伴う血液疾患の病態に対する薬剤を包含する。例えば、抗癌剤の投与により血小板数が減少した場合には治療剤として、抗癌剤投与による血小板数の減少が予測される場合には予防剤として使用することができる。
本明細書中、「血小板産生を調節する」とは、１）抗癌剤の投与等により減少した血小板数を増加させる、２）抗癌剤の投与等により減少するであろう血小板数を維持させる、３）抗癌剤の投与等による血小板数の減少度を低下させることを包含する。

本発明化合物（Ｉ）は、以下のＡ法ならびにＢ法、およびそれらに類似の方法で合成することができる。
（Ａ法）

（式中、Ｒ^１、Ｒ^２、Ｒ^３、およびＸ^１は前記と同意義）
（第１工程）
本工程は、４−ホルミルまたは４−アシル置換安息香酸誘導体のカルボン酸をR^Eで保護する工程である。第３工程において２つのカルボン酸保護基を選択的に脱保護する必要があることから、R^Fとの組み合わせが重要となる。例えばR^Fがメチル、エチル等のアルカリ条件で脱保護が可能な保護基である場合、R^Eはアルカリ条件以外での脱保護が可能な保護基である必要があり、具体的にはアリル基（Pd(0)錯体にて脱保護）、tert-ブチル基、p-メトキシベンジル基、トリフェニルメチル基、ジフェニルメチル基（酸性条件で脱保護）、トリメチルシリルエチル基、トリメチルシリルエトキシメチル基、tert-ブチルジメチルシリル基（フッ素イオンで脱保護）等が挙げられる。
エステル化の条件としては適当な塩基の存在下、相当するハロゲン化物と反応させる方法を用いることができる。またはアルコール誘導体を出発原料として用いた縮合反応等によっても合成することができる。
（第２工程）
本工程は、アルデヒドまたはケトンをオレフィンに変換する工程である。Wittig反応、Horner-Emmons反応等のリンイリドを用いる反応、またはクネフェネーゲル（Knoevenagel）反応等の脱水縮合反応を行うことにより合成することができる。
（第３工程）
本工程は、R^Eの脱保護反応を行う工程である。Protective Groups in Organic Synthesis, Theodora W Green (John Wiley & Sons)等に記載の方法を用いて、保護基であるR^Eを適当な反応条件で脱保護する。
（第４工程）
本工程は、カルボン酸誘導体（ＶＩＩ）とアミン誘導体（X¹-NH₂）を、活性エステル法、酸クロリド法、混合酸無水物法等により反応させることにより、アミド誘導体（ＶＩＩＩ）を得る工程である。本工程は、テトラヒドロフラン、ジオキサン、ジクロロメタン、トルエン、ベンゼン等の溶媒中で行われる。活性エステル法では、１−ヒドロキシベンゾトリアゾール、ヒドロキシスクシンイミド、ジメチルアミノピリジン等と、ジシクロヘキシルカルボジイミド、１−エチル−３−（３−ジメチルアミノプロピル）カルボジイミド塩酸塩等を縮合剤として用いることにより行うことができる。酸クロリド法ではチオニルクロリドやオキザリルクロリドを試薬として遊離のカルボン酸を一旦酸クロリドとすることにより行うことができる。混合酸無水物法では、カルボン酸にエチルクロロホルメート、イソブチルクロロホルメート等を反応させ、混合酸無水物とすることにより行うことができる。反応には必要に応じてトリエチルアミン、ピリジン等の塩基が用いられる。
（第５工程）
本工程は、R^Fの脱保護反応を行う工程である。Protective Groups in Organic Synthesis, Theodora W Green (John Wiley & Sons)等に記載の方法を用いて、保護基であるR^Fを適当な反応条件で脱保護する。
（第６工程）
本工程は、カルボン酸誘導体（ＩＸ）とアミン誘導体（R³-NH₂）を、活性エステル法、酸クロリド法、混合酸無水物法等により反応させることにより、アミド誘導体（Ｉ−Ａ）を得る工程である。本工程は、テトラヒドロフラン、ジオキサン、ジクロロメタン、トルエン、ベンゼン等の溶媒中で行われる。活性エステル法では、１−ヒドロキシベンゾトリアゾール、ヒドロキシスクシンイミド、ジメチルアミノピリジン等と、ジシクロヘキシルカルボジイミド、１−エチル−３−（３−ジメチルアミノプロピル）カルボジイミド塩酸塩等を縮合剤として用いることにより行うことができる。酸クロリド法ではチオニルクロリドやオキザリルクロリドを試薬として遊離のカルボン酸を一旦酸クロリドとすることにより行うことができる。混合酸無水物法では、カルボン酸にエチルクロロホルメート、イソブチルクロロホルメート等を反応させ、混合酸無水物とすることにより行うことができる。反応には必要に応じてトリエチルアミン、ピリジン等の塩基が用いられる。

（Ｂ法）
本法は、Ａ法における化合物（ＶＩＩＩ）を合成するための別法である。

（式中、Ｒ^１、Ｒ^２、およびＸ^１は前記と同意義）
（第１工程）
本工程は、Ａ法第４工程と同様の方法を用いることにより、カルボン酸アミド誘導体（ＸＩ）を合成する工程である。
（第２工程）
本工程は、Ａ法第２工程と同様の方法を用いることにより、アルデヒド誘導体（ＸＩ）をオレフィン誘導体（ＸＩＩ）に変換する工程である。化合物（ＸＩＩ）は、Ａ法第５工程および第６工程と同様の反応を行うことにより化合物（Ｉ−Ａ）へと変換することができる。
Ｙ^１が−Ｎ（−アルキル）−ＣＯ−であり、Ｚ^１が置換されていてもよいチアゾール等である化合物：

（Ｗ^１およびＺ^１は前記と同意義、Ａｌｋは低級アルキル）
を合成する際のアルキル化の条件によっては、以下に示す化合物を得る場合がある。

（Ｗ^１、Ｚ^１、およびＡｌｋは前記と同意義）
一般式（Ｉ）、（ＩＩ）、および（ＩＩＩ）において破線が結合の存在を示す場合は、シス体、トランス体、およびそれらの混合物を包含する。例えば、Ｗ^１がアミドタイプの化合物である場合は以下のようなシス体およびトランス体が存在しうる。Ｗ^１がアミドタイプ以外の置換基である場合も同様である。

（式中、Ｒ^１、Ｒ^２、Ｒ^３、Ｒ^４、Ｘ^１、Ｙ^１、およびＺ^１は前記と同意義）

本明細書中、「溶媒和物」とは、例えば有機溶媒との溶媒和物、水和物等を包含する。
「本発明化合物」という場合には、製薬上許容される塩、またはその水和物も抱合される。例えば、アルカリ金属（リチウム、ナトリウム、カリウム等）、アルカリ土類金属（マグネシウム、カルシウム等）、アンモニウム、有機塩基およびアミノ酸との塩、または無機酸（塩酸、臭化水素酸、リン酸、硫酸等）、および有機酸（酢酸、クエン酸、マレイン酸、フマル酸、ベンゼンスルホン酸、ｐ−トルエンスルホン酸等）との塩が挙げられる。これらの塩は、通常行われる方法によって形成させることができる。水和物を形成する時は、任意の数の水分子と配位していてもよい。
プロドラッグは、化学的または代謝的に分解できる基を有する本発明化合物の誘導体であり、加溶媒分解によりまたは生理学的条件下でインビボにおいて薬学的に活性な本発明化合物となる化合物である。適当なプロドラッグ誘導体を選択する方法および製造する方法は、例えばＤｅｓｉｇｎｏｆＰｒｏｄｒｕｇｓ，Ｅｌｓｅｖｉｅｒ，Ａｍｓｔｅｒｄａｍ１９８５に記載されている。本発明化合物がカルボキシル基を有する場合は、もとになる酸性化合物と適当なアルコールを反応させることによって製造されるエステル誘導体、またはもとになる酸性化合物と適当なアミンを反応させることによって製造されるアミド誘導体のようなプロドラッグが例示される。プロドラッグとして特に好ましいエステルとしては、メチルエステル、エチルエステル、ｎ−プロピルエステル、イソプロピルエステル、ｎ−ブチルエステル、イソブチルエステル、ｔｅｒｔ−ブチルエステル、モルホリノエチルエステル、Ｎ，Ｎ−ジエチルグリコールアミドエステル等が挙げられる。本発明化合物がヒドロキシル基を有する場合は、例えばヒドロキシル基を有する化合物と適当なアシルハライドまたは適当な酸無水物とを反応させることに製造されるアシルオキシ誘導体のようなプロドラッグが例示される。プロドラッグとして特に好ましいアシルオキシとしては、−ＯＣＯＣ_２Ｈ_５、−ＯＣＯ（ｔ−Ｂｕ）、−ＯＣＯＣ_１５Ｈ_３１、−ＯＣＯ（ｍ−ＣＯＯＮａ−Ｐｈ）、−ＯＣＯＣＨ_２ＣＨ_２ＣＯＯＮａ、−ＯＣＯＣＨ（ＮＨ_２）ＣＨ_３、−ＯＣＯＣＨ_２Ｎ（ＣＨ_３）_２等が挙げられる。本発明化合物がアミノ基を有する場合は、アミノ基を有する化合物と適当な酸ハロゲン化物または適当な混合酸無水物とを反応させることにより製造されるアミド誘導体のようなプロドラッグが例示される。プロドラッグとして特に好ましいアミドとしては、−ＮＨＣＯ（ＣＨ_２）_２０ＣＨ_３、−ＮＨＣＯＣＨ（ＮＨ_２）ＣＨ_３等が挙げられる。
また、本発明化合物は特定の異性体に限定するものではなく、全ての可能な異性体やラセミ体を含むものである。

本発明化合物は後述する実験例の記載の通り、優れたトロンボポエチンアゴニスト活性を示し、血小板減少症（骨髄移植後、化学療法後、再生不良性貧血、骨髄異形成症候群、難治性突発性血小板減少性紫斑病等の後天性血小板減少症、トロンボポエチン欠損症等の先天性血小板減少症）等の血小板数の異常を伴う血液疾患の病態に対する薬剤（血小板産生調節剤）として使用しうる。抗癌剤投与による血小板数の異常の治療および／または予防に対して使用することができる。
本発明化合物を、上記の疾患の治療を目的としてヒトに投与する場合は、散剤、顆粒剤、錠剤、カプセル剤、丸剤、液剤等として経口的に、または注射剤、坐剤、経皮吸収剤、吸入剤等として非経口的に投与することができる。また、本化合物の有効量にその剤型に適した賦形剤、結合剤、湿潤剤、崩壊剤、滑沢剤等の医薬用添加剤を必要に応じて混合し、医薬製剤とすることができる。注射剤の場合には、適当な担体と共に滅菌処理を行って製剤とする。
投与量は疾患の状態、投与ルート、患者の年齢、または体重によっても異なるが、成人に経口で投与する場合、通常０．１〜１００mg／kg／日であり、好ましくは１〜２０mg／kg／日である。

以下に実施例および試験例を挙げて本発明をさらに詳しく説明するが、本発明はこれらにより限定されるものではない。
実施例中、以下の略号を使用する。
Ｍｅ：メチル
Ｅｔ：エチル
ｎ−Ｐｒ：ｎ−プロピル
ｉ−Ｐｒ：イソプロピル
ｃ−Ｐｒ：シクロプロピル
ｎ−Ｂｕ：ｎ−ブチル
ｉ−Ｂｕ：イソブチル
ｓｅｃ−Ｂｕ：ｓｅｃ−ブチル
ｔ−Ｂｕ：ｔｅｒｔ−ブチル
ｉ−Ｂｕ：イソブチル
ｎ−Ｐｅｎ：ｎ−ペンチル
ｃ−Ｐｅｎ：シクロペンチル
ｎ−Ｈｅｘ：ｎ−ヘキシル
ｃ−Ｈｅｘ：シクロヘキシル
ｉ−Ｈｅｘ：イソヘキシル
Ｐｈ：フェニル
Ｂｎ：ベンジル
Ｂｚ：ベンゾイル
Ｐｙ：ピリジル
Ｔｈ：チエニル
Ａｃ：アセチル
Ｚ：ベンジルオキシカルボニル
ＤＭＦ：Ｎ，Ｎ−ジメチルホルムアミド
ＴＨＦ：テトラヒドロフラン
propargyl：プロパルギル、allyl：アリル、pyrazole：ピラゾール、pyrimidine：ピリミジン、piperidine：ピペリジン、methyl：メチル、cyclohexylmethyl：シクロヘキシルメチル
実施例

実施例１化合物(A-1、A-2、およびB-1)の調製

（第１工程）
テレフタルアルデヒド酸(7.5 g)、臭化アリル(4.41 ml)、および炭酸カリウム(7.0 g)のDMF(100 ml)溶液を60℃にて１６時間攪拌した。反応溶媒を減圧下留去し、残留物を酢酸エチル−水に分配した。酢酸エチル層を重曹水、水、飽和食塩水にて洗浄し、硫酸マグネシウムにて乾燥した。溶媒を減圧留去することによって化合物(２)を無色透明油状化合物として(9.2 g)得た。
¹H NMR(CDCl₃, δ ppm): 4.87 (2H, dt, J = 1.2, 5.7 Hz), 5.30 - 5.47 (2H, m), 5.99 - 6.12 (1H, m), 7.94 - 7.98 (2H, m), 8.20 - 8.25 (2H, m), 10.11 (1H, s).
（第２工程）
化合物(２) (4.37 g)、２−（トリフェニルホスホルアニリデン）プロピオン酸エチル(10.63 g)のトルエン(100 ml)溶液を70℃にて１時間加熱攪拌した。反応溶媒をおよそ30〜40 mlまで減圧留去し、析出するトリフェニルホスフィンオキシドを濾去した。濾液を濃縮後、残留物をシリカゲルカラムクロマトグラフィー（酢酸エチル：n−ヘキサン＝１：１０）にて精製することによって化合物(３)を無色透明油状化合物として(6.9 g)得た。
¹H NMR (CDCl₃, δ ppm): 1.36 (3H, t, J = 7.2 Hz), 2.11 (3H, d, J = 1.5 Hz), 4.29 (2H, q, J = 7.2 Hz), 4.84 (2H, dt, J = 1.2, 5.7 Hz), 5.28 - 5.46 (2H, m), 5.98 - 6.11 (1H, m), 7.43 - 7.47 (2H, m), 7.69 (1H, d, J = 1.5 Hz), 8.06 - 8.10 (2H, m).
（第３工程）
化合物(３) (6 g)、テトラキストリフェニルホスフィンパラジウム(1.27 g)、およびモルホリン(2.68g)のTHF(100 ml)溶液を60℃にて30分攪拌した。反応溶媒をおよそ30〜40 mlまで減圧留去し、残留物に酢酸エチルを加え、重曹水にて３回抽出操作を行った。全ての重曹抽出溶液を３Ｍ−塩酸水溶液によって酸性とし、析出する結晶を酢酸エチルにて抽出した。酢酸エチル層を飽和食塩水にて洗浄し、硫酸マグネシウムにて乾燥した。溶媒を減圧留去することによって化合物(４)を白色結晶として(4.5 g)得た。
¹H NMR (CDCl₃, δ ppm): 1.37 (3H, t, J = 7.2 Hz), 2.13 (3H, d, J = 1.2 Hz), 4.30 (2H, q, J = 7.2 Hz), 7.49 (2H, d, J = 8.4 Hz), 7.71 (1H, s), 8.14 (2H, d, J = 8.4 Hz).
（第４工程）
化合物(４) (1.05 g)およびオキサリルクロリド(1.3 ml)のTHF(100 ml)溶液に触媒量のDMFを加え、２時間室温にて攪拌した。反応溶液を減圧溜去し、得られた残渣にトルエンを加えて、トルエンを減圧溜去した。得られたカルボン酸塩化物をジオキサン(70 ml)に溶解し、２−アミノ−４−（３，４−ジクロロフェニル）チアゾール(1 g)およびピリジン(970μl)を加えた。反応溶液を100℃にて１６時間加熱攪拌後、反応溶液を酢酸エチル−水に分配した。酢酸エチル層を希塩酸水、重曹水、水、飽和食塩水にて洗浄し、硫酸マグネシウムにて乾燥した。溶媒を減圧留去することによって化合物(A-1)を白色結晶として(1.5 g)得た。
¹H NMR (DMSO-d₆, δ ppm): 1.29 (3H, t, J = 7.2 Hz), 2.10 (3H, d, J = 1.2 Hz), 4.23 (2H, q, J = 7.2 Hz), 7.62 - 7.68 (3H, m), 7.72 (1H, d, J = 8.4 Hz), 7.91 (1H, s), 7.94 (1H, dd, J = 1.8, 8.4 Hz), 8.15 - 8.20 (2H, m), 8.21 (1H, d, J = 1.8 Hz), 12.84 (1H, br).
（第５工程）
化合物(A-1) (1.7 g)、4M−水酸化ナトリウム水溶液(5.5 ml)、THF(150 ml)の溶液を１８時間８５℃にて加熱攪拌した。反応溶液を希塩酸水溶液にて酸性とし、析出する結晶を濾取する。得られた粉末をメタノール、酢酸エチルにて洗浄することによって化合物(A-2)を白色粉末として(1.5 g)得た。
¹H NMR (DMSO-d₆, δ ppm): 2.08 (3H, d, J = 0.9 Hz), 7.62 - 7.68 (3H, m), 7.72 (1H, d, J = 8.7 Hz), 7.92 (1H, s), 7.95 (1H, dd, J = 2.1, 8.7 Hz), 8.16 - 8.20 (2H, m), 8.22 (1H, d, J = 1.8 Hz), 12.84 (1H, br).
（第６工程）
化合物(A-2) (690 mg)、オキサリルクロリド(420μl)のTHF(150 ml)溶液に触媒量のDMFを加え、７０℃にて1時間攪拌した。反応溶液を減圧溜去し、得られた残渣にトルエンを加えてトルエンを減圧溜去した。得られたカルボン酸塩化物にTHF(100 ml)を加え、氷冷した。別途に28％アンモニア水溶液(20 ml)に、氷冷下エーテル及び水酸化ナトリウム(5 g)を加えて10分間攪拌し静置した。このエーテル溶液を酸塩化物のTHF溶液に加えて氷冷下1時間攪拌した。反応溶液を酢酸エチル−THF−水に分配した。有機溶媒層を希塩酸水、重曹水、水、飽和食塩水にて洗浄し、硫酸マグネシウムにて乾燥した。溶媒を減圧留去して得られる残留物をシリカゲルカラムコロマトグラフィー（酢酸エチル：n−ヘキサン＝１０：１〜酢酸エチル）にて精製することによって化合物(B-1)を無色結晶として(400 mg)得た。
¹H NMR (DMSO-d₆, δ ppm): 2.04 (3H, d, J = 1.5 Hz), 7.18 (1H, br), 7.32 (1H, s), 7.52 - 7.58 (2H, m), 7.60 (1H, br), 7.72 (1H, d, J = 8.1 Hz), 7.91 (1H, s), 7.94 (1H, dd, J = 2.1, 8.4 Hz), 8.14 - 8.19 (2H, m), 8.22 (1H, d, J = 2.4 Hz), 12.81 (1H, br).
実施例２化合物(A-7)の調製

（第１工程）
４−アセチル安息香酸(1.64 g)、オキサリルクロリド(1.31 ml)のTHF(30 ml)溶液に触媒量のDMFを加え、２時間室温にて攪拌した。反応溶液を減圧溜去し、得られた残渣にトルエンを加えて、トルエンを減圧溜去する。こうして得られたカルボン酸塩化物にTHF(50 ml)、tert-ブチルアルコール(1.15 ml)、ピリジン(1.21 ml)を加え、40時間加熱還流した。反応溶液を塩酸酸性氷水−酢酸エチルに分配した後、酢酸エチル層を重曹水、水、飽和食塩水にて洗浄し、硫酸マグネシウムにて乾燥した。溶媒を濃縮後、残留物をシリカゲルカラムクロマトグラフィー（酢酸エチル：n−ヘキサン＝１：５）にて精製し、化合物(７)を白色結晶として(2.0 g)得た。
¹H NMR(CDCl₃, δ ppm): 1.61 (9H, s), 2.64 (3H, s), 7.96 - 7.00 (2H, m), 8.04 - 8.09 (2H, m).
（第２工程）
水素化ナトリウム(60% 360 mg)のTHF(10 ml)懸濁溶液に２−ホスホノプロピオン酸トリエチル(2.14 g)を氷冷下加える。30分攪拌後、化合物(７) (1.9 g)のTHF(15 ml)溶液を氷冷下、滴下した。反応溶液を50℃にて3時間攪拌後、塩酸酸性氷水−酢酸エチルに分配した。酢酸エチル層を重曹水、水、飽和食塩水にて洗浄し、硫酸マグネシウムにて乾燥した。溶媒を濃縮後、残留物をシリカゲルカラムクロマトグラフィー（酢酸エチル：n−ヘキサン＝１：１５）にて精製し、化合物(８)を無色油状物質として(1.0 g)得た。
¹H NMR(CDCl₃, δ ppm): 1.35 (3H, t, J = 7.2 Hz), 1.60 (9H, s), 1.74 (3H, q, J = 1.5 Hz), 2.24 (3H, q, J = 1.5 Hz), 4.27 (2H, q, J = 6.9 Hz), 7.18 - 7.22 (2H, m), 7.97 - 8.10 (2H, m).
（第３工程）
化合物(８) (900 mg)のぎ酸(98〜100%, 10 ml)溶液を室温にて3時間攪拌した。反応溶液を濃縮後、残渣にトルエンを加え再び濃縮した。得られた残渣をn−ヘキサンにて濾取することによって化合物(９)を白色結晶として(680 mg)得た。
¹H NMR(CDCl₃, δ ppm): 1.36 (3H, t, J = 7.2 Hz), 1.74 (3H, q, J = 1.5 Hz), 2.26 (3H, q, J = 1.5 Hz), 4.28 (2H, q, J = 7.2 Hz), 7.25 - 7.29 (2H, m), 8.10 - 8.14 (2H, m).
（第４工程）
化合物(９)を原料として、実施例１−第４工程と同様の反応を行うことにより化合物(A-7)を合成した。
¹H NMR(CDCl₃, δ ppm): 1.36 (3H, t, J = 7.2 Hz), 1.74 (3H, q, J = 1.5 Hz), 2.25 (3H, q, J = 1.5 Hz), 4.28 (2H, q, J = 7.2 Hz), 7.26 - 7.29 (2H, m), 7.44 (1H, d, J = 8.4 Hz), 7.61 (1H, dd, J = 2.1, 8.4 Hz), 7.91 (1H, d, J = 2.1 Hz), 7.91 - 7.95 (2H, m), 10.09 (1H, br).

化合物(A-3)〜(A-6)、(A-8)〜(A-107)、(B-2)〜(B-46)、(C-1)〜(C-5)、(D-1)、(E-1)〜(E-2)、(F-1)〜(F-3)、(F-1)〜(F-3)、(G-1)〜(G-8)、(H-1)〜(H-8)、および(I-1)〜(I-6)を実施例１および２に記載の方法と同様の方法で合成した。化合物群Ａの物理恒数を表１〜１０に、化合物群Ｂの物理恒数を表１１〜１７に、化合物Ｃ群の物理恒数を表１８に、化合物Ｄ群の物理恒数を表１９に、化合物Ｅ群の物理恒数を表２０に、化合物Ｆ群の化合物の物理恒数を表２１に、化合物Ｇ群の化合物の物理恒数を表２２〜２３に、化合物Ｈ群の化合物の物理恒数を表２４〜２５に、化合物Ｉ群の化合物の物理恒数を表２６に示した。

実施例３化合物(A-15)の調製

メトキシ-メトキシカルボニルメチル-トリフェニルホスホニウムクロリド (152 mg)と2-(4-ホルミルベンゾイルアミノ)-4-(3, 4-ジクロロフェニル)チアゾール（57 mg）を塩化メチレン(3 ml)に懸濁させトリエチルアミン (38 mg)を加えた。室温で一夜攪拌した。濃縮後、シリカゲルカラムクロマトグラフィーにより精製し目的とする化合物（A-15）を30 mg得た。
融点203〜205℃
¹H-NMR (CDCl₃) δppm: 3.85 (s, 3H), 3.89 (s, 3H), 6.96 (s, 1H), 7.22 (s, 1H), 7.46 (dd, 1H, J = 8.2, 1.9 Hz), 7.63 (d, 1H, J = 8.2 Hz) 7.86 (d, 2H, J = 8.6 Hz), 7.92 (d, 1H, J = 1.9 Hz), 7.94 (d, 2H, J = 8.6 Hz), 9.82 (brs, 1H).

実施例４化合物(J-3)の調製
(E)-3-(4-ヨードフェニル)-2-メチルアクリル酸エチルエステル(200mg)、ジクロロビス(トリフェニルホスフィン)パラジウム(II)(22mg)、2-アミノ-4-(4'-クロロフェニル)-1H-イミダゾール(277mg)、トリエチルアミン(0.27ml)のDMF(7ml)溶液を一酸化炭素ガス雰囲気下90℃にて15分間攪拌した。反応液を放冷後水にあけ、析出する結晶を濾取しDMFで再結晶して化合物(J-3)を淡黄色結晶として117mg得た。

実施例５化合物(J-16)の調製
化合物(A-53)のエチルエステル体(300mg)のアセトニトリル-テトラヒドロフラン(1:1)溶液(80ml)に1-フルオロ-4-ヒドロキシ-1,4-ジアゾニアビシクロ[2.2.2]オクタンビステトラフルオロボレート(50% onアルミナ1.24 g)を加えて80℃にて30分間攪拌した。アルミナを濾別後、濾液を減圧濃縮し、クロロホルムを加えて懸濁させ、再度不溶物を濾別し減圧濃縮した。分取用TLCプレートで精製後、フッ素化体を黄色結晶として20mg得た。得られたエステル体を化合物(A-2)の調製と同様の方法にて加水分解し、化合物(J-16)を得た。
実施例４および５と同様の方法で化合物(J-1)〜(J-2)、(J-4)〜(J-15)、および(J-17)を合成した。物理恒数を表２７および２８に示した。

実施例６
化合物(K-14, 15, 18)の調製

（第１工程）
化合物(11)(1.1 g)、(12)(760 mg)、炭酸カリウム(1.44 g)、テトラキストリフェニルホスフィンパラジウム(250 mg)のDMF溶液を110℃にて2時間攪拌した。反応溶液を酢酸エチルに注ぎ、水にて4回、飽和食塩水にて洗浄し、硫酸マグネシウムにて乾燥した。溶媒を濃縮後、残留物をシリカゲルカラムクロマトグラフィー（酢酸エチル：n−ヘキサン＝２：３）にて精製し、化合物(13)をアモルファスとして（870 mg）得た。
¹H NMR(CDCl₃, δ ppm): 4.06 (3H, s), 7.16 (1H, s), 7.28 - 7.50 (10H, m), 7.72 (1H, dd, J = 4.8 Hz, 1.8 Hz), 7.75 - 7.80 (2H, m), 8.25 - 8.30 (2H, m), 8.40 (1H, d, J = 2.1 Hz).
（第２工程）
化合物(13) (870 mg)のぎ酸(98〜100%, 20 ml)溶液を50℃にて3時間攪拌した。反応溶液を濃縮後、残渣にトルエンを加え再び濃縮した。得られた残渣をイソプロピルエーテルにて濾取することによって化合物(4)を白色結晶として(473 mg)得た。
¹H NMR(CDCl₃, δ ppm): 3.93 (3H, s), 7.97 - 8.02 (2H, m), 8.04 (1H, dd, J = 7.8 Hz, 1.8 Hz), 8.07 - 8.12 (2H, m), 8.35 (1H, d, J = 1.5 Hz), 8.82 (1H, d, J = 4.8 Hz).
（第３工程）
化合物(K-14)は、化合物(4)を原料とし実施例１の第４工程と同様の反応を行うことによって合成した。物理恒数は表２９に示した。
（第４工程）
化合物(K-15)は、化合物(K-14)を原料とし実施例１の第５工程と同様の反応を行うことによって合成した。物理恒数は表２９に示した。
（第５工程）
化合物(K-15) (100 mg)、ジフェニルリン酸アジド (55 μl)、トリエチルアミン (35l μl)、tert-ブタノール (1 ml)のジメチルホルムアミド (15 ml)溶液を100℃にて1時間攪拌した。反応溶液を酢酸エチルに注ぎ（析出した場合は必要に応じてTHFを加えた）、水にて２回、炭酸水素ナトリウム水溶液、飽和食塩水にて洗浄し、硫酸マグネシウムにて乾燥した。溶媒を濃縮後、残留物をシリカゲルカラムクロマトグラフィー（酢酸エチル：n−ヘキサン＝１：１）にて精製し、化合物(K-18)を白色結晶として（60 mg）得た。物理恒数は表２９に示した。
実施例６と同様の方法を用いて(K-16)〜(K-17)および(K-19)を合成した。実施例１と同様の方法を用いて化合物(K-1)〜(K-13)を合成した。物理恒数を表２９〜３１に示した。

実施例７化合物(L-1、L-２)の調製

（第１工程）
化合物(15)(6.3 g)、(16)(2.0 ml)、トリエチルアミン(6.3 ml)、テトラキストリフェニルホスフィンパラジウム(870 mg)、よう化銅(I) (290 mg)のDMF(70 ml)溶液を90℃にて4時間攪拌した。反応溶液を酢酸エチルに注ぎ、水にて4回、飽和食塩水にて洗浄し、硫酸マグネシウムにて乾燥した。溶媒を濃縮後、残留物をシリカゲルカラムクロマトグラフィー（酢酸エチル：n−ヘキサン＝１：４）にて精製し、化合物(17)をアモルファスとして（2.25 g）得た。
¹H NMR(CDCl₃, δ ppm): 3.81 (3H, s), 7.06 (1H, s), 7.28 - 7.42 (6H, m), 7.51 - 7.55 (4H, m), 7.85 (2H, d, J = 8.7 Hz), 8.17 (2H, d, J = 8.7 Hz).
（第２工程）
化合物(17) (180 mg)のぎ酸(98〜100%, 4 ml)、THF(4 ml)の溶液を室温にて18時間攪拌した。反応溶液を濃縮後、残渣にトルエンを加え再び濃縮した。得られた残渣をイソプロピルエーテルにて濾取することによって化合物(18)を白色針状晶として(95 mg)得た。
¹H NMR(CDCl₃, δ ppm): 3.80 (3H, s), 7.79 (2H, d, J = 8.1 Hz), 8.00 (2H, d, J = 8.1 Hz), 13.33 (1H, bs).
（第３工程）
化合物(L-1)は、化合物(4)を原料とし実施例１の第４工程と同様の反応を行うことによって合成した。物理恒数は表３２に示した。
（第４工程）
化合物(L-2)は、化合物(L-1)を原料とし実施例１の第５工程と同様の反応を行うことによって合成した。物理恒数は表３２に示した。
実施例７と同様の方法で化合物(L-3)〜(L-4)を合成した。物理恒数を表３２に示した。

上記の方法と同様の反応を行うことにより、以下に示す化合物を合成することができる。

(化合物No., R^a, R^b, R^c, R^d, R^e) = (M-1, H, H, H, H, H), (M-2, H, H, H, H, Cl), (M-3, H, H, H, H, F), (M-4, H, H, H, H, CF₃), (M-5, H, H, H, H, Br), (M-6, H, H, H, H, CH₃), (M-7, H, H, H, F, H), (M-8, H, H, H, F, Cl), (M-9, H, H, H, F, F), (M-10, H, H, H, F, CF₃), (M-11, H, H, H, F, Br), (M-12, H, H, H, F, CH₃), (M-13, H, H, H, Cl, H), (M-14, MeO, H, H, Cl, Cl), (M-15, H, H, H, Cl, F), (M-16, H, H, H, Cl, CF₃), (M-17, H, H, H, Cl, Br), (M-18, H, H, H, Cl, CH₃), (M-19, H, H, H, CH₃, H), (M-20, H, H, H, CH₃, Cl), (M-21, H, H, H, CH₃, F), (M-22, H, H, H, CH₃, CF₃), (M-23, H, H, H, CH₃, Br), (M-24, H, H, H, CH₃, CH₃), (M-25, H, H, H, Et, H), (M-26, H, H, H, Et, Cl), (M-27, H, H, H, Et, F), (M-28, H, H, H, Et, CF₃), (M-29, H, H, H, Et, Br), (M-30, H, H, H, Et, CH₃), (M-31, H, H, H, n-Pr, H), (M-32, H, H, H, n-Pr, Cl), (M-33, H, H, H, n-Pr, F), (M-34, H, H, H, n-Pr, CF₃), (M-35, H, H, H, n-Pr, Br), (M-36, H, H, H, n-Pr, CH₃), (M-37, H, H, H, c-Pr, H), (M-38, H, H, H, c-Pr, Cl), (M-39, H, H, H, c-Pr, F), (M-40, H, H, H, c-Pr, CF₃), (M-41, H, H, H, c-Pr, Br), (M-42, H, H, H, c-Pr, CH₃), (M-43, H, H, H, i-Pr, H), (M-44, H, H, H, i-Pr, Cl), (M-45, H, H, H, i-Pr, F), (M-46, H, H, H, i-Pr, CF₃), (M-47, H, H, H, i-Pr, Br), (M-48, H, H, H, i-Pr, CH₃), (M-49, H, H, H, n-Bu, H), (M-50, H, H, H, n-Bu, Cl), (M-51, H, H, H, n-Bu, F), (M-52, H, H, H, n-Bu, CF₃), (M-53, H, H, H, n-Bu, Br), (M-54, H, H, H, n-Bu, CH₃), (M-55, H, H, H, i-Bu, H), (M-56, H, H, H, i-Bu, Cl), (M-57, H, H, H, i-Bu, F), (M-58, H, H, H, i-Bu, CF₃), (M-59, H, H, H, i-Bu, Br), (M-60, H, H, H, i-Bu, CH₃), (M-61, H, H, H, sec-Bu, H), (M-62, H, H, H, sec-Bu, Cl), (M-63, H, H, H, sec-Bu, F), (M-64, H, H, H, sec-Bu, CF₃), (M-65, H, H, H, sec-Bu, Br), (M-66, H, H, H, sec-Bu, CH₃), (M-67, H, H, H, n-Pen, H), (M-68, H, H, H, n-Pen, Cl), (M-69, H, H, H, n-Pen, F), (M-70, H, H, H, n-Pen, CF₃), (M-71, H, H, H, n-Pen, Br), (M-72, H, H, H, n-Pen, CH₃), (M-73, H, H, H, c-Pen, H), (M-74, H, H, H, c-Pen, Cl), (M-75, H, H, H, c-Pen, F), (M-76, H, H, H, c-Pen, CF₃), (M-77, H, H, H, c-Pen, Br), (M-78, H, H, H, c-Pen, CH₃), (M-79, H, H, H, n-Hex, H), (M-80, H, H, H, n-Hex, Cl), (M-81, H, H, H, n-Hex, F), (M-82, H, H, H, n-Hex, CF₃), (M-83, H, H, H, n-Hex, Br), (M-84, H, H, H, n-Hex, CH₃), (M-85, H, H, H, c-Hex, H), (M-86, H, H, H, c-Hex, Cl), (M-87, H, H, H, c-Hex, F), (M-88, H, H, H, c-Hex, CF₃), (M-89, H, H, H, c-Hex, Br), (M-90, H, H, H, c-Hex, CH₃), (M-91, H, H, H, OH, H), (M-92, H, H, H, OH, Cl), (M-93, H, H, H, OH, F), (M-94, H, H, H, OH, CF₃), (M-95, H, H, H, OH, Br), (M-96, H, H, H, OH, CH₃), (M-97, H, H, H, EtO, H), (M-98, H, H, H, EtO, Cl), (M-99, H, H, H, EtO, F), (M-100, H, H, H, EtO, CF₃), (M-101, H, H, H, EtO, Br), (M-102, H, H, H, EtO, CH₃), (M-103, H, H, H, n-PrO, H), (M-104, H, H, H, n-PrO, Cl), (M-105, H, H, H, n-PrO, F), (M-106, H, H, H, n-PrO, CF₃), (M-107, H, H, H, n-PrO, Br), (M-108, H, H, H, n-PrO, CH₃), (M-109, H, H, H, PhO, H), (M-110, H, H, H, PhO, Cl), (M-111, H, H, H, PhO, F), (M-112, H, H, H, PhO, CF₃), (M-113, H, H, H, PhO, Br), (M-114, H, H, H, PhO, CH₃), (M-115, H, H, H, BnO, H), (M-116, H, H, H, BnO, Cl), (M-117, H, H, H, BnO, F), (M-118, H, H, H, BnO, CF₃), (M-119, H, H, H, BnO, Br), (M-120, H, H, H, BnO, CH₃), (M-121, H, H, H, PhCH₂CH₂O, H), (M-122, H, H, H, PhCH₂CH₂O, Cl), (M-123, H, H, H, PhCH₂CH₂O, F), (M-124, H, H, H, PhCH₂CH₂O, CF₃), (M-125, H, H, H, PhCH₂CH₂O, Br), (M-126, H, H, H, PhCH₂CH₂O, CH₃), (M-127, H, H, H, CF₃O, H), (M-128, H, H, H, CF₃O, Cl), (M-129, H, H, H, CF₃O, F), (M-130, H, H, H, CF₃O, CF₃), (M-131, H, H, H, CF₃O, Br), (M-132, H, H, H, CF₃O, CH₃), (M-133, H, H, H, Ph, H), (M-134, H, H, H, Ph, Cl), (M-135, H, H, H, Ph, F), (M-136, H, H, H, Ph, CF₃), (M-137, H, H, H, Ph, Br), (M-138, H, H, H, Ph, CH₃), (M-139, H, H, H, 4-F-Ph, H), (M-140, H, H, H, 4-F-Ph, Cl), (M-141, H, H, H, 4-F-Ph, F), (M-142, H, H, H, 4-F-Ph, CF₃), (M-143, H, H, H, 4-F-Ph, Br), (M-144, H, H, H, 4-F-Ph, CH₃), (M-145, H, H, H, 4-CF₃-Ph, H), (M-146, H, H, H, 4-CF₃-Ph, Cl), (M-147, H, H, H, 4-CF₃-Ph, F), (M-148, H, H, H, 4-CF₃-Ph, CF₃), (M-149, H, H, H, 4-CF₃-Ph, Br), (M-150, H, H, H, 4-CF₃-Ph, CH₃), (M-151, H, H, H, 4-(Me)₂N-Ph, H), (M-152, H, H, H, 4-(Me)₂N-Ph, Cl), (M-153, H, H, H, 4-(Me)₂N-Ph, F), (M-154, H, H, H, 4-(Me)₂N-Ph, CF₃), (M-155, H, H, H, 4-(Me)₂N-Ph, Br), (M-156, H, H, H, 4-(Me)₂N-Ph, CH₃), (M-157, H, H, H, 4-OH-Ph, H), (M-158, H, H, H, 4-OH-Ph, Cl), (M-159, H, H, H, 4-OH-Ph, F), (M-160, H, H, H, 4-OH-Ph, CF₃), (M-161, H, H, H, 4-OH-Ph, Br), (M-162, H, H, H, 4-OH-Ph, CH₃), (M-163, H, H, H, 3,4-di-F-Ph, H), (M-164, H, H, H, 3,4-di-F-Ph, Cl), (M-165, H, H, H, 3,4-di-F-Ph, F), (M-166, H, H, H, 3,4-di-F-Ph, CF₃), (M-167, H, H, H, 3,4-di-F-Ph, Br), (M-168, H, H, H, 3,4-di-F-Ph, CH₃), (M-169, H, H, H, 4-COOH-Ph, H), (M-170, H, H, H, 4-COOH-Ph, Cl), (M-171, H, H, H, 4-COOH-Ph, F), (M-172, H, H, H, 4-COOH-Ph, CF₃), (M-173, H, H, H, 4-COOH-Ph, Br), (M-174, H, H, H, 4-COOH-Ph, CH₃), (M-175, H, H, H, Bn, H), (M-176, H, H, H, Bn, Cl), (M-177, H, H, H, Bn, F), (M-178, H, H, H, Bn, CF₃), (M-179, H, H, H, Bn, Br), (M-180, H, H, H, Bn, CH₃), (M-181, H, H, H, 4-F-Bn, H), (M-182, H, H, H, 4-F-Bn, Cl), (M-183, H, H, H, 4-F-Bn, F), (M-184, H, H, H, 4-F-Bn, CF₃), (M-185, H, H, H, 4-F-Bn, Br), (M-186, H, H, H, 4-F-Bn, CH₃), (M-187, H, H, H, 2-Py, H), (M-188, H, H, H, 2-Py, Cl), (M-189, H, H, H, 2-Py, F), (M-190, H, H, H, 2-Py, CF₃), (M-191, H, H, H, 2-Py, Br), (M-192, H, H, H, 2-Py, CH₃), (M-193, H, H, H, 3-Py, H), (M-194, H, H, H, 3-Py, Cl), (M-195, H, H, H, 3-Py, F), (M-196, H, H, H, 3-Py, CF₃), (M-197, H, H, H, 3-Py, Br), (M-198, H, H, H, 3-Py, CH₃), (M-199, H, H, H, 4-Py, H), (M-200, H, H, H, 4-Py, Cl), (M-201, H, H, H, 4-Py, F), (M-202, H, H, H, 4-Py, CF₃), (M-203, H, H, H, 4-Py, Br), (M-204, H, H, H, 4-Py, CH₃), (M-205, H, H, H, 2-Th, H), (M-206, H, H, H, 2-Th, Cl), (M-207, H, H, H, 2-Th, F), (M-208, H, H, H, 2-Th, CF₃), (M-209, H, H, H, 2-Th, Br), (M-210, H, H, H, 2-Th, CH₃), (M-211, H, H, H, 3-Th, H), (M-212, H, H, H, 3-Th, Cl), (M-213, H, H, H, 3-Th, F), (M-214, H, H, H, 3-Th, CF₃), (M-215, H, H, H, 3-Th, Br), (M-216, H, H, H, 3-Th, CH₃), (M-217, H, H, H, pyrazol-2-yl, H), (M-218, H, H, H, pyrazol-2-yl, Cl), (M-219, H, H, H, pyrazol-2-yl, F), (M-220, H, H, H, pyrazol-2-yl, CF₃), (M-221, H, H, H, pyrazol-2-yl, Br), (M-222, H, H, H, pyrazol-2-yl, CH₃), (M-223, H, H, H, pyrazol-3-yl, H), (M-224, H, H, H, pyrazol-3-yl, Cl), (M-225, H, H, H, pyrazol-3-yl, F), (M-226, H, H, H, pyrazol-3-yl, CF₃), (M-227, H, H, H, pyrazol-3-yl, Br), (M-228, H, H, H, pyrazol-3-yl, CH₃), (M-229, H, H, H, pyrimidin-2-yl, H), (M-230, H, H, H, pyrimidin-2-yl, Cl), (M-231, H, H, H, pyrimidin-2-yl, F), (M-232, H, H, H, pyrimidin-2-yl, CF₃), (M-233, H, H, H, pyrimidin-2-yl, Br), (M-234, H, H, H, pyrimidin-2-yl, CH₃), (M-235, H, H, H, pyrimidin-4-yl, H), (M-236, H, H, H, pyrimidin-4-yl, Cl), (M-237, H, H, H, pyrimidin-4-yl, F), (M-238, H, H, H, pyrimidin-4-yl, CF₃), (M-239, H, H, H, pyrimidin-4-yl, Br), (M-240, H, H, H, pyrimidin-4-yl, CH₃), (M-241, H, H, H, pyrimidin-5-yl, H), (M-242, H, H, H, pyrimidin-5-yl, Cl), (M-243, H, H, H, pyrimidin-5-yl, F), (M-244, H, H, H, pyrimidin-5-yl, CF₃), (M-245, H, H, H, pyrimidin-5-yl, Br), (M-246, H, H, H, pyrimidin-5-yl, CH₃), (M-247, H, H, H, HOOCCH₂CH₂CH₂, H), (M-248, H, H, H, HOOCCH₂CH₂CH₂, Cl), (M-249, H, H, H, HOOCCH₂CH₂CH₂, F), (M-250, H, H, H, HOOCCH₂CH₂CH₂, CF₃), (M-251, H, H, H, HOOCCH₂CH₂CH₂, Br), (M-252, H, H, H, HOOCCH₂CH₂CH₂, CH₃), (M-253, H, H, H, HOOCCH₂CH₂CH₂CH₂, H), (M-254, H, H, H, HOOCCH₂CH₂CH₂CH₂, Cl), (M-255, H, H, H, HOOCCH₂CH₂CH₂CH₂, F), (M-256, H, H, H, HOOCCH₂CH₂CH₂CH₂, CF₃), (M-257, H, H, H, HOOCCH₂CH₂CH₂CH₂, Br), (M-258, H, H, H, HOOCCH₂CH₂CH₂CH₂, CH₃), (M-259, H, H, H, (Me)₂NCOCH₂CH₂CH₂CH₂, H), (M-260, H, H, H, (Me)₂NCOCH₂CH₂CH₂CH₂, Cl), (M-261, H, H, H, (Me)₂NCOCH₂CH₂CH₂CH₂, F), (M-262, H, H, H, (Me)₂NCOCH₂CH₂CH₂CH₂, CF₃), (M-263, H, H, H, (Me)₂NCOCH₂CH₂CH₂CH₂, Br), (M-264, H, H, H, (Me)₂NCOCH₂CH₂CH₂CH₂, CH₃), (M-265, H, H, H, (Me)₂NCOCH₂CH₂CH₂CH
₂CH₂, H), (M-266, H, H, H, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, Cl), (M-267, H, H, H, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, F), (M-268, H, H, H, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, CF₃), (M-269, H, H, H, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, Br), (M-270, H, H, H, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, CH₃), (M-271, H, H, H, MeOCH₂, H), (M-272, H, H, H, MeOCH₂, Cl), (M-273, H, H, H, MeOCH₂, F), (M-274, H, H, H, MeOCH₂, CF₃), (M-275, H, H, H, MeOCH₂, Br), (M-276, H, H, H, MeOCH₂, CH₃), (M-277, H, H, H, EtOCH₂, H), (M-278, H, H, H, EtOCH₂, Cl), (M-279, H, H, H, EtOCH₂, F), (M-280, H, H, H, EtOCH₂, CF₃), (M-281, H, H, H, EtOCH₂, Br), (M-282, H, H, H, EtOCH₂, CH₃), (M-283, H, H, H, EtOCH₂CH₂, H), (M-284, H, H, H, EtOCH₂CH₂, Cl), (M-285, H, H, H, EtOCH₂CH₂, F), (M-286, H, H, H, EtOCH₂CH₂, CF₃), (M-287, H, H, H, EtOCH₂CH₂, Br), (M-288, H, H, H, EtOCH₂CH₂, CH₃), (M-289, H, H, H, MeOCH₂CH₂OCH₂CH₂, H), (M-290, H, H, H, MeOCH₂CH₂OCH₂CH₂, Cl), (M-291, H, H, H, MeOCH₂CH₂OCH₂CH₂, F), (M-292, H, H, H, MeOCH₂CH₂OCH₂CH₂, CF₃), (M-293, H, H, H, MeOCH₂CH₂OCH₂CH₂, Br), (M-294, H, H, H, MeOCH₂CH₂OCH₂CH₂, CH₃), (M-295, H, H, H, MeOCH₂CH₂, H), (M-296, H, H, H, MeOCH₂CH₂, Cl), (M-297, H, H, H, MeOCH₂CH₂, F), (M-298, H, H, H, MeOCH₂CH₂, CF₃), (M-299, H, H, H, MeOCH₂CH₂, Br), (M-300, H, H, H, MeOCH₂CH₂, CH₃), (M-301, H, H, H, HOCH₂, H), (M-302, H, H, H, HOCH₂, Cl), (M-303, H, H, H, HOCH₂, F), (M-304, H, H, H, HOCH₂, CF₃), (M-305, H, H, H, HOCH₂, Br), (M-306, H, H, H, HOCH₂, CH₃), (M-307, H, H, H, HOCH₂CH₂, H), (M-308, H, H, H, HOCH₂CH₂, Cl), (M-309, H, H, H, HOCH₂CH₂, F), (M-310, H, H, H, HOCH₂CH₂, CF₃), (M-311, H, H, H, HOCH₂CH₂, Br), (M-312, H, H, H, HOCH₂CH₂, CH₃), (M-313, H, H, H, HOCH₂CH₂CH₂, H), (M-314, H, H, H, HOCH₂CH₂CH₂, Cl), (M-315, H, H, H, HOCH₂CH₂CH₂, F), (M-316, H, H, H, HOCH₂CH₂CH₂, CF₃), (M-317, H, H, H, HOCH₂CH₂CH₂, Br), (M-318, H, H, H, HOCH₂CH₂CH₂, CH₃), (M-319, H, H, H, HOCH₂CH₂CH₂CH₂, H), (M-320, H, H, H, HOCH₂CH₂CH₂CH₂, Cl), (M-321, H, H, H, HOCH₂CH₂CH₂CH₂, F), (M-322, H, H, H, HOCH₂CH₂CH₂CH₂, CF₃), (M-323, H, H, H, HOCH₂CH₂CH₂CH₂, Br), (M-324, H, H, H, HOCH₂CH₂CH₂CH₂, CH₃), (M-325, H, H, H, HOCH₂CH₂CH₂CH₂CH₂, H), (M-326, H, H, H, HOCH₂CH₂CH₂CH₂CH₂, Cl), (M-327, H, H, H, HOCH₂CH₂CH₂CH₂CH₂, F), (M-328, H, H, H, HOCH₂CH₂CH₂CH₂CH₂, CF₃), (M-329, H, H, H, HOCH₂CH₂CH₂CH₂CH₂, Br), (M-330, H, H, H, HOCH₂CH₂CH₂CH₂CH₂, CH₃), (M-331, H, H, H, HOCH₂CH₂OCH₂CH₂, H), (M-332, H, H, H, HOCH₂CH₂OCH₂CH₂, Cl), (M-333, H, H, H, HOCH₂CH₂OCH₂CH₂, F), (M-334, H, H, H, HOCH₂CH₂OCH₂CH₂, CF₃), (M-335, H, H, H, HOCH₂CH₂OCH₂CH₂, Br), (M-336, H, H, H, HOCH₂CH₂OCH₂CH₂, CH₃), (M-337, H, H, H, (Me)₂N, H), (M-338, H, H, H, (Me)₂N, Cl), (M-339, H, H, H, (Me)₂N, F), (M-340, H, H, H, (Me)₂N, CF₃), (M-341, H, H, H, (Me)₂N, Br), (M-342, H, H, H, (Me)₂N, CH₃), (M-343, H, H, H, piperidin-4-yl-methyl, H), (M-344, H, H, H, piperidin-4-yl-methyl, Cl), (M-345, H, H, H, piperidin-4-yl-methyl, F), (M-346, H, H, H, piperidin-4-yl-methyl, CF₃), (M-347, H, H, H, piperidin-4-yl-methyl, Br), (M-348, H, H, H, piperidin-4-yl-methyl, CH₃), (M-349, H, H, H, cyclohexylmethyl, H), (M-350, H, H, H, cyclohexylmethyl, Cl), (M-351, H, H, H, cyclohexylmethyl, F), (M-352, H, H, H, cyclohexylmethyl, CF₃), (M-353, H, H, H, cyclohexylmethyl, Br), (M-354, H, H, H, cyclohexylmethyl, CH₃), (M-355, H, H, F, H, H), (M-356, H, H, F, H, Cl), (M-357, H, H, F, H, F), (M-358, H, H, F, H, CF₃), (M-359, H, H, F, H, Br), (M-360, H, H, F, H, CH₃), (M-361, H, H, F, F, H), (M-362, H, H, F, F, Cl), (M-363, H, H, F, F, F), (M-364, H, H, F, F, CF₃), (M-365, H, H, F, F, Br), (M-366, H, H, F, F, CH₃), (M-367, H, H, F, Cl, H), (M-368, H, H, F, Cl, Cl), (M-369, H, H, F, Cl, F), (M-370, H, H, F, Cl, CF₃), (M-371, H, H, F, Cl, Br), (M-372, H, H, F, Cl, CH₃), (M-373, H, H, F, CH₃, H), (M-374, H, H, F, CH₃, Cl), (M-375, H, H, F, CH₃, F), (M-376, H, H, F, CH₃, CF₃), (M-377, H, H, F, CH₃, Br), (M-378, H, H, F, CH₃, CH₃), (M-379, H, H, F, Et, H), (M-380, H, H, F, Et, Cl), (M-381, H, H, F, Et, F), (M-382, H, H, F, Et, CF₃), (M-383, H, H, F, Et, Br), (M-384, H, H, F, Et, CH₃), (M-385, H, H, F, n-Pr, H), (M-386, H, H, F, n-Pr, Cl), (M-387, H, H, F, n-Pr, F), (M-388, H, H, F, n-Pr, CF₃), (M-389, H, H, F, n-Pr, Br), (M-390, H, H, F, n-Pr, CH₃), (M-391, H, H, F, c-Pr, H), (M-392, H, H, F, c-Pr, Cl), (M-393, H, H, F, c-Pr, F), (M-394, H, H, F, c-Pr, CF₃), (M-395, H, H, F, c-Pr, Br), (M-396, H, H, F, c-Pr, CH₃), (M-397, H, H, F, i-Pr, H), (M-398, H, H, F, i-Pr, Cl), (M-399, H, H, F, i-Pr, F), (M-400, H, H, F, i-Pr, CF₃), (M-401, H, H, F, i-Pr, Br), (M-402, H, H, F, i-Pr, CH₃), (M-403, H, H, F, n-Bu, H), (M-404, H, H, F, n-Bu, Cl), (M-405, H, H, F, n-Bu, F), (M-406, H, H, F, n-Bu, CF₃), (M-407, H, H, F, n-Bu, Br), (M-408, H, H, F, n-Bu, CH₃), (M-409, H, H, F, i-Bu, H), (M-410, H, H, F, i-Bu, Cl), (M-411, H, H, F, i-Bu, F), (M-412, H, H, F, i-Bu, CF₃), (M-413, H, H, F, i-Bu, Br), (M-414, H, H, F, i-Bu, CH₃), (M-415, H, H, F, sec-Bu, H), (M-416, H, H, F, sec-Bu, Cl), (M-417, H, H, F, sec-Bu, F), (M-418, H, H, F, sec-Bu, CF₃), (M-419, H, H, F, sec-Bu, Br), (M-420, H, H, F, sec-Bu, CH₃), (M-421, H, H, F, n-Pen, H), (M-422, H, H, F, n-Pen, Cl), (M-423, H, H, F, n-Pen, F), (M-424, H, H, F, n-Pen, CF₃), (M-425, H, H, F, n-Pen, Br), (M-426, H, H, F, n-Pen, CH₃), (M-427, H, H, F, c-Pen, H), (M-428, H, H, F, c-Pen, Cl), (M-429, H, H, F, c-Pen, F), (M-430, H, H, F, c-Pen, CF₃), (M-431, H, H, F, c-Pen, Br), (M-432, H, H, F, c-Pen, CH₃), (M-433, H, H, F, n-Hex, H), (M-434, H, H, F, n-Hex, Cl), (M-435, H, H, F, n-Hex, F), (M-436, H, H, F, n-Hex, CF₃), (M-437, H, H, F, n-Hex, Br), (M-438, H, H, F, n-Hex, CH₃), (M-439, H, H, F, c-Hex, H), (M-440, H, H, F, c-Hex, Cl), (M-441, H, H, F, c-Hex, F), (M-442, H, H, F, c-Hex, CF₃), (M-443, H, H, F, c-Hex, Br), (M-444, H, H, F, c-Hex, CH₃), (M-445, H, H, F, OH, H), (M-446, H, H, F, OH, Cl), (M-447, H, H, F, OH, F), (M-448, H, H, F, OH, CF₃), (M-449, H, H, F, OH, Br), (M-450, H, H, F, OH, CH₃), (M-451, H, H, F, EtO, H), (M-452, H, H, F, EtO, Cl), (M-453, H, H, F, EtO, F), (M-454, H, H, F, EtO, CF₃), (M-455, H, H, F, EtO, Br), (M-456, H, H, F, EtO, CH₃), (M-457, H, H, F, n-PrO, H), (M-458, H, H, F, n-PrO, Cl), (M-459, H, H, F, n-PrO, F), (M-460, H, H, F, n-PrO, CF₃), (M-461, H, H, F, n-PrO, Br), (M-462, H, H, F, n-PrO, CH₃), (M-463, H, H, F, PhO, H), (M-464, H, H, F, PhO, Cl), (M-465, H, H, F, PhO, F), (M-466, H, H, F, PhO, CF₃), (M-467, H, H, F, PhO, Br), (M-468, H, H, F, PhO, CH₃), (M-469, H, H, F, BnO, H), (M-470, H, H, F, BnO, Cl), (M-471, H, H, F, BnO, F), (M-472, H, H, F, BnO, CF₃), (M-473, H, H, F, BnO, Br), (M-474, H, H, F, BnO, CH₃), (M-475, H, H, F, PhCH₂CH₂O, H), (M-476, H, H, F, PhCH₂CH₂O, Cl), (M-477, H, H, F, PhCH₂CH₂O, F), (M-478, H, H, F, PhCH₂CH₂O, CF₃), (M-479, H, H, F, PhCH₂CH₂O, Br), (M-480, H, H, F, PhCH₂CH₂O, CH₃), (M-481, H, H, F, CF₃O, H), (M-482, H, H, F, CF₃O, Cl), (M-483, H, H, F, CF₃O, F), (M-484, H, H, F, CF₃O, CF₃), (M-485, H, H, F, CF₃O,
Br), (M-486, H, H, F, CF₃O, CH₃), (M-487, H, H, F, Ph, H), (M-488, H, H, F, Ph, Cl), (M-489, H, H, F, Ph, F), (M-490, H, H, F, Ph, CF₃), (M-491, H, H, F, Ph, Br), (M-492, H, H, F, Ph, CH₃), (M-493, H, H, F, 4-F-Ph, H), (M-494, H, H, F, 4-F-Ph, Cl), (M-495, H, H, F, 4-F-Ph, F), (M-496, H, H, F, 4-F-Ph, CF₃), (M-497, H, H, F, 4-F-Ph, Br), (M-498, H, H, F, 4-F-Ph, CH₃), (M-499, H, H, F, 4-CF₃-Ph, H), (M-500, H, H, F, 4-CF₃-Ph, Cl), (M-501, H, H, F, 4-CF₃-Ph, F), (M-502, H, H, F, 4-CF₃-Ph, CF₃), (M-503, H, H, F, 4-CF₃-Ph, Br), (M-504, H, H, F, 4-CF₃-Ph, CH₃), (M-505, H, H, F, 4-(Me)₂N-Ph, H), (M-506, H, H, F, 4-(Me)₂N-Ph, Cl), (M-507, H, H, F, 4-(Me)₂N-Ph, F), (M-508, H, H, F, 4-(Me)₂N-Ph, CF₃), (M-509, H, H, F, 4-(Me)₂N-Ph, Br), (M-510, H, H, F, 4-(Me)₂N-Ph, CH₃), (M-511, H, H, F, 4-OH-Ph, H), (M-512, H, H, F, 4-OH-Ph, Cl), (M-513, H, H, F, 4-OH-Ph, F), (M-514, H, H, F, 4-OH-Ph, CF₃), (M-515, H, H, F, 4-OH-Ph, Br), (M-516, H, H, F, 4-OH-Ph, CH₃), (M-517, H, H, F, 3,4-di-F-Ph, H), (M-518, H, H, F, 3,4-di-F-Ph, Cl), (M-519, H, H, F, 3,4-di-F-Ph, F), (M-520, H, H, F, 3,4-di-F-Ph, CF₃), (M-521, H, H, F, 3,4-di-F-Ph, Br), (M-522, H, H, F, 3,4-di-F-Ph, CH₃), (M-523, H, H, F, 4-COOH-Ph, H), (M-524, H, H, F, 4-COOH-Ph, Cl), (M-525, H, H, F, 4-COOH-Ph, F), (M-526, H, H, F, 4-COOH-Ph, CF₃), (M-527, H, H, F, 4-COOH-Ph, Br), (M-528, H, H, F, 4-COOH-Ph, CH₃), (M-529, H, H, F, Bn, H), (M-530, H, H, F, Bn, Cl), (M-531, H, H, F, Bn, F), (M-532, H, H, F, Bn, CF₃), (M-533, H, H, F, Bn, Br), (M-534, H, H, F, Bn, CH₃), (M-535, H, H, F, 4-F-Bn, H), (M-536, H, H, F, 4-F-Bn, Cl), (M-537, H, H, F, 4-F-Bn, F), (M-538, H, H, F, 4-F-Bn, CF₃), (M-539, H, H, F, 4-F-Bn, Br), (M-540, H, H, F, 4-F-Bn, CH₃), (M-541, H, H, F, 2-Py, H), (M-542, H, H, F, 2-Py, Cl), (M-543, H, H, F, 2-Py, F), (M-544, H, H, F, 2-Py, CF₃), (M-545, H, H, F, 2-Py, Br), (M-546, H, H, F, 2-Py, CH₃), (M-547, H, H, F, 3-Py, H), (M-548, H, H, F, 3-Py, Cl), (M-549, H, H, F, 3-Py, F), (M-550, H, H, F, 3-Py, CF₃), (M-551, H, H, F, 3-Py, Br), (M-552, H, H, F, 3-Py, CH₃), (M-553, H, H, F, 4-Py, H), (M-554, H, H, F, 4-Py, Cl), (M-555, H, H, F, 4-Py, F), (M-556, H, H, F, 4-Py, CF₃), (M-557, H, H, F, 4-Py, Br), (M-558, H, H, F, 4-Py, CH₃), (M-559, H, H, F, 2-Th, H), (M-560, H, H, F, 2-Th, Cl), (M-561, H, H, F, 2-Th, F), (M-562, H, H, F, 2-Th, CF₃), (M-563, H, H, F, 2-Th, Br), (M-564, H, H, F, 2-Th, CH₃), (M-565, H, H, F, 3-Th, H), (M-566, H, H, F, 3-Th, Cl), (M-567, H, H, F, 3-Th, F), (M-568, H, H, F, 3-Th, CF₃), (M-569, H, H, F, 3-Th, Br), (M-570, H, H, F, 3-Th, CH₃), (M-571, H, H, F, pyrazol-2-yl, H), (M-572, H, H, F, pyrazol-2-yl, Cl), (M-573, H, H, F, pyrazol-2-yl, F), (M-574, H, H, F, pyrazol-2-yl, CF₃), (M-575, H, H, F, pyrazol-2-yl, Br), (M-576, H, H, F, pyrazol-2-yl, CH₃), (M-577, H, H, F, pyrazol-3-yl, H), (M-578, H, H, F, pyrazol-3-yl, Cl), (M-579, H, H, F, pyrazol-3-yl, F), (M-580, H, H, F, pyrazol-3-yl, CF₃), (M-581, H, H, F, pyrazol-3-yl, Br), (M-582, H, H, F, pyrazol-3-yl, CH₃), (M-583, H, H, F, pyrimidin-2-yl, H), (M-584, H, H, F, pyrimidin-2-yl, Cl), (M-585, H, H, F, pyrimidin-2-yl, F), (M-586, H, H, F, pyrimidin-2-yl, CF₃), (M-587, H, H, F, pyrimidin-2-yl, Br), (M-588, H, H, F, pyrimidin-2-yl, CH₃), (M-589, H, H, F, pyrimidin-4-yl, H), (M-590, H, H, F, pyrimidin-4-yl, Cl), (M-591, H, H, F, pyrimidin-4-yl, F), (M-592, H, H, F, pyrimidin-4-yl, CF₃), (M-593, H, H, F, pyrimidin-4-yl, Br), (M-594, H, H, F, pyrimidin-4-yl, CH₃), (M-595, H, H, F, pyrimidin-5-yl, H), (M-596, H, H, F, pyrimidin-5-yl, Cl), (M-597, H, H, F, pyrimidin-5-yl, F), (M-598, H, H, F, pyrimidin-5-yl, CF₃), (M-599, H, H, F, pyrimidin-5-yl, Br), (M-600, H, H, F, pyrimidin-5-yl, CH₃), (M-601, H, H, F, HOOCCH₂CH₂CH₂, H), (M-602, H, H, F, HOOCCH₂CH₂CH₂, Cl), (M-603, H, H, F, HOOCCH₂CH₂CH₂, F), (M-604, H, H, F, HOOCCH₂CH₂CH₂, CF₃), (M-605, H, H, F, HOOCCH₂CH₂CH₂, Br), (M-606, H, H, F, HOOCCH₂CH₂CH₂, CH₃), (M-607, H, H, F, HOOCCH₂CH₂CH₂CH₂, H), (M-608, H, H, F, HOOCCH₂CH₂CH₂CH₂, Cl), (M-609, H, H, F, HOOCCH₂CH₂CH₂CH₂, F), (M-610, H, H, F, HOOCCH₂CH₂CH₂CH₂, CF₃), (M-611, H, H, F, HOOCCH₂CH₂CH₂CH₂, Br), (M-612, H, H, F, HOOCCH₂CH₂CH₂CH₂, CH₃), (M-613, H, H, F, (Me)₂NCOCH₂CH₂CH₂CH₂, H), (M-614, H, H, F, (Me)₂NCOCH₂CH₂CH₂CH₂, Cl), (M-615, H, H, F, (Me)₂NCOCH₂CH₂CH₂CH₂, F), (M-616, H, H, F, (Me)₂NCOCH₂CH₂CH₂CH₂, CF₃), (M-617, H, H, F, (Me)₂NCOCH₂CH₂CH₂CH₂, Br), (M-618, H, H, F, (Me)₂NCOCH₂CH₂CH₂CH₂, CH₃), (M-619, H, H, F, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, H), (M-620, H, H, F, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, Cl), (M-621, H, H, F, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, F), (M-622, H, H, F, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, CF₃), (M-623, H, H, F, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, Br), (M-624, H, H, F, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, CH₃), (M-625, H, H, F, MeOCH₂, H), (M-626, H, H, F, MeOCH₂, Cl), (M-627, H, H, F, MeOCH₂, F), (M-628, H, H, F, MeOCH₂, CF₃), (M-629, H, H, F, MeOCH₂, Br), (M-630, H, H, F, MeOCH₂, CH₃), (M-631, H, H, F, EtOCH₂, H), (M-632, H, H, F, EtOCH₂, Cl), (M-633, H, H, F, EtOCH₂, F), (M-634, H, H, F, EtOCH₂, CF₃), (M-635, H, H, F, EtOCH₂, Br), (M-636, H, H, F, EtOCH₂, CH₃), (M-637, H, H, F, EtOCH₂CH₂, H), (M-638, H, H, F, EtOCH₂CH₂, Cl), (M-639, H, H, F, EtOCH₂CH₂, F), (M-640, H, H, F, EtOCH₂CH₂, CF₃), (M-641, H, H, F, EtOCH₂CH₂, Br), (M-642, H, H, F, EtOCH₂CH₂, CH₃), (M-643, H, H, F, MeOCH₂CH₂OCH₂CH₂, H), (M-644, H, H, F, MeOCH₂CH₂OCH₂CH₂, Cl), (M-645, H, H, F, MeOCH₂CH₂OCH₂CH₂, F), (M-646, H, H, F, MeOCH₂CH₂OCH₂CH₂, CF₃), (M-647, H, H, F, MeOCH₂CH₂OCH₂CH₂, Br), (M-648, H, H, F, MeOCH₂CH₂OCH₂CH₂, CH₃), (M-649, H, H, F, MeOCH₂CH₂, H), (M-650, H, H, F, MeOCH₂CH₂, Cl), (M-651, H, H, F, MeOCH₂CH₂, F), (M-652, H, H, F, MeOCH₂CH₂, CF₃), (M-653, H, H, F, MeOCH₂CH₂, Br), (M-654, H, H, F, MeOCH₂CH₂, CH₃), (M-655, H, H, F, HOCH₂, H), (M-656, H, H, F, HOCH₂, Cl), (M-657, H, H, F, HOCH₂, F), (M-658, H, H, F, HOCH₂, CF₃), (M-659, H, H, F, HOCH₂, Br), (M-660, H, H, F, HOCH₂, CH₃), (M-661, H, H, F, HOCH₂CH₂, H), (M-662, H, H, F, HOCH₂CH₂, Cl), (M-663, H, H, F, HOCH₂CH₂, F), (M-664, H, H, F, HOCH₂CH₂, CF₃), (M-665, H, H, F, HOCH₂CH₂, Br), (M-666, H, H, F, HOCH₂CH₂, CH₃), (M-667, H, H, F, HOCH₂CH₂CH₂, H), (M-668, H, H, F, HOCH₂CH₂CH₂, Cl), (M-669, H, H, F, HOCH₂CH₂CH₂, F), (M-670, H, H, F, HOCH₂CH₂CH₂, CF₃), (M-671, H, H, F, HOCH₂CH₂CH₂, Br), (M-672, H, H, F, HOCH₂CH₂CH₂, CH₃), (M-673, H, H, F, HOCH₂CH₂CH₂CH₂, H), (M-674, H, H, F, HOCH₂CH₂CH₂CH₂, Cl), (M-675, H, H, F, HOCH₂CH₂CH₂CH₂, F), (M-676, H, H, F, HOCH₂CH₂CH₂CH₂, CF₃), (M-677, H, H, F, HOCH₂CH₂CH₂CH₂, Br), (M-678, H, H, F, HOCH₂CH₂CH₂CH₂, CH₃), (M-679, H, H, F, HOCH₂CH₂CH₂CH₂CH₂, H), (M-680, H, H, F, HOCH₂CH₂CH₂CH₂CH₂, Cl), (M-681, H, H, F, HOCH₂CH₂CH₂CH₂CH₂, F), (M-682, H, H, F, HOCH₂CH₂CH₂CH₂CH₂, CF₃), (M-683, H, H,
F, HOCH₂CH₂CH₂CH₂CH₂, Br), (M-684, H, H, F, HOCH₂CH₂CH₂CH₂CH₂, CH₃), (M-685, H, H, F, HOCH₂CH₂OCH₂CH₂, H), (M-686, H, H, F, HOCH₂CH₂OCH₂CH₂, Cl), (M-687, H, H, F, HOCH₂CH₂OCH₂CH₂, F), (M-688, H, H, F, HOCH₂CH₂OCH₂CH₂, CF₃), (M-689, H, H, F, HOCH₂CH₂OCH₂CH₂, Br), (M-690, H, H, F, HOCH₂CH₂OCH₂CH₂, CH₃), (M-691, H, H, F, (Me)₂N, H), (M-692, H, H, F, (Me)₂N, Cl), (M-693, H, H, F, (Me)₂N, F), (M-694, H, H, F, (Me)₂N, CF₃), (M-695, H, H, F, (Me)₂N, Br), (M-696, H, H, F, (Me)₂N, CH₃), (M-697, H, H, F, piperidin-4-yl-methyl, H), (M-698, H, H, F, piperidin-4-yl-methyl, Cl), (M-699, H, H, F, piperidin-4-yl-methyl, F), (M-700, H, H, F, piperidin-4-yl-methyl, CF₃), (M-701, H, H, F, piperidin-4-yl-methyl, Br), (M-702, H, H, F, piperidin-4-yl-methyl, CH₃), (M-703, H, H, F, cyclohexylmethyl, H), (M-704, H, H, F, cyclohexylmethyl, Cl), (M-705, H, H, F, cyclohexylmethyl, F), (M-706, H, H, F, cyclohexylmethyl, CF₃), (M-707, H, H, F, cyclohexylmethyl, Br), (M-708, H, H, F, cyclohexylmethyl, CH₃), (M-709, H, H, Cl, H, H), (M-710, H, H, Cl, H, Cl), (M-711, H, H, Cl, H, F), (M-712, H, H, Cl, H, CF₃), (M-713, H, H, Cl, H, Br), (M-714, H, H, Cl, H, CH₃), (M-715, H, H, Cl, F, H), (M-716, H, H, Cl, F, Cl), (M-717, H, H, Cl, F, F), (M-718, H, H, Cl, F, CF₃), (M-719, H, H, Cl, F, Br), (M-720, H, H, Cl, F, CH₃), (M-721, H, H, Cl, Cl, H), (M-722, H, H, Cl, Cl, Cl), (M-723, H, H, Cl, Cl, F), (M-724, H, H, Cl, Cl, CF₃), (M-725, H, H, Cl, Cl, Br), (M-726, H, H, Cl, Cl, CH₃), (M-727, H, H, Cl, CH₃, H), (M-728, H, H, Cl, CH₃, Cl), (M-729, H, H, Cl, CH₃, F), (M-730, H, H, Cl, CH₃, CF₃), (M-731, H, H, Cl, CH₃, Br), (M-732, H, H, Cl, CH₃, CH₃), (M-733, H, H, Cl, Et, H), (M-734, H, H, Cl, Et, Cl), (M-735, H, H, Cl, Et, F), (M-736, H, H, Cl, Et, CF₃), (M-737, H, H, Cl, Et, Br), (M-738, H, H, Cl, Et, CH₃), (M-739, H, H, Cl, n-Pr, H), (M-740, H, H, Cl, n-Pr, Cl), (M-741, H, H, Cl, n-Pr, F), (M-742, H, H, Cl, n-Pr, CF₃), (M-743, H, H, Cl, n-Pr, Br), (M-744, H, H, Cl, n-Pr, CH₃), (M-745, H, H, Cl, c-Pr, H), (M-746, H, H, Cl, c-Pr, Cl), (M-747, H, H, Cl, c-Pr, F), (M-748, H, H, Cl, c-Pr, CF₃), (M-749, H, H, Cl, c-Pr, Br), (M-750, H, H, Cl, c-Pr, CH₃), (M-751, H, H, Cl, i-Pr, H), (M-752, H, H, Cl, i-Pr, Cl), (M-753, H, H, Cl, i-Pr, F), (M-754, H, H, Cl, i-Pr, CF₃), (M-755, H, H, Cl, i-Pr, Br), (M-756, H, H, Cl, i-Pr, CH₃), (M-757, H, H, Cl, n-Bu, H), (M-758, H, H, Cl, n-Bu, Cl), (M-759, H, H, Cl, n-Bu, F), (M-760, H, H, Cl, n-Bu, CF₃), (M-761, H, H, Cl, n-Bu, Br), (M-762, H, H, Cl, n-Bu, CH₃), (M-763, H, H, Cl, i-Bu, H), (M-764, H, H, Cl, i-Bu, Cl), (M-765, H, H, Cl, i-Bu, F), (M-766, H, H, Cl, i-Bu, CF₃), (M-767, H, H, Cl, i-Bu, Br), (M-768, H, H, Cl, i-Bu, CH₃), (M-769, H, H, Cl, sec-Bu, H), (M-770, H, H, Cl, sec-Bu, Cl), (M-771, H, H, Cl, sec-Bu, F), (M-772, H, H, Cl, sec-Bu, CF₃), (M-773, H, H, Cl, sec-Bu, Br), (M-774, H, H, Cl, sec-Bu, CH₃), (M-775, H, H, Cl, n-Pen, H), (M-776, H, H, Cl, n-Pen, Cl), (M-777, H, H, Cl, n-Pen, F), (M-778, H, H, Cl, n-Pen, CF₃), (M-779, H, H, Cl, n-Pen, Br), (M-780, H, H, Cl, n-Pen, CH₃), (M-781, H, H, Cl, c-Pen, H), (M-782, H, H, Cl, c-Pen, Cl), (M-783, H, H, Cl, c-Pen, F), (M-784, H, H, Cl, c-Pen, CF₃), (M-785, H, H, Cl, c-Pen, Br), (M-786, H, H, Cl, c-Pen, CH₃), (M-787, H, H, Cl, n-Hex, H), (M-788, H, H, Cl, n-Hex, Cl), (M-789, H, H, Cl, n-Hex, F), (M-790, H, H, Cl, n-Hex, CF₃), (M-791, H, H, Cl, n-Hex, Br), (M-792, H, H, Cl, n-Hex, CH₃), (M-793, H, H, Cl, c-Hex, H), (M-794, H, H, Cl, c-Hex, Cl), (M-795, H, H, Cl, c-Hex, F), (M-796, H, H, Cl, c-Hex, CF₃), (M-797, H, H, Cl, c-Hex, Br), (M-798, H, H, Cl, c-Hex, CH₃), (M-799, H, H, Cl, OH, H), (M-800, H, H, Cl, OH, Cl), (M-801, H, H, Cl, OH, F), (M-802, H, H, Cl, OH, CF₃), (M-803, H, H, Cl, OH, Br), (M-804, H, H, Cl, OH, CH₃), (M-805, H, H, Cl, EtO, H), (M-806, H, H, Cl, EtO, Cl), (M-807, H, H, Cl, EtO, F), (M-808, H, H, Cl, EtO, CF₃), (M-809, H, H, Cl, EtO, Br), (M-810, H, H, Cl, EtO, CH₃), (M-811, H, H, Cl, n-PrO, H), (M-812, H, H, Cl, n-PrO, Cl), (M-813, H, H, Cl, n-PrO, F), (M-814, H, H, Cl, n-PrO, CF₃), (M-815, H, H, Cl, n-PrO, Br), (M-816, H, H, Cl, n-PrO, CH₃), (M-817, H, H, Cl, PhO, H), (M-818, H, H, Cl, PhO, Cl), (M-819, H, H, Cl, PhO, F), (M-820, H, H, Cl, PhO, CF₃), (M-821, H, H, Cl, PhO, Br), (M-822, H, H, Cl, PhO, CH₃), (M-823, H, H, Cl, BnO, H), (M-824, H, H, Cl, BnO, Cl), (M-825, H, H, Cl, BnO, F), (M-826, H, H, Cl, BnO, CF₃), (M-827, H, H, Cl, BnO, Br), (M-828, H, H, Cl, BnO, CH₃), (M-829, H, H, Cl, PhCH₂CH₂O, H), (M-830, H, H, Cl, PhCH₂CH₂O, Cl), (M-831, H, H, Cl, PhCH₂CH₂O, F), (M-832, H, H, Cl, PhCH₂CH₂O, CF₃), (M-833, H, H, Cl, PhCH₂CH₂O, Br), (M-834, H, H, Cl, PhCH₂CH₂O, CH₃), (M-835, H, H, Cl, CF₃O, H), (M-836, H, H, Cl, CF₃O, Cl), (M-837, H, H, Cl, CF₃O, F), (M-838, H, H, Cl, CF₃O, CF₃), (M-839, H, H, Cl, CF₃O, Br), (M-840, H, H, Cl, CF₃O, CH₃), (M-841, H, H, Cl, Ph, H), (M-842, H, H, Cl, Ph, Cl), (M-843, H, H, Cl, Ph, F), (M-844, H, H, Cl, Ph, CF₃), (M-845, H, H, Cl, Ph, Br), (M-846, H, H, Cl, Ph, CH₃), (M-847, H, H, Cl, 4-F-Ph, H), (M-848, H, H, Cl, 4-F-Ph, Cl), (M-849, H, H, Cl, 4-F-Ph, F), (M-850, H, H, Cl, 4-F-Ph, CF₃), (M-851, H, H, Cl, 4-F-Ph, Br), (M-852, H, H, Cl, 4-F-Ph, CH₃), (M-853, H, H, Cl, 4-CF₃-Ph, H), (M-854, H, H, Cl, 4-CF₃-Ph, Cl), (M-855, H, H, Cl, 4-CF₃-Ph, F), (M-856, H, H, Cl, 4-CF₃-Ph, CF₃), (M-857, H, H, Cl, 4-CF₃-Ph, Br), (M-858, H, H, Cl, 4-CF₃-Ph, CH₃), (M-859, H, H, Cl, 4-(Me)₂N-Ph, H), (M-860, H, H, Cl, 4-(Me)₂N-Ph, Cl), (M-861, H, H, Cl, 4-(Me)₂N-Ph, F), (M-862, H, H, Cl, 4-(Me)₂N-Ph, CF₃), (M-863, H, H, Cl, 4-(Me)₂N-Ph, Br), (M-864, H, H, Cl, 4-(Me)₂N-Ph, CH₃), (M-865, H, H, Cl, 4-OH-Ph, H), (M-866, H, H, Cl, 4-OH-Ph, Cl), (M-867, H, H, Cl, 4-OH-Ph, F), (M-868, H, H, Cl, 4-OH-Ph, CF₃), (M-869, H, H, Cl, 4-OH-Ph, Br), (M-870, H, H, Cl, 4-OH-Ph, CH₃), (M-871, H, H, Cl, 3,4-di-F-Ph, H), (M-872, H, H, Cl, 3,4-di-F-Ph, Cl), (M-873, H, H, Cl, 3,4-di-F-Ph, F), (M-874, H, H, Cl, 3,4-di-F-Ph, CF₃), (M-875, H, H, Cl, 3,4-di-F-Ph, Br), (M-876, H, H, Cl, 3,4-di-F-Ph, CH₃), (M-877, H, H, Cl, 4-COOH-Ph, H), (M-878, H, H, Cl, 4-COOH-Ph, Cl), (M-879, H, H, Cl, 4-COOH-Ph, F), (M-880, H, H, Cl, 4-COOH-Ph, CF₃), (M-881, H, H, Cl, 4-COOH-Ph, Br), (M-882, H, H, Cl, 4-COOH-Ph, CH₃), (M-883, H, H, Cl, Bn, H), (M-884, H, H, Cl, Bn, Cl), (M-885, H, H, Cl, Bn, F), (M-886, H, H, Cl, Bn, CF₃), (M-887, H, H, Cl, Bn, Br), (M-888, H, H, Cl, Bn, CH₃), (M-889, H, H, Cl, 4-F-Bn, H), (M-890, H, H, Cl, 4-F-Bn, Cl), (M-891, H, H, Cl, 4-F-Bn, F), (M-892, H, H, Cl, 4-F-Bn, CF₃), (M-893, H, H, Cl, 4-F-Bn, Br), (M-894, H, H, Cl, 4-F-Bn, CH₃), (M-895, H, H, Cl, 2-Py, H), (M-896, H, H, Cl, 2-Py, Cl), (M-897, H, H, Cl, 2-Py, F), (M-898, H, H, Cl, 2-Py, CF₃), (M-899, H, H, Cl, 2-Py, Br), (M-900, H, H, Cl, 2-Py, CH₃), (M-901, H, H, Cl, 3-Py, H), (M-902, H, H, Cl, 3-Py, Cl), (M-903, H, H, Cl, 3-Py, F), (M-904, H, H, Cl, 3-Py, CF₃), (M-905, H, H, Cl, 3-Py, Br), (M-906, H, H, Cl, 3-Py, CH₃), (M-907, H, H, Cl, 4-Py, H), (M-908, H, H, Cl, 4-Py, Cl), (M-909, H, H, Cl, 4-Py, F), (M-910, H, H, Cl, 4-Py, CF₃), (M-911, H, H, Cl, 4-Py, Br), (M-912, H, H, Cl, 4-Py, CH₃), (M-913, H, H, Cl, 2-Th, H), (M-914, H, H, Cl, 2-Th, Cl), (M-915, H, H, Cl, 2-Th, F), (M-916, H, H, Cl, 2-Th, CF₃), (M-917, H, H, Cl, 2-Th, Br), (M-918, H, H, Cl, 2-Th, CH₃), (M-919, H, H, Cl, 3-Th, H), (M-920, H, H, Cl, 3-Th, Cl), (M-921, H, H, Cl, 3-Th, F), (M-922, H, H, Cl, 3-Th, CF₃), (M-923, H, H, Cl, 3-Th, Br), (M-924, H, H, Cl, 3-Th, CH₃), (M-925, H, H, Cl, pyrazol-2-yl, H), (M-926, H, H, Cl, pyrazol-2-yl, Cl), (M-927, H, H, Cl, pyrazol-2-yl, F), (M-928, H, H, Cl, pyrazol-2-yl, CF₃), (M-929, H, H, Cl, pyrazol-2-yl, Br), (M-930, H, H, Cl, pyrazol-2-yl, CH₃), (M-931, H, H, Cl, pyrazol-3-yl, H), (M-932, H, H, Cl, pyrazol-3-yl, Cl), (M-933, H, H, Cl, pyrazol-3-yl, F), (M-934, H, H, Cl, pyrazol-3-yl, CF₃), (M-935, H, H, Cl, pyrazol-3-yl, Br), (M-936, H, H, Cl, pyrazol-3-yl, CH₃), (M-937, H, H, Cl, pyrimidin-2-yl, H), (M-938, H, H, Cl, pyrimidin-2-yl, Cl), (M-939, H, H, Cl, pyrimidin-2-yl, F), (M-940, H, H, Cl, pyrimidin-2-yl, CF₃), (M-941, H, H, Cl, pyrimidin-2-yl, Br), (M-942, H, H, Cl, pyrimidin-2-yl, CH₃), (M-943, H, H, Cl, pyrimidin-4-yl, H), (M-944, H, H, Cl, pyrimidin-4-yl, Cl), (M-945, H, H, Cl, pyrimidin-4-yl, F), (M-946, H, H, Cl, pyrimidin-4-yl, CF₃), (M-947, H, H, Cl, pyrimidin-4-yl, Br), (M-948, H, H, Cl, pyrimidin-4-yl, CH₃), (M-949, H, H, Cl, pyrimidin-5-yl, H), (M-950, H, H, Cl, pyrimidin-5-yl, Cl), (M-951, H, H, Cl, pyrimidin-5-yl, F), (M-952, H,
H, Cl, pyrimidin-5-yl, CF₃), (M-953, H, H, Cl, pyrimidin-5-yl, Br), (M-954, H, H, Cl, pyrimidin-5-yl, CH₃), (M-955, H, H, Cl, HOOCCH₂CH₂CH₂, H), (M-956, H, H, Cl, HOOCCH₂CH₂CH₂, Cl), (M-957, H, H, Cl, HOOCCH₂CH₂CH₂, F), (M-958, H, H, Cl, HOOCCH₂CH₂CH₂, CF₃), (M-959, H, H, Cl, HOOCCH₂CH₂CH₂, Br), (M-960, H, H, Cl, HOOCCH₂CH₂CH₂, CH₃), (M-961, H, H, Cl, HOOCCH₂CH₂CH₂CH₂, H), (M-962, H, H, Cl, HOOCCH₂CH₂CH₂CH₂, Cl), (M-963, H, H, Cl, HOOCCH₂CH₂CH₂CH₂, F), (M-964, H, H, Cl, HOOCCH₂CH₂CH₂CH₂, CF₃), (M-965, H, H, Cl, HOOCCH₂CH₂CH₂CH₂, Br), (M-966, H, H, Cl, HOOCCH₂CH₂CH₂CH₂, CH₃), (M-967, H, H, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂, H), (M-968, H, H, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂, Cl), (M-969, H, H, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂, F), (M-970, H, H, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂, CF₃), (M-971, H, H, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂, Br), (M-972, H, H, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂, CH₃), (M-973, H, H, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, H), (M-974, H, H, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, Cl), (M-975, H, H, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, F), (M-976, H, H, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, CF₃), (M-977, H, H, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, Br), (M-978, H, H, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, CH₃), (M-979, H, H, Cl, MeOCH₂, H), (M-980, H, H, Cl, MeOCH₂, Cl), (M-981, H, H, Cl, MeOCH₂, F), (M-982, H, H, Cl, MeOCH₂, CF₃), (M-983, H, H, Cl, MeOCH₂, Br), (M-984, H, H, Cl, MeOCH₂, CH₃), (M-985, H, H, Cl, EtOCH₂, H), (M-986, H, H, Cl, EtOCH₂, Cl), (M-987, H, H, Cl, EtOCH₂, F), (M-988, H, H, Cl, EtOCH₂, CF₃), (M-989, H, H, Cl, EtOCH₂, Br), (M-990, H, H, Cl, EtOCH₂, CH₃), (M-991, H, H, Cl, EtOCH₂CH₂, H), (M-992, H, H, Cl, EtOCH₂CH₂, Cl), (M-993, H, H, Cl, EtOCH₂CH₂, F), (M-994, H, H, Cl, EtOCH₂CH₂, CF₃), (M-995, H, H, Cl, EtOCH₂CH₂, Br), (M-996, H, H, Cl, EtOCH₂CH₂, CH₃), (M-997, H, H, Cl, MeOCH₂CH₂OCH₂CH₂, H), (M-998, H, H, Cl, MeOCH₂CH₂OCH₂CH₂, Cl), (M-999, H, H, Cl, MeOCH₂CH₂OCH₂CH₂, F), (M-1000, H, H, Cl, MeOCH₂CH₂OCH₂CH₂, CF₃), (M-1001, H, H, Cl, MeOCH₂CH₂OCH₂CH₂, Br), (M-1002, H, H, Cl, MeOCH₂CH₂OCH₂CH₂, CH₃), (M-1003, H, H, Cl, MeOCH₂CH₂, H), (M-1004, H, H, Cl, MeOCH₂CH₂, Cl), (M-1005, H, H, Cl, MeOCH₂CH₂, F), (M-1006, H, H, Cl, MeOCH₂CH₂, CF₃), (M-1007, H, H, Cl, MeOCH₂CH₂, Br), (M-1008, H, H, Cl, MeOCH₂CH₂, CH₃), (M-1009, H, H, Cl, HOCH₂, H), (M-1010, H, H, Cl, HOCH₂, Cl), (M-1011, H, H, Cl, HOCH₂, F), (M-1012, H, H, Cl, HOCH₂, CF₃), (M-1013, H, H, Cl, HOCH₂, Br), (M-1014, H, H, Cl, HOCH₂, CH₃), (M-1015, H, H, Cl, HOCH₂CH₂, H), (M-1016, H, H, Cl, HOCH₂CH₂, Cl), (M-1017, H, H, Cl, HOCH₂CH₂, F), (M-1018, H, H, Cl, HOCH₂CH₂, CF₃), (M-1019, H, H, Cl, HOCH₂CH₂, Br), (M-1020, H, H, Cl, HOCH₂CH₂, CH₃), (M-1021, H, H, Cl, HOCH₂CH₂CH₂, H), (M-1022, H, H, Cl, HOCH₂CH₂CH₂, Cl), (M-1023, H, H, Cl, HOCH₂CH₂CH₂, F), (M-1024, H, H, Cl, HOCH₂CH₂CH₂, CF₃), (M-1025, H, H, Cl, HOCH₂CH₂CH₂, Br), (M-1026, H, H, Cl, HOCH₂CH₂CH₂, CH₃), (M-1027, H, H, Cl, HOCH₂CH₂CH₂CH₂, H), (M-1028, H, H, Cl, HOCH₂CH₂CH₂CH₂, Cl), (M-1029, H, H, Cl, HOCH₂CH₂CH₂CH₂, F), (M-1030, H, H, Cl, HOCH₂CH₂CH₂CH₂, CF₃), (M-1031, H, H, Cl, HOCH₂CH₂CH₂CH₂, Br), (M-1032, H, H, Cl, HOCH₂CH₂CH₂CH₂, CH₃), (M-1033, H, H, Cl, HOCH₂CH₂CH₂CH₂CH₂, H), (M-1034, H, H, Cl, HOCH₂CH₂CH₂CH₂CH₂, Cl), (M-1035, H, H, Cl, HOCH₂CH₂CH₂CH₂CH₂, F), (M-1036, H, H, Cl, HOCH₂CH₂CH₂CH₂CH₂, CF₃), (M-1037, H, H, Cl, HOCH₂CH₂CH₂CH₂CH₂, Br), (M-1038, H, H, Cl, HOCH₂CH₂CH₂CH₂CH₂, CH₃), (M-1039, H, H, Cl, HOCH₂CH₂OCH₂CH₂, H), (M-1040, H, H, Cl, HOCH₂CH₂OCH₂CH₂, Cl), (M-1041, H, H, Cl, HOCH₂CH₂OCH₂CH₂, F), (M-1042, H, H, Cl, HOCH₂CH₂OCH₂CH₂, CF₃), (M-1043, H, H, Cl, HOCH₂CH₂OCH₂CH₂, Br), (M-1044, H, H, Cl, HOCH₂CH₂OCH₂CH₂, CH₃), (M-1045, H, H, Cl, (Me)₂N, H), (M-1046, H, H, Cl, (Me)₂N, Cl), (M-1047, H, H, Cl, (Me)₂N, F), (M-1048, H, H, Cl, (Me)₂N, CF₃), (M-1049, H, H, Cl, (Me)₂N, Br), (M-1050, H, H, Cl, (Me)₂N, CH₃), (M-1051, H, H, Cl, piperidin-4-yl-methyl, H), (M-1052, H, H, Cl, piperidin-4-yl-methyl, Cl), (M-1053, H, H, Cl, piperidin-4-yl-methyl, F), (M-1054, H, H, Cl, piperidin-4-yl-methyl, CF₃), (M-1055, H, H, Cl, piperidin-4-yl-methyl, Br), (M-1056, H, H, Cl, piperidin-4-yl-methyl, CH₃), (M-1057, H, H, Cl, cyclohexylmethyl, H), (M-1058, H, H, Cl, cyclohexylmethyl, Cl), (M-1059, H, H, Cl, cyclohexylmethyl, F), (M-1060, H, H, Cl, cyclohexylmethyl, CF₃), (M-1061, H, H, Cl, cyclohexylmethyl, Br), (M-1062, H, H, Cl, cyclohexylmethyl, CH₃), (M-1063, H, F, H, H, H), (M-1064, H, F, H, H, Cl), (M-1065, H, F, H, H, F), (M-1066, H, F, H, H, CF₃), (M-1067, H, F, H, H, Br), (M-1068, H, F, H, H, CH₃), (M-1069, H, F, H, F, H), (M-1070, H, F, H, F, Cl), (M-1071, H, F, H, F, F), (M-1072, H, F, H, F, CF₃), (M-1073, H, F, H, F, Br), (M-1074, H, F, H, F, CH₃), (M-1075, H, F, H, Cl, H), (M-1076, H, F, H, Cl, Cl), (M-1077, H, F, H, Cl, F), (M-1078, H, F, H, Cl, CF₃), (M-1079, H, F, H, Cl, Br), (M-1080, H, F, H, Cl, CH₃), (M-1081, H, F, H, CH₃, H), (M-1082, H, F, H, CH₃, Cl), (M-1083, H, F, H, CH₃, F), (M-1084, H, F, H, CH₃, CF₃), (M-1085, H, F, H, CH₃, Br), (M-1086, H, F, H, CH₃, CH₃), (M-1087, H, F, H, Et, H), (M-1088, H, F, H, Et, Cl), (M-1089, H, F, H, Et, F), (M-1090, H, F, H, Et, CF₃), (M-1091, H, F, H, Et, Br), (M-1092, H, F, H, Et, CH₃), (M-1093, H, F, H, n-Pr, H), (M-1094, H, F, H, n-Pr, Cl), (M-1095, H, F, H, n-Pr, F), (M-1096, H, F, H, n-Pr, CF₃), (M-1097, H, F, H, n-Pr, Br), (M-1098, H, F, H, n-Pr, CH₃), (M-1099, H, F, H, c-Pr, H), (M-1100, H, F, H, c-Pr, Cl), (M-1101, H, F, H, c-Pr, F), (M-1102, H, F, H, c-Pr, CF₃), (M-1103, H, F, H, c-Pr, Br), (M-1104, H, F, H, c-Pr, CH₃), (M-1105, H, F, H, i-Pr, H), (M-1106, H, F, H, i-Pr, Cl), (M-1107, H, F, H, i-Pr, F), (M-1108, H, F, H, i-Pr, CF₃), (M-1109, H, F, H, i-Pr, Br), (M-1110, H, F, H, i-Pr, CH₃), (M-1111, H, F, H, n-Bu, H), (M-1112, H, F, H, n-Bu, Cl), (M-1113, H, F, H, n-Bu, F), (M-1114, H, F, H, n-Bu, CF₃), (M-1115, H, F, H, n-Bu, Br), (M-1116, H, F, H, n-Bu, CH₃), (M-1117, H, F, H, i-Bu, H), (M-1118, H, F, H, i-Bu, Cl), (M-1119, H, F, H, i-Bu, F), (M-1120, H, F, H, i-Bu, CF₃), (M-1121, H, F, H, i-Bu, Br), (M-1122, H, F, H, i-Bu, CH₃), (M-1123, H, F, H, sec-Bu, H), (M-1124, H, F, H, sec-Bu, Cl), (M-1125, H, F, H, sec-Bu, F), (M-1126, H, F, H, sec-Bu, CF₃), (M-1127, H, F, H, sec-Bu, Br), (M-1128, H, F, H, sec-Bu, CH₃), (M-1129, H, F, H, n-Pen, H), (M-1130, H, F, H, n-Pen, Cl), (M-1131, H, F, H, n-Pen, F), (M-1132, H, F, H, n-Pen, CF₃), (M-1133, H, F, H, n-Pen, Br), (M-1134, H, F, H, n-Pen, CH₃), (M-1135, H, F, H, c-Pen, H)
, (M-1136, H, F, H, c-Pen, Cl), (M-1137, H, F, H, c-Pen, F), (M-1138, H, F, H, c-Pen, CF₃), (M-1139, H, F, H, c-Pen, Br), (M-1140, H, F, H, c-Pen, CH₃), (M-1141, H, F, H, n-Hex, H), (M-1142, H, F, H, n-Hex, Cl), (M-1143, H, F, H, n-Hex, F), (M-1144, H, F, H, n-Hex, CF₃), (M-1145, H, F, H, n-Hex, Br), (M-1146, H, F, H, n-Hex, CH₃), (M-1147, H, F, H, c-Hex, H), (M-1148, H, F, H, c-Hex, Cl), (M-1149, H, F, H, c-Hex, F), (M-1150, H, F, H, c-Hex, CF₃), (M-1151, H, F, H, c-Hex, Br), (M-1152, H, F, H, c-Hex, CH₃), (M-1153, H, F, H, OH, H), (M-1154, H, F, H, OH, Cl), (M-1155, H, F, H, OH, F), (M-1156, H, F, H, OH, CF₃), (M-1157, H, F, H, OH, Br), (M-1158, H, F, H, OH, CH₃), (M-1159, H, F, H, EtO, H), (M-1160, H, F, H, EtO, Cl), (M-1161, H, F, H, EtO, F), (M-1162, H, F, H, EtO, CF₃), (M-1163, H, F, H, EtO, Br), (M-1164, H, F, H, EtO, CH₃), (M-1165, H, F, H, n-PrO, H), (M-1166, H, F, H, n-PrO, Cl), (M-1167, H, F, H, n-PrO, F), (M-1168, H, F, H, n-PrO, CF₃), (M-1169, H, F, H, n-PrO, Br), (M-1170, H, F, H, n-PrO, CH₃), (M-1171, H, F, H, PhO, H), (M-1172, H, F, H, PhO, Cl), (M-1173, H, F, H, PhO, F), (M-1174, H, F, H, PhO, CF₃), (M-1175, H, F, H, PhO, Br), (M-1176, H, F, H, PhO, CH₃), (M-1177, H, F, H, BnO, H), (M-1178, H, F, H, BnO, Cl), (M-1179, H, F, H, BnO, F), (M-1180, H, F, H, BnO, CF₃), (M-1181, H, F, H, BnO, Br), (M-1182, H, F, H, BnO, CH₃), (M-1183, H, F, H, PhCH₂CH₂O, H), (M-1184, H, F, H, PhCH₂CH₂O, Cl), (M-1185, H, F, H, PhCH₂CH₂O, F), (M-1186, H, F, H, PhCH₂CH₂O, CF₃), (M-1187, H, F, H, PhCH₂CH₂O, Br), (M-1188, H, F, H, PhCH₂CH₂O, CH₃), (M-1189, H, F, H, CF₃O, H), (M-1190, H, F, H, CF₃O, Cl), (M-1191, H, F, H, CF₃O, F), (M-1192, H, F, H, CF₃O, CF₃), (M-1193, H, F, H, CF₃O, Br), (M-1194, H, F, H, CF₃O, CH₃), (M-1195, H, F, H, Ph, H), (M-1196, H, F, H, Ph, Cl), (M-1197, H, F, H, Ph, F), (M-1198, H, F, H, Ph, CF₃), (M-1199, H, F, H, Ph, Br), (M-1200, H, F, H, Ph, CH₃), (M-1201, H, F, H, 4-F-Ph, H), (M-1202, H, F, H, 4-F-Ph, Cl), (M-1203, H, F, H, 4-F-Ph, F), (M-1204, H, F, H, 4-F-Ph, CF₃), (M-1205, H, F, H, 4-F-Ph, Br), (M-1206, H, F, H, 4-F-Ph, CH₃), (M-1207, H, F, H, 4-CF₃-Ph, H), (M-1208, H, F, H, 4-CF₃-Ph, Cl), (M-1209, H, F, H, 4-CF₃-Ph, F), (M-1210, H, F, H, 4-CF₃-Ph, CF₃), (M-1211, H, F, H, 4-CF₃-Ph, Br), (M-1212, H, F, H, 4-CF₃-Ph, CH₃), (M-1213, H, F, H, 4-(Me)₂N-Ph, H), (M-1214, H, F, H, 4-(Me)₂N-Ph, Cl), (M-1215, H, F, H, 4-(Me)₂N-Ph, F), (M-1216, H, F, H, 4-(Me)₂N-Ph, CF₃), (M-1217, H, F, H, 4-(Me)₂N-Ph, Br), (M-1218, H, F, H, 4-(Me)₂N-Ph, CH₃), (M-1219, H, F, H, 4-OH-Ph, H), (M-1220, H, F, H, 4-OH-Ph, Cl), (M-1221, H, F, H, 4-OH-Ph, F), (M-1222, H, F, H, 4-OH-Ph, CF₃), (M-1223, H, F, H, 4-OH-Ph, Br), (M-1224, H, F, H, 4-OH-Ph, CH₃), (M-1225, H, F, H, 3,4-di-F-Ph, H), (M-1226, H, F, H, 3,4-di-F-Ph, Cl), (M-1227, H, F, H, 3,4-di-F-Ph, F), (M-1228, H, F, H, 3,4-di-F-Ph, CF₃), (M-1229, H, F, H, 3,4-di-F-Ph, Br), (M-1230, H, F, H, 3,4-di-F-Ph, CH₃), (M-1231, H, F, H, 4-COOH-Ph, H), (M-1232, H, F, H, 4-COOH-Ph, Cl), (M-1233, H, F, H, 4-COOH-Ph, F), (M-1234, H, F, H, 4-COOH-Ph, CF₃), (M-1235, H, F, H, 4-COOH-Ph, Br), (M-1236, H, F, H, 4-COOH-Ph, CH₃), (M-1237, H, F, H, Bn, H), (M-1238, H, F, H, Bn, Cl), (M-1239, H, F, H, Bn, F), (M-1240, H, F, H, Bn, CF₃), (M-1241, H, F, H, Bn, Br), (M-1242, H, F, H, Bn, CH₃), (M-1243, H, F, H, 4-F-Bn, H), (M-1244, H, F, H, 4-F-Bn, Cl), (M-1245, H, F, H, 4-F-Bn, F), (M-1246, H, F, H, 4-F-Bn, CF₃), (M-1247, H, F, H, 4-F-Bn, Br), (M-1248, H, F, H, 4-F-Bn, CH₃), (M-1249, H, F, H, 2-Py, H), (M-1250, H, F, H, 2-Py, Cl), (M-1251, H, F, H, 2-Py, F), (M-1252, H, F, H, 2-Py, CF₃), (M-1253, H, F, H, 2-Py, Br), (M-1254, H, F, H, 2-Py, CH₃), (M-1255, H, F, H, 3-Py, H), (M-1256, H, F, H, 3-Py, Cl), (M-1257, H, F, H, 3-Py, F), (M-1258, H, F, H, 3-Py, CF₃), (M-1259, H, F, H, 3-Py, Br), (M-1260, H, F, H, 3-Py, CH₃), (M-1261, H, F, H, 4-Py, H), (M-1262, H, F, H, 4-Py, Cl), (M-1263, H, F, H, 4-Py, F), (M-1264, H, F, H, 4-Py, CF₃), (M-1265, H, F, H, 4-Py, Br), (M-1266, H, F, H, 4-Py, CH₃), (M-1267, H, F, H, 2-Th, H), (M-1268, H, F, H, 2-Th, Cl), (M-1269, H, F, H, 2-Th, F), (M-1270, H, F, H, 2-Th, CF₃), (M-1271, H, F, H, 2-Th, Br), (M-1272, H, F, H, 2-Th, CH₃), (M-1273, H, F, H, 3-Th, H), (M-1274, H, F, H, 3-Th, Cl), (M-1275, H, F, H, 3-Th, F), (M-1276, H, F, H, 3-Th, CF₃), (M-1277, H, F, H, 3-Th, Br), (M-1278, H, F, H, 3-Th, CH₃), (M-1279, H, F, H, pyrazol-2-yl, H), (M-1280, H, F, H, pyrazol-2-yl, Cl), (M-1281, H, F, H, pyrazol-2-yl, F), (M-1282, H, F, H, pyrazol-2-yl, CF₃), (M-1283, H, F, H, pyrazol-2-yl, Br), (M-1284, H, F, H, pyrazol-2-yl, CH₃), (M-1285, H, F, H, pyrazol-3-yl, H), (M-1286, H, F, H, pyrazol-3-yl, Cl), (M-1287, H, F, H, pyrazol-3-yl, F), (M-1288, H, F, H, pyrazol-3-yl, CF₃), (M-1289, H, F, H, pyrazol-3-yl, Br), (M-1290, H, F, H, pyrazol-3-yl, CH₃), (M-1291, H, F, H, pyrimidin-2-yl, H), (M-1292, H, F, H, pyrimidin-2-yl, Cl), (M-1293, H, F, H, pyrimidin-2-yl, F), (M-1294, H, F, H, pyrimidin-2-yl, CF₃), (M-1295, H, F, H, pyrimidin-2-yl, Br), (M-1296, H, F, H, pyrimidin-2-yl, CH₃), (M-1297, H, F, H, pyrimidin-4-yl, H), (M-1298, H, F, H, pyrimidin-4-yl, Cl), (M-1299, H, F, H, pyrimidin-4-yl, F), (M-1300, H, F, H, pyrimidin-4-yl, CF₃), (M-1301, H, F, H, pyrimidin-4-yl, Br), (M-1302, H, F, H, pyrimidin-4-yl, CH₃), (M-1303, H, F, H, pyrimidin-5-yl, H), (M-1304, H, F, H, pyrimidin-5-yl, Cl), (M-1305, H, F, H, pyrimidin-5-yl, F), (M-1306, H, F, H, pyrimidin-5-yl, CF₃), (M-1307, H, F, H, pyrimidin-5-yl, Br), (M-1308, H, F, H, pyrimidin-5-yl, CH₃), (M-1309, H, F, H, HOOCCH₂CH₂CH₂, H), (M-1310, H, F, H, HOOCCH₂CH₂CH₂, Cl), (M-1311, H, F, H, HOOCCH₂CH₂CH₂, F), (M-1312, H, F, H, HOOCCH₂CH₂CH₂, CF₃), (M-1313, H, F, H, HOOCCH₂CH₂CH₂, Br), (M-1314, H, F, H, HOOCCH₂CH₂CH₂, CH₃), (M-1315, H, F, H, HOOCCH₂CH₂CH₂CH₂, H), (M-1316, H, F, H, HOOCCH₂CH₂CH₂CH₂, Cl), (M-1317, H, F, H, HOOCCH₂CH₂CH₂CH₂, F), (M-1318, H, F, H, HOOCCH₂CH₂CH₂CH₂, CF₃), (M-1319, H, F, H, HOOCCH₂CH₂CH₂CH₂, Br), (M-1320, H, F, H, HOOCCH₂CH₂CH₂CH₂, CH₃), (M-1321, H, F, H, (Me)₂NCOCH₂CH₂CH₂CH₂, H), (M-1322, H, F, H, (Me)₂NCOCH₂CH₂CH₂CH₂, Cl), (M-1323, H, F, H, (Me)₂NCOCH₂CH₂CH₂CH₂, F), (M-1324, H, F, H, (Me)₂NCOCH₂CH₂CH₂CH₂, CF₃), (M-1325, H, F, H, (Me)₂NCOCH₂CH₂CH₂CH₂, Br), (M-1326, H, F, H, (Me)₂NCOCH₂CH₂CH₂CH₂, CH₃), (M-1327, H, F, H, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, H), (M-1328, H, F, H, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, Cl), (M-1329, H, F, H, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, F), (M-1330, H, F, H, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, CF₃), (M-1331, H, F, H, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, Br), (M-1332, H, F, H, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, CH₃), (M-1333, H, F, H, MeOCH₂, H), (M-1334, H, F, H, MeOCH₂, Cl), (M-1335, H, F, H, MeOCH₂, F), (M-1336, H, F, H, MeOCH₂, CF₃), (M-1337, H, F, H, MeOCH₂, Br), (M-1338, H, F, H, MeOCH₂, CH₃), (M-1339, H, F, H, EtOCH₂, H), (M-1340, H, F, H, EtOCH₂, Cl), (M-1341, H, F, H, EtOCH₂, F), (M-1342, H, F, H, EtOCH₂, CF₃), (M-1343, H, F, H, EtOCH₂, Br), (M-1344, H, F, H, EtOCH₂, CH₃), (M-1345, H, F, H, EtOCH₂CH₂, H), (M-1346, H, F, H, EtOCH₂CH₂, Cl), (M-1347, H, F, H, EtOCH₂CH₂, F), (M-1348, H, F, H, EtOCH₂CH₂, CF₃), (M-1349, H, F, H, EtOCH₂CH₂, Br), (M-1350, H, F, H, EtOCH₂CH₂, CH₃), (M-1351, H, F, H, MeOCH₂CH₂OCH₂CH₂, H), (M-1352, H, F, H, MeOCH₂CH₂OCH₂CH₂, Cl), (M-1353, H, F, H, MeOCH₂CH₂OCH₂CH₂, F), (M-1354, H, F, H, MeOCH₂CH₂OCH₂CH₂, CF₃), (M-1355, H, F, H, MeOCH₂CH₂OCH₂CH₂, Br), (M-1356, H, F, H, MeOCH₂CH₂OCH₂CH₂, CH₃), (M-1357, H, F, H, MeOCH₂CH₂, H
), (M-1358, H, F, H, MeOCH₂CH₂, Cl), (M-1359, H, F, H, MeOCH₂CH₂, F), (M-1360, H, F, H, MeOCH₂CH₂, CF₃), (M-1361, H, F, H, MeOCH₂CH₂, Br), (M-1362, H, F, H, MeOCH₂CH₂, CH₃), (M-1363, H, F, H, HOCH₂, H), (M-1364, H, F, H, HOCH₂, Cl), (M-1365, H, F, H, HOCH₂, F), (M-1366, H, F, H, HOCH₂, CF₃), (M-1367, H, F, H, HOCH₂, Br), (M-1368, H, F, H, HOCH₂, CH₃), (M-1369, H, F, H, HOCH₂CH₂, H), (M-1370, H, F, H, HOCH₂CH₂, Cl), (M-1371, H, F, H, HOCH₂CH₂, F), (M-1372, H, F, H, HOCH₂CH₂, CF₃), (M-1373, H, F, H, HOCH₂CH₂, Br), (M-1374, H, F, H, HOCH₂CH₂, CH₃), (M-1375, H, F, H, HOCH₂CH₂CH₂, H), (M-1376, H, F, H, HOCH₂CH₂CH₂, Cl), (M-1377, H, F, H, HOCH₂CH₂CH₂, F), (M-1378, H, F, H, HOCH₂CH₂CH₂, CF₃), (M-1379, H, F, H, HOCH₂CH₂CH₂, Br), (M-1380, H, F, H, HOCH₂CH₂CH₂, CH₃), (M-1381, H, F, H, HOCH₂CH₂CH₂CH₂, H), (M-1382, H, F, H, HOCH₂CH₂CH₂CH₂, Cl), (M-1383, H, F, H, HOCH₂CH₂CH₂CH₂, F), (M-1384, H, F, H, HOCH₂CH₂CH₂CH₂, CF₃), (M-1385, H, F, H, HOCH₂CH₂CH₂CH₂, Br), (M-1386, H, F, H, HOCH₂CH₂CH₂CH₂, CH₃), (M-1387, H, F, H, HOCH₂CH₂CH₂CH₂CH₂, H), (M-1388, H, F, H, HOCH₂CH₂CH₂CH₂CH₂, Cl), (M-1389, H, F, H, HOCH₂CH₂CH₂CH₂CH₂, F), (M-1390, H, F, H, HOCH₂CH₂CH₂CH₂CH₂, CF₃), (M-1391, H, F, H, HOCH₂CH₂CH₂CH₂CH₂, Br), (M-1392, H, F, H, HOCH₂CH₂CH₂CH₂CH₂, CH₃), (M-1393, H, F, H, HOCH₂CH₂OCH₂CH₂, H), (M-1394, H, F, H, HOCH₂CH₂OCH₂CH₂, Cl), (M-1395, H, F, H, HOCH₂CH₂OCH₂CH₂, F), (M-1396, H, F, H, HOCH₂CH₂OCH₂CH₂, CF₃), (M-1397, H, F, H, HOCH₂CH₂OCH₂CH₂, Br), (M-1398, H, F, H, HOCH₂CH₂OCH₂CH₂, CH₃), (M-1399, H, F, H, (Me)₂N, H), (M-1400, H, F, H, (Me)₂N, Cl), (M-1401, H, F, H, (Me)₂N, F), (M-1402, H, F, H, (Me)₂N, CF₃), (M-1403, H, F, H, (Me)₂N, Br), (M-1404, H, F, H, (Me)₂N, CH₃), (M-1405, H, F, H, piperidin-4-yl-methyl, H), (M-1406, H, F, H, piperidin-4-yl-methyl, Cl), (M-1407, H, F, H, piperidin-4-yl-methyl, F), (M-1408, H, F, H, piperidin-4-yl-methyl, CF₃), (M-1409, H, F, H, piperidin-4-yl-methyl, Br), (M-1410, H, F, H, piperidin-4-yl-methyl, CH₃), (M-1411, H, F, H, cyclohexylmethyl, H), (M-1412, H, F, H, cyclohexylmethyl, Cl), (M-1413, H, F, H, cyclohexylmethyl, F), (M-1414, H, F, H, cyclohexylmethyl, CF₃), (M-1415, H, F, H, cyclohexylmethyl, Br), (M-1416, H, F, H, cyclohexylmethyl, CH₃), (M-1417, H, F, F, H, H), (M-1418, H, F, F, H, Cl), (M-1419, H, F, F, H, F), (M-1420, H, F, F, H, CF₃), (M-1421, H, F, F, H, Br), (M-1422, H, F, F, H, CH₃), (M-1423, H, F, F, F, H), (M-1424, H, F, F, F, Cl), (M-1425, H, F, F, F, F), (M-1426, H, F, F, F, CF₃), (M-1427, H, F, F, F, Br), (M-1428, H, F, F, F, CH₃), (M-1429, H, F, F, Cl, H), (M-1430, H, F, F, Cl, Cl), (M-1431, H, F, F, Cl, F), (M-1432, H, F, F, Cl, CF₃), (M-1433, H, F, F, Cl, Br), (M-1434, H, F, F, Cl, CH₃), (M-1435, H, F, F, CH₃, H), (M-1436, H, F, F, CH₃, Cl), (M-1437, H, F, F, CH₃, F), (M-1438, H, F, F, CH₃, CF₃), (M-1439, H, F, F, CH₃, Br), (M-1440, H, F, F, CH₃, CH₃), (M-1441, H, F, F, Et, H), (M-1442, H, F, F, Et, Cl), (M-1443, H, F, F, Et, F), (M-1444, H, F, F, Et, CF₃), (M-1445, H, F, F, Et, Br), (M-1446, H, F, F, Et, CH₃), (M-1447, H, F, F, n-Pr, H), (M-1448, H, F, F, n-Pr, Cl), (M-1449, H, F, F, n-Pr, F), (M-1450, H, F, F, n-Pr, CF₃), (M-1451, H, F, F, n-Pr, Br), (M-1452, H, F, F, n-Pr, CH₃), (M-1453, H, F, F, c-Pr, H), (M-1454, H, F, F, c-Pr, Cl), (M-1455, H, F, F, c-Pr, F), (M-1456, H, F, F, c-Pr, CF₃), (M-1457, H, F, F, c-Pr, Br), (M-1458, H, F, F, c-Pr, CH₃), (M-1459, H, F, F, i-Pr, H), (M-1460, H, F, F, i-Pr, Cl), (M-1461, H, F, F, i-Pr, F), (M-1462, H, F, F, i-Pr, CF₃), (M-1463, H, F, F, i-Pr, Br), (M-1464, H, F, F, i-Pr, CH₃), (M-1465, H, F, F, n-Bu, H), (M-1466, H, F, F, n-Bu, Cl), (M-1467, H, F, F, n-Bu, F), (M-1468, H, F, F, n-Bu, CF₃), (M-1469, H, F, F, n-Bu, Br), (M-1470, H, F, F, n-Bu, CH₃), (M-1471, H, F, F, i-Bu, H), (M-1472, H, F, F, i-Bu, Cl), (M-1473, H, F, F, i-Bu, F), (M-1474, H, F, F, i-Bu, CF₃), (M-1475, H, F, F, i-Bu, Br), (M-1476, H, F, F, i-Bu, CH₃), (M-1477, H, F, F, sec-Bu, H), (M-1478, H, F, F, sec-Bu, Cl), (M-1479, H, F, F, sec-Bu, F), (M-1480, H, F, F, sec-Bu, CF₃), (M-1481, H, F, F, sec-Bu, Br), (M-1482, H, F, F, sec-Bu, CH₃), (M-1483, H, F, F, n-Pen, H), (M-1484, H, F, F, n-Pen, Cl), (M-1485, H, F, F, n-Pen, F), (M-1486, H, F, F, n-Pen, CF₃), (M-1487, H, F, F, n-Pen, Br), (M-1488, H, F, F, n-Pen, CH₃), (M-1489, H, F, F, c-Pen, H), (M-1490, H, F, F, c-Pen, Cl), (M-1491, H, F, F, c-Pen, F), (M-1492, H, F, F, c-Pen, CF₃), (M-1493, H, F, F, c-Pen, Br), (M-1494, H, F, F, c-Pen, CH₃), (M-1495, H, F, F, n-Hex, H), (M-1496, H, F, F, n-Hex, Cl), (M-1497, H, F, F, n-Hex, F), (M-1498, H, F, F, n-Hex, CF₃), (M-1499, H, F, F, n-Hex, Br), (M-1500, H, F, F, n-Hex, CH₃), (M-1501, H, F, F, c-Hex, H), (M-1502, H, F, F, c-Hex, Cl), (M-1503, H, F, F, c-Hex, F), (M-1504, H, F, F, c-Hex, CF₃), (M-1505, H, F, F, c-Hex, Br), (M-1506, H, F, F, c-Hex, CH₃), (M-1507, H, F, F, OH, H), (M-1508, H, F, F, OH, Cl), (M-1509, H, F, F, OH, F), (M-1510, H, F, F, OH, CF₃), (M-1511, H, F, F, OH, Br), (M-1512, H, F, F, OH, CH₃), (M-1513, H, F, F, EtO, H), (M-1514, H, F, F, EtO, Cl), (M-1515, H, F, F, EtO, F), (M-1516, H, F, F, EtO, CF₃), (M-1517, H, F, F, EtO, Br), (M-1518, H, F, F, EtO, CH₃), (M-1519, H, F, F, n-PrO, H), (M-1520, H, F, F, n-PrO, Cl), (M-1521, H, F, F, n-PrO, F), (M-1522, H, F, F, n-PrO, CF₃), (M-1523, H, F, F, n-PrO, Br), (M-1524, H, F, F, n-PrO, CH₃), (M-1525, H, F, F, PhO, H), (M-1526, H, F, F, PhO, Cl), (M-1527, H, F, F, PhO, F), (M-1528, H, F, F, PhO, CF₃), (M-1529, H, F, F, PhO, Br), (M-1530, H, F, F, PhO, CH₃), (M-1531, H, F, F, BnO, H), (M-1532, H, F, F, BnO, Cl), (M-1533, H, F, F, BnO, F), (M-1534, H, F, F, BnO, CF₃), (M-1535, H, F, F, BnO, Br), (M-1536, H, F, F, BnO, CH₃), (M-1537, H, F, F, PhCH₂CH₂O, H), (M-1538, H, F, F, PhCH₂CH₂O, Cl), (M-1539, H, F, F, PhCH₂CH₂O, F), (M-1540, H, F, F, PhCH₂CH₂O, CF₃), (M-1541, H, F, F, PhCH₂CH₂O, Br), (M-1542, H, F, F, PhCH₂CH₂O, CH₃), (M-1543, H, F, F, CF₃O, H), (M-1544, H, F, F, CF₃O, Cl), (M-1545, H, F, F, CF₃O, F), (M-1546, H, F, F, CF₃O, CF₃), (M-1547, H, F, F, CF₃O, Br), (M-1548, H, F, F, CF₃O, CH₃), (M-1549, H, F, F, Ph, H), (M-1550, H, F, F, Ph, Cl), (M-1551, H, F, F, Ph, F), (M-1552, H, F, F, Ph, CF₃), (M-1553, H, F, F, Ph, Br), (M-1554, H, F, F, Ph, CH₃), (M-1555, H, F, F, 4-F-Ph, H), (M-1556, H, F, F, 4-F-Ph, Cl), (M-1557, H, F, F, 4-F-Ph, F), (M-1558, H, F, F, 4-F-Ph, CF₃), (M-1559, H, F, F, 4-F-Ph, Br), (M-1560, H, F, F, 4-F-Ph, CH₃), (M-1561, H, F, F, 4-CF₃-Ph, H), (M-1562, H, F, F, 4-CF₃-Ph, Cl), (M-1563, H, F, F, 4-CF₃-Ph, F), (M-1564, H, F, F, 4-CF₃-Ph, CF₃), (M-1565, H, F, F, 4-CF₃-Ph, Br), (M-1566, H, F, F, 4-CF₃-Ph, CH₃), (M-1567, H, F, F, 4-(Me)₂N-Ph, H), (M-1568, H, F, F, 4-(Me)₂N-Ph, Cl), (M-1569, H, F, F, 4-(Me)₂N-Ph, F), (M-1570, H, F, F, 4-(Me)₂N-Ph, CF₃), (M-1571, H, F, F, 4-(Me)₂N-Ph, Br), (M-1572, H, F, F, 4-(Me)₂N-Ph, CH₃), (M-1573, H, F, F, 4-OH-Ph, H), (M-1574, H, F, F, 4-OH-Ph, Cl), (M-1575, H, F, F, 4-OH-Ph, F), (M-1576, H, F, F, 4-OH-Ph, CF₃), (M-1577, H, F, F, 4-OH-Ph, Br), (M-1578, H, F, F, 4-OH-Ph, CH₃), (M-1579, H, F, F, 3,4-di-F-Ph, H), (M-1580, H, F, F, 3,4-di-F-Ph, Cl), (M-1581, H, F, F, 3,4-di-F-Ph, F), (M-1582, H, F, F, 3,4-di-F-Ph, CF₃), (M-1583, H, F, F, 3,4-di-F-Ph, Br), (M-1584, H, F, F, 3,4-di-F-Ph, CH₃), (M-1585, H, F, F, 4-COOH-Ph, H), (M-1586, H, F, F, 4-COOH-Ph, Cl), (M-1587, H, F, F, 4-COOH-Ph, F), (M-1588, H, F, F, 4-COOH-Ph, CF₃), (M-1589, H, F, F, 4-COOH-Ph, Br), (M-1590, H, F, F, 4-COOH-Ph, CH₃), (M-1591, H, F, F, Bn, H), (M-1592, H, F, F, Bn, Cl), (M-1593, H, F, F, Bn, F), (M-1594, H, F, F, Bn, CF₃), (M-1595, H, F, F, Bn, Br), (M-1596, H, F, F, Bn, CH₃
), (M-1597, H, F, F, 4-F-Bn, H), (M-1598, H, F, F, 4-F-Bn, Cl), (M-1599, H, F, F, 4-F-Bn, F), (M-1600, H, F, F, 4-F-Bn, CF₃), (M-1601, H, F, F, 4-F-Bn, Br), (M-1602, H, F, F, 4-F-Bn, CH₃), (M-1603, H, F, F, 2-Py, H), (M-1604, H, F, F, 2-Py, Cl), (M-1605, H, F, F, 2-Py, F), (M-1606, H, F, F, 2-Py, CF₃), (M-1607, H, F, F, 2-Py, Br), (M-1608, H, F, F, 2-Py, CH₃), (M-1609, H, F, F, 3-Py, H), (M-1610, H, F, F, 3-Py, Cl), (M-1611, H, F, F, 3-Py, F), (M-1612, H, F, F, 3-Py, CF₃), (M-1613, H, F, F, 3-Py, Br), (M-1614, H, F, F, 3-Py, CH₃), (M-1615, H, F, F, 4-Py, H), (M-1616, H, F, F, 4-Py, Cl), (M-1617, H, F, F, 4-Py, F), (M-1618, H, F, F, 4-Py, CF₃), (M-1619, H, F, F, 4-Py, Br), (M-1620, H, F, F, 4-Py, CH₃), (M-1621, H, F, F, 2-Th, H), (M-1622, H, F, F, 2-Th, Cl), (M-1623, H, F, F, 2-Th, F), (M-1624, H, F, F, 2-Th, CF₃), (M-1625, H, F, F, 2-Th, Br), (M-1626, H, F, F, 2-Th, CH₃), (M-1627, H, F, F, 3-Th, H), (M-1628, H, F, F, 3-Th, Cl), (M-1629, H, F, F, 3-Th, F), (M-1630, H, F, F, 3-Th, CF₃), (M-1631, H, F, F, 3-Th, Br), (M-1632, H, F, F, 3-Th, CH₃), (M-1633, H, F, F, pyrazol-2-yl, H), (M-1634, H, F, F, pyrazol-2-yl, Cl), (M-1635, H, F, F, pyrazol-2-yl, F), (M-1636, H, F, F, pyrazol-2-yl, CF₃), (M-1637, H, F, F, pyrazol-2-yl, Br), (M-1638, H, F, F, pyrazol-2-yl, CH₃), (M-1639, H, F, F, pyrazol-3-yl, H), (M-1640, H, F, F, pyrazol-3-yl, Cl), (M-1641, H, F, F, pyrazol-3-yl, F), (M-1642, H, F, F, pyrazol-3-yl, CF₃), (M-1643, H, F, F, pyrazol-3-yl, Br), (M-1644, H, F, F, pyrazol-3-yl, CH₃), (M-1645, H, F, F, pyrimidin-2-yl, H), (M-1646, H, F, F, pyrimidin-2-yl, Cl), (M-1647, H, F, F, pyrimidin-2-yl, F), (M-1648, H, F, F, pyrimidin-2-yl, CF₃), (M-1649, H, F, F, pyrimidin-2-yl, Br), (M-1650, H, F, F, pyrimidin-2-yl, CH₃), (M-1651, H, F, F, pyrimidin-4-yl, H), (M-1652, H, F, F, pyrimidin-4-yl, Cl), (M-1653, H, F, F, pyrimidin-4-yl, F), (M-1654, H, F, F, pyrimidin-4-yl, CF₃), (M-1655, H, F, F, pyrimidin-4-yl, Br), (M-1656, H, F, F, pyrimidin-4-yl, CH₃), (M-1657, H, F, F, pyrimidin-5-yl, H), (M-1658, H, F, F, pyrimidin-5-yl, Cl), (M-1659, H, F, F, pyrimidin-5-yl, F), (M-1660, H, F, F, pyrimidin-5-yl, CF₃), (M-1661, H, F, F, pyrimidin-5-yl, Br), (M-1662, H, F, F, pyrimidin-5-yl, CH₃), (M-1663, H, F, F, HOOCCH₂CH₂CH₂, H), (M-1664, H, F, F, HOOCCH₂CH₂CH₂, Cl), (M-1665, H, F, F, HOOCCH₂CH₂CH₂, F), (M-1666, H, F, F, HOOCCH₂CH₂CH₂, CF₃), (M-1667, H, F, F, HOOCCH₂CH₂CH₂, Br), (M-1668, H, F, F, HOOCCH₂CH₂CH₂, CH₃), (M-1669, H, F, F, HOOCCH₂CH₂CH₂CH₂, H), (M-1670, H, F, F, HOOCCH₂CH₂CH₂CH₂, Cl), (M-1671, H, F, F, HOOCCH₂CH₂CH₂CH₂, F), (M-1672, H, F, F, HOOCCH₂CH₂CH₂CH₂, CF₃), (M-1673, H, F, F, HOOCCH₂CH₂CH₂CH₂, Br), (M-1674, H, F, F, HOOCCH₂CH₂CH₂CH₂, CH₃), (M-1675, H, F, F, (Me)₂NCOCH₂CH₂CH₂CH₂, H), (M-1676, H, F, F, (Me)₂NCOCH₂CH₂CH₂CH₂, Cl), (M-1677, H, F, F, (Me)₂NCOCH₂CH₂CH₂CH₂, F), (M-1678, H, F, F, (Me)₂NCOCH₂CH₂CH₂CH₂, CF₃), (M-1679, H, F, F, (Me)₂NCOCH₂CH₂CH₂CH₂, Br), (M-1680, H, F, F, (Me)₂NCOCH₂CH₂CH₂CH₂, CH₃), (M-1681, H, F, F, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, H), (M-1682, H, F, F, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, Cl), (M-1683, H, F, F, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, F), (M-1684, H, F, F, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, CF₃), (M-1685, H, F, F, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, Br), (M-1686, H, F, F, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, CH₃), (M-1687, H, F, F, MeOCH₂, H), (M-1688, H, F, F, MeOCH₂, Cl), (M-1689, H, F, F, MeOCH₂, F), (M-1690, H, F, F, MeOCH₂, CF₃), (M-1691, H, F, F, MeOCH₂, Br), (M-1692, H, F, F, MeOCH₂, CH₃), (M-1693, H, F, F, EtOCH₂, H), (M-1694, H, F, F, EtOCH₂, Cl), (M-1695, H, F, F, EtOCH₂, F), (M-1696, H, F, F, EtOCH₂, CF₃), (M-1697, H, F, F, EtOCH₂, Br), (M-1698, H, F, F, EtOCH₂, CH₃), (M-1699, H, F, F, EtOCH₂CH₂, H), (M-1700, H, F, F, EtOCH₂CH₂, Cl), (M-1701, H, F, F, EtOCH₂CH₂, F), (M-1702, H, F, F, EtOCH₂CH₂, CF₃), (M-1703, H, F, F, EtOCH₂CH₂, Br), (M-1704, H, F, F, EtOCH₂CH₂, CH₃), (M-1705, H, F, F, MeOCH₂CH₂OCH₂CH₂, H), (M-1706, H, F, F, MeOCH₂CH₂OCH₂CH₂, Cl), (M-1707, H, F, F, MeOCH₂CH₂OCH₂CH₂, F), (M-1708, H, F, F, MeOCH₂CH₂OCH₂CH₂, CF₃), (M-1709, H, F, F, MeOCH₂CH₂OCH₂CH₂, Br), (M-1710, H, F, F, MeOCH₂CH₂OCH₂CH₂, CH₃), (M-1711, H, F, F, MeOCH₂CH₂, H), (M-1712, H, F, F, MeOCH₂CH₂, Cl), (M-1713, H, F, F, MeOCH₂CH₂, F), (M-1714, H, F, F, MeOCH₂CH₂, CF₃), (M-1715, H, F, F, MeOCH₂CH₂, Br), (M-1716, H, F, F, MeOCH₂CH₂, CH₃), (M-1717, H, F, F, HOCH₂, H), (M-1718, H, F, F, HOCH₂, Cl), (M-1719, H, F, F, HOCH₂, F), (M-1720, H, F, F, HOCH₂, CF₃), (M-1721, H, F, F, HOCH₂, Br), (M-1722, H, F, F, HOCH₂, CH₃), (M-1723, H, F, F, HOCH₂CH₂, H), (M-1724, H, F, F, HOCH₂CH₂, Cl), (M-1725, H, F, F, HOCH₂CH₂, F), (M-1726, H, F, F, HOCH₂CH₂, CF₃), (M-1727, H, F, F, HOCH₂CH₂, Br), (M-1728, H, F, F, HOCH₂CH₂, CH₃), (M-1729, H, F, F, HOCH₂CH₂CH₂, H), (M-1730, H, F, F, HOCH₂CH₂CH₂, Cl), (M-1731, H, F, F, HOCH₂CH₂CH₂, F), (M-1732, H, F, F, HOCH₂CH₂CH₂, CF₃), (M-1733, H, F, F, HOCH₂CH₂CH₂, Br), (M-1734, H, F, F, HOCH₂CH₂CH₂, CH₃), (M-1735, H, F, F, HOCH₂CH₂CH₂CH₂, H), (M-1736, H, F, F, HOCH₂CH₂CH₂CH₂, Cl), (M-1737, H, F, F, HOCH₂CH₂CH₂CH₂, F), (M-1738, H, F, F, HOCH₂CH₂CH₂CH₂, CF₃), (M-1739, H, F, F, HOCH₂CH₂CH₂CH₂, Br), (M-1740, H, F, F, HOCH₂CH₂CH₂CH₂, CH₃), (M-1741, H, F, F, HOCH₂CH₂CH₂CH₂CH₂, H), (M-1742, H, F, F, HOCH₂CH₂CH₂CH₂CH₂, Cl), (M-1743, H, F, F, HOCH₂CH₂CH₂CH₂CH₂, F), (M-1744, H, F, F, HOCH₂CH₂CH₂CH₂CH₂, CF₃), (M-1745, H, F, F, HOCH₂CH₂CH₂CH₂CH₂, Br), (M-1746, H, F, F, HOCH₂CH₂CH₂CH₂CH₂, CH₃), (M-1747, H, F, F, HOCH₂CH₂OCH₂CH₂, H), (M-1748, H, F, F, HOCH₂CH₂OCH₂CH₂, Cl), (M-1749, H, F, F, HOCH₂CH₂OCH₂CH₂, F), (M-1750, H, F, F, HOCH₂CH₂OCH₂CH₂, CF₃), (M-1751, H, F, F, HOCH₂CH₂OCH₂CH₂, Br), (M-1752, H, F, F, HOCH₂CH₂OCH₂CH₂, CH₃), (M-1753, H, F, F, (Me)₂N, H), (M-1754, H, F, F, (Me)₂N, Cl), (M-1755, H, F, F, (Me)₂N, F), (M-1756, H, F, F, (Me)₂N, CF₃), (M-1757, H, F, F, (Me)₂N, Br), (M-1758, H, F, F, (Me)₂N, CH₃), (M-1759, H, F, F, piperidin-4-yl-methyl, H), (M-1760, H, F, F, piperidin-4-yl-methyl, Cl), (M-1761, H, F, F, piperidin-4-yl-methyl, F), (M-1762, H, F, F, piperidin-4-yl-methyl, CF₃), (M-1763, H, F, F, piperidin-4-yl-methyl, Br), (M-1764, H, F, F, piperidin-4-yl-methyl, CH₃), (M-1765, H, F, F, cyclohexylmethyl, H), (M-1766, H, F, F, cyclohexylmethyl, Cl), (M-1767, H, F, F, cyclohexylmethyl, F), (M-1768, H, F, F, cyclohexylmethyl, CF₃), (M-1769, H, F, F, cyclohexylmethyl, Br), (M-1770, H, F, F, cyclohexylmethyl, CH₃), (M-1771, H, F, Cl, H, H), (M-1772, H, F, Cl, H, Cl), (M-1773, H, F, Cl, H, F), (M-1774, H, F, Cl, H, CF₃), (M-1775, H, F, Cl, H, Br),
(M-1776, H, F, Cl, H, CH₃), (M-1777, H, F, Cl, F, H), (M-1778, H, F, Cl, F, Cl), (M-1779, H, F, Cl, F, F), (M-1780, H, F, Cl, F, CF₃), (M-1781, H, F, Cl, F, Br), (M-1782, H, F, Cl, F, CH₃), (M-1783, H, F, Cl, Cl, H), (M-1784, H, F, Cl, Cl, Cl), (M-1785, H, F, Cl, Cl, F), (M-1786, H, F, Cl, Cl, CF₃), (M-1787, H, F, Cl, Cl, Br), (M-1788, H, F, Cl, Cl, CH₃), (M-1789, H, F, Cl, CH₃, H), (M-1790, H, F, Cl, CH₃, Cl), (M-1791, H, F, Cl, CH₃, F), (M-1792, H, F, Cl, CH₃, CF₃), (M-1793, H, F, Cl, CH₃, Br), (M-1794, H, F, Cl, CH₃, CH₃), (M-1795, H, F, Cl, Et, H), (M-1796, H, F, Cl, Et, Cl), (M-1797, H, F, Cl, Et, F), (M-1798, H, F, Cl, Et, CF₃), (M-1799, H, F, Cl, Et, Br), (M-1800, H, F, Cl, Et, CH₃), (M-1801, H, F, Cl, n-Pr, H), (M-1802, H, F, Cl, n-Pr, Cl), (M-1803, H, F, Cl, n-Pr, F), (M-1804, H, F, Cl, n-Pr, CF₃), (M-1805, H, F, Cl, n-Pr, Br), (M-1806, H, F, Cl, n-Pr, CH₃), (M-1807, H, F, Cl, c-Pr, H), (M-1808, H, F, Cl, c-Pr, Cl), (M-1809, H, F, Cl, c-Pr, F), (M-1810, H, F, Cl, c-Pr, CF₃), (M-1811, H, F, Cl, c-Pr, Br), (M-1812, H, F, Cl, c-Pr, CH₃), (M-1813, H, F, Cl, i-Pr, H), (M-1814, H, F, Cl, i-Pr, Cl), (M-1815, H, F, Cl, i-Pr, F), (M-1816, H, F, Cl, i-Pr, CF₃), (M-1817, H, F, Cl, i-Pr, Br), (M-1818, H, F, Cl, i-Pr, CH₃), (M-1819, H, F, Cl, n-Bu, H), (M-1820, H, F, Cl, n-Bu, Cl), (M-1821, H, F, Cl, n-Bu, F), (M-1822, H, F, Cl, n-Bu, CF₃), (M-1823, H, F, Cl, n-Bu, Br), (M-1824, H, F, Cl, n-Bu, CH₃), (M-1825, H, F, Cl, i-Bu, H), (M-1826, H, F, Cl, i-Bu, Cl), (M-1827, H, F, Cl, i-Bu, F), (M-1828, H, F, Cl, i-Bu, CF₃), (M-1829, H, F, Cl, i-Bu, Br), (M-1830, H, F, Cl, i-Bu, CH₃), (M-1831, H, F, Cl, sec-Bu, H), (M-1832, H, F, Cl, sec-Bu, Cl), (M-1833, H, F, Cl, sec-Bu, F), (M-1834, H, F, Cl, sec-Bu, CF₃), (M-1835, H, F, Cl, sec-Bu, Br), (M-1836, H, F, Cl, sec-Bu, CH₃), (M-1837, H, F, Cl, n-Pen, H), (M-1838, H, F, Cl, n-Pen, Cl), (M-1839, H, F, Cl, n-Pen, F), (M-1840, H, F, Cl, n-Pen, CF₃), (M-1841, H, F, Cl, n-Pen, Br), (M-1842, H, F, Cl, n-Pen, CH₃), (M-1843, H, F, Cl, c-Pen, H), (M-1844, H, F, Cl, c-Pen, Cl), (M-1845, H, F, Cl, c-Pen, F), (M-1846, H, F, Cl, c-Pen, CF₃), (M-1847, H, F, Cl, c-Pen, Br), (M-1848, H, F, Cl, c-Pen, CH₃), (M-1849, H, F, Cl, n-Hex, H), (M-1850, H, F, Cl, n-Hex, Cl), (M-1851, H, F, Cl, n-Hex, F), (M-1852, H, F, Cl, n-Hex, CF₃), (M-1853, H, F, Cl, n-Hex, Br), (M-1854, H, F, Cl, n-Hex, CH₃), (M-1855, H, F, Cl, c-Hex, H), (M-1856, H, F, Cl, c-Hex, Cl), (M-1857, H, F, Cl, c-Hex, F), (M-1858, H, F, Cl, c-Hex, CF₃), (M-1859, H, F, Cl, c-Hex, Br), (M-1860, H, F, Cl, c-Hex, CH₃), (M-1861, H, F, Cl, OH, H), (M-1862, H, F, Cl, OH, Cl), (M-1863, H, F, Cl, OH, F), (M-1864, H, F, Cl, OH, CF₃), (M-1865, H, F, Cl, OH, Br), (M-1866, H, F, Cl, OH, CH₃), (M-1867, H, F, Cl, EtO, H), (M-1868, H, F, Cl, EtO, Cl), (M-1869, H, F, Cl, EtO, F), (M-1870, H, F, Cl, EtO, CF₃), (M-1871, H, F, Cl, EtO, Br), (M-1872, H, F, Cl, EtO, CH₃), (M-1873, H, F, Cl, n-PrO, H), (M-1874, H, F, Cl, n-PrO, Cl), (M-1875, H, F, Cl, n-PrO, F), (M-1876, H, F, Cl, n-PrO, CF₃), (M-1877, H, F, Cl, n-PrO, Br), (M-1878, H, F, Cl, n-PrO, CH₃), (M-1879, H, F, Cl, PhO, H), (M-1880, H, F, Cl, PhO, Cl), (M-1881, H, F, Cl, PhO, F), (M-1882, H, F, Cl, PhO, CF₃), (M-1883, H, F, Cl, PhO, Br), (M-1884, H, F, Cl, PhO, CH₃), (M-1885, H, F, Cl, BnO, H), (M-1886, H, F, Cl, BnO, Cl), (M-1887, H, F, Cl, BnO, F), (M-1888, H, F, Cl, BnO, CF₃), (M-1889, H, F, Cl, BnO, Br), (M-1890, H, F, Cl, BnO, CH₃), (M-1891, H, F, Cl, PhCH₂CH₂O, H), (M-1892, H, F, Cl, PhCH₂CH₂O, Cl), (M-1893, H, F, Cl, PhCH₂CH₂O, F), (M-1894, H, F, Cl, PhCH₂CH₂O, CF₃), (M-1895, H, F, Cl, PhCH₂CH₂O, Br), (M-1896, H, F, Cl, PhCH₂CH₂O, CH₃), (M-1897, H, F, Cl, CF₃O, H), (M-1898, H, F, Cl, CF₃O, Cl), (M-1899, H, F, Cl, CF₃O, F), (M-1900, H, F, Cl, CF₃O, CF₃), (M-1901, H, F, Cl, CF₃O, Br), (M-1902, H, F, Cl, CF₃O, CH₃), (M-1903, H, F, Cl, Ph, H), (M-1904, H, F, Cl, Ph, Cl), (M-1905, H, F, Cl, Ph, F), (M-1906, H, F, Cl, Ph, CF₃), (M-1907, H, F, Cl, Ph, Br), (M-1908, H, F, Cl, Ph, CH₃), (M-1909, H, F, Cl, 4-F-Ph, H), (M-1910, H, F, Cl, 4-F-Ph, Cl), (M-1911, H, F, Cl, 4-F-Ph, F), (M-1912, H, F, Cl, 4-F-Ph, CF₃), (M-1913, H, F, Cl, 4-F-Ph, Br), (M-1914, H, F, Cl, 4-F-Ph, CH₃), (M-1915, H, F, Cl, 4-CF₃-Ph, H), (M-1916, H, F, Cl, 4-CF₃-Ph, Cl), (M-1917, H, F, Cl, 4-CF₃-Ph, F), (M-1918, H, F, Cl, 4-CF₃-Ph, CF₃), (M-1919, H, F, Cl, 4-CF₃-Ph, Br), (M-1920, H, F, Cl, 4-CF₃-Ph, CH₃), (M-1921, H, F, Cl, 4-(Me)₂N-Ph, H), (M-1922, H, F, Cl, 4-(Me)₂N-Ph, Cl), (M-1923, H, F, Cl, 4-(Me)₂N-Ph, F), (M-1924, H, F, Cl, 4-(Me)₂N-Ph, CF₃), (M-1925, H, F, Cl, 4-(Me)₂N-Ph, Br), (M-1926, H, F, Cl, 4-(Me)₂N-Ph, CH₃), (M-1927, H, F, Cl, 4-OH-Ph, H), (M-1928, H, F, Cl, 4-OH-Ph, Cl), (M-1929, H, F, Cl, 4-OH-Ph, F), (M-1930, H, F, Cl, 4-OH-Ph, CF₃), (M-1931, H, F, Cl, 4-OH-Ph, Br), (M-1932, H, F, Cl, 4-OH-Ph, CH₃), (M-1933, H, F, Cl, 3,4-di-F-Ph, H), (M-1934, H, F, Cl, 3,4-di-F-Ph, Cl), (M-1935, H, F, Cl, 3,4-di-F-Ph, F), (M-1936, H, F, Cl, 3,4-di-F-Ph, CF₃), (M-1937, H, F, Cl, 3,4-di-F-Ph, Br), (M-1938, H, F, Cl, 3,4-di-F-Ph, CH₃), (M-1939, H, F, Cl, 4-COOH-Ph, H), (M-1940, H, F, Cl, 4-COOH-Ph, Cl), (M-1941, H, F, Cl, 4-COOH-Ph, F), (M-1942, H, F, Cl, 4-COOH-Ph, CF₃), (M-1943, H, F, Cl, 4-COOH-Ph, Br), (M-1944, H, F, Cl, 4-COOH-Ph, CH₃), (M-1945, H, F, Cl, Bn, H), (M-1946, H, F, Cl, Bn, Cl), (M-1947, H, F, Cl, Bn, F), (M-1948, H, F, Cl, Bn, CF₃), (M-1949, H, F, Cl, Bn, Br), (M-1950, H, F, Cl, Bn, CH₃), (M-1951, H, F, Cl, 4-F-Bn, H), (M-1952, H, F, Cl, 4-F-Bn, Cl), (M-1953, H, F, Cl, 4-F-Bn, F), (M-1954, H, F, Cl, 4-F-Bn, CF₃), (M-1955, H, F, Cl, 4-F-Bn, Br), (M-1956, H, F, Cl, 4-F-Bn, CH₃), (M-1957, H, F, Cl, 2-Py, H), (M-1958, H, F, Cl, 2-Py, Cl), (M-1959, H, F, Cl, 2-Py, F), (M-1960, H, F, Cl, 2-Py, CF₃), (M-1961, H, F, Cl, 2-Py, Br), (M-1962, H, F, Cl, 2-Py, CH₃), (M-1963, H, F, Cl, 3-Py, H), (M-1964, H, F, Cl, 3-Py, Cl), (M-1965, H, F, Cl, 3-Py, F), (M-1966, H, F, Cl, 3-Py, CF₃), (M-1967, H, F, Cl, 3-Py, Br), (M-1968, H, F, Cl, 3-Py, CH₃), (M-1969, H, F, Cl, 4-Py, H), (M-1970, H, F, Cl, 4-Py, Cl), (M-1971, H, F, Cl, 4-Py, F), (M-1972, H, F, Cl, 4-Py, CF₃), (M-1973, H, F, Cl, 4-Py, Br), (M-1974, H, F, Cl, 4-Py, CH₃), (M-1975, H, F, Cl, 2-Th, H), (M-1976, H, F, Cl, 2-Th, Cl), (M-1977, H, F, Cl, 2-Th, F), (M-1978, H, F, Cl, 2-Th, CF₃), (M-1979, H, F, Cl, 2-Th, Br), (M-1980, H, F, Cl, 2-Th, CH₃), (M-1981, H, F, Cl, 3-Th, H), (M-1982, H, F, Cl, 3-Th, Cl), (M-1983, H, F, Cl, 3-Th, F), (M-1984, H, F, Cl, 3-Th, CF₃), (M-1985, H, F, Cl, 3-Th, Br), (M-1986, H, F, Cl, 3-Th, CH₃), (M-1987, H, F, Cl, pyrazol-2-yl, H), (M-1988, H, F, Cl, pyrazol-2-yl, Cl), (M-1989, H, F, Cl, pyrazol-2-yl, F), (M-1990, H, F, Cl, pyrazol-2-yl, CF₃), (M-1991, H, F, Cl, pyrazol-2-yl, Br), (M-1992, H, F, Cl, pyrazol-2-yl, CH₃), (M-1993, H, F, Cl, pyrazol-3-yl, H), (M-1994, H, F, Cl, pyrazol-3-yl, Cl), (M-1995, H, F, Cl, pyrazol-3-yl, F), (M-1996, H, F, Cl, pyrazol-3-yl, CF₃), (M-1997, H, F, Cl, pyrazol-3-yl, Br), (M-1998, H, F, Cl, pyrazol-3-yl, CH₃), (M-1999, H, F, Cl, pyrimidin-2-yl, H), (M-2000, H, F, Cl, pyrimidin-2-yl, Cl), (M-2001, H, F, Cl, pyrimidin-2-yl, F), (M-2002, H, F, Cl, pyrimidin-2-yl, CF₃), (M-2003, H, F, Cl, pyrimidin-2-yl, Br), (M-2004, H, F, Cl, pyrimidin-2-yl, CH₃), (M-2005, H, F, Cl, pyrimidin-4-yl, H), (M-2006, H, F, Cl, pyrimidin-4-yl, Cl), (M-2007, H, F, Cl, pyrimidin-4-yl, F), (M-2008, H, F, Cl, pyrimidin-4-yl, CF₃), (M-2009, H, F, Cl, pyrimidin-4-yl, Br), (M-2010, H, F, Cl, pyrimidin-4-yl, CH₃), (M-2011, H, F, Cl, pyrimidin-5-yl, H), (M-2012, H, F, Cl, pyrimidin-5-yl, Cl), (M-2013, H, F, Cl, pyrimidin-5-yl, F), (M-2014, H, F, Cl, pyrimidin-5-yl, CF₃), (M-2015, H, F, Cl, pyrimidin-5-yl, Br), (M-2016, H, F, Cl, pyrimidin-5-yl, CH₃), (M-2017, H, F, Cl, HOOCCH₂CH₂CH₂, H), (M-2018, H, F, Cl, HOOCCH₂CH₂CH₂, Cl), (M-2019, H, F, Cl, HOOCCH₂CH₂CH₂, F), (M-2020, H, F, Cl, HOOCCH₂CH₂CH₂, CF₃), (M-2021, H, F, Cl, HOOCCH₂CH₂CH₂, Br), (M-2022, H, F, Cl, HOOCCH₂CH₂CH₂, CH₃), (M-2023, H, F, Cl, HOOCCH₂CH₂CH₂CH₂, H), (M-2024, H, F, Cl, HOOCCH₂CH₂CH₂CH₂, Cl), (M-2025, H, F, Cl, HOOCCH₂CH₂CH₂CH₂, F), (M-2026, H, F, Cl, HOOCCH₂CH₂CH₂CH₂, CF₃), (M-2027, H, F, Cl, HOOCCH₂CH₂CH₂CH₂, Br), (M-2028, H, F, Cl, HOOCCH₂CH₂CH₂CH₂, CH₃), (M-2029, H, F, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂, H), (M-2030, H, F, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂, Cl), (M-2031, H, F, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂, F), (M-203
2, H, F, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂, CF₃), (M-2033, H, F, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂, Br), (M-2034, H, F, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂, CH₃), (M-2035, H, F, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, H), (M-2036, H, F, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, Cl), (M-2037, H, F, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, F), (M-2038, H, F, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, CF₃), (M-2039, H, F, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, Br), (M-2040, H, F, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, CH₃), (M-2041, H, F, Cl, MeOCH₂, H), (M-2042, H, F, Cl, MeOCH₂, Cl), (M-2043, H, F, Cl, MeOCH₂, F), (M-2044, H, F, Cl, MeOCH₂, CF₃), (M-2045, H, F, Cl, MeOCH₂, Br), (M-2046, H, F, Cl, MeOCH₂, CH₃), (M-2047, H, F, Cl, EtOCH₂, H), (M-2048, H, F, Cl, EtOCH₂, Cl), (M-2049, H, F, Cl, EtOCH₂, F), (M-2050, H, F, Cl, EtOCH₂, CF₃), (M-2051, H, F, Cl, EtOCH₂, Br), (M-2052, H, F, Cl, EtOCH₂, CH₃), (M-2053, H, F, Cl, EtOCH₂CH₂, H), (M-2054, H, F, Cl, EtOCH₂CH₂, Cl), (M-2055, H, F, Cl, EtOCH₂CH₂, F), (M-2056, H, F, Cl, EtOCH₂CH₂, CF₃), (M-2057, H, F, Cl, EtOCH₂CH₂, Br), (M-2058, H, F, Cl, EtOCH₂CH₂, CH₃), (M-2059, H, F, Cl, MeOCH₂CH₂OCH₂CH₂, H), (M-2060, H, F, Cl, MeOCH₂CH₂OCH₂CH₂, Cl), (M-2061, H, F, Cl, MeOCH₂CH₂OCH₂CH₂, F), (M-2062, H, F, Cl, MeOCH₂CH₂OCH₂CH₂, CF₃), (M-2063, H, F, Cl, MeOCH₂CH₂OCH₂CH₂, Br), (M-2064, H, F, Cl, MeOCH₂CH₂OCH₂CH₂, CH₃), (M-2065, H, F, Cl, MeOCH₂CH₂, H), (M-2066, H, F, Cl, MeOCH₂CH₂, Cl), (M-2067, H, F, Cl, MeOCH₂CH₂, F), (M-2068, H, F, Cl, MeOCH₂CH₂, CF₃), (M-2069, H, F, Cl, MeOCH₂CH₂, Br), (M-2070, H, F, Cl, MeOCH₂CH₂, CH₃), (M-2071, H, F, Cl, HOCH₂, H), (M-2072, H, F, Cl, HOCH₂, Cl), (M-2073, H, F, Cl, HOCH₂, F), (M-2074, H, F, Cl, HOCH₂, CF₃), (M-2075, H, F, Cl, HOCH₂, Br), (M-2076, H, F, Cl, HOCH₂, CH₃), (M-2077, H, F, Cl, HOCH₂CH₂, H), (M-2078, H, F, Cl, HOCH₂CH₂, Cl), (M-2079, H, F, Cl, HOCH₂CH₂, F), (M-2080, H, F, Cl, HOCH₂CH₂, CF₃), (M-2081, H, F, Cl, HOCH₂CH₂, Br), (M-2082, H, F, Cl, HOCH₂CH₂, CH₃), (M-2083, H, F, Cl, HOCH₂CH₂CH₂, H), (M-2084, H, F, Cl, HOCH₂CH₂CH₂, Cl), (M-2085, H, F, Cl, HOCH₂CH₂CH₂, F), (M-2086, H, F, Cl, HOCH₂CH₂CH₂, CF₃), (M-2087, H, F, Cl, HOCH₂CH₂CH₂, Br), (M-2088, H, F, Cl, HOCH₂CH₂CH₂, CH₃), (M-2089, H, F, Cl, HOCH₂CH₂CH₂CH₂, H), (M-2090, H, F, Cl, HOCH₂CH₂CH₂CH₂, Cl), (M-2091, H, F, Cl, HOCH₂CH₂CH₂CH₂, F), (M-2092, H, F, Cl, HOCH₂CH₂CH₂CH₂, CF₃), (M-2093, H, F, Cl, HOCH₂CH₂CH₂CH₂, Br), (M-2094, H, F, Cl, HOCH₂CH₂CH₂CH₂, CH₃), (M-2095, H, F, Cl, HOCH₂CH₂CH₂CH₂CH₂, H), (M-2096, H, F, Cl, HOCH₂CH₂CH₂CH₂CH₂, Cl), (M-2097, H, F, Cl, HOCH₂CH₂CH₂CH₂CH₂, F), (M-2098, H, F, Cl, HOCH₂CH₂CH₂CH₂CH₂, CF₃), (M-2099, H, F, Cl, HOCH₂CH₂CH₂CH₂CH₂, Br), (M-2100, H, F, Cl, HOCH₂CH₂CH₂CH₂CH₂, CH₃), (M-2101, H, F, Cl, HOCH₂CH₂OCH₂CH₂, H), (M-2102, H, F, Cl, HOCH₂CH₂OCH₂CH₂, Cl), (M-2103, H, F, Cl, HOCH₂CH₂OCH₂CH₂, F), (M-2104, H, F, Cl, HOCH₂CH₂OCH₂CH₂, CF₃), (M-2105, H, F, Cl, HOCH₂CH₂OCH₂CH₂, Br), (M-2106, H, F, Cl, HOCH₂CH₂OCH₂CH₂, CH₃), (M-2107, H, F, Cl, (Me)₂N, H), (M-2108, H, F, Cl, (Me)₂N, Cl), (M-2109, H, F, Cl, (Me)₂N, F), (M-2110, H, F, Cl, (Me)₂N, CF₃), (M-2111, H, F, Cl, (Me)₂N, Br), (M-2112, H, F, Cl, (Me)₂N, CH₃), (M-2113, H, F, Cl, piperidin-4-yl-methyl, H), (M-2114, H, F, Cl, piperidin-4-yl-methyl, Cl), (M-2115, H, F, Cl, piperidin-4-yl-methyl, F), (M-2116, H, F, Cl, piperidin-4-yl-methyl, CF₃), (M-2117, H, F, Cl, piperidin-4-yl-methyl, Br), (M-2118, H, F, Cl, piperidin-4-yl-methyl, CH₃), (M-2119, H, F, Cl, cyclohexylmethyl, H), (M-2120, H, F, Cl, cyclohexylmethyl, Cl), (M-2121, H, F, Cl, cyclohexylmethyl, F), (M-2122, H, F, Cl, cyclohexylmethyl, CF₃), (M-2123, H, F, Cl, cyclohexylmethyl, Br), (M-2124, H, F, Cl, cyclohexylmethyl, CH₃), (M-2125, H, CH₃, H, H, H), (M-2126, H, CH₃, H, H, Cl), (M-2127, H, CH₃, H, H, F), (M-2128, H, CH₃, H, H, CF₃), (M-2129, H, CH₃, H, H, Br), (M-2130, H, CH₃, H, H, CH₃), (M-2131, H, CH₃, H, F, H), (M-2132, H, CH₃, H, F, Cl), (M-2133, H, CH₃, H, F, F), (M-2134, H, CH₃, H, F, CF₃), (M-2135, H, CH₃, H, F, Br), (M-2136, H, CH₃, H, F, CH₃), (M-2137, H, CH₃, H, Cl, H), (M-2138, H, CH₃, H, Cl, Cl), (M-2139, H, CH₃, H, Cl, F), (M-2140, H, CH₃, H, Cl, CF₃), (M-2141, H, CH₃, H, Cl, Br), (M-2142, H, CH₃, H, Cl, CH₃), (M-2143, H, CH₃, H, CH₃, H), (M-2144, H, CH₃, H, CH₃, Cl), (M-2145, H, CH₃, H, CH₃, F), (M-2146, H, CH₃, H, CH₃, CF₃), (M-2147, H, CH₃, H, CH₃, Br), (M-2148, H, CH₃, H, CH₃, CH₃), (M-2149, H, CH₃, H, Et, H), (M-2150, H, CH₃, H, Et, Cl), (M-2151, H, CH₃, H, Et, F), (M-2152, H, CH₃, H, Et, CF₃), (M-2153, H, CH₃, H, Et, Br), (M-2154, H, CH₃, H, Et, CH₃), (M-2155, H, CH₃, H, n-Pr, H), (M-2156, H, CH₃, H, n-Pr, Cl), (M-2157, H, CH₃, H, n-Pr, F), (M-2158, H, CH₃, H, n-Pr, CF₃), (M-2159, H, CH₃, H, n-Pr, Br), (M-2160, H, CH₃, H, n-Pr, CH₃), (M-2161, H, CH₃, H, c-Pr, H), (M-2162, H, CH₃, H, c-Pr, Cl), (M-2163, H, CH₃, H, c-Pr, F), (M-2164, H, CH₃, H, c-Pr, CF₃), (M-2165, H, CH₃, H, c-Pr, Br), (M-2166, H, CH₃, H, c-Pr, CH₃), (M-2167, H, CH₃, H, i-Pr, H), (M-2168, H, CH₃, H, i-Pr, Cl), (M-2169, H, CH₃, H, i-Pr, F), (M-2170, H, CH₃, H, i-Pr, CF₃), (M-2171, H, CH₃, H, i-Pr, Br), (M-2172, H, CH₃, H, i-Pr, CH₃), (M-2173, H, CH₃, H, n-Bu, H), (M-2174, H, CH₃, H, n-Bu, Cl), (M-2175, H, CH₃, H, n-Bu, F), (M-2176, H, CH₃, H, n-Bu, CF₃), (M-2177, H, CH₃, H, n-Bu, Br), (M-2178, H, CH₃, H, n-Bu, CH₃), (M-2179, H, CH₃, H, i-Bu, H), (M-2180, H, CH₃, H, i-Bu, Cl), (M-2181, H, CH₃, H, i-Bu, F), (M-2182, H, CH₃, H, i-Bu, CF₃), (M-2183, H, CH₃, H, i-Bu, Br), (M-2184, H, CH₃, H, i-Bu, CH₃), (M-2185, H, CH₃, H, sec-Bu, H), (M-2186, H, CH₃, H, sec-Bu, Cl), (M-2187, H, CH₃, H, sec-Bu, F), (M-2188, H, CH₃, H, sec-Bu, CF₃), (M-2189, H, CH₃, H, sec-Bu, Br), (M-2190, H, CH₃, H, sec-Bu, CH₃), (M-2191, H, CH₃, H, n-Pen, H), (M-2192, H, CH₃, H, n-Pen, Cl), (M-2193, H, CH₃, H, n-Pen, F), (M-2194, H, CH₃, H, n-Pen, CF₃), (M-2195, H, CH₃, H, n-Pen, Br), (M-2196, H, CH₃, H, n-Pen, CH₃), (M-2197, H, CH₃, H, c-Pen, H), (M-2198, H, CH₃, H, c-Pen, Cl), (M-2199, H, CH₃, H, c-Pen, F), (M-2200, H, CH₃, H, c-Pen, CF₃), (M-2201, H, CH₃, H, c-Pen, Br), (M-2202, H, CH₃, H, c-Pen, CH₃), (M-2203, H, CH₃, H, n-Hex, H), (M-2204, H, CH₃, H, n-Hex, Cl), (M-2205, H, CH₃, H, n-Hex, F), (M-2206, H, CH₃, H, n-Hex, CF₃), (M-2207, H, CH
₃, H, n-Hex, Br), (M-2208, H, CH₃, H, n-Hex, CH₃), (M-2209, H, CH₃, H, c-Hex, H), (M-2210, H, CH₃, H, c-Hex, Cl), (M-2211, H, CH₃, H, c-Hex, F), (M-2212, H, CH₃, H, c-Hex, CF₃), (M-2213, H, CH₃, H, c-Hex, Br), (M-2214, H, CH₃, H, c-Hex, CH₃), (M-2215, H, CH₃, H, OH, H), (M-2216, H, CH₃, H, OH, Cl), (M-2217, H, CH₃, H, OH, F), (M-2218, H, CH₃, H, OH, CF₃), (M-2219, H, CH₃, H, OH, Br), (M-2220, H, CH₃, H, OH, CH₃), (M-2221, H, CH₃, H, EtO, H), (M-2222, H, CH₃, H, EtO, Cl), (M-2223, H, CH₃, H, EtO, F), (M-2224, H, CH₃, H, EtO, CF₃), (M-2225, H, CH₃, H, EtO, Br), (M-2226, H, CH₃, H, EtO, CH₃), (M-2227, H, CH₃, H, n-PrO, H), (M-2228, H, CH₃, H, n-PrO, Cl), (M-2229, H, CH₃, H, n-PrO, F), (M-2230, H, CH₃, H, n-PrO, CF₃), (M-2231, H, CH₃, H, n-PrO, Br), (M-2232, H, CH₃, H, n-PrO, CH₃), (M-2233, H, CH₃, H, PhO, H), (M-2234, H, CH₃, H, PhO, Cl), (M-2235, H, CH₃, H, PhO, F), (M-2236, H, CH₃, H, PhO, CF₃), (M-2237, H, CH₃, H, PhO, Br), (M-2238, H, CH₃, H, PhO, CH₃), (M-2239, H, CH₃, H, BnO, H), (M-2240, H, CH₃, H, BnO, Cl), (M-2241, H, CH₃, H, BnO, F), (M-2242, H, CH₃, H, BnO, CF₃), (M-2243, H, CH₃, H, BnO, Br), (M-2244, H, CH₃, H, BnO, CH₃), (M-2245, H, CH₃, H, PhCH₂CH₂O, H), (M-2246, H, CH₃, H, PhCH₂CH₂O, Cl), (M-2247, H, CH₃, H, PhCH₂CH₂O, F), (M-2248, H, CH₃, H, PhCH₂CH₂O, CF₃), (M-2249, H, CH₃, H, PhCH₂CH₂O, Br), (M-2250, H, CH₃, H, PhCH₂CH₂O, CH₃), (M-2251, H, CH₃, H, CF₃O, H), (M-2252, H, CH₃, H, CF₃O, Cl), (M-2253, H, CH₃, H, CF₃O, F), (M-2254, H, CH₃, H, CF₃O, CF₃), (M-2255, H, CH₃, H, CF₃O, Br), (M-2256, H, CH₃, H, CF₃O, CH₃), (M-2257, H, CH₃, H, Ph, H), (M-2258, H, CH₃, H, Ph, Cl), (M-2259, H, CH₃, H, Ph, F), (M-2260, H, CH₃, H, Ph, CF₃), (M-2261, H, CH₃, H, Ph, Br), (M-2262, H, CH₃, H, Ph, CH₃), (M-2263, H, CH₃, H, 4-F-Ph, H), (M-2264, H, CH₃, H, 4-F-Ph, Cl), (M-2265, H, CH₃, H, 4-F-Ph, F), (M-2266, H, CH₃, H, 4-F-Ph, CF₃), (M-2267, H, CH₃, H, 4-F-Ph, Br), (M-2268, H, CH₃, H, 4-F-Ph, CH₃), (M-2269, H, CH₃, H, 4-CF₃-Ph, H), (M-2270, H, CH₃, H, 4-CF₃-Ph, Cl), (M-2271, H, CH₃, H, 4-CF₃-Ph, F), (M-2272, H, CH₃, H, 4-CF₃-Ph, CF₃), (M-2273, H, CH₃, H, 4-CF₃-Ph, Br), (M-2274, H, CH₃, H, 4-CF₃-Ph, CH₃), (M-2275, H, CH₃, H, 4-(Me)₂N-Ph, H), (M-2276, H, CH₃, H, 4-(Me)₂N-Ph, Cl), (M-2277, H, CH₃, H, 4-(Me)₂N-Ph, F), (M-2278, H, CH₃, H, 4-(Me)₂N-Ph, CF₃), (M-2279, H, CH₃, H, 4-(Me)₂N-Ph, Br), (M-2280, H, CH₃, H, 4-(Me)₂N-Ph, CH₃), (M-2281, H, CH₃, H, 4-OH-Ph, H), (M-2282, H, CH₃, H, 4-OH-Ph, Cl), (M-2283, H, CH₃, H, 4-OH-Ph, F), (M-2284, H, CH₃, H, 4-OH-Ph, CF₃), (M-2285, H, CH₃, H, 4-OH-Ph, Br), (M-2286, H, CH₃, H, 4-OH-Ph, CH₃), (M-2287, H, CH₃, H, 3,4-di-F-Ph, H), (M-2288, H, CH₃, H, 3,4-di-F-Ph, Cl), (M-2289, H, CH₃, H, 3,4-di-F-Ph, F), (M-2290, H, CH₃, H, 3,4-di-F-Ph, CF₃), (M-2291, H, CH₃, H, 3,4-di-F-Ph, Br), (M-2292, H, CH₃, H, 3,4-di-F-Ph, CH₃), (M-2293, H, CH₃, H, 4-COOH-Ph, H), (M-2294, H, CH₃, H, 4-COOH-Ph, Cl), (M-2295, H, CH₃, H, 4-COOH-Ph, F), (M-2296, H, CH₃, H, 4-COOH-Ph, CF₃), (M-2297, H, CH₃, H, 4-COOH-Ph, Br), (M-2298, H, CH₃, H, 4-COOH-Ph, CH₃), (M-2299, H, CH₃, H, Bn, H), (M-2300, H, CH₃, H, Bn, Cl), (M-2301, H, CH₃, H, Bn, F), (M-2302, H, CH₃, H, Bn, CF₃), (M-2303, H, CH₃, H, Bn, Br), (M-2304, H, CH₃, H, Bn, CH₃), (M-2305, H, CH₃, H, 4-F-Bn, H), (M-2306, H, CH₃, H, 4-F-Bn, Cl), (M-2307, H, CH₃, H, 4-F-Bn, F), (M-2308, H, CH₃, H, 4-F-Bn, CF₃), (M-2309, H, CH₃, H, 4-F-Bn, Br), (M-2310, H, CH₃, H, 4-F-Bn, CH₃), (M-2311, H, CH₃, H, 2-Py, H), (M-2312, H, CH₃, H, 2-Py, Cl), (M-2313, H, CH₃, H, 2-Py, F), (M-2314, H, CH₃, H, 2-Py, CF₃), (M-2315, H, CH₃, H, 2-Py, Br), (M-2316, H, CH₃, H, 2-Py, CH₃), (M-2317, H, CH₃, H, 3-Py, H), (M-2318, H, CH₃, H, 3-Py, Cl), (M-2319, H, CH₃, H, 3-Py, F), (M-2320, H, CH₃, H, 3-Py, CF₃), (M-2321, H, CH₃, H, 3-Py, Br), (M-2322, H, CH₃, H, 3-Py, CH₃), (M-2323, H, CH₃, H, 4-Py, H), (M-2324, H, CH₃, H, 4-Py, Cl), (M-2325, H, CH₃, H, 4-Py, F), (M-2326, H, CH₃, H, 4-Py, CF₃), (M-2327, H, CH₃, H, 4-Py, Br), (M-2328, H, CH₃, H, 4-Py, CH₃), (M-2329, H, CH₃, H, 2-Th, H), (M-2330, H, CH₃, H, 2-Th, Cl), (M-2331, H, CH₃, H, 2-Th, F), (M-2332, H, CH₃, H, 2-Th, CF₃), (M-2333, H, CH₃, H, 2-Th, Br), (M-2334, H, CH₃, H, 2-Th, CH₃), (M-2335, H, CH₃, H, 3-Th, H), (M-2336, H, CH₃, H, 3-Th, Cl), (M-2337, H, CH₃, H, 3-Th, F), (M-2338, H, CH₃, H, 3-Th, CF₃), (M-2339, H, CH₃, H, 3-Th, Br), (M-2340, H, CH₃, H, 3-Th, CH₃), (M-2341, H, CH₃, H, pyrazol-2-yl, H), (M-2342, H, CH₃, H, pyrazol-2-yl, Cl), (M-2343, H, CH₃, H, pyrazol-2-yl, F), (M-2344, H, CH₃, H, pyrazol-2-yl, CF₃), (M-2345, H, CH₃, H, pyrazol-2-yl, Br), (M-2346, H, CH₃, H, pyrazol-2-yl, CH₃), (M-2347, H, CH₃, H, pyrazol-3-yl, H), (M-2348, H, CH₃, H, pyrazol-3-yl, Cl), (M-2349, H, CH₃, H, pyrazol-3-yl, F), (M-2350, H, CH₃, H, pyrazol-3-yl, CF₃), (M-2351, H, CH₃, H, pyrazol-3-yl, Br), (M-2352, H, CH₃, H, pyrazol-3-yl, CH₃), (M-2353, H, CH₃, H, pyrimidin-2-yl, H), (M-2354, H, CH₃, H, pyrimidin-2-yl, Cl), (M-2355, H, CH₃, H, pyrimidin-2-yl, F), (M-2356, H, CH₃, H, pyrimidin-2-yl, CF₃), (M-2357, H, CH₃, H, pyrimidin-2-yl, Br), (M-2358, H, CH₃, H, pyrimidin-2-yl, CH₃), (M-2359, H, CH₃, H, pyrimidin-4-yl, H), (M-2360, H, CH₃, H, pyrimidin-4-yl, Cl), (M-2361, H, CH₃, H, pyrimidin-4-yl, F), (M-2362, H, CH₃, H, pyrimidin-4-yl, CF₃), (M-2363, H, CH₃, H, pyrimidin-4-yl, Br), (M-2364, H, CH₃, H, pyrimidin-4-yl, CH₃), (M-2365, H, CH₃, H, pyrimidin-5-yl, H), (M-2366, H, CH₃, H, pyrimidin-5-yl, Cl), (M-2367, H, CH₃, H, pyrimidin-5-yl, F), (M-2368, H, CH₃, H, pyrimidin-5-yl, CF₃), (M-2369, H, CH₃, H, pyrimidin-5-yl, Br), (M-2370, H, CH₃, H, pyrimidin-5-yl, CH₃), (M-2371, H, CH₃, H, HOOCCH₂CH₂CH₂, H), (M-2372, H, CH₃, H, HOOCCH₂CH₂CH₂, Cl), (M-2373, H, CH₃, H, HOOCCH₂CH₂CH₂, F), (M-2374, H, CH₃, H, HOOCCH₂CH₂CH₂, CF₃), (M-2375, H, CH₃, H, HOOCCH₂CH₂CH₂, Br), (M-2376, H, CH₃, H, HOOCCH₂CH₂CH₂, CH₃), (M-2377, H, CH₃, H, HOOCCH₂CH₂CH₂CH₂, H), (M-2378, H, CH₃, H, HOOCCH₂CH₂CH₂CH₂, Cl), (M-2379, H, CH₃, H, HOOCCH₂CH₂CH₂CH₂, F), (M-2380, H, CH₃, H, HOOCCH₂CH₂CH₂CH₂, CF₃), (M-2381, H, CH₃, H, HOOCCH₂CH₂CH₂CH₂, Br), (M-2382, H, CH₃, H, HOOCCH₂CH₂CH₂CH₂, CH₃), (M-2383, H, CH₃, H, (Me)₂NCOCH₂CH₂CH₂CH₂, H), (M-2384, H, CH₃, H, (Me)₂NCOCH₂CH₂CH₂CH₂, Cl), (M-2385, H, CH₃, H, (Me)₂NCOCH₂CH₂CH₂CH₂, F), (M-2386, H, CH₃, H, (Me)₂NCOCH₂CH₂CH₂CH₂, CF₃), (M-2387, H, CH₃, H, (Me)₂NCOCH₂CH₂CH₂CH₂, Br), (M-2388, H, CH₃, H, (Me)₂NCOCH₂CH₂CH₂CH₂, CH₃), (M-2389, H, CH₃, H, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, H), (M-2390, H, CH₃
, H, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, Cl), (M-2391, H, CH₃, H, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, F), (M-2392, H, CH₃, H, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, CF₃), (M-2393, H, CH₃, H, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, Br), (M-2394, H, CH₃, H, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, CH₃), (M-2395, H, CH₃, H, MeOCH₂, H), (M-2396, H, CH₃, H, MeOCH₂, Cl), (M-2397, H, CH₃, H, MeOCH₂, F), (M-2398, H, CH₃, H, MeOCH₂, CF₃), (M-2399, H, CH₃, H, MeOCH₂, Br), (M-2400, H, CH₃, H, MeOCH₂, CH₃), (M-2401, H, CH₃, H, EtOCH₂, H), (M-2402, H, CH₃, H, EtOCH₂, Cl), (M-2403, H, CH₃, H, EtOCH₂, F), (M-2404, H, CH₃, H, EtOCH₂, CF₃), (M-2405, H, CH₃, H, EtOCH₂, Br), (M-2406, H, CH₃, H, EtOCH₂, CH₃), (M-2407, H, CH₃, H, EtOCH₂CH₂, H), (M-2408, H, CH₃, H, EtOCH₂CH₂, Cl), (M-2409, H, CH₃, H, EtOCH₂CH₂, F), (M-2410, H, CH₃, H, EtOCH₂CH₂, CF₃), (M-2411, H, CH₃, H, EtOCH₂CH₂, Br), (M-2412, H, CH₃, H, EtOCH₂CH₂, CH₃), (M-2413, H, CH₃, H, MeOCH₂CH₂OCH₂CH₂, H), (M-2414, H, CH₃, H, MeOCH₂CH₂OCH₂CH₂, Cl), (M-2415, H, CH₃, H, MeOCH₂CH₂OCH₂CH₂, F), (M-2416, H, CH₃, H, MeOCH₂CH₂OCH₂CH₂, CF₃), (M-2417, H, CH₃, H, MeOCH₂CH₂OCH₂CH₂, Br), (M-2418, H, CH₃, H, MeOCH₂CH₂OCH₂CH₂, CH₃), (M-2419, H, CH₃, H, MeOCH₂CH₂, H), (M-2420, H, CH₃, H, MeOCH₂CH₂, Cl), (M-2421, H, CH₃, H, MeOCH₂CH₂, F), (M-2422, H, CH₃, H, MeOCH₂CH₂, CF₃), (M-2423, H, CH₃, H, MeOCH₂CH₂, Br), (M-2424, H, CH₃, H, MeOCH₂CH₂, CH₃), (M-2425, H, CH₃, H, HOCH₂, H), (M-2426, H, CH₃, H, HOCH₂, Cl), (M-2427, H, CH₃, H, HOCH₂, F), (M-2428, H, CH₃, H, HOCH₂, CF₃), (M-2429, H, CH₃, H, HOCH₂, Br), (M-2430, H, CH₃, H, HOCH₂, CH₃), (M-2431, H, CH₃, H, HOCH₂CH₂, H), (M-2432, H, CH₃, H, HOCH₂CH₂, Cl), (M-2433, H, CH₃, H, HOCH₂CH₂, F), (M-2434, H, CH₃, H, HOCH₂CH₂, CF₃), (M-2435, H, CH₃, H, HOCH₂CH₂, Br), (M-2436, H, CH₃, H, HOCH₂CH₂, CH₃), (M-2437, H, CH₃, H, HOCH₂CH₂CH₂, H), (M-2438, H, CH₃, H, HOCH₂CH₂CH₂, Cl), (M-2439, H, CH₃, H, HOCH₂CH₂CH₂, F), (M-2440, H, CH₃, H, HOCH₂CH₂CH₂, CF₃), (M-2441, H, CH₃, H, HOCH₂CH₂CH₂, Br), (M-2442, H, CH₃, H, HOCH₂CH₂CH₂, CH₃), (M-2443, H, CH₃, H, HOCH₂CH₂CH₂CH₂, H), (M-2444, H, CH₃, H, HOCH₂CH₂CH₂CH₂, Cl), (M-2445, H, CH₃, H, HOCH₂CH₂CH₂CH₂, F), (M-2446, H, CH₃, H, HOCH₂CH₂CH₂CH₂, CF₃), (M-2447, H, CH₃, H, HOCH₂CH₂CH₂CH₂, Br), (M-2448, H, CH₃, H, HOCH₂CH₂CH₂CH₂, CH₃), (M-2449, H, CH₃, H, HOCH₂CH₂CH₂CH₂CH₂, H), (M-2450, H, CH₃, H, HOCH₂CH₂CH₂CH₂CH₂, Cl), (M-2451, H, CH₃, H, HOCH₂CH₂CH₂CH₂CH₂, F), (M-2452, H, CH₃, H, HOCH₂CH₂CH₂CH₂CH₂, CF₃), (M-2453, H, CH₃, H, HOCH₂CH₂CH₂CH₂CH₂, Br), (M-2454, H, CH₃, H, HOCH₂CH₂CH₂CH₂CH₂, CH₃), (M-2455, H, CH₃, H, HOCH₂CH₂OCH₂CH₂, H), (M-2456, H, CH₃, H, HOCH₂CH₂OCH₂CH₂, Cl), (M-2457, H, CH₃, H, HOCH₂CH₂OCH₂CH₂, F), (M-2458, H, CH₃, H, HOCH₂CH₂OCH₂CH₂, CF₃), (M-2459, H, CH₃, H, HOCH₂CH₂OCH₂CH₂, Br), (M-2460, H, CH₃, H, HOCH₂CH₂OCH₂CH₂, CH₃), (M-2461, H, CH₃, H, (Me)₂N, H), (M-2462, H, CH₃, H, (Me)₂N, Cl), (M-2463, H, CH₃, H, (Me)₂N, F), (M-2464, H, CH₃, H, (Me)₂N, CF₃), (M-2465, H, CH₃, H, (Me)₂N, Br), (M-2466, H, CH₃, H, (Me)₂N, CH₃), (M-2467, H, CH₃, H, piperidin-4-yl-methyl, H), (M-2468, H, CH₃, H, piperidin-4-yl-methyl, Cl), (M-2469, H, CH₃, H, piperidin-4-yl-methyl, F), (M-2470, H, CH₃, H, piperidin-4-yl-methyl, CF₃), (M-2471, H, CH₃, H, piperidin-4-yl-methyl, Br), (M-2472, H, CH₃, H, piperidin-4-yl-methyl, CH₃), (M-2473, H, CH₃, H, cyclohexylmethyl, H), (M-2474, H, CH₃, H, cyclohexylmethyl, Cl), (M-2475, H, CH₃, H, cyclohexylmethyl, F), (M-2476, H, CH₃, H, cyclohexylmethyl, CF₃), (M-2477, H, CH₃, H, cyclohexylmethyl, Br), (M-2478, H, CH₃, H, cyclohexylmethyl, CH₃), (M-2479, H, CH₃, F, H, H), (M-2480, H, CH₃, F, H, Cl), (M-2481, H, CH₃, F, H, F), (M-2482, H, CH₃, F, H, CF₃), (M-2483, H, CH₃, F, H, Br), (M-2484, H, CH₃, F, H, CH₃), (M-2485, H, CH₃, F, F, H), (M-2486, H, CH₃, F, F, Cl), (M-2487, H, CH₃, F, F, F), (M-2488, H, CH₃, F, F, CF₃), (M-2489, H, CH₃, F, F, Br), (M-2490, H, CH₃, F, F, CH₃), (M-2491, H, CH₃, F, Cl, H), (M-2492, H, CH₃, F, Cl, Cl), (M-2493, H, CH₃, F, Cl, F), (M-2494, H, CH₃, F, Cl, CF₃), (M-2495, H, CH₃, F, Cl, Br), (M-2496, H, CH₃, F, Cl, CH₃), (M-2497, H, CH₃, F, CH₃, H), (M-2498, H, CH₃, F, CH₃, Cl), (M-2499, H, CH₃, F, CH₃, F), (M-2500, H, CH₃, F, CH₃, CF₃), (M-2501, H, CH₃, F, CH₃, Br), (M-2502, H, CH₃, F, CH₃, CH₃), (M-2503, H, CH₃, F, Et, H), (M-2504, H, CH₃, F, Et, Cl), (M-2505, H, CH₃, F, Et, F), (M-2506, H, CH₃, F, Et, CF₃), (M-2507, H, CH₃, F, Et, Br), (M-2508, H, CH₃, F, Et, CH₃), (M-2509, H, CH₃, F, n-Pr, H), (M-2510, H, CH₃, F, n-Pr, Cl), (M-2511, H, CH₃, F, n-Pr, F), (M-2512, H, CH₃, F, n-Pr, CF₃), (M-2513, H, CH₃, F, n-Pr, Br), (M-2514, H, CH₃, F, n-Pr, CH₃), (M-2515, H, CH₃, F, c-Pr, H), (M-2516, H, CH₃, F, c-Pr, Cl), (M-2517, H, CH₃, F, c-Pr, F), (M-2518, H, CH₃, F, c-Pr, CF₃), (M-2519, H, CH₃, F, c-Pr, Br), (M-2520, H, CH₃, F, c-Pr, CH₃), (M-2521, H, CH₃, F, i-Pr, H), (M-2522, H, CH₃, F, i-Pr, Cl), (M-2523, H, CH₃, F, i-Pr, F), (M-2524, H, CH₃, F, i-Pr, CF₃), (M-2525, H, CH₃, F, i-Pr, Br), (M-2526, H, CH₃, F, i-Pr, CH₃), (M-2527, H, CH₃, F, n-Bu, H), (M-2528, H, CH₃, F, n-Bu, Cl), (M-2529, H, CH₃, F, n-Bu, F), (M-2530, H, CH₃, F, n-Bu, CF₃), (M-2531, H, CH₃, F, n-Bu, Br), (M-2532, H, CH₃, F, n-Bu, CH₃), (M-2533, H, CH₃, F, i-Bu, H), (M-2534, H, CH₃, F, i-Bu, Cl), (M-2535, H, CH₃, F, i-Bu, F), (M-2536, H, CH₃, F, i-Bu, CF₃), (M-2537, H, CH₃, F, i-Bu, Br), (M-2538, H, CH₃, F, i-Bu, CH₃), (M-2539, H, CH₃, F, sec-Bu, H), (M-2540, H, CH₃, F, sec-Bu, Cl), (M-2541, H, CH₃, F, sec-Bu, F), (M-2542, H, CH₃, F, sec-Bu, CF₃), (M-2543, H, CH₃, F, sec-Bu, Br), (M-2544, H, CH₃, F, sec-Bu, CH₃), (M-2545, H, CH₃, F, n-Pen, H), (M-2546, H, CH₃, F, n-Pen, Cl), (M-2547, H, CH₃, F, n-Pen, F), (M-2548, H, CH₃
, F, n-Pen, CF₃), (M-2549, H, CH₃, F, n-Pen, Br), (M-2550, H, CH₃, F, n-Pen, CH₃), (M-2551, H, CH₃, F, c-Pen, H), (M-2552, H, CH₃, F, c-Pen, Cl), (M-2553, H, CH₃, F, c-Pen, F), (M-2554, H, CH₃, F, c-Pen, CF₃), (M-2555, H, CH₃, F, c-Pen, Br), (M-2556, H, CH₃, F, c-Pen, CH₃), (M-2557, H, CH₃, F, n-Hex, H), (M-2558, H, CH₃, F, n-Hex, Cl), (M-2559, H, CH₃, F, n-Hex, F), (M-2560, H, CH₃, F, n-Hex, CF₃), (M-2561, H, CH₃, F, n-Hex, Br), (M-2562, H, CH₃, F, n-Hex, CH₃), (M-2563, H, CH₃, F, c-Hex, H), (M-2564, H, CH₃, F, c-Hex, Cl), (M-2565, H, CH₃, F, c-Hex, F), (M-2566, H, CH₃, F, c-Hex, CF₃), (M-2567, H, CH₃, F, c-Hex, Br), (M-2568, H, CH₃, F, c-Hex, CH₃), (M-2569, H, CH₃, F, OH, H), (M-2570, H, CH₃, F, OH, Cl), (M-2571, H, CH₃, F, OH, F), (M-2572, H, CH₃, F, OH, CF₃), (M-2573, H, CH₃, F, OH, Br), (M-2574, H, CH₃, F, OH, CH₃), (M-2575, H, CH₃, F, EtO, H), (M-2576, H, CH₃, F, EtO, Cl), (M-2577, H, CH₃, F, EtO, F), (M-2578, H, CH₃, F, EtO, CF₃), (M-2579, H, CH₃, F, EtO, Br), (M-2580, H, CH₃, F, EtO, CH₃), (M-2581, H, CH₃, F, n-PrO, H), (M-2582, H, CH₃, F, n-PrO, Cl), (M-2583, H, CH₃, F, n-PrO, F), (M-2584, H, CH₃, F, n-PrO, CF₃), (M-2585, H, CH₃, F, n-PrO, Br), (M-2586, H, CH₃, F, n-PrO, CH₃), (M-2587, H, CH₃, F, PhO, H), (M-2588, H, CH₃, F, PhO, Cl), (M-2589, H, CH₃, F, PhO, F), (M-2590, H, CH₃, F, PhO, CF₃), (M-2591, H, CH₃, F, PhO, Br), (M-2592, H, CH₃, F, PhO, CH₃), (M-2593, H, CH₃, F, BnO, H), (M-2594, H, CH₃, F, BnO, Cl), (M-2595, H, CH₃, F, BnO, F), (M-2596, H, CH₃, F, BnO, CF₃), (M-2597, H, CH₃, F, BnO, Br), (M-2598, H, CH₃, F, BnO, CH₃), (M-2599, H, CH₃, F, PhCH₂CH₂O, H), (M-2600, H, CH₃, F, PhCH₂CH₂O, Cl), (M-2601, H, CH₃, F, PhCH₂CH₂O, F), (M-2602, H, CH₃, F, PhCH₂CH₂O, CF₃), (M-2603, H, CH₃, F, PhCH₂CH₂O, Br), (M-2604, H, CH₃, F, PhCH₂CH₂O, CH₃), (M-2605, H, CH₃, F, CF₃O, H), (M-2606, H, CH₃, F, CF₃O, Cl), (M-2607, H, CH₃, F, CF₃O, F), (M-2608, H, CH₃, F, CF₃O, CF₃), (M-2609, H, CH₃, F, CF₃O, Br), (M-2610, H, CH₃, F, CF₃O, CH₃), (M-2611, H, CH₃, F, Ph, H), (M-2612, H, CH₃, F, Ph, Cl), (M-2613, H, CH₃, F, Ph, F), (M-2614, H, CH₃, F, Ph, CF₃), (M-2615, H, CH₃, F, Ph, Br), (M-2616, H, CH₃, F, Ph, CH₃), (M-2617, H, CH₃, F, 4-F-Ph, H), (M-2618, H, CH₃, F, 4-F-Ph, Cl), (M-2619, H, CH₃, F, 4-F-Ph, F), (M-2620, H, CH₃, F, 4-F-Ph, CF₃), (M-2621, H, CH₃, F, 4-F-Ph, Br), (M-2622, H, CH₃, F, 4-F-Ph, CH₃), (M-2623, H, CH₃, F, 4-CF₃-Ph, H), (M-2624, H, CH₃, F, 4-CF₃-Ph, Cl), (M-2625, H, CH₃, F, 4-CF₃-Ph, F), (M-2626, H, CH₃, F, 4-CF₃-Ph, CF₃), (M-2627, H, CH₃, F, 4-CF₃-Ph, Br), (M-2628, H, CH₃, F, 4-CF₃-Ph, CH₃), (M-2629, H, CH₃, F, 4-(Me)₂N-Ph, H), (M-2630, H, CH₃, F, 4-(Me)₂N-Ph, Cl), (M-2631, H, CH₃, F, 4-(Me)₂N-Ph, F), (M-2632, H, CH₃, F, 4-(Me)₂N-Ph, CF₃), (M-2633, H, CH₃, F, 4-(Me)₂N-Ph, Br), (M-2634, H, CH₃, F, 4-(Me)₂N-Ph, CH₃), (M-2635, H, CH₃, F, 4-OH-Ph, H), (M-2636, H, CH₃, F, 4-OH-Ph, Cl), (M-2637, H, CH₃, F, 4-OH-Ph, F), (M-2638, H, CH₃, F, 4-OH-Ph, CF₃), (M-2639, H, CH₃, F, 4-OH-Ph, Br), (M-2640, H, CH₃, F, 4-OH-Ph, CH₃), (M-2641, H, CH₃, F, 3,4-di-F-Ph, H), (M-2642, H, CH₃, F, 3,4-di-F-Ph, Cl), (M-2643, H, CH₃, F, 3,4-di-F-Ph, F), (M-2644, H, CH₃, F, 3,4-di-F-Ph, CF₃), (M-2645, H, CH₃, F, 3,4-di-F-Ph, Br), (M-2646, H, CH₃, F, 3,4-di-F-Ph, CH₃), (M-2647, H, CH₃, F, 4-COOH-Ph, H), (M-2648, H, CH₃, F, 4-COOH-Ph, Cl), (M-2649, H, CH₃, F, 4-COOH-Ph, F), (M-2650, H, CH₃, F, 4-COOH-Ph, CF₃), (M-2651, H, CH₃, F, 4-COOH-Ph, Br), (M-2652, H, CH₃, F, 4-COOH-Ph, CH₃), (M-2653, H, CH₃, F, Bn, H), (M-2654, H, CH₃, F, Bn, Cl), (M-2655, H, CH₃, F, Bn, F), (M-2656, H, CH₃, F, Bn, CF₃), (M-2657, H, CH₃, F, Bn, Br), (M-2658, H, CH₃, F, Bn, CH₃), (M-2659, H, CH₃, F, 4-F-Bn, H), (M-2660, H, CH₃, F, 4-F-Bn, Cl), (M-2661, H, CH₃, F, 4-F-Bn, F), (M-2662, H, CH₃, F, 4-F-Bn, CF₃), (M-2663, H, CH₃, F, 4-F-Bn, Br), (M-2664, H, CH₃, F, 4-F-Bn, CH₃), (M-2665, H, CH₃, F, 2-Py, H), (M-2666, H, CH₃, F, 2-Py, Cl), (M-2667, H, CH₃, F, 2-Py, F), (M-2668, H, CH₃, F, 2-Py, CF₃), (M-2669, H, CH₃, F, 2-Py, Br), (M-2670, H, CH₃, F, 2-Py, CH₃), (M-2671, H, CH₃, F, 3-Py, H), (M-2672, H, CH₃, F, 3-Py, Cl), (M-2673, H, CH₃, F, 3-Py, F), (M-2674, H, CH₃, F, 3-Py, CF₃), (M-2675, H, CH₃, F, 3-Py, Br), (M-2676, H, CH₃, F, 3-Py, CH₃), (M-2677, H, CH₃, F, 4-Py, H), (M-2678, H, CH₃, F, 4-Py, Cl), (M-2679, H, CH₃, F, 4-Py, F), (M-2680, H, CH₃, F, 4-Py, CF₃), (M-2681, H, CH₃, F, 4-Py, Br), (M-2682, H, CH₃, F, 4-Py, CH₃), (M-2683, H, CH₃, F, 2-Th, H), (M-2684, H, CH₃, F, 2-Th, Cl), (M-2685, H, CH₃, F, 2-Th, F), (M-2686, H, CH₃, F, 2-Th, CF₃), (M-2687, H, CH₃, F, 2-Th, Br), (M-2688, H, CH₃, F, 2-Th, CH₃), (M-2689, H, CH₃, F, 3-Th, H), (M-2690, H, CH₃, F, 3-Th, Cl), (M-2691, H, CH₃, F, 3-Th, F), (M-2692, H, CH₃, F, 3-Th, CF₃), (M-2693, H, CH₃, F, 3-Th, Br), (M-2694, H, CH₃, F, 3-Th, CH₃), (M-2695, H, CH₃, F, pyrazol-2-yl, H), (M-2696, H, CH₃, F, pyrazol-2-yl, Cl), (M-2697, H, CH₃, F, pyrazol-2-yl, F), (M-2698, H, CH₃, F, pyrazol-2-yl, CF₃), (M-2699, H, CH₃, F, pyrazol-2-yl, Br), (M-2700, H, CH₃, F, pyrazol-2-yl, CH₃), (M-2701, H, CH₃, F, pyrazol-3-yl, H), (M-2702, H, CH₃, F, pyrazol-3-yl, Cl), (M-2703, H, CH₃, F, pyrazol-3-yl, F), (M-2704, H, CH₃, F, pyrazol-3-yl, CF₃), (M-2705, H, CH₃, F, pyrazol-3-yl, Br), (M-2706, H, CH₃, F, pyrazol-3-yl, CH₃), (M-2707, H, CH₃, F, pyrimidin-2-yl, H), (M-2708, H, CH₃, F, pyrimidin-2-yl, Cl), (M-2709, H, CH₃, F, pyrimidin-2-yl, F), (M-2710, H, CH₃, F, pyrimidin-2-yl, CF₃), (M-2711, H, CH₃, F, pyrimidin-2-yl, Br), (M-2712, H, CH₃, F, pyrimidin-2-yl, CH₃), (M-2713, H, CH₃, F, pyrimidin-4-yl, H), (M-2714, H, CH₃, F, pyrimidin-4-yl, Cl), (M-2715, H, CH₃, F, pyrimidin-4-yl, F), (M-2716, H, CH₃, F, pyrimidin-4-yl, CF₃), (M-2717, H, CH₃, F, pyrimidin-4-yl, Br), (M-2718, H, CH₃, F, pyrimidin-4-yl, CH₃), (M-2719, H, CH₃, F, pyrimidin-5-yl, H), (M-2720, H, CH₃, F, pyrimidin-5-yl, Cl), (M-2721, H, CH₃, F, pyrimidin-5-yl, F), (M-2722, H, CH₃, F, pyrimidin-5-yl, CF₃), (M-2723, H, CH₃, F, pyrimidin-5-yl, Br), (M-2724, H, CH₃, F, pyrimidin-5-yl, CH₃), (M-2725, H, CH₃, F, HOOCCH₂CH₂CH₂, H), (M-2726, H, CH₃, F, HOOCCH₂CH₂CH₂, Cl), (M-2727, H, CH₃, F, HOOCCH₂CH₂CH₂, F), (M-2728, H, CH₃, F, HOOCCH₂CH₂CH₂, CF₃), (M-2729, H, CH₃, F, HOOCCH₂CH₂CH₂, Br), (M-2730, H, CH₃, F, HOOCCH₂CH₂CH₂, CH₃), (M-2731, H, CH₃, F, HOOCCH₂CH₂CH₂CH₂, H), (M-2732, H, CH₃, F, HOOCCH₂CH₂CH₂CH₂, Cl), (M-2733, H, CH₃, F, HOOCCH₂CH₂CH₂CH₂, F), (M-2734, H, CH₃, F, HOOCCH₂CH₂CH₂CH₂, CF₃), (M-2735, H, CH₃, F, HOOCCH₂CH₂CH₂CH₂, Br), (M-2736, H, CH₃, F, HOOCCH₂CH₂CH₂CH₂, CH₃), (M-2737, H, CH₃, F, (Me)₂NCOCH₂CH₂CH₂CH₂, H), (M-2738, H, CH₃, F, (Me)₂NCOCH₂CH₂CH₂CH₂, Cl), (M-2739, H, CH₃
, F, (Me)₂NCOCH₂CH₂CH₂CH₂, F), (M-2740, H, CH₃, F, (Me)₂NCOCH₂CH₂CH₂CH₂, CF₃), (M-2741, H, CH₃, F, (Me)₂NCOCH₂CH₂CH₂CH₂, Br), (M-2742, H, CH₃, F, (Me)₂NCOCH₂CH₂CH₂CH₂, CH₃), (M-2743, H, CH₃, F, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, H), (M-2744, H, CH₃, F, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, Cl), (M-2745, H, CH₃, F, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, F), (M-2746, H, CH₃, F, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, CF₃), (M-2747, H, CH₃, F, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, Br), (M-2748, H, CH₃, F, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, CH₃), (M-2749, H, CH₃, F, MeOCH₂, H), (M-2750, H, CH₃, F, MeOCH₂, Cl), (M-2751, H, CH₃, F, MeOCH₂, F), (M-2752, H, CH₃, F, MeOCH₂, CF₃), (M-2753, H, CH₃, F, MeOCH₂, Br), (M-2754, H, CH₃, F, MeOCH₂, CH₃), (M-2755, H, CH₃, F, EtOCH₂, H), (M-2756, H, CH₃, F, EtOCH₂, Cl), (M-2757, H, CH₃, F, EtOCH₂, F), (M-2758, H, CH₃, F, EtOCH₂, CF₃), (M-2759, H, CH₃, F, EtOCH₂, Br), (M-2760, H, CH₃, F, EtOCH₂, CH₃), (M-2761, H, CH₃, F, EtOCH₂CH₂, H), (M-2762, H, CH₃, F, EtOCH₂CH₂, Cl), (M-2763, H, CH₃, F, EtOCH₂CH₂, F), (M-2764, H, CH₃, F, EtOCH₂CH₂, CF₃), (M-2765, H, CH₃, F, EtOCH₂CH₂, Br), (M-2766, H, CH₃, F, EtOCH₂CH₂, CH₃), (M-2767, H, CH₃, F, MeOCH₂CH₂OCH₂CH₂, H), (M-2768, H, CH₃, F, MeOCH₂CH₂OCH₂CH₂, Cl), (M-2769, H, CH₃, F, MeOCH₂CH₂OCH₂CH₂, F), (M-2770, H, CH₃, F, MeOCH₂CH₂OCH₂CH₂, CF₃), (M-2771, H, CH₃, F, MeOCH₂CH₂OCH₂CH₂, Br), (M-2772, H, CH₃, F, MeOCH₂CH₂OCH₂CH₂, CH₃), (M-2773, H, CH₃, F, MeOCH₂CH₂, H), (M-2774, H, CH₃, F, MeOCH₂CH₂, Cl), (M-2775, H, CH₃, F, MeOCH₂CH₂, F), (M-2776, H, CH₃, F, MeOCH₂CH₂, CF₃), (M-2777, H, CH₃, F, MeOCH₂CH₂, Br), (M-2778, H, CH₃, F, MeOCH₂CH₂, CH₃), (M-2779, H, CH₃, F, HOCH₂, H), (M-2780, H, CH₃, F, HOCH₂, Cl), (M-2781, H, CH₃, F, HOCH₂, F), (M-2782, H, CH₃, F, HOCH₂, CF₃), (M-2783, H, CH₃, F, HOCH₂, Br), (M-2784, H, CH₃, F, HOCH₂, CH₃), (M-2785, H, CH₃, F, HOCH₂CH₂, H), (M-2786, H, CH₃, F, HOCH₂CH₂, Cl), (M-2787, H, CH₃, F, HOCH₂CH₂, F), (M-2788, H, CH₃, F, HOCH₂CH₂, CF₃), (M-2789, H, CH₃, F, HOCH₂CH₂, Br), (M-2790, H, CH₃, F, HOCH₂CH₂, CH₃), (M-2791, H, CH₃, F, HOCH₂CH₂CH₂, H), (M-2792, H, CH₃, F, HOCH₂CH₂CH₂, Cl), (M-2793, H, CH₃, F, HOCH₂CH₂CH₂, F), (M-2794, H, CH₃, F, HOCH₂CH₂CH₂, CF₃), (M-2795, H, CH₃, F, HOCH₂CH₂CH₂, Br), (M-2796, H, CH₃, F, HOCH₂CH₂CH₂, CH₃), (M-2797, H, CH₃, F, HOCH₂CH₂CH₂CH₂, H), (M-2798, H, CH₃, F, HOCH₂CH₂CH₂CH₂, Cl), (M-2799, H, CH₃, F, HOCH₂CH₂CH₂CH₂, F), (M-2800, H, CH₃, F, HOCH₂CH₂CH₂CH₂, CF₃), (M-2801, H, CH₃, F, HOCH₂CH₂CH₂CH₂, Br), (M-2802, H, CH₃, F, HOCH₂CH₂CH₂CH₂, CH₃), (M-2803, H, CH₃, F, HOCH₂CH₂CH₂CH₂CH₂, H), (M-2804, H, CH₃, F, HOCH₂CH₂CH₂CH₂CH₂, Cl), (M-2805, H, CH₃, F, HOCH₂CH₂CH₂CH₂CH₂, F), (M-2806, H, CH₃, F, HOCH₂CH₂CH₂CH₂CH₂, CF₃), (M-2807, H, CH₃, F, HOCH₂CH₂CH₂CH₂CH₂, Br), (M-2808, H, CH₃, F, HOCH₂CH₂CH₂CH₂CH₂, CH₃), (M-2809, H, CH₃, F, HOCH₂CH₂OCH₂CH₂, H), (M-2810, H, CH₃, F, HOCH₂CH₂OCH₂CH₂, Cl), (M-2811, H, CH₃, F, HOCH₂CH₂OCH₂CH₂, F), (M-2812, H, CH₃, F, HOCH₂CH₂OCH₂CH₂, CF₃), (M-2813, H, CH₃, F, HOCH₂CH₂OCH₂CH₂, Br), (M-2814, H, CH₃, F, HOCH₂CH₂OCH₂CH₂, CH₃), (M-2815, H, CH₃, F, (Me)₂N, H), (M-2816, H, CH₃, F, (Me)₂N, Cl), (M-2817, H, CH₃, F, (Me)₂N, F), (M-2818, H, CH₃, F, (Me)₂N, CF₃), (M-2819, H, CH₃, F, (Me)₂N, Br), (M-2820, H, CH₃, F, (Me)₂N, CH₃), (M-2821, H, CH₃, F, piperidin-4-yl-methyl, H), (M-2822, H, CH₃, F, piperidin-4-yl-methyl, Cl), (M-2823, H, CH₃, F, piperidin-4-yl-methyl, F), (M-2824, H, CH₃, F, piperidin-4-yl-methyl, CF₃), (M-2825, H, CH₃, F, piperidin-4-yl-methyl, Br), (M-2826, H, CH₃, F, piperidin-4-yl-methyl, CH₃), (M-2827, H, CH₃, F, cyclohexylmethyl, H), (M-2828, H, CH₃, F, cyclohexylmethyl, Cl), (M-2829, H, CH₃, F, cyclohexylmethyl, F), (M-2830, H, CH₃, F, cyclohexylmethyl, CF₃), (M-2831, H, CH₃, F, cyclohexylmethyl, Br), (M-2832, H, CH₃, F, cyclohexylmethyl, CH₃), (M-2833, H, CH₃, Cl, H, H), (M-2834, H, CH₃, Cl, H, Cl), (M-2835, H, CH₃, Cl, H, F), (M-2836, H, CH₃, Cl, H, CF₃), (M-2837, H, CH₃, Cl, H, Br), (M-2838, H, CH₃, Cl, H, CH₃), (M-2839, H, CH₃, Cl, F, H), (M-2840, H, CH₃, Cl, F, Cl), (M-2841, H, CH₃, Cl, F, F), (M-2842, H, CH₃, Cl, F, CF₃), (M-2843, H, CH₃, Cl, F, Br), (M-2844, H, CH₃, Cl, F, CH₃), (M-2845, H, CH₃, Cl, Cl, H), (M-2846, H, CH₃, Cl, Cl, Cl), (M-2847, H, CH₃, Cl, Cl, F), (M-2848, H, CH₃, Cl, Cl, CF₃), (M-2849, H, CH₃, Cl, Cl, Br), (M-2850, H, CH₃, Cl, Cl, CH₃), (M-2851, H, CH₃, Cl, CH₃, H), (M-2852, H, CH₃, Cl, CH₃, Cl), (M-2853, H, CH₃, Cl, CH₃, F), (M-2854, H, CH₃, Cl, CH₃, CF₃), (M-2855, H, CH₃, Cl, CH₃, Br), (M-2856, H, CH₃, Cl, CH₃, CH₃), (M-2857, H, CH₃, Cl, Et, H), (M-2858, H, CH₃, Cl, Et, Cl), (M-2859, H, CH₃, Cl, Et, F), (M-2860, H, CH₃, Cl, Et, CF₃), (M-2861, H, CH₃, Cl, Et, Br), (M-2862, H, CH₃, Cl, Et, CH₃), (M-2863, H, CH₃, Cl, n-Pr, H), (M-2864, H, CH₃, Cl, n-Pr, Cl), (M-2865, H, CH₃, Cl, n-Pr, F), (M-2866, H, CH₃, Cl, n-Pr, CF₃), (M-2867, H, CH₃, Cl, n-Pr, Br), (M-2868, H, CH₃, Cl, n-Pr, CH₃), (M-2869, H, CH₃, Cl, c-Pr, H), (M-2870, H, CH₃, Cl, c-Pr, Cl), (M-2871, H, CH₃, Cl, c-Pr, F), (M-2872, H, CH₃, Cl, c-Pr, CF₃), (M-2873, H, CH₃, Cl, c-Pr, Br), (M-2874, H, CH₃, Cl, c-Pr, CH₃), (M-2875, H, CH₃, Cl, i-Pr, H), (M-2876, H, CH₃, Cl, i-Pr, Cl), (M-2877, H, CH₃, Cl, i-Pr, F), (M-2878, H, CH₃, Cl, i-Pr, CF₃), (M-2879, H, CH₃, Cl, i-Pr, Br), (M-2880, H, CH₃, Cl, i-Pr, CH₃), (M-2881, H, CH₃, Cl, n-Bu, H), (M-2882, H, CH₃, Cl, n-Bu, Cl), (M-2883, H, CH₃, Cl, n-Bu, F), (M-2884, H, CH₃, Cl, n-Bu, CF₃), (M-2885, H, CH₃, Cl, n-Bu, Br), (M-2886, H, CH₃, Cl, n-Bu, CH₃), (M-2887, H, CH₃, Cl, i-Bu, H), (M-2888, H,
CH₃, Cl, i-Bu, Cl), (M-2889, H, CH₃, Cl, i-Bu, F), (M-2890, H, CH₃, Cl, i-Bu, CF₃), (M-2891, H, CH₃, Cl, i-Bu, Br), (M-2892, H, CH₃, Cl, i-Bu, CH₃), (M-2893, H, CH₃, Cl, sec-Bu, H), (M-2894, H, CH₃, Cl, sec-Bu, Cl), (M-2895, H, CH₃, Cl, sec-Bu, F), (M-2896, H, CH₃, Cl, sec-Bu, CF₃), (M-2897, H, CH₃, Cl, sec-Bu, Br), (M-2898, H, CH₃, Cl, sec-Bu, CH₃), (M-2899, H, CH₃, Cl, n-Pen, H), (M-2900, H, CH₃, Cl, n-Pen, Cl), (M-2901, H, CH₃, Cl, n-Pen, F), (M-2902, H, CH₃, Cl, n-Pen, CF₃), (M-2903, H, CH₃, Cl, n-Pen, Br), (M-2904, H, CH₃, Cl, n-Pen, CH₃), (M-2905, H, CH₃, Cl, c-Pen, H), (M-2906, H, CH₃, Cl, c-Pen, Cl), (M-2907, H, CH₃, Cl, c-Pen, F), (M-2908, H, CH₃, Cl, c-Pen, CF₃), (M-2909, H, CH₃, Cl, c-Pen, Br), (M-2910, H, CH₃, Cl, c-Pen, CH₃), (M-2911, H, CH₃, Cl, n-Hex, H), (M-2912, H, CH₃, Cl, n-Hex, Cl), (M-2913, H, CH₃, Cl, n-Hex, F), (M-2914, H, CH₃, Cl, n-Hex, CF₃), (M-2915, H, CH₃, Cl, n-Hex, Br), (M-2916, H, CH₃, Cl, n-Hex, CH₃), (M-2917, H, CH₃, Cl, c-Hex, H), (M-2918, H, CH₃, Cl, c-Hex, Cl), (M-2919, H, CH₃, Cl, c-Hex, F), (M-2920, H, CH₃, Cl, c-Hex, CF₃), (M-2921, H, CH₃, Cl, c-Hex, Br), (M-2922, H, CH₃, Cl, c-Hex, CH₃), (M-2923, H, CH₃, Cl, OH, H), (M-2924, H, CH₃, Cl, OH, Cl), (M-2925, H, CH₃, Cl, OH, F), (M-2926, H, CH₃, Cl, OH, CF₃), (M-2927, H, CH₃, Cl, OH, Br), (M-2928, H, CH₃, Cl, OH, CH₃), (M-2929, H, CH₃, Cl, EtO, H), (M-2930, H, CH₃, Cl, EtO, Cl), (M-2931, H, CH₃, Cl, EtO, F), (M-2932, H, CH₃, Cl, EtO, CF₃), (M-2933, H, CH₃, Cl, EtO, Br), (M-2934, H, CH₃, Cl, EtO, CH₃), (M-2935, H, CH₃, Cl, n-PrO, H), (M-2936, H, CH₃, Cl, n-PrO, Cl), (M-2937, H, CH₃, Cl, n-PrO, F), (M-2938, H, CH₃, Cl, n-PrO, CF₃), (M-2939, H, CH₃, Cl, n-PrO, Br), (M-2940, H, CH₃, Cl, n-PrO, CH₃), (M-2941, H, CH₃, Cl, PhO, H), (M-2942, H, CH₃, Cl, PhO, Cl), (M-2943, H, CH₃, Cl, PhO, F), (M-2944, H, CH₃, Cl, PhO, CF₃), (M-2945, H, CH₃, Cl, PhO, Br), (M-2946, H, CH₃, Cl, PhO, CH₃), (M-2947, H, CH₃, Cl, BnO, H), (M-2948, H, CH₃, Cl, BnO, Cl), (M-2949, H, CH₃, Cl, BnO, F), (M-2950, H, CH₃, Cl, BnO, CF₃), (M-2951, H, CH₃, Cl, BnO, Br), (M-2952, H, CH₃, Cl, BnO, CH₃), (M-2953, H, CH₃, Cl, PhCH₂CH₂O, H), (M-2954, H, CH₃, Cl, PhCH₂CH₂O, Cl), (M-2955, H, CH₃, Cl, PhCH₂CH₂O, F), (M-2956, H, CH₃, Cl, PhCH₂CH₂O, CF₃), (M-2957, H, CH₃, Cl, PhCH₂CH₂O, Br), (M-2958, H, CH₃, Cl, PhCH₂CH₂O, CH₃), (M-2959, H, CH₃, Cl, CF₃O, H), (M-2960, H, CH₃, Cl, CF₃O, Cl), (M-2961, H, CH₃, Cl, CF₃O, F), (M-2962, H, CH₃, Cl, CF₃O, CF₃), (M-2963, H, CH₃, Cl, CF₃O, Br), (M-2964, H, CH₃, Cl, CF₃O, CH₃), (M-2965, H, CH₃, Cl, Ph, H), (M-2966, H, CH₃, Cl, Ph, Cl), (M-2967, H, CH₃, Cl, Ph, F), (M-2968, H, CH₃, Cl, Ph, CF₃), (M-2969, H, CH₃, Cl, Ph, Br), (M-2970, H, CH₃, Cl, Ph, CH₃), (M-2971, H, CH₃, Cl, 4-F-Ph, H), (M-2972, H, CH₃, Cl, 4-F-Ph, Cl), (M-2973, H, CH₃, Cl, 4-F-Ph, F), (M-2974, H, CH₃, Cl, 4-F-Ph, CF₃), (M-2975, H, CH₃, Cl, 4-F-Ph, Br), (M-2976, H, CH₃, Cl, 4-F-Ph, CH₃), (M-2977, H, CH₃, Cl, 4-CF₃-Ph, H), (M-2978, H, CH₃, Cl, 4-CF₃-Ph, Cl), (M-2979, H, CH₃, Cl, 4-CF₃-Ph, F), (M-2980, H, CH₃, Cl, 4-CF₃-Ph, CF₃), (M-2981, H, CH₃, Cl, 4-CF₃-Ph, Br), (M-2982, H, CH₃, Cl, 4-CF₃-Ph, CH₃), (M-2983, H, CH₃, Cl, 4-(Me)₂N-Ph, H), (M-2984, H, CH₃, Cl, 4-(Me)₂N-Ph, Cl), (M-2985, H, CH₃, Cl, 4-(Me)₂N-Ph, F), (M-2986, H, CH₃, Cl, 4-(Me)₂N-Ph, CF₃), (M-2987, H, CH₃, Cl, 4-(Me)₂N-Ph, Br), (M-2988, H, CH₃, Cl, 4-(Me)₂N-Ph, CH₃), (M-2989, H, CH₃, Cl, 4-OH-Ph, H), (M-2990, H, CH₃, Cl, 4-OH-Ph, Cl), (M-2991, H, CH₃, Cl, 4-OH-Ph, F), (M-2992, H, CH₃, Cl, 4-OH-Ph, CF₃), (M-2993, H, CH₃, Cl, 4-OH-Ph, Br), (M-2994, H, CH₃, Cl, 4-OH-Ph, CH₃), (M-2995, H, CH₃, Cl, 3,4-di-F-Ph, H), (M-2996, H, CH₃, Cl, 3,4-di-F-Ph, Cl), (M-2997, H, CH₃, Cl, 3,4-di-F-Ph, F), (M-2998, H, CH₃, Cl, 3,4-di-F-Ph, CF₃), (M-2999, H, CH₃, Cl, 3,4-di-F-Ph, Br), (M-3000, H, CH₃, Cl, 3,4-di-F-Ph, CH₃), (M-3001, H, CH₃, Cl, 4-COOH-Ph, H), (M-3002, H, CH₃, Cl, 4-COOH-Ph, Cl), (M-3003, H, CH₃, Cl, 4-COOH-Ph, F), (M-3004, H, CH₃, Cl, 4-COOH-Ph, CF₃), (M-3005, H, CH₃, Cl, 4-COOH-Ph, Br), (M-3006, H, CH₃, Cl, 4-COOH-Ph, CH₃), (M-3007, H, CH₃, Cl, Bn, H), (M-3008, H, CH₃, Cl, Bn, Cl), (M-3009, H, CH₃, Cl, Bn, F), (M-3010, H, CH₃, Cl, Bn, CF₃), (M-3011, H, CH₃, Cl, Bn, Br), (M-3012, H, CH₃, Cl, Bn, CH₃), (M-3013, H, CH₃, Cl, 4-F-Bn, H), (M-3014, H, CH₃, Cl, 4-F-Bn, Cl), (M-3015, H, CH₃, Cl, 4-F-Bn, F), (M-3016, H, CH₃, Cl, 4-F-Bn, CF₃), (M-3017, H, CH₃, Cl, 4-F-Bn, Br), (M-3018, H, CH₃, Cl, 4-F-Bn, CH₃), (M-3019, H, CH₃, Cl, 2-Py, H), (M-3020, H, CH₃, Cl, 2-Py, Cl), (M-3021, H, CH₃, Cl, 2-Py, F), (M-3022, H, CH₃, Cl, 2-Py, CF₃), (M-3023, H, CH₃, Cl, 2-Py, Br), (M-3024, H, CH₃, Cl, 2-Py, CH₃), (M-3025, H, CH₃, Cl, 3-Py, H), (M-3026, H, CH₃, Cl, 3-Py, Cl), (M-3027, H, CH₃, Cl, 3-Py, F), (M-3028, H, CH₃, Cl, 3-Py, CF₃), (M-3029, H, CH₃, Cl, 3-Py, Br), (M-3030, H, CH₃, Cl, 3-Py, CH₃), (M-3031, H, CH₃, Cl, 4-Py, H), (M-3032, H, CH₃, Cl, 4-Py, Cl), (M-3033, H, CH₃, Cl, 4-Py, F), (M-3034, H, CH₃, Cl, 4-Py, CF₃), (M-3035, H, CH₃, Cl, 4-Py, Br), (M-3036, H, CH₃, Cl, 4-Py, CH₃), (M-3037, H, CH₃, Cl, 2-Th, H), (M-3038, H, CH₃, Cl, 2-Th, Cl), (M-3039, H, CH₃, Cl, 2-Th, F), (M-3040, H, CH₃, Cl, 2-Th, CF₃), (M-3041, H, CH₃, Cl, 2-Th, Br), (M-3042, H, CH₃, Cl, 2-Th, CH₃), (M-3043, H, CH₃, Cl, 3-Th, H), (M-3044, H, CH₃, Cl, 3-Th, Cl), (M-3045, H, CH₃, Cl, 3-Th, F), (M-3046, H, CH₃, Cl, 3-Th, CF₃), (M-3047, H, CH₃, Cl, 3-Th, Br), (M-3048, H, CH₃, Cl, 3-Th, CH₃), (M-3049, H, CH₃, Cl, pyrazol-2-yl, H), (M-3050, H, CH₃, Cl, pyrazol-2-yl, Cl), (M-3051, H, CH₃, Cl, pyrazol-2-yl, F), (M-3052, H, CH₃, Cl, pyrazol-2-yl, CF₃), (M-3053, H, CH₃, Cl, pyrazol-2-yl, Br), (M-3054, H, CH₃, Cl, pyrazol-2-yl, CH₃), (M-3055, H, CH₃, Cl, pyrazol-3-yl, H), (M-3056, H, CH₃, Cl, pyrazol-3-yl, Cl), (M-3057, H, CH₃, Cl, pyrazol-3-yl, F), (M-3058, H, CH₃, Cl, pyrazol-3-yl, CF₃), (M-3059, H, CH₃, Cl, pyrazol-3-yl, Br), (M-3060, H, CH₃, Cl, pyrazol-3-yl, CH₃), (M-3061, H, CH₃, Cl, pyrimidin-2-yl, H), (M-3062, H, CH₃, Cl, pyrimidin-2-yl, Cl), (M-3063, H, CH₃, Cl, pyrimidin-2-yl, F), (M-3064, H, CH₃, Cl, pyrimidin-2-yl, CF₃), (M-3065, H, CH₃, Cl, pyrimidin-2-yl, Br), (M-3066, H, CH₃, Cl, pyrimidin-2-yl, CH₃), (M-3067, H, CH₃, Cl, pyrimidin-4-yl, H), (M-3068, H, CH₃, Cl, pyrimidin-4-yl, Cl), (M-3069, H, CH₃, Cl, pyrimidin-4-yl, F), (M-3070, H, CH₃, Cl, pyrimidin-4-yl, CF₃), (M-3071, H, CH₃, Cl, pyrimidin-4-yl, Br), (M-3072, H, CH₃, Cl, pyrimidin-4-yl, CH₃), (M-3073, H, CH₃, Cl, pyrimidin-5-yl, H), (M-3074, H, CH₃, Cl, pyrimidin-5-yl, Cl), (M-3075, H, CH₃, Cl, pyrimidin-5-yl, F), (M-3076, H, CH₃, Cl, pyrimidin-5-yl, CF₃), (M-3077, H, CH₃, Cl, pyrimidin-5-yl, Br), (M-3078, H, CH₃, Cl, pyrimidin-5-yl, CH₃), (M-3079, H, CH₃, Cl, HOOCCH₂CH₂CH₂, H), (M-3080, H, CH₃, Cl, HOOCCH₂CH₂CH₂, Cl), (M-3081, H, CH₃, Cl, HOOCCH₂CH₂CH₂, F), (M-3082, H, CH₃, Cl, HOOCCH₂CH₂CH₂, CF₃), (M-3083, H, CH₃, Cl, HOOCCH₂CH₂CH₂, Br), (M-3084, H, CH₃, Cl, HOOCCH₂CH₂CH₂, CH₃),
(M-3085, H, CH₃, Cl, HOOCCH₂CH₂CH₂CH₂, H), (M-3086, H, CH₃, Cl, HOOCCH₂CH₂CH₂CH₂, Cl), (M-3087, H, CH₃, Cl, HOOCCH₂CH₂CH₂CH₂, F), (M-3088, H, CH₃, Cl, HOOCCH₂CH₂CH₂CH₂, CF₃), (M-3089, H, CH₃, Cl, HOOCCH₂CH₂CH₂CH₂, Br), (M-3090, H, CH₃, Cl, HOOCCH₂CH₂CH₂CH₂, CH₃), (M-3091, H, CH₃, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂, H), (M-3092, H, CH₃, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂, Cl), (M-3093, H, CH₃, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂, F), (M-3094, H, CH₃, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂, CF₃), (M-3095, H, CH₃, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂, Br), (M-3096, H, CH₃, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂, CH₃), (M-3097, H, CH₃, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, H), (M-3098, H, CH₃, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, Cl), (M-3099, H, CH₃, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, F), (M-3100, H, CH₃, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, CF₃), (M-3101, H, CH₃, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, Br), (M-3102, H, CH₃, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, CH₃), (M-3103, H, CH₃, Cl, MeOCH₂, H), (M-3104, H, CH₃, Cl, MeOCH₂, Cl), (M-3105, H, CH₃, Cl, MeOCH₂, F), (M-3106, H, CH₃, Cl, MeOCH₂, CF₃), (M-3107, H, CH₃, Cl, MeOCH₂, Br), (M-3108, H, CH₃, Cl, MeOCH₂, CH₃), (M-3109, H, CH₃, Cl, EtOCH₂, H), (M-3110, H, CH₃, Cl, EtOCH₂, Cl), (M-3111, H, CH₃, Cl, EtOCH₂, F), (M-3112, H, CH₃, Cl, EtOCH₂, CF₃), (M-3113, H, CH₃, Cl, EtOCH₂, Br), (M-3114, H, CH₃, Cl, EtOCH₂, CH₃), (M-3115, H, CH₃, Cl, EtOCH₂CH₂, H), (M-3116, H, CH₃, Cl, EtOCH₂CH₂, Cl), (M-3117, H, CH₃, Cl, EtOCH₂CH₂, F), (M-3118, H, CH₃, Cl, EtOCH₂CH₂, CF₃), (M-3119, H, CH₃, Cl, EtOCH₂CH₂, Br), (M-3120, H, CH₃, Cl, EtOCH₂CH₂, CH₃), (M-3121, H, CH₃, Cl, MeOCH₂CH₂OCH₂CH₂, H), (M-3122, H, CH₃, Cl, MeOCH₂CH₂OCH₂CH₂, Cl), (M-3123, H, CH₃, Cl, MeOCH₂CH₂OCH₂CH₂, F), (M-3124, H, CH₃, Cl, MeOCH₂CH₂OCH₂CH₂, CF₃), (M-3125, H, CH₃, Cl, MeOCH₂CH₂OCH₂CH₂, Br), (M-3126, H, CH₃, Cl, MeOCH₂CH₂OCH₂CH₂, CH₃), (M-3127, H, CH₃, Cl, MeOCH₂CH₂, H), (M-3128, H, CH₃, Cl, MeOCH₂CH₂, Cl), (M-3129, H, CH₃, Cl, MeOCH₂CH₂, F), (M-3130, H, CH₃, Cl, MeOCH₂CH₂, CF₃), (M-3131, H, CH₃, Cl, MeOCH₂CH₂, Br), (M-3132, H, CH₃, Cl, MeOCH₂CH₂, CH₃), (M-3133, H, CH₃, Cl, HOCH₂, H), (M-3134, H, CH₃, Cl, HOCH₂, Cl), (M-3135, H, CH₃, Cl, HOCH₂, F), (M-3136, H, CH₃, Cl, HOCH₂, CF₃), (M-3137, H, CH₃, Cl, HOCH₂, Br), (M-3138, H, CH₃, Cl, HOCH₂, CH₃), (M-3139, H, CH₃, Cl, HOCH₂CH₂, H), (M-3140, H, CH₃, Cl, HOCH₂CH₂, Cl), (M-3141, H, CH₃, Cl, HOCH₂CH₂, F), (M-3142, H, CH₃, Cl, HOCH₂CH₂, CF₃), (M-3143, H, CH₃, Cl, HOCH₂CH₂, Br), (M-3144, H, CH₃, Cl, HOCH₂CH₂, CH₃), (M-3145, H, CH₃, Cl, HOCH₂CH₂CH₂, H), (M-3146, H, CH₃, Cl, HOCH₂CH₂CH₂, Cl), (M-3147, H, CH₃, Cl, HOCH₂CH₂CH₂, F), (M-3148, H, CH₃, Cl, HOCH₂CH₂CH₂, CF₃), (M-3149, H, CH₃, Cl, HOCH₂CH₂CH₂, Br), (M-3150, H, CH₃, Cl, HOCH₂CH₂CH₂, CH₃), (M-3151, H, CH₃, Cl, HOCH₂CH₂CH₂CH₂, H), (M-3152, H, CH₃, Cl, HOCH₂CH₂CH₂CH₂, Cl), (M-3153, H, CH₃, Cl, HOCH₂CH₂CH₂CH₂, F), (M-3154, H, CH₃, Cl, HOCH₂CH₂CH₂CH₂, CF₃), (M-3155, H, CH₃, Cl, HOCH₂CH₂CH₂CH₂, Br), (M-3156, H, CH₃, Cl, HOCH₂CH₂CH₂CH₂, CH₃), (M-3157, H, CH₃, Cl, HOCH₂CH₂CH₂CH₂CH₂, H), (M-3158, H, CH₃, Cl, HOCH₂CH₂CH₂CH₂CH₂, Cl), (M-3159, H, CH₃, Cl, HOCH₂CH₂CH₂CH₂CH₂, F), (M-3160, H, CH₃, Cl, HOCH₂CH₂CH₂CH₂CH₂, CF₃), (M-3161, H, CH₃, Cl, HOCH₂CH₂CH₂CH₂CH₂, Br), (M-3162, H, CH₃, Cl, HOCH₂CH₂CH₂CH₂CH₂, CH₃), (M-3163, H, CH₃, Cl, HOCH₂CH₂OCH₂CH₂, H), (M-3164, H, CH₃, Cl, HOCH₂CH₂OCH₂CH₂, Cl), (M-3165, H, CH₃, Cl, HOCH₂CH₂OCH₂CH₂, F), (M-3166, H, CH₃, Cl, HOCH₂CH₂OCH₂CH₂, CF₃), (M-3167, H, CH₃, Cl, HOCH₂CH₂OCH₂CH₂, Br), (M-3168, H, CH₃, Cl, HOCH₂CH₂OCH₂CH₂, CH₃), (M-3169, H, CH₃, Cl, (Me)₂N, H), (M-3170, H, CH₃, Cl, (Me)₂N, Cl), (M-3171, H, CH₃, Cl, (Me)₂N, F), (M-3172, H, CH₃, Cl, (Me)₂N, CF₃), (M-3173, H, CH₃, Cl, (Me)₂N, Br), (M-3174, H, CH₃, Cl, (Me)₂N, CH₃), (M-3175, H, CH₃, Cl, piperidin-4-yl-methyl, H), (M-3176, H, CH₃, Cl, piperidin-4-yl-methyl, Cl), (M-3177, H, CH₃, Cl, piperidin-4-yl-methyl, F), (M-3178, H, CH₃, Cl, piperidin-4-yl-methyl, CF₃), (M-3179, H, CH₃, Cl, piperidin-4-yl-methyl, Br), (M-3180, H, CH₃, Cl, piperidin-4-yl-methyl, CH₃), (M-3181, H, CH₃, Cl, cyclohexylmethyl, H), (M-3182, H, CH₃, Cl, cyclohexylmethyl, Cl), (M-3183, H, CH₃, Cl, cyclohexylmethyl, F), (M-3184, H, CH₃, Cl, cyclohexylmethyl, CF₃), (M-3185, H, CH₃, Cl, cyclohexylmethyl, Br), (M-3186, H, CH₃, Cl, cyclohexylmethyl, CH₃), (M-3187, F, H, H, H, H), (M-3188, F, H, H, H, Cl), (M-3189, MeO, F, H, H, CF₃), (M-3190, MeO, F, F, H, CF₃), (M-3191, F, H, H, H, Br), (M-3192, F, H, H, H, CH₃), (M-3193, F, H, H, F, H), (M-3194, F, H, H, F, Cl), (M-3195, F, H, H, F, F), (M-3196, F, H, H, F, CF₃), (M-3197, F, H, H, F, Br), (M-3198, F, H, H, F, CH₃), (M-3199, F, H, H, Cl, H), (M-3200, MeO, F, H, H, n-Pr), (M-3201, F, H, H, Cl, F), (M-3202, F, H, H, Cl, CF₃), (M-3203, F, H, H, Cl, Br), (M-3204, F, H, H, Cl, CH₃), (M-3205, F, H, H, CH₃, H), (M-3206, F, H, H, CH₃, Cl), (M-3207, F, H, H, CH₃, F), (M-3208, F, H, H, CH₃, CF₃), (M-3209, F, H, H, CH₃, Br), (M-3210, F, H, H, CH₃, CH₃), (M-3211, F, H, H, Et, H), (M-3212, F, H, H, Et, Cl), (M-3213, F, H, H, Et, F), (M-3214, F, H, H, Et, CF₃), (M-3215, F, H, H, Et, Br), (M-3216, F, H, H, Et, CH₃), (M-3217, F, H, H, n-Pr, H), (M-3218, F, H, H, n-Pr, Cl), (M-3219, F, H, H, n-Pr, F), (M-3220, F, H, H, n-Pr, CF₃), (M-3221, F, H, H, n-Pr, Br), (M-3222, F, H, H, n-Pr, CH₃), (M-3223, F, H, H, c-Pr, H), (M-3224, F, H, H, c-Pr, Cl), (M-3225, F, H, H, c-Pr, F), (M-3226, F, H, H, c-Pr, CF₃), (M-3227, F, H, H, c-Pr, Br), (M-3228, F, H, H, c-Pr, CH₃), (M-3229, F, H, H, i-Pr, H), (M-3230, F, H, H, i-Pr, Cl), (M-3231, F, H, H, i-Pr, F), (M-3232, F, H, H, i-Pr, CF₃), (M-3233, F, H, H, i-Pr, Br), (M-3234, F, H, H, i-Pr, CH₃), (M-3235, F, H, H, n-Bu
, H), (M-3236, F, H, H, n-Bu, Cl), (M-3237, F, H, H, n-Bu, F), (M-3238, F, H, H, n-Bu, CF₃), (M-3239, F, H, H, n-Bu, Br), (M-3240, F, H, H, n-Bu, CH₃), (M-3241, F, H, H, i-Bu, H), (M-3242, F, H, H, i-Bu, Cl), (M-3243, F, H, H, i-Bu, F), (M-3244, F, H, H, i-Bu, CF₃), (M-3245, F, H, H, i-Bu, Br), (M-3246, F, H, H, i-Bu, CH₃), (M-3247, F, H, H, sec-Bu, H), (M-3248, F, H, H, sec-Bu, Cl), (M-3249, F, H, H, sec-Bu, F), (M-3250, F, H, H, sec-Bu, CF₃), (M-3251, F, H, H, sec-Bu, Br), (M-3252, F, H, H, sec-Bu, CH₃), (M-3253, F, H, H, n-Pen, H), (M-3254, F, H, H, n-Pen, Cl), (M-3255, F, H, H, n-Pen, F), (M-3256, F, H, H, n-Pen, CF₃), (M-3257, F, H, H, n-Pen, Br), (M-3258, F, H, H, n-Pen, CH₃), (M-3259, F, H, H, c-Pen, H), (M-3260, F, H, H, c-Pen, Cl), (M-3261, F, H, H, c-Pen, F), (M-3262, F, H, H, c-Pen, CF₃), (M-3263, F, H, H, c-Pen, Br), (M-3264, F, H, H, c-Pen, CH₃), (M-3265, F, H, H, n-Hex, H), (M-3266, F, H, H, n-Hex, Cl), (M-3267, F, H, H, n-Hex, F), (M-3268, F, H, H, n-Hex, CF₃), (M-3269, F, H, H, n-Hex, Br), (M-3270, F, H, H, n-Hex, CH₃), (M-3271, F, H, H, c-Hex, H), (M-3272, F, H, H, c-Hex, Cl), (M-3273, F, H, H, c-Hex, F), (M-3274, F, H, H, c-Hex, CF₃), (M-3275, F, H, H, c-Hex, Br), (M-3276, F, H, H, c-Hex, CH₃), (M-3277, F, H, H, OH, H), (M-3278, F, H, H, OH, Cl), (M-3279, F, H, H, OH, F), (M-3280, F, H, H, OH, CF₃), (M-3281, F, H, H, OH, Br), (M-3282, F, H, H, OH, CH₃), (M-3283, F, H, H, EtO, H), (M-3284, F, H, H, EtO, Cl), (M-3285, F, H, H, EtO, F), (M-3286, F, H, H, EtO, CF₃), (M-3287, F, H, H, EtO, Br), (M-3288, F, H, H, EtO, CH₃), (M-3289, F, H, H, n-PrO, H), (M-3290, F, H, H, n-PrO, Cl), (M-3291, F, H, H, n-PrO, F), (M-3292, F, H, H, n-PrO, CF₃), (M-3293, F, H, H, n-PrO, Br), (M-3294, F, H, H, n-PrO, CH₃), (M-3295, F, H, H, PhO, H), (M-3296, F, H, H, PhO, Cl), (M-3297, F, H, H, PhO, F), (M-3298, F, H, H, PhO, CF₃), (M-3299, F, H, H, PhO, Br), (M-3300, F, H, H, PhO, CH₃), (M-3301, F, H, H, BnO, H), (M-3302, F, H, H, BnO, Cl), (M-3303, F, H, H, BnO, F), (M-3304, F, H, H, BnO, CF₃), (M-3305, F, H, H, BnO, Br), (M-3306, F, H, H, BnO, CH₃), (M-3307, F, H, H, PhCH₂CH₂O, H), (M-3308, F, H, H, PhCH₂CH₂O, Cl), (M-3309, F, H, H, PhCH₂CH₂O, F), (M-3310, F, H, H, PhCH₂CH₂O, CF₃), (M-3311, F, H, H, PhCH₂CH₂O, Br), (M-3312, F, H, H, PhCH₂CH₂O, CH₃), (M-3313, MeO, H, H, CF3O, CH3), (M-3314, F, H, H, CF₃O, Cl), (M-3315, F, H, H, CF₃O, F), (M-3316, F, H, H, CF₃O, CF₃), (M-3317, F, H, H, CF₃O, Br), (M-3318, F, H, H, CF₃O, CH₃), (M-3319, F, H, H, Ph, H), (M-3320, F, H, H, Ph, Cl), (M-3321, F, H, H, Ph, F), (M-3322, F, H, H, Ph, CF₃), (M-3323, F, H, H, Ph, Br), (M-3324, F, H, H, Ph, CH₃), (M-3325, F, H, H, 4-F-Ph, H), (M-3326, F, H, H, 4-F-Ph, Cl), (M-3327, F, H, H, 4-F-Ph, F), (M-3328, F, H, H, 4-F-Ph, CF₃), (M-3329, F, H, H, 4-F-Ph, Br), (M-3330, F, H, H, 4-F-Ph, CH₃), (M-3331, F, H, H, 4-CF₃-Ph, H), (M-3332, F, H, H, 4-CF₃-Ph, Cl), (M-3333, F, H, H, 4-CF₃-Ph, F), (M-3334, F, H, H, 4-CF₃-Ph, CF₃), (M-3335, F, H, H, 4-CF₃-Ph, Br), (M-3336, F, H, H, 4-CF₃-Ph, CH₃), (M-3337, F, H, H, 4-(Me)₂N-Ph, H), (M-3338, F, H, H, 4-(Me)₂N-Ph, Cl), (M-3339, F, H, H, 4-(Me)₂N-Ph, F), (M-3340, F, H, H, 4-(Me)₂N-Ph, CF₃), (M-3341, F, H, H, 4-(Me)₂N-Ph, Br), (M-3342, F, H, H, 4-(Me)₂N-Ph, CH₃), (M-3343, F, H, H, 4-OH-Ph, H), (M-3344, F, H, H, 4-OH-Ph, Cl), (M-3345, F, H, H, 4-OH-Ph, F), (M-3346, F, H, H, 4-OH-Ph, CF₃), (M-3347, F, H, H, 4-OH-Ph, Br), (M-3348, F, H, H, 4-OH-Ph, CH₃), (M-3349, F, H, H, 3,4-di-F-Ph, H), (M-3350, F, H, H, 3,4-di-F-Ph, Cl), (M-3351, F, H, H, 3,4-di-F-Ph, F), (M-3352, F, H, H, 3,4-di-F-Ph, CF₃), (M-3353, F, H, H, 3,4-di-F-Ph, Br), (M-3354, F, H, H, 3,4-di-F-Ph, CH₃), (M-3355, F, H, H, 4-COOH-Ph, H), (M-3356, F, H, H, 4-COOH-Ph, Cl), (M-3357, F, H, H, 4-COOH-Ph, F), (M-3358, F, H, H, 4-COOH-Ph, CF₃), (M-3359, F, H, H, 4-COOH-Ph, Br), (M-3360, F, H, H, 4-COOH-Ph, CH₃), (M-3361, F, H, H, Bn, H), (M-3362, F, H, H, Bn, Cl), (M-3363, F, H, H, Bn, F), (M-3364, F, H, H, Bn, CF₃), (M-3365, F, H, H, Bn, Br), (M-3366, F, H, H, Bn, CH₃), (M-3367, F, H, H, 4-F-Bn, H), (M-3368, F, H, H, 4-F-Bn, Cl), (M-3369, F, H, H, 4-F-Bn, F), (M-3370, F, H, H, 4-F-Bn, CF₃), (M-3371, F, H, H, 4-F-Bn, Br), (M-3372, F, H, H, 4-F-Bn, CH₃), (M-3373, F, H, H, 2-Py, H), (M-3374, F, H, H, 2-Py, Cl), (M-3375, F, H, H, 2-Py, F), (M-3376, F, H, H, 2-Py, CF₃), (M-3377, F, H, H, 2-Py, Br), (M-3378, F, H, H, 2-Py, CH₃), (M-3379, F, H, H, 3-Py, H), (M-3380, F, H, H, 3-Py, Cl), (M-3381, F, H, H, 3-Py, F), (M-3382, F, H, H, 3-Py, CF₃), (M-3383, F, H, H, 3-Py, Br), (M-3384, F, H, H, 3-Py, CH₃), (M-3385, F, H, H, 4-Py, H), (M-3386, F, H, H, 4-Py, Cl), (M-3387, F, H, H, 4-Py, F), (M-3388, F, H, H, 4-Py, CF₃), (M-3389, F, H, H, 4-Py, Br), (M-3390, F, H, H, 4-Py, CH₃), (M-3391, F, H, H, 2-Th, H), (M-3392, F, H, H, 2-Th, Cl), (M-3393, F, H, H, 2-Th, F), (M-3394, F, H, H, 2-Th, CF₃), (M-3395, F, H, H, 2-Th, Br), (M-3396, F, H, H, 2-Th, CH₃), (M-3397, F, H, H, 3-Th, H), (M-3398, F, H, H, 3-Th, Cl), (M-3399, F, H, H, 3-Th, F), (M-3400, F, H, H, 3-Th, CF₃), (M-3401, F, H, H, 3-Th, Br), (M-3402, F, H, H, 3-Th, CH₃), (M-3403, F, H, H, pyrazol-2-yl, H), (M-3404, F, H, H, pyrazol-2-yl, Cl), (M-3405, F, H, H, pyrazol-2-yl, F), (M-3406, F, H, H, pyrazol-2-yl, CF₃), (M-3407, F, H, H, pyrazol-2-yl, Br), (M-3408, F, H, H, pyrazol-2-yl, CH₃), (M-3409, F, H, H, pyrazol-3-yl, H), (M-3410, F, H, H, pyrazol-3-yl, Cl), (M-3411, F, H, H, pyrazol-3-yl, F), (M-3412, F, H, H, pyrazol-3-yl, CF₃), (M-3413, F, H, H, pyrazol-3-yl, Br), (M-3414, F, H, H, pyrazol-3-yl, CH₃), (M-3415, F, H, H, pyrimidin-2-yl, H), (M-3416, F, H, H, pyrimidin-2-yl, Cl), (M-3417, F, H, H, pyrimidin-2-yl, F), (M-3418, F, H, H, pyrimidin-2-yl, CF₃), (M-3419, F, H, H, pyrimidin-2-yl, Br), (M-3420, F, H, H, pyrimidin-2-yl, CH₃), (M-3421, F, H, H, pyrimidin-4-yl, H), (M-3422, F, H, H, pyrimidin-4-yl, Cl), (M-3423, F, H, H, pyrimidin-4-yl, F), (M-3424, F, H, H, pyrimidin-4-yl, CF₃), (M-3425, F, H, H, pyrimidin-4-yl, Br), (M-3426, F, H, H, pyrimidin-4-yl, CH₃), (M-3427, F, H, H, pyrimidin-5-yl, H), (M-3428, F, H, H, pyrimidin-5-yl, Cl), (M-3429, F, H, H, pyrimidin-5-yl, F), (M-3430, F, H, H, pyrimidin-5-yl, CF₃), (M-3431, F, H, H, pyrimidin-5-yl, Br), (M-3432, F, H, H, pyrimidin-5-yl, CH₃), (M-3433, F, H, H, HOOCCH₂CH₂CH₂, H), (M-3434, F, H, H, HOOCCH₂CH₂CH₂, Cl), (M-3435, F, H, H, HOOCCH₂CH₂CH₂, F), (M-3436, F, H, H, HOOCCH₂CH₂CH₂, CF₃), (M-3437, F, H, H, HOOCCH₂CH₂CH₂, Br), (M-3438, F, H, H, HOOCCH₂CH₂CH₂, CH₃), (M-3439, F, H, H, HOOCCH₂CH₂CH₂CH₂, H), (M-3440, F, H, H, HOOCCH₂CH₂CH₂CH₂, Cl), (M-3441, F, H, H, HOOCCH₂CH₂CH₂CH₂, F), (M-3442, F, H, H, HOOCCH₂CH₂CH₂CH₂, CF₃), (M-3443, F, H, H, HOOCCH₂CH₂CH₂CH₂, Br), (M-3444, F, H, H, HOOCCH₂CH₂CH₂CH₂, CH₃), (M-3445, F, H, H, (Me)₂NCOCH₂CH₂CH₂CH₂, H), (M-3446, F, H, H, (Me)₂NCOCH₂CH₂CH₂CH₂, Cl), (M-3447, F, H, H, (Me)₂NCOCH₂CH₂CH₂CH₂, F), (M-3448, F, H, H, (Me)₂NCOCH₂CH₂CH₂CH₂, CF₃), (M-3449, F, H, H, (Me)₂NCOCH₂CH₂CH₂CH₂, Br), (M-3450, F, H, H, (Me)₂NCOCH₂CH₂CH₂CH₂, CH₃), (M-3451, F, H, H, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, H), (M-3452, F, H, H, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, Cl), (M-3453, F, H, H, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, F), (M-3454, F, H, H, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, CF₃), (M-3455, F, H, H, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, Br), (M-3456, F, H, H, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, CH₃), (M-3457, F, H, H, MeOCH₂, H), (M-3458, F, H, H, MeOCH₂, Cl), (M-3459, F, H, H, MeOCH₂, F), (M-3460, F, H, H, MeOCH₂, CF₃), (M-3461, F, H, H, MeOCH₂, Br), (M-3462, F, H, H, MeOCH₂, CH₃), (M-3463, F, H, H, EtOCH₂, H), (M-3464, F, H, H, EtOCH₂, Cl), (M-3465, F, H, H, EtOCH₂, F), (M-3466, F, H, H, EtOCH₂, CF₃), (M-3467, F, H, H, EtOCH₂, Br), (M-3468, F, H, H, EtOCH₂, CH₃), (M-3469, F, H, H, EtOCH₂CH₂, H), (M-3470, F, H, H, EtOCH₂CH₂, Cl), (M-3471, F, H, H, EtOCH₂
CH₂, F), (M-3472, F, H, H, EtOCH₂CH₂, CF₃), (M-3473, F, H, H, EtOCH₂CH₂, Br), (M-3474, F, H, H, EtOCH₂CH₂, CH₃), (M-3475, F, H, H, MeOCH₂CH₂OCH₂CH₂, H), (M-3476, F, H, H, MeOCH₂CH₂OCH₂CH₂, Cl), (M-3477, F, H, H, MeOCH₂CH₂OCH₂CH₂, F), (M-3478, F, H, H, MeOCH₂CH₂OCH₂CH₂, CF₃), (M-3479, F, H, H, MeOCH₂CH₂OCH₂CH₂, Br), (M-3480, F, H, H, MeOCH₂CH₂OCH₂CH₂, CH₃), (M-3481, F, H, H, MeOCH₂CH₂, H), (M-3482, F, H, H, MeOCH₂CH₂, Cl), (M-3483, F, H, H, MeOCH₂CH₂, F), (M-3484, F, H, H, MeOCH₂CH₂, CF₃), (M-3485, F, H, H, MeOCH₂CH₂, Br), (M-3486, F, H, H, MeOCH₂CH₂, CH₃), (M-3487, F, H, H, HOCH₂, H), (M-3488, F, H, H, HOCH₂, Cl), (M-3489, F, H, H, HOCH₂, F), (M-3490, F, H, H, HOCH₂, CF₃), (M-3491, F, H, H, HOCH₂, Br), (M-3492, F, H, H, HOCH₂, CH₃), (M-3493, F, H, H, HOCH₂CH₂, H), (M-3494, F, H, H, HOCH₂CH₂, Cl), (M-3495, F, H, H, HOCH₂CH₂, F), (M-3496, F, H, H, HOCH₂CH₂, CF₃), (M-3497, F, H, H, HOCH₂CH₂, Br), (M-3498, F, H, H, HOCH₂CH₂, CH₃), (M-3499, F, H, H, HOCH₂CH₂CH₂, H), (M-3500, F, H, H, HOCH₂CH₂CH₂, Cl), (M-3501, F, H, H, HOCH₂CH₂CH₂, F), (M-3502, F, H, H, HOCH₂CH₂CH₂, CF₃), (M-3503, F, H, H, HOCH₂CH₂CH₂, Br), (M-3504, F, H, H, HOCH₂CH₂CH₂, CH₃), (M-3505, F, H, H, HOCH₂CH₂CH₂CH₂, H), (M-3506, F, H, H, HOCH₂CH₂CH₂CH₂, Cl), (M-3507, F, H, H, HOCH₂CH₂CH₂CH₂, F), (M-3508, F, H, H, HOCH₂CH₂CH₂CH₂, CF₃), (M-3509, F, H, H, HOCH₂CH₂CH₂CH₂, Br), (M-3510, F, H, H, HOCH₂CH₂CH₂CH₂, CH₃), (M-3511, F, H, H, HOCH₂CH₂CH₂CH₂CH₂, H), (M-3512, F, H, H, HOCH₂CH₂CH₂CH₂CH₂, Cl), (M-3513, F, H, H, HOCH₂CH₂CH₂CH₂CH₂, F), (M-3514, F, H, H, HOCH₂CH₂CH₂CH₂CH₂, CF₃), (M-3515, F, H, H, HOCH₂CH₂CH₂CH₂CH₂, Br), (M-3516, F, H, H, HOCH₂CH₂CH₂CH₂CH₂, CH₃), (M-3517, F, H, H, HOCH₂CH₂OCH₂CH₂, H), (M-3518, F, H, H, HOCH₂CH₂OCH₂CH₂, Cl), (M-3519, F, H, H, HOCH₂CH₂OCH₂CH₂, F), (M-3520, F, H, H, HOCH₂CH₂OCH₂CH₂, CF₃), (M-3521, F, H, H, HOCH₂CH₂OCH₂CH₂, Br), (M-3522, F, H, H, HOCH₂CH₂OCH₂CH₂, CH₃), (M-3523, F, H, H, (Me)₂N, H), (M-3524, F, H, H, (Me)₂N, Cl), (M-3525, F, H, H, (Me)₂N, F), (M-3526, F, H, H, (Me)₂N, CF₃), (M-3527, F, H, H, (Me)₂N, Br), (M-3528, F, H, H, (Me)₂N, CH₃), (M-3529, F, H, H, piperidin-4-yl-methyl, H), (M-3530, F, H, H, piperidin-4-yl-methyl, Cl), (M-3531, F, H, H, piperidin-4-yl-methyl, F), (M-3532, F, H, H, piperidin-4-yl-methyl, CF₃), (M-3533, F, H, H, piperidin-4-yl-methyl, Br), (M-3534, F, H, H, piperidin-4-yl-methyl, CH₃), (M-3535, F, H, H, cyclohexylmethyl, H), (M-3536, F, H, H, cyclohexylmethyl, Cl), (M-3537, F, H, H, cyclohexylmethyl, F), (M-3538, F, H, H, cyclohexylmethyl, CF₃), (M-3539, F, H, H, cyclohexylmethyl, Br), (M-3540, F, H, H, cyclohexylmethyl, CH₃), (M-3541, F, H, F, H, H), (M-3542, F, H, F, H, Cl), (M-3543, F, H, F, H, F), (M-3544, F, H, F, H, CF₃), (M-3545, F, H, F, H, Br), (M-3546, F, H, F, H, CH₃), (M-3547, F, H, F, F, H), (M-3548, F, H, F, F, Cl), (M-3549, F, H, F, F, F), (M-3550, F, H, F, F, CF₃), (M-3551, F, H, F, F, Br), (M-3552, F, H, F, F, CH₃), (M-3553, F, H, F, Cl, H), (M-3554, F, H, F, Cl, Cl), (M-3555, F, H, F, Cl, F), (M-3556, F, H, F, Cl, CF₃), (M-3557, F, H, F, Cl, Br), (M-3558, F, H, F, Cl, CH₃), (M-3559, F, H, F, CH₃, H), (M-3560, F, H, F, CH₃, Cl), (M-3561, F, H, F, CH₃, F), (M-3562, F, H, F, CH₃, CF₃), (M-3563, F, H, F, CH₃, Br), (M-3564, F, H, F, CH₃, CH₃), (M-3565, F, H, F, Et, H), (M-3566, F, H, F, Et, Cl), (M-3567, F, H, F, Et, F), (M-3568, F, H, F, Et, CF₃), (M-3569, F, H, F, Et, Br), (M-3570, F, H, F, Et, CH₃), (M-3571, F, H, F, n-Pr, H), (M-3572, F, H, F, n-Pr, Cl), (M-3573, F, H, F, n-Pr, F), (M-3574, F, H, F, n-Pr, CF₃), (M-3575, F, H, F, n-Pr, Br), (M-3576, F, H, F, n-Pr, CH₃), (M-3577, F, H, F, c-Pr, H), (M-3578, F, H, F, c-Pr, Cl), (M-3579, F, H, F, c-Pr, F), (M-3580, F, H, F, c-Pr, CF₃), (M-3581, F, H, F, c-Pr, Br), (M-3582, F, H, F, c-Pr, CH₃), (M-3583, F, H, F, i-Pr, H), (M-3584, F, H, F, i-Pr, Cl), (M-3585, F, H, F, i-Pr, F), (M-3586, F, H, F, i-Pr, CF₃), (M-3587, F, H, F, i-Pr, Br), (M-3588, F, H, F, i-Pr, CH₃), (M-3589, F, H, F, n-Bu, H), (M-3590, F, H, F, n-Bu, Cl), (M-3591, F, H, F, n-Bu, F), (M-3592, F, H, F, n-Bu, CF₃), (M-3593, F, H, F, n-Bu, Br), (M-3594, F, H, F, n-Bu, CH₃), (M-3595, F, H, F, i-Bu, H), (M-3596, F, H, F, i-Bu, Cl), (M-3597, F, H, F, i-Bu, F), (M-3598, F, H, F, i-Bu, CF₃), (M-3599, F, H, F, i-Bu, Br), (M-3600, F, H, F, i-Bu, CH₃), (M-3601, F, H, F, sec-Bu, H), (M-3602, F, H, F, sec-Bu, Cl), (M-3603, F, H, F, sec-Bu, F), (M-3604, F, H, F, sec-Bu, CF₃), (M-3605, F, H, F, sec-Bu, Br), (M-3606, F, H, F, sec-Bu, CH₃), (M-3607, F, H, F, n-Pen, H), (M-3608, F, H, F, n-Pen, Cl), (M-3609, F, H, F, n-Pen, F), (M-3610, F, H, F, n-Pen, CF₃), (M-3611, F, H, F, n-Pen, Br), (M-3612, F, H, F, n-Pen, CH₃), (M-3613, F, H, F, c-Pen, H), (M-3614, F, H, F, c-Pen, Cl), (M-3615, F, H, F, c-Pen, F), (M-3616, F, H, F, c-Pen, CF₃), (M-3617, F, H, F, c-Pen, Br), (M-3618, F, H, F, c-Pen, CH₃), (M-3619, F, H, F, n-Hex, H), (M-3620, F, H, F, n-Hex, Cl), (M-3621, F, H, F, n-Hex, F), (M-3622, F, H, F, n-Hex, CF₃), (M-3623, F, H, F, n-Hex, Br), (M-3624, F, H, F, n-Hex, CH₃), (M-3625, F, H, F, c-Hex, H), (M-3626, F, H, F, c-Hex, Cl), (M-3627, F, H, F, c-Hex, F), (M-3628, F, H, F, c-Hex, CF₃), (M-3629, F, H, F, c-Hex, Br), (M-3630, F, H, F, c-Hex, CH₃), (M-3631, F, H, F, OH, H), (M-3632, F, H, F, OH, Cl), (M-3633, F, H, F, OH, F), (M-3634, F, H, F, OH, CF₃), (M-3635, F, H, F, OH, Br), (M-3636, F, H, F, OH, CH₃), (M-3637, F, H, F, EtO, H), (M-3638, F, H, F, EtO, Cl), (M-3639, F, H, F, EtO, F), (M-3640, F, H, F, EtO, CF₃), (M-3641, F, H, F, EtO, Br), (M-3642, F, H, F, EtO, CH₃), (M-3643, F, H, F, n-PrO, H), (M-3644, F, H, F, n-PrO, Cl), (M-3645, F, H, F, n-PrO, F), (M-3646, F, H, F, n-PrO, CF₃), (M-3647, F, H, F, n-PrO, Br), (M-3648, F, H, F, n-PrO, CH₃), (M-3649, F, H, F, PhO, H), (M-3650, F, H, F, PhO, Cl), (M-3651, F, H, F, PhO, F), (M-3652, F, H, F, PhO, CF₃), (M-3653, F, H, F, PhO, Br), (M-3654, F, H, F, PhO, CH₃), (M-3655, F, H, F, BnO, H), (M-3656, F, H, F, BnO, Cl), (M-3657, F, H, F, BnO, F), (M-3658, F, H, F, BnO, CF₃), (M-3659, F, H, F, BnO, Br), (M-3660, F, H, F, BnO, CH₃), (M-3661, F, H, F, PhCH₂CH₂O, H), (M-3662, F, H, F, PhCH₂CH₂O, Cl), (M-3663, F, H, F, PhCH₂CH₂O, F), (M-3664, F, H, F, PhCH₂CH₂O, CF₃), (M-3665, F, H, F, PhCH₂CH₂O, Br), (M-3666, F, H, F, PhCH₂CH₂O, CH₃), (M-3667, F, H, F, CF₃O, H), (M-3668, F, H, F, CF₃O, Cl), (M-3669, F, H, F, CF₃O, F), (M-3670, F, H, F, CF₃O, CF₃), (M-3671, F, H, F, CF₃O, Br), (M-3672, F, H, F, CF₃O, CH₃), (M-3673, F, H, F, Ph, H), (M-3674, F, H, F, Ph, Cl), (M-3675, F, H, F, Ph, F), (M-3676, F, H, F, Ph, CF₃), (M-3677, F, H, F, Ph, Br), (M-3678, F, H, F, Ph, CH₃), (M-3679, F, H, F, 4-F-Ph, H), (M-3680, F, H, F, 4-F-Ph, Cl), (M-3681, F, H, F, 4-F-Ph, F), (M-3682, F, H, F, 4-F-Ph, CF₃), (M-3683, F, H, F, 4-F-Ph, Br), (M-3684, F, H, F, 4-F-Ph, CH₃), (M-3685, F, H, F, 4-CF₃-Ph, H), (M-3686, F, H, F, 4-CF₃-Ph, Cl), (M-3687, F, H, F, 4-CF₃-Ph, F), (M-3688, F, H, F, 4-CF₃-Ph, CF₃), (M-3689, F, H, F, 4-CF₃-Ph, Br), (M-3690, F, H, F, 4-CF₃-Ph, CH₃), (M-3691, F, H, F, 4-(Me)₂N-Ph, H), (M-3692, F, H, F, 4-(Me)₂N-Ph, Cl), (M-3693, F, H, F, 4-(Me)₂N-Ph, F), (M-3694, F, H, F, 4-(Me)₂N-Ph, CF₃), (M-3695, F, H, F, 4-(Me)₂N-Ph, Br), (M-3696, F, H, F, 4-(Me)₂N-Ph, CH₃), (M-3697, F, H, F, 4-OH-Ph, H), (M-3698, F, H, F, 4-OH-Ph, C
l), (M-3699, F, H, F, 4-OH-Ph, F), (M-3700, F, H, F, 4-OH-Ph, CF₃), (M-3701, F, H, F, 4-OH-Ph, Br), (M-3702, F, H, F, 4-OH-Ph, CH₃), (M-3703, F, H, F, 3,4-di-F-Ph, H), (M-3704, F, H, F, 3,4-di-F-Ph, Cl), (M-3705, F, H, F, 3,4-di-F-Ph, F), (M-3706, F, H, F, 3,4-di-F-Ph, CF₃), (M-3707, F, H, F, 3,4-di-F-Ph, Br), (M-3708, F, H, F, 3,4-di-F-Ph, CH₃), (M-3709, F, H, F, 4-COOH-Ph, H), (M-3710, F, H, F, 4-COOH-Ph, Cl), (M-3711, F, H, F, 4-COOH-Ph, F), (M-3712, F, H, F, 4-COOH-Ph, CF₃), (M-3713, F, H, F, 4-COOH-Ph, Br), (M-3714, F, H, F, 4-COOH-Ph, CH₃), (M-3715, F, H, F, Bn, H), (M-3716, F, H, F, Bn, Cl), (M-3717, F, H, F, Bn, F), (M-3718, F, H, F, Bn, CF₃), (M-3719, F, H, F, Bn, Br), (M-3720, F, H, F, Bn, CH₃), (M-3721, F, H, F, 4-F-Bn, H), (M-3722, F, H, F, 4-F-Bn, Cl), (M-3723, F, H, F, 4-F-Bn, F), (M-3724, F, H, F, 4-F-Bn, CF₃), (M-3725, F, H, F, 4-F-Bn, Br), (M-3726, F, H, F, 4-F-Bn, CH₃), (M-3727, F, H, F, 2-Py, H), (M-3728, F, H, F, 2-Py, Cl), (M-3729, F, H, F, 2-Py, F), (M-3730, F, H, F, 2-Py, CF₃), (M-3731, F, H, F, 2-Py, Br), (M-3732, F, H, F, 2-Py, CH₃), (M-3733, F, H, F, 3-Py, H), (M-3734, F, H, F, 3-Py, Cl), (M-3735, F, H, F, 3-Py, F), (M-3736, F, H, F, 3-Py, CF₃), (M-3737, F, H, F, 3-Py, Br), (M-3738, F, H, F, 3-Py, CH₃), (M-3739, F, H, F, 4-Py, H), (M-3740, F, H, F, 4-Py, Cl), (M-3741, F, H, F, 4-Py, F), (M-3742, F, H, F, 4-Py, CF₃), (M-3743, F, H, F, 4-Py, Br), (M-3744, F, H, F, 4-Py, CH₃), (M-3745, F, H, F, 2-Th, H), (M-3746, F, H, F, 2-Th, Cl), (M-3747, F, H, F, 2-Th, F), (M-3748, F, H, F, 2-Th, CF₃), (M-3749, F, H, F, 2-Th, Br), (M-3750, F, H, F, 2-Th, CH₃), (M-3751, F, H, F, 3-Th, H), (M-3752, F, H, F, 3-Th, Cl), (M-3753, F, H, F, 3-Th, F), (M-3754, F, H, F, 3-Th, CF₃), (M-3755, F, H, F, 3-Th, Br), (M-3756, F, H, F, 3-Th, CH₃), (M-3757, F, H, F, pyrazol-2-yl, H), (M-3758, F, H, F, pyrazol-2-yl, Cl), (M-3759, F, H, F, pyrazol-2-yl, F), (M-3760, F, H, F, pyrazol-2-yl, CF₃), (M-3761, F, H, F, pyrazol-2-yl, Br), (M-3762, F, H, F, pyrazol-2-yl, CH₃), (M-3763, F, H, F, pyrazol-3-yl, H), (M-3764, F, H, F, pyrazol-3-yl, Cl), (M-3765, F, H, F, pyrazol-3-yl, F), (M-3766, F, H, F, pyrazol-3-yl, CF₃), (M-3767, F, H, F, pyrazol-3-yl, Br), (M-3768, F, H, F, pyrazol-3-yl, CH₃), (M-3769, F, H, F, pyrimidin-2-yl, H), (M-3770, F, H, F, pyrimidin-2-yl, Cl), (M-3771, F, H, F, pyrimidin-2-yl, F), (M-3772, F, H, F, pyrimidin-2-yl, CF₃), (M-3773, F, H, F, pyrimidin-2-yl, Br), (M-3774, F, H, F, pyrimidin-2-yl, CH₃), (M-3775, F, H, F, pyrimidin-4-yl, H), (M-3776, F, H, F, pyrimidin-4-yl, Cl), (M-3777, F, H, F, pyrimidin-4-yl, F), (M-3778, F, H, F, pyrimidin-4-yl, CF₃), (M-3779, F, H, F, pyrimidin-4-yl, Br), (M-3780, F, H, F, pyrimidin-4-yl, CH₃), (M-3781, F, H, F, pyrimidin-5-yl, H), (M-3782, F, H, F, pyrimidin-5-yl, Cl), (M-3783, F, H, F, pyrimidin-5-yl, F), (M-3784, F, H, F, pyrimidin-5-yl, CF₃), (M-3785, F, H, F, pyrimidin-5-yl, Br), (M-3786, F, H, F, pyrimidin-5-yl, CH₃), (M-3787, F, H, F, HOOCCH₂CH₂CH₂, H), (M-3788, F, H, F, HOOCCH₂CH₂CH₂, Cl), (M-3789, F, H, F, HOOCCH₂CH₂CH₂, F), (M-3790, F, H, F, HOOCCH₂CH₂CH₂, CF₃), (M-3791, F, H, F, HOOCCH₂CH₂CH₂, Br), (M-3792, F, H, F, HOOCCH₂CH₂CH₂, CH₃), (M-3793, F, H, F, HOOCCH₂CH₂CH₂CH₂, H), (M-3794, F, H, F, HOOCCH₂CH₂CH₂CH₂, Cl), (M-3795, F, H, F, HOOCCH₂CH₂CH₂CH₂, F), (M-3796, F, H, F, HOOCCH₂CH₂CH₂CH₂, CF₃), (M-3797, F, H, F, HOOCCH₂CH₂CH₂CH₂, Br), (M-3798, F, H, F, HOOCCH₂CH₂CH₂CH₂, CH₃), (M-3799, F, H, F, (Me)₂NCOCH₂CH₂CH₂CH₂, H), (M-3800, F, H, F, (Me)₂NCOCH₂CH₂CH₂CH₂, Cl), (M-3801, F, H, F, (Me)₂NCOCH₂CH₂CH₂CH₂, F), (M-3802, F, H, F, (Me)₂NCOCH₂CH₂CH₂CH₂, CF₃), (M-3803, F, H, F, (Me)₂NCOCH₂CH₂CH₂CH₂, Br), (M-3804, F, H, F, (Me)₂NCOCH₂CH₂CH₂CH₂, CH₃), (M-3805, F, H, F, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, H), (M-3806, F, H, F, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, Cl), (M-3807, F, H, F, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, F), (M-3808, F, H, F, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, CF₃), (M-3809, F, H, F, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, Br), (M-3810, F, H, F, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, CH₃), (M-3811, F, H, F, MeOCH₂, H), (M-3812, F, H, F, MeOCH₂, Cl), (M-3813, F, H, F, MeOCH₂, F), (M-3814, F, H, F, MeOCH₂, CF₃), (M-3815, F, H, F, MeOCH₂, Br), (M-3816, F, H, F, MeOCH₂, CH₃), (M-3817, F, H, F, EtOCH₂, H), (M-3818, F, H, F, EtOCH₂, Cl), (M-3819, F, H, F, EtOCH₂, F), (M-3820, F, H, F, EtOCH₂, CF₃), (M-3821, F, H, F, EtOCH₂, Br), (M-3822, F, H, F, EtOCH₂, CH₃), (M-3823, F, H, F, EtOCH₂CH₂, H), (M-3824, F, H, F, EtOCH₂CH₂, Cl), (M-3825, F, H, F, EtOCH₂CH₂, F), (M-3826, F, H, F, EtOCH₂CH₂, CF₃), (M-3827, F, H, F, EtOCH₂CH₂, Br), (M-3828, F, H, F, EtOCH₂CH₂, CH₃), (M-3829, F, H, F, MeOCH₂CH₂OCH₂CH₂, H), (M-3830, F, H, F, MeOCH₂CH₂OCH₂CH₂, Cl), (M-3831, F, H, F, MeOCH₂CH₂OCH₂CH₂, F), (M-3832, F, H, F, MeOCH₂CH₂OCH₂CH₂, CF₃), (M-3833, F, H, F, MeOCH₂CH₂OCH₂CH₂, Br), (M-3834, F, H, F, MeOCH₂CH₂OCH₂CH₂, CH₃), (M-3835, F, H, F, MeOCH₂CH₂, H), (M-3836, F, H, F, MeOCH₂CH₂, Cl), (M-3837, F, H, F, MeOCH₂CH₂, F), (M-3838, F, H, F, MeOCH₂CH₂, CF₃), (M-3839, F, H, F, MeOCH₂CH₂, Br), (M-3840, F, H, F, MeOCH₂CH₂, CH₃), (M-3841, F, H, F, HOCH₂, H), (M-3842, F, H, F, HOCH₂, Cl), (M-3843, F, H, F, HOCH₂, F), (M-3844, F, H, F, HOCH₂, CF₃), (M-3845, F, H, F, HOCH₂, Br), (M-3846, F, H, F, HOCH₂, CH₃), (M-3847, F, H, F, HOCH₂CH₂, H), (M-3848, F, H, F, HOCH₂CH₂, Cl), (M-3849, F, H, F, HOCH₂CH₂, F), (M-3850, F, H, F, HOCH₂CH₂, CF₃), (M-3851, F, H, F, HOCH₂CH₂, Br), (M-3852, F, H, F, HOCH₂CH₂, CH₃), (M-3853, F, H, F, HOCH₂CH₂CH₂, H), (M-3854, F, H, F, HOCH₂CH₂CH₂, Cl), (M-3855, F, H, F, HOCH₂CH₂CH₂, F), (M-3856, F, H, F, HOCH₂CH₂CH₂, CF₃), (M-3857, F, H, F, HOCH₂CH₂CH₂, Br), (M-3858, F, H, F, HOCH₂CH₂CH₂, CH₃), (M-3859, F, H, F, HOCH₂CH₂CH₂CH₂, H), (M-3860, F, H, F, HOCH₂CH₂CH₂CH₂, Cl), (M-3861, F, H, F, HOCH₂CH₂CH₂CH₂, F), (M-3862, F, H, F, HOCH₂CH₂CH₂CH₂, CF₃), (M-3863, F, H, F, HOCH₂CH₂CH₂CH₂, Br), (M-3864, F, H, F, HOCH₂CH₂CH₂CH₂, CH₃), (M-3865, F, H, F, HOCH₂CH₂CH₂CH₂CH₂, H), (M-3866, F, H, F, HOCH₂CH₂CH₂CH₂CH₂, Cl), (M-3867, F, H, F, HOCH₂CH₂CH₂CH₂CH₂, F), (M-3868, F, H, F, HOCH₂CH₂CH₂CH₂CH₂, CF₃), (M-3869, F, H, F, HOCH₂CH₂CH₂CH₂CH₂, Br), (M-3870, F, H, F, HOCH₂CH₂CH₂CH₂CH₂, CH₃), (M-3871, F, H, F, HOCH₂CH₂OCH₂CH₂, H), (M-3872, F, H, F, HOCH₂CH₂OCH₂CH₂, Cl), (M-3873, F, H, F, HOCH₂CH₂OCH₂CH₂, F), (M-3874, F, H, F, HOCH₂CH₂OCH₂CH₂, CF₃), (M-3875, F, H, F, HOCH₂CH₂OCH₂CH₂, Br), (M-3876, F, H, F, HOCH₂CH₂OCH₂CH₂, CH₃), (M-3877, F, H, F, (Me)₂N, H), (M-3878, F, H, F, (Me)₂N, Cl), (M-3879, F, H, F, (Me)₂N, F), (M-3880, F, H, F, (Me)₂N, CF₃), (M-388
1, F, H, F, (Me)₂N, Br), (M-3882, F, H, F, (Me)₂N, CH₃), (M-3883, F, H, F, piperidin-4-yl-methyl, H), (M-3884, F, H, F, piperidin-4-yl-methyl, Cl), (M-3885, F, H, F, piperidin-4-yl-methyl, F), (M-3886, F, H, F, piperidin-4-yl-methyl, CF₃), (M-3887, F, H, F, piperidin-4-yl-methyl, Br), (M-3888, F, H, F, piperidin-4-yl-methyl, CH₃), (M-3889, F, H, F, cyclohexylmethyl, H), (M-3890, F, H, F, cyclohexylmethyl, Cl), (M-3891, F, H, F, cyclohexylmethyl, F), (M-3892, F, H, F, cyclohexylmethyl, CF₃), (M-3893, F, H, F, cyclohexylmethyl, Br), (M-3894, F, H, F, cyclohexylmethyl, CH₃), (M-3895, F, H, Cl, H, H), (M-3896, F, H, Cl, H, Cl), (M-3897, F, H, Cl, H, F), (M-3898, F, H, Cl, H, CF₃), (M-3899, F, H, Cl, H, Br), (M-3900, F, H, Cl, H, CH₃), (M-3901, F, H, Cl, F, H), (M-3902, F, H, Cl, F, Cl), (M-3903, F, H, Cl, F, F), (M-3904, F, H, Cl, F, CF₃), (M-3905, F, H, Cl, F, Br), (M-3906, F, H, Cl, F, CH₃), (M-3907, F, H, Cl, Cl, H), (M-3908, F, H, Cl, Cl, Cl), (M-3909, F, H, Cl, Cl, F), (M-3910, F, H, Cl, Cl, CF₃), (M-3911, F, H, Cl, Cl, Br), (M-3912, F, H, Cl, Cl, CH₃), (M-3913, F, H, Cl, CH₃, H), (M-3914, F, H, Cl, CH₃, Cl), (M-3915, F, H, Cl, CH₃, F), (M-3916, F, H, Cl, CH₃, CF₃), (M-3917, F, H, Cl, CH₃, Br), (M-3918, F, H, Cl, CH₃, CH₃), (M-3919, F, H, Cl, Et, H), (M-3920, F, H, Cl, Et, Cl), (M-3921, F, H, Cl, Et, F), (M-3922, F, H, Cl, Et, CF₃), (M-3923, F, H, Cl, Et, Br), (M-3924, F, H, Cl, Et, CH₃), (M-3925, F, H, Cl, n-Pr, H), (M-3926, F, H, Cl, n-Pr, Cl), (M-3927, F, H, Cl, n-Pr, F), (M-3928, F, H, Cl, n-Pr, CF₃), (M-3929, F, H, Cl, n-Pr, Br), (M-3930, F, H, Cl, n-Pr, CH₃), (M-3931, F, H, Cl, c-Pr, H), (M-3932, F, H, Cl, c-Pr, Cl), (M-3933, F, H, Cl, c-Pr, F), (M-3934, F, H, Cl, c-Pr, CF₃), (M-3935, F, H, Cl, c-Pr, Br), (M-3936, F, H, Cl, c-Pr, CH₃), (M-3937, F, H, Cl, i-Pr, H), (M-3938, F, H, Cl, i-Pr, Cl), (M-3939, F, H, Cl, i-Pr, F), (M-3940, F, H, Cl, i-Pr, CF₃), (M-3941, F, H, Cl, i-Pr, Br), (M-3942, F, H, Cl, i-Pr, CH₃), (M-3943, F, H, Cl, n-Bu, H), (M-3944, F, H, Cl, n-Bu, Cl), (M-3945, F, H, Cl, n-Bu, F), (M-3946, F, H, Cl, n-Bu, CF₃), (M-3947, F, H, Cl, n-Bu, Br), (M-3948, F, H, Cl, n-Bu, CH₃), (M-3949, F, H, Cl, i-Bu, H), (M-3950, F, H, Cl, i-Bu, Cl), (M-3951, F, H, Cl, i-Bu, F), (M-3952, F, H, Cl, i-Bu, CF₃), (M-3953, F, H, Cl, i-Bu, Br), (M-3954, F, H, Cl, i-Bu, CH₃), (M-3955, F, H, Cl, sec-Bu, H), (M-3956, F, H, Cl, sec-Bu, Cl), (M-3957, F, H, Cl, sec-Bu, F), (M-3958, F, H, Cl, sec-Bu, CF₃), (M-3959, F, H, Cl, sec-Bu, Br), (M-3960, F, H, Cl, sec-Bu, CH₃), (M-3961, F, H, Cl, n-Pen, H), (M-3962, F, H, Cl, n-Pen, Cl), (M-3963, F, H, Cl, n-Pen, F), (M-3964, F, H, Cl, n-Pen, CF₃), (M-3965, F, H, Cl, n-Pen, Br), (M-3966, F, H, Cl, n-Pen, CH₃), (M-3967, F, H, Cl, c-Pen, H), (M-3968, F, H, Cl, c-Pen, Cl), (M-3969, F, H, Cl, c-Pen, F), (M-3970, F, H, Cl, c-Pen, CF₃), (M-3971, F, H, Cl, c-Pen, Br), (M-3972, F, H, Cl, c-Pen, CH₃), (M-3973, F, H, Cl, n-Hex, H), (M-3974, F, H, Cl, n-Hex, Cl), (M-3975, F, H, Cl, n-Hex, F), (M-3976, F, H, Cl, n-Hex, CF₃), (M-3977, F, H, Cl, n-Hex, Br), (M-3978, F, H, Cl, n-Hex, CH₃), (M-3979, F, H, Cl, c-Hex, H), (M-3980, F, H, Cl, c-Hex, Cl), (M-3981, F, H, Cl, c-Hex, F), (M-3982, F, H, Cl, c-Hex, CF₃), (M-3983, F, H, Cl, c-Hex, Br), (M-3984, F, H, Cl, c-Hex, CH₃), (M-3985, F, H, Cl, OH, H), (M-3986, F, H, Cl, OH, Cl), (M-3987, F, H, Cl, OH, F), (M-3988, F, H, Cl, OH, CF₃), (M-3989, F, H, Cl, OH, Br), (M-3990, F, H, Cl, OH, CH₃), (M-3991, F, H, Cl, EtO, H), (M-3992, F, H, Cl, EtO, Cl), (M-3993, F, H, Cl, EtO, F), (M-3994, F, H, Cl, EtO, CF₃), (M-3995, F, H, Cl, EtO, Br), (M-3996, F, H, Cl, EtO, CH₃), (M-3997, F, H, Cl, n-PrO, H), (M-3998, F, H, Cl, n-PrO, Cl), (M-3999, F, H, Cl, n-PrO, F), (M-4000, F, H, Cl, n-PrO, CF₃), (M-4001, F, H, Cl, n-PrO, Br), (M-4002, F, H, Cl, n-PrO, CH₃), (M-4003, F, H, Cl, PhO, H), (M-4004, F, H, Cl, PhO, Cl), (M-4005, F, H, Cl, PhO, F), (M-4006, F, H, Cl, PhO, CF₃), (M-4007, F, H, Cl, PhO, Br), (M-4008, F, H, Cl, PhO, CH₃), (M-4009, F, H, Cl, BnO, H), (M-4010, F, H, Cl, BnO, Cl), (M-4011, F, H, Cl, BnO, F), (M-4012, F, H, Cl, BnO, CF₃), (M-4013, F, H, Cl, BnO, Br), (M-4014, F, H, Cl, BnO, CH₃), (M-4015, F, H, Cl, PhCH₂CH₂O, H), (M-4016, F, H, Cl, PhCH₂CH₂O, Cl), (M-4017, F, H, Cl, PhCH₂CH₂O, F), (M-4018, F, H, Cl, PhCH₂CH₂O, CF₃), (M-4019, F, H, Cl, PhCH₂CH₂O, Br), (M-4020, F, H, Cl, PhCH₂CH₂O, CH₃), (M-4021, F, H, Cl, CF₃O, H), (M-4022, F, H, Cl, CF₃O, Cl), (M-4023, F, H, Cl, CF₃O, F), (M-4024, F, H, Cl, CF₃O, CF₃), (M-4025, F, H, Cl, CF₃O, Br), (M-4026, F, H, Cl, CF₃O, CH₃), (M-4027, F, H, Cl, Ph, H), (M-4028, F, H, Cl, Ph, Cl), (M-4029, F, H, Cl, Ph, F), (M-4030, F, H, Cl, Ph, CF₃), (M-4031, F, H, Cl, Ph, Br), (M-4032, F, H, Cl, Ph, CH₃), (M-4033, F, H, Cl, 4-F-Ph, H), (M-4034, F, H, Cl, 4-F-Ph, Cl), (M-4035, F, H, Cl, 4-F-Ph, F), (M-4036, F, H, Cl, 4-F-Ph, CF₃), (M-4037, F, H, Cl, 4-F-Ph, Br), (M-4038, F, H, Cl, 4-F-Ph, CH₃), (M-4039, F, H, Cl, 4-CF₃-Ph, H), (M-4040, F, H, Cl, 4-CF₃-Ph, Cl), (M-4041, F, H, Cl, 4-CF₃-Ph, F), (M-4042, F, H, Cl, 4-CF₃-Ph, CF₃), (M-4043, F, H, Cl, 4-CF₃-Ph, Br), (M-4044, F, H, Cl, 4-CF₃-Ph, CH₃), (M-4045, F, H, Cl, 4-(Me)₂N-Ph, H), (M-4046, F, H, Cl, 4-(Me)₂N-Ph, Cl), (M-4047, F, H, Cl, 4-(Me)₂N-Ph, F), (M-4048, F, H, Cl, 4-(Me)₂N-Ph, CF₃), (M-4049, F, H, Cl, 4-(Me)₂N-Ph, Br), (M-4050, F, H, Cl, 4-(Me)₂N-Ph, CH₃), (M-4051, F, H, Cl, 4-OH-Ph, H), (M-4052, F, H, Cl, 4-OH-Ph, Cl), (M-4053, F, H, Cl, 4-OH-Ph, F), (M-4054, F, H, Cl, 4-OH-Ph, CF₃), (M-4055, F, H, Cl, 4-OH-Ph, Br), (M-4056, F, H, Cl, 4-OH-Ph, CH₃), (M-4057, F, H, Cl, 3,4-di-F-Ph, H), (M-4058, F, H, Cl, 3,4-di-F-Ph, Cl), (M-4059, F, H, Cl, 3,4-di-F-Ph, F), (M-4060, F, H, Cl, 3,4-di-F-Ph, CF₃), (M-4061, F, H, Cl, 3,4-di-F-Ph, Br), (M-4062, F, H, Cl, 3,4-di-F-Ph, CH₃), (M-4063, F, H, Cl, 4-COOH-Ph, H), (M-4064, F, H, Cl, 4-COOH-Ph, Cl), (M-4065, F, H, Cl, 4-COOH-Ph, F), (M-4066, F, H, Cl, 4-COOH-Ph, CF₃), (M-4067, F, H, Cl, 4-COOH-Ph, Br), (M-4068, F, H, Cl, 4-COOH-Ph, CH₃), (M-4069, F, H, Cl, Bn, H), (M-4070, F, H, Cl, Bn, Cl), (M-4071, F, H, Cl, Bn, F), (M-4072, F, H, Cl, Bn, CF₃), (M-4073, F, H, Cl, Bn, Br), (M-4074, F, H, Cl, Bn, CH₃), (M-4075, F, H, Cl, 4-F-Bn, H), (M-4076, F, H, Cl, 4-F-Bn, Cl), (M-4077, F, H, Cl, 4-F-Bn, F), (M-4078, F, H, Cl, 4-F-Bn, CF₃), (M-4079, F, H, Cl, 4-F-Bn, Br), (M-4080, F, H, Cl, 4-F-Bn, CH₃), (M-4081, F, H, Cl, 2-Py, H), (M-4082, F, H, Cl, 2-Py, Cl), (M-4083, F, H, Cl, 2-Py, F), (M-4084, F, H, Cl, 2-Py, CF₃), (M-4085, F, H, Cl, 2-Py, Br), (M-4086, F, H, Cl, 2-Py, CH₃), (M-4087, F, H, Cl, 3-Py, H), (M-4088, F, H, Cl, 3-Py, Cl), (M-4089, F, H, Cl, 3-Py, F), (M-4090, F, H, Cl, 3-Py, CF₃), (M-4091, F, H, Cl, 3-Py, Br), (M-4092, F, H, Cl, 3-Py, CH₃), (M-4093, F, H, Cl, 4-Py, H), (M-4094, F, H, Cl, 4-Py, Cl), (M-4095, F, H, Cl, 4-Py, F), (M-4096, F, H, Cl, 4-Py, CF₃), (M-4097, F, H, Cl, 4-Py, Br), (M-4098, F, H, Cl, 4-Py, CH₃), (M-4099, F, H, Cl, 2-Th, H), (M-4100, F, H, Cl, 2-Th, Cl), (M-4101, F, H, Cl, 2-Th, F), (M-4102, F, H, Cl, 2-Th, CF₃), (M-4103, F, H, Cl, 2-Th, Br), (M-4104, F, H, Cl, 2-Th, CH₃), (M-4105, F, H, Cl, 3-Th, H), (M-4106, F, H, Cl, 3-Th, Cl), (M-4107, F, H, Cl, 3-Th, F), (M-4108, F, H, Cl, 3-Th, CF₃), (M-4109, F, H, Cl, 3-Th, Br), (M-4110, F, H, Cl, 3-Th, CH₃), (M-4111, F, H, Cl, pyrazol-2-yl, H), (M-4112, F, H, Cl, pyrazol-2-yl, Cl), (M-4113, F, H, Cl, pyrazol-2-yl, F), (M-4114, F, H, Cl, pyrazol-2-yl, CF₃), (M-4115, F, H, Cl, pyrazol-2-yl, Br), (M-4116, F, H, Cl, pyrazol-2-yl, CH₃), (M-4117, F, H, Cl, pyrazol-3-yl, H), (M-4118, F, H, Cl, pyrazol-3-yl, Cl), (M-4119, F, H, Cl, pyrazol-3-yl, F), (M-4120, F, H, Cl, pyrazol-3-yl, CF₃), (M-4121, F, H, Cl, pyrazol-3-yl, Br), (M-4122, F, H, Cl, pyrazol-3-yl, CH₃), (M-4123, F, H, Cl, pyrimidin-2-yl, H), (M-4124, F, H, Cl, pyrimidin-2-yl, Cl), (M-4125, F, H, Cl, pyrimidin-2-yl, F), (M-4126, F, H, Cl, pyrimidin-2-yl, CF₃), (M-4127, F, H, Cl, pyrimidin-2-yl, Br), (M-4128, F, H, Cl, pyrimidin-2-yl, CH₃), (M-4129, F, H, Cl, pyrimidin-4-yl, H), (M-4130, F, H, Cl, pyrimidin-4-yl, Cl), (M-4131, F, H, Cl, pyrimidin-4-yl, F), (M-4132, F, H, Cl, pyrimidin-4-yl, CF₃), (M-4133, F, H, Cl, pyrimidin-4-yl, Br), (M-4134, F, H, Cl, pyrimidin-4-yl, CH₃), (M-4135, F, H, Cl, pyrimidin-5-yl, H), (M-4136, F, H, Cl, pyrimidin-5-yl, Cl), (M-4137, F, H, Cl, pyrimidin-5-yl, F), (M-4138, F, H, Cl, pyrimidin-5-yl, CF₃), (M-4139, F, H, Cl, pyrimidin-5-yl, Br), (M-4140, F, H, Cl, pyrimidin-5-yl, CH₃), (M-4141, F, H, Cl, HOOCCH₂CH₂CH₂, H), (M-4142, F, H, Cl, HOOCCH₂CH₂CH₂, Cl), (M-4143, F, H, Cl, HOOCCH₂CH₂CH₂, F), (M-4144, F, H, Cl, HOOCCH₂CH₂CH₂, CF₃), (M-4145, F, H, Cl, HOOCCH₂CH₂CH₂, Br), (M-4146, F, H, Cl, HOOCCH₂CH₂CH₂, CH₃), (M-4147, F, H, Cl, HOOCCH₂CH₂
CH₂CH₂, H), (M-4148, F, H, Cl, HOOCCH₂CH₂CH₂CH₂, Cl), (M-4149, F, H, Cl, HOOCCH₂CH₂CH₂CH₂, F), (M-4150, F, H, Cl, HOOCCH₂CH₂CH₂CH₂, CF₃), (M-4151, F, H, Cl, HOOCCH₂CH₂CH₂CH₂, Br), (M-4152, F, H, Cl, HOOCCH₂CH₂CH₂CH₂, CH₃), (M-4153, F, H, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂, H), (M-4154, F, H, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂, Cl), (M-4155, F, H, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂, F), (M-4156, F, H, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂, CF₃), (M-4157, F, H, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂, Br), (M-4158, F, H, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂, CH₃), (M-4159, F, H, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, H), (M-4160, F, H, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, Cl), (M-4161, F, H, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, F), (M-4162, F, H, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, CF₃), (M-4163, F, H, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, Br), (M-4164, F, H, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, CH₃), (M-4165, F, H, Cl, MeOCH₂, H), (M-4166, F, H, Cl, MeOCH₂, Cl), (M-4167, F, H, Cl, MeOCH₂, F), (M-4168, F, H, Cl, MeOCH₂, CF₃), (M-4169, F, H, Cl, MeOCH₂, Br), (M-4170, F, H, Cl, MeOCH₂, CH₃), (M-4171, F, H, Cl, EtOCH₂, H), (M-4172, F, H, Cl, EtOCH₂, Cl), (M-4173, F, H, Cl, EtOCH₂, F), (M-4174, F, H, Cl, EtOCH₂, CF₃), (M-4175, F, H, Cl, EtOCH₂, Br), (M-4176, F, H, Cl, EtOCH₂, CH₃), (M-4177, F, H, Cl, EtOCH₂CH₂, H), (M-4178, F, H, Cl, EtOCH₂CH₂, Cl), (M-4179, F, H, Cl, EtOCH₂CH₂, F), (M-4180, F, H, Cl, EtOCH₂CH₂, CF₃), (M-4181, F, H, Cl, EtOCH₂CH₂, Br), (M-4182, F, H, Cl, EtOCH₂CH₂, CH₃), (M-4183, F, H, Cl, MeOCH₂CH₂OCH₂CH₂, H), (M-4184, F, H, Cl, MeOCH₂CH₂OCH₂CH₂, Cl), (M-4185, F, H, Cl, MeOCH₂CH₂OCH₂CH₂, F), (M-4186, F, H, Cl, MeOCH₂CH₂OCH₂CH₂, CF₃), (M-4187, F, H, Cl, MeOCH₂CH₂OCH₂CH₂, Br), (M-4188, F, H, Cl, MeOCH₂CH₂OCH₂CH₂, CH₃), (M-4189, F, H, Cl, MeOCH₂CH₂, H), (M-4190, F, H, Cl, MeOCH₂CH₂, Cl), (M-4191, F, H, Cl, MeOCH₂CH₂, F), (M-4192, F, H, Cl, MeOCH₂CH₂, CF₃), (M-4193, F, H, Cl, MeOCH₂CH₂, Br), (M-4194, F, H, Cl, MeOCH₂CH₂, CH₃), (M-4195, F, H, Cl, HOCH₂, H), (M-4196, F, H, Cl, HOCH₂, Cl), (M-4197, F, H, Cl, HOCH₂, F), (M-4198, F, H, Cl, HOCH₂, CF₃), (M-4199, F, H, Cl, HOCH₂, Br), (M-4200, F, H, Cl, HOCH₂, CH₃), (M-4201, F, H, Cl, HOCH₂CH₂, H), (M-4202, F, H, Cl, HOCH₂CH₂, Cl), (M-4203, F, H, Cl, HOCH₂CH₂, F), (M-4204, F, H, Cl, HOCH₂CH₂, CF₃), (M-4205, F, H, Cl, HOCH₂CH₂, Br), (M-4206, F, H, Cl, HOCH₂CH₂, CH₃), (M-4207, F, H, Cl, HOCH₂CH₂CH₂, H), (M-4208, F, H, Cl, HOCH₂CH₂CH₂, Cl), (M-4209, F, H, Cl, HOCH₂CH₂CH₂, F), (M-4210, F, H, Cl, HOCH₂CH₂CH₂, CF₃), (M-4211, F, H, Cl, HOCH₂CH₂CH₂, Br), (M-4212, F, H, Cl, HOCH₂CH₂CH₂, CH₃), (M-4213, F, H, Cl, HOCH₂CH₂CH₂CH₂, H), (M-4214, F, H, Cl, HOCH₂CH₂CH₂CH₂, Cl), (M-4215, F, H, Cl, HOCH₂CH₂CH₂CH₂, F), (M-4216, F, H, Cl, HOCH₂CH₂CH₂CH₂, CF₃), (M-4217, F, H, Cl, HOCH₂CH₂CH₂CH₂, Br), (M-4218, F, H, Cl, HOCH₂CH₂CH₂CH₂, CH₃), (M-4219, F, H, Cl, HOCH₂CH₂CH₂CH₂CH₂, H), (M-4220, F, H, Cl, HOCH₂CH₂CH₂CH₂CH₂, Cl), (M-4221, F, H, Cl, HOCH₂CH₂CH₂CH₂CH₂, F), (M-4222, F, H, Cl, HOCH₂CH₂CH₂CH₂CH₂, CF₃), (M-4223, F, H, Cl, HOCH₂CH₂CH₂CH₂CH₂, Br), (M-4224, F, H, Cl, HOCH₂CH₂CH₂CH₂CH₂, CH₃), (M-4225, F, H, Cl, HOCH₂CH₂OCH₂CH₂, H), (M-4226, F, H, Cl, HOCH₂CH₂OCH₂CH₂, Cl), (M-4227, F, H, Cl, HOCH₂CH₂OCH₂CH₂, F), (M-4228, F, H, Cl, HOCH₂CH₂OCH₂CH₂, CF₃), (M-4229, F, H, Cl, HOCH₂CH₂OCH₂CH₂, Br), (M-4230, F, H, Cl, HOCH₂CH₂OCH₂CH₂, CH₃), (M-4231, F, H, Cl, (Me)₂N, H), (M-4232, F, H, Cl, (Me)₂N, Cl), (M-4233, F, H, Cl, (Me)₂N, F), (M-4234, F, H, Cl, (Me)₂N, CF₃), (M-4235, F, H, Cl, (Me)₂N, Br), (M-4236, F, H, Cl, (Me)₂N, CH₃), (M-4237, F, H, Cl, piperidin-4-yl-methyl, H), (M-4238, F, H, Cl, piperidin-4-yl-methyl, Cl), (M-4239, F, H, Cl, piperidin-4-yl-methyl, F), (M-4240, F, H, Cl, piperidin-4-yl-methyl, CF₃), (M-4241, F, H, Cl, piperidin-4-yl-methyl, Br), (M-4242, F, H, Cl, piperidin-4-yl-methyl, CH₃), (M-4243, F, H, Cl, cyclohexylmethyl, H), (M-4244, F, H, Cl, cyclohexylmethyl, Cl), (M-4245, F, H, Cl, cyclohexylmethyl, F), (M-4246, F, H, Cl, cyclohexylmethyl, CF₃), (M-4247, F, H, Cl, cyclohexylmethyl, Br), (M-4248, F, H, Cl, cyclohexylmethyl, CH₃), (M-4249, F, F, H, H, H), (M-4250, F, F, H, H, Cl), (M-4251, F, F, H, H, F), (M-4252, F, F, H, H, CF₃), (M-4253, F, F, H, H, Br), (M-4254, F, F, H, H, CH₃), (M-4255, F, F, H, F, H), (M-4256, F, F, H, F, Cl), (M-4257, F, F, H, F, F), (M-4258, F, F, H, F, CF₃), (M-4259, F, F, H, F, Br), (M-4260, F, F, H, F, CH₃), (M-4261, F, F, H, Cl, H), (M-4262, F, F, H, Cl, Cl), (M-4263, F, F, H, Cl, F), (M-4264, F, F, H, Cl, CF₃), (M-4265, F, F, H, Cl, Br), (M-4266, F, F, H, Cl, CH₃), (M-4267, F, F, H, CH₃, H), (M-4268, F, F, H, CH₃, Cl), (M-4269, F, F, H, CH₃, F), (M-4270, F, F, H, CH₃, CF₃), (M-4271, F, F, H, CH₃, Br), (M-4272, F, F, H, CH₃, CH₃), (M-4273, F, F, H, Et, H), (M-4274, F, F, H, Et, Cl), (M-4275, F, F, H, Et, F), (M-4276, F, F, H, Et, CF₃), (M-4277, F, F, H, Et, Br), (M-4278, F, F, H, Et, CH₃), (M-4279, F, F, H, n-Pr, H), (M-4280, F, F, H, n-Pr, Cl), (M-4281, F, F, H, n-Pr, F), (M-4282, F, F, H, n-Pr, CF₃), (M-4283, F, F, H, n-Pr, Br), (M-4284, F, F, H, n-Pr, CH₃), (M-4285, F, F, H, c-Pr, H), (M-4286, F, F, H, c-Pr, Cl), (M-4287, F, F, H, c-Pr, F), (M-4288, F, F, H, c-Pr, CF₃), (M-4289, F, F, H, c-Pr, Br), (M-4290, F, F, H, c-Pr, CH₃), (M-4291, F, F, H, i-Pr, H), (M-4292, F, F, H, i-Pr, Cl), (M-4293, F, F, H, i-Pr, F), (M-4294, F, F, H, i-Pr, CF₃), (M-4295, F, F, H, i-Pr, Br), (M-4296, F, F, H, i-Pr, CH₃), (M-4297, F, F, H, n-Bu, H), (M-4298, F, F, H, n-Bu, Cl), (M-4299, F, F, H, n-Bu, F), (M-4300, F, F, H, n-Bu, CF₃), (M-4301, F, F, H, n-Bu, Br), (M-4302, F, F, H, n-Bu, CH₃), (M-4303, F, F, H, i-Bu, H), (M-4304, F, F, H, i-Bu, Cl), (M-4305, F, F, H, i-Bu, F), (M-4306, F, F, H, i-Bu, CF₃), (M-4307, F, F, H, i-Bu, Br), (M-4308, F, F, H, i-Bu, CH₃), (M-4309, F, F, H, sec-Bu, H), (M-4310, F, F, H, sec-Bu, Cl), (M-4311, F, F, H, sec-Bu, F), (M-4312, F, F, H, sec-Bu, CF₃), (M-4313, F, F, H, sec-Bu, Br), (M-4314, F, F, H, sec-Bu, CH₃), (M-4315, F, F, H, n-Pen, H), (M-4316, F, F, H, n-Pen, Cl), (M-4317, F, F, H, n-Pen, F), (M-4318, F, F, H, n-Pen, CF₃), (M-4319, F, F, H, n-Pen, Br), (M-4320, F, F, H, n-Pen, CH₃), (M-4321, F, F, H, c-Pen, H), (M-4322, F, F, H, c-Pen, Cl), (M-4323, F, F, H, c-Pen, F), (M-4324, F, F, H, c-Pen, CF₃), (M-4325, F, F, H, c-Pen, Br), (M-4326, F, F, H, c-Pen, CH₃), (M-4327, F, F, H, n-Hex, H), (M-4328, F, F, H, n-Hex, Cl), (M-4329, F, F, H, n-Hex, F), (M-4330, F, F, H, n-Hex, CF₃), (M-4331, F, F, H, n-Hex, Br), (M-4332, F, F, H, n-Hex, CH₃), (M-4333, F, F, H, c-Hex, H), (M-4334, F, F, H, c-Hex, Cl), (M-4335, F, F, H, c-Hex, F), (M-4336, F, F, H, c-Hex, CF₃), (M-4337, F, F, H, c-Hex, Br), (M-4338, F, F, H, c-Hex, CH₃), (M-433
9, F, F, H, OH, H), (M-4340, F, F, H, OH, Cl), (M-4341, F, F, H, OH, F), (M-4342, F, F, H, OH, CF₃), (M-4343, F, F, H, OH, Br), (M-4344, F, F, H, OH, CH₃), (M-4345, F, F, H, EtO, H), (M-4346, F, F, H, EtO, Cl), (M-4347, F, F, H, EtO, F), (M-4348, F, F, H, EtO, CF₃), (M-4349, F, F, H, EtO, Br), (M-4350, F, F, H, EtO, CH₃), (M-4351, F, F, H, n-PrO, H), (M-4352, F, F, H, n-PrO, Cl), (M-4353, F, F, H, n-PrO, F), (M-4354, F, F, H, n-PrO, CF₃), (M-4355, F, F, H, n-PrO, Br), (M-4356, F, F, H, n-PrO, CH₃), (M-4357, F, F, H, PhO, H), (M-4358, F, F, H, PhO, Cl), (M-4359, F, F, H, PhO, F), (M-4360, F, F, H, PhO, CF₃), (M-4361, F, F, H, PhO, Br), (M-4362, F, F, H, PhO, CH₃), (M-4363, F, F, H, BnO, H), (M-4364, F, F, H, BnO, Cl), (M-4365, F, F, H, BnO, F), (M-4366, F, F, H, BnO, CF₃), (M-4367, F, F, H, BnO, Br), (M-4368, F, F, H, BnO, CH₃), (M-4369, F, F, H, PhCH₂CH₂O, H), (M-4370, F, F, H, PhCH₂CH₂O, Cl), (M-4371, F, F, H, PhCH₂CH₂O, F), (M-4372, F, F, H, PhCH₂CH₂O, CF₃), (M-4373, F, F, H, PhCH₂CH₂O, Br), (M-4374, F, F, H, PhCH₂CH₂O, CH₃), (M-4375, F, F, H, CF₃O, H), (M-4376, F, F, H, CF₃O, Cl), (M-4377, F, F, H, CF₃O, F), (M-4378, F, F, H, CF₃O, CF₃), (M-4379, F, F, H, CF₃O, Br), (M-4380, F, F, H, CF₃O, CH₃), (M-4381, F, F, H, Ph, H), (M-4382, F, F, H, Ph, Cl), (M-4383, F, F, H, Ph, F), (M-4384, F, F, H, Ph, CF₃), (M-4385, F, F, H, Ph, Br), (M-4386, F, F, H, Ph, CH₃), (M-4387, F, F, H, 4-F-Ph, H), (M-4388, F, F, H, 4-F-Ph, Cl), (M-4389, F, F, H, 4-F-Ph, F), (M-4390, F, F, H, 4-F-Ph, CF₃), (M-4391, F, F, H, 4-F-Ph, Br), (M-4392, F, F, H, 4-F-Ph, CH₃), (M-4393, F, F, H, 4-CF₃-Ph, H), (M-4394, F, F, H, 4-CF₃-Ph, Cl), (M-4395, F, F, H, 4-CF₃-Ph, F), (M-4396, F, F, H, 4-CF₃-Ph, CF₃), (M-4397, F, F, H, 4-CF₃-Ph, Br), (M-4398, F, F, H, 4-CF₃-Ph, CH₃), (M-4399, F, F, H, 4-(Me)₂N-Ph, H), (M-4400, F, F, H, 4-(Me)₂N-Ph, Cl), (M-4401, F, F, H, 4-(Me)₂N-Ph, F), (M-4402, F, F, H, 4-(Me)₂N-Ph, CF₃), (M-4403, F, F, H, 4-(Me)₂N-Ph, Br), (M-4404, F, F, H, 4-(Me)₂N-Ph, CH₃), (M-4405, F, F, H, 4-OH-Ph, H), (M-4406, F, F, H, 4-OH-Ph, Cl), (M-4407, F, F, H, 4-OH-Ph, F), (M-4408, F, F, H, 4-OH-Ph, CF₃), (M-4409, F, F, H, 4-OH-Ph, Br), (M-4410, F, F, H, 4-OH-Ph, CH₃), (M-4411, F, F, H, 3,4-di-F-Ph, H), (M-4412, F, F, H, 3,4-di-F-Ph, Cl), (M-4413, F, F, H, 3,4-di-F-Ph, F), (M-4414, F, F, H, 3,4-di-F-Ph, CF₃), (M-4415, F, F, H, 3,4-di-F-Ph, Br), (M-4416, F, F, H, 3,4-di-F-Ph, CH₃), (M-4417, F, F, H, 4-COOH-Ph, H), (M-4418, F, F, H, 4-COOH-Ph, Cl), (M-4419, F, F, H, 4-COOH-Ph, F), (M-4420, F, F, H, 4-COOH-Ph, CF₃), (M-4421, F, F, H, 4-COOH-Ph, Br), (M-4422, F, F, H, 4-COOH-Ph, CH₃), (M-4423, F, F, H, Bn, H), (M-4424, F, F, H, Bn, Cl), (M-4425, F, F, H, Bn, F), (M-4426, F, F, H, Bn, CF₃), (M-4427, F, F, H, Bn, Br), (M-4428, F, F, H, Bn, CH₃), (M-4429, F, F, H, 4-F-Bn, H), (M-4430, F, F, H, 4-F-Bn, Cl), (M-4431, F, F, H, 4-F-Bn, F), (M-4432, F, F, H, 4-F-Bn, CF₃), (M-4433, F, F, H, 4-F-Bn, Br), (M-4434, F, F, H, 4-F-Bn, CH₃), (M-4435, F, F, H, 2-Py, H), (M-4436, F, F, H, 2-Py, Cl), (M-4437, F, F, H, 2-Py, F), (M-4438, F, F, H, 2-Py, CF₃), (M-4439, F, F, H, 2-Py, Br), (M-4440, F, F, H, 2-Py, CH₃), (M-4441, F, F, H, 3-Py, H), (M-4442, F, F, H, 3-Py, Cl), (M-4443, F, F, H, 3-Py, F), (M-4444, F, F, H, 3-Py, CF₃), (M-4445, F, F, H, 3-Py, Br), (M-4446, F, F, H, 3-Py, CH₃), (M-4447, F, F, H, 4-Py, H), (M-4448, F, F, H, 4-Py, Cl), (M-4449, F, F, H, 4-Py, F), (M-4450, F, F, H, 4-Py, CF₃), (M-4451, F, F, H, 4-Py, Br), (M-4452, F, F, H, 4-Py, CH₃), (M-4453, F, F, H, 2-Th, H), (M-4454, F, F, H, 2-Th, Cl), (M-4455, F, F, H, 2-Th, F), (M-4456, F, F, H, 2-Th, CF₃), (M-4457, F, F, H, 2-Th, Br), (M-4458, F, F, H, 2-Th, CH₃), (M-4459, F, F, H, 3-Th, H), (M-4460, F, F, H, 3-Th, Cl), (M-4461, F, F, H, 3-Th, F), (M-4462, F, F, H, 3-Th, CF₃), (M-4463, F, F, H, 3-Th, Br), (M-4464, F, F, H, 3-Th, CH₃), (M-4465, F, F, H, pyrazol-2-yl, H), (M-4466, F, F, H, pyrazol-2-yl, Cl), (M-4467, F, F, H, pyrazol-2-yl, F), (M-4468, F, F, H, pyrazol-2-yl, CF₃), (M-4469, F, F, H, pyrazol-2-yl, Br), (M-4470, F, F, H, pyrazol-2-yl, CH₃), (M-4471, F, F, H, pyrazol-3-yl, H), (M-4472, F, F, H, pyrazol-3-yl, Cl), (M-4473, F, F, H, pyrazol-3-yl, F), (M-4474, F, F, H, pyrazol-3-yl, CF₃), (M-4475, F, F, H, pyrazol-3-yl, Br), (M-4476, F, F, H, pyrazol-3-yl, CH₃), (M-4477, F, F, H, pyrimidin-2-yl, H), (M-4478, F, F, H, pyrimidin-2-yl, Cl), (M-4479, F, F, H, pyrimidin-2-yl, F), (M-4480, F, F, H, pyrimidin-2-yl, CF₃), (M-4481, F, F, H, pyrimidin-2-yl, Br), (M-4482, F, F, H, pyrimidin-2-yl, CH₃), (M-4483, F, F, H, pyrimidin-4-yl, H), (M-4484, F, F, H, pyrimidin-4-yl, Cl), (M-4485, F, F, H, pyrimidin-4-yl, F), (M-4486, F, F, H, pyrimidin-4-yl, CF₃), (M-4487, F, F, H, pyrimidin-4-yl, Br), (M-4488, F, F, H, pyrimidin-4-yl, CH₃), (M-4489, F, F, H, pyrimidin-5-yl, H), (M-4490, F, F, H, pyrimidin-5-yl, Cl), (M-4491, F, F, H, pyrimidin-5-yl, F), (M-4492, F, F, H, pyrimidin-5-yl, CF₃), (M-4493, F, F, H, pyrimidin-5-yl, Br), (M-4494, F, F, H, pyrimidin-5-yl, CH₃), (M-4495, F, F, H, HOOCCH₂CH₂CH₂, H), (M-4496, F, F, H, HOOCCH₂CH₂CH₂, Cl), (M-4497, F, F, H, HOOCCH₂CH₂CH₂, F), (M-4498, F, F, H, HOOCCH₂CH₂CH₂, CF₃), (M-4499, F, F, H, HOOCCH₂CH₂CH₂, Br), (M-4500, F, F, H, HOOCCH₂CH₂CH₂, CH₃), (M-4501, F, F, H, HOOCCH₂CH₂CH₂CH₂, H), (M-4502, F, F, H, HOOCCH₂CH₂CH₂CH₂, Cl), (M-4503, F, F, H, HOOCCH₂CH₂CH₂CH₂, F), (M-4504, F, F, H, HOOCCH₂CH₂CH₂CH₂, CF₃), (M-4505, F, F, H, HOOCCH₂CH₂CH₂CH₂, Br), (M-4506, F, F, H, HOOCCH₂CH₂CH₂CH₂, CH₃), (M-4507, F, F, H, (Me)₂NCOCH₂CH₂CH₂CH₂, H), (M-4508, F, F, H, (Me)₂NCOCH₂CH₂CH₂CH₂, Cl), (M-4509, F, F, H, (Me)₂NCOCH₂CH₂CH₂CH₂, F), (M-4510, F, F, H, (Me)₂NCOCH₂CH₂CH₂CH₂, CF₃), (M-4511, F, F, H, (Me)₂NCOCH₂CH₂CH₂CH₂, Br), (M-4512, F, F, H, (Me)₂NCOCH₂CH₂CH₂CH₂, CH₃), (M-4513, F, F, H, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, H), (M-4514, F, F, H, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, Cl), (M-4515, F, F, H, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, F), (M-4516, F, F, H, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, CF₃), (M-4517, F, F, H, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, Br), (M-4518, F, F, H, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, CH₃), (M-4519, F, F, H, MeOCH₂, H), (M-4520, F, F, H, MeOCH₂, Cl), (M-4521, F, F, H, MeOCH₂, F), (M-4522, F, F, H, MeOCH₂, CF₃), (M-4523, F, F, H, MeOCH₂, Br), (M-4524, F, F, H, MeOCH₂, CH₃), (M-4525, F, F, H, EtOCH₂, H), (M-4526, F, F, H, EtOCH₂, Cl), (M-4527, F, F, H, EtOCH₂, F), (M-4528, F, F, H, EtOCH₂, CF₃), (M-4529, F, F, H, EtOCH₂, Br), (M-4530, F, F, H, EtOCH₂, CH₃), (M-4531, F, F, H, EtOCH₂CH₂, H), (M-4532, F, F, H, EtOCH₂CH₂, Cl), (M-4533, F, F, H, EtOCH₂CH₂, F), (M-4534, F, F, H, EtOCH₂CH₂, CF₃), (M-4535, F, F, H, EtOCH₂CH₂, Br), (M-4536, F, F, H, EtOCH₂CH₂, CH₃), (M-4537, F, F, H, MeOCH₂CH₂OCH₂CH₂, H), (M-4538, F, F, H, MeOCH₂CH₂OCH₂CH₂, Cl), (M-4539, F, F, H, MeOCH₂CH₂OCH₂CH₂, F), (M-4540, F, F, H, MeOCH₂CH₂OCH₂CH₂, CF₃), (M-4541, F, F, H, MeOCH₂CH₂OCH₂CH₂, Br), (M-4542, F, F, H, MeOCH₂CH₂OCH₂CH₂, CH₃), (M-4543, F, F, H, MeOCH₂CH₂, H), (M-4544, F, F, H, MeOCH₂CH₂, Cl), (M-4545, F, F, H, MeOCH₂CH₂, F), (M-4546, F, F, H, MeOCH₂CH₂, CF₃), (M-4547, F, F, H, MeOCH₂CH₂, Br), (M-4548, F, F, H, MeOCH₂CH₂, CH₃), (M-4549, F, F, H, HOCH₂, H), (M-4550, F, F, H, HOCH₂, Cl), (M-4551, F, F, H, HOCH₂, F), (M-4552, F, F, H, HOCH₂, CF₃), (M-4553, F, F, H, HOCH₂, Br), (M-4554, F, F, H, HOCH₂, CH₃), (M-4555, F,
F, H, HOCH₂CH₂, H), (M-4556, F, F, H, HOCH₂CH₂, Cl), (M-4557, F, F, H, HOCH₂CH₂, F), (M-4558, F, F, H, HOCH₂CH₂, CF₃), (M-4559, F, F, H, HOCH₂CH₂, Br), (M-4560, F, F, H, HOCH₂CH₂, CH₃), (M-4561, F, F, H, HOCH₂CH₂CH₂, H), (M-4562, F, F, H, HOCH₂CH₂CH₂, Cl), (M-4563, F, F, H, HOCH₂CH₂CH₂, F), (M-4564, F, F, H, HOCH₂CH₂CH₂, CF₃), (M-4565, F, F, H, HOCH₂CH₂CH₂, Br), (M-4566, F, F, H, HOCH₂CH₂CH₂, CH₃), (M-4567, F, F, H, HOCH₂CH₂CH₂CH₂, H), (M-4568, F, F, H, HOCH₂CH₂CH₂CH₂, Cl), (M-4569, F, F, H, HOCH₂CH₂CH₂CH₂, F), (M-4570, F, F, H, HOCH₂CH₂CH₂CH₂, CF₃), (M-4571, F, F, H, HOCH₂CH₂CH₂CH₂, Br), (M-4572, F, F, H, HOCH₂CH₂CH₂CH₂, CH₃), (M-4573, F, F, H, HOCH₂CH₂CH₂CH₂CH₂, H), (M-4574, F, F, H, HOCH₂CH₂CH₂CH₂CH₂, Cl), (M-4575, F, F, H, HOCH₂CH₂CH₂CH₂CH₂, F), (M-4576, F, F, H, HOCH₂CH₂CH₂CH₂CH₂, CF₃), (M-4577, F, F, H, HOCH₂CH₂CH₂CH₂CH₂, Br), (M-4578, F, F, H, HOCH₂CH₂CH₂CH₂CH₂, CH₃), (M-4579, F, F, H, HOCH₂CH₂OCH₂CH₂, H), (M-4580, F, F, H, HOCH₂CH₂OCH₂CH₂, Cl), (M-4581, F, F, H, HOCH₂CH₂OCH₂CH₂, F), (M-4582, F, F, H, HOCH₂CH₂OCH₂CH₂, CF₃), (M-4583, F, F, H, HOCH₂CH₂OCH₂CH₂, Br), (M-4584, F, F, H, HOCH₂CH₂OCH₂CH₂, CH₃), (M-4585, F, F, H, (Me)₂N, H), (M-4586, F, F, H, (Me)₂N, Cl), (M-4587, F, F, H, (Me)₂N, F), (M-4588, F, F, H, (Me)₂N, CF₃), (M-4589, F, F, H, (Me)₂N, Br), (M-4590, F, F, H, (Me)₂N, CH₃), (M-4591, F, F, H, piperidin-4-yl-methyl, H), (M-4592, F, F, H, piperidin-4-yl-methyl, Cl), (M-4593, F, F, H, piperidin-4-yl-methyl, F), (M-4594, F, F, H, piperidin-4-yl-methyl, CF₃), (M-4595, F, F, H, piperidin-4-yl-methyl, Br), (M-4596, F, F, H, piperidin-4-yl-methyl, CH₃), (M-4597, F, F, H, cyclohexylmethyl, H), (M-4598, F, F, H, cyclohexylmethyl, Cl), (M-4599, F, F, H, cyclohexylmethyl, F), (M-4600, F, F, H, cyclohexylmethyl, CF₃), (M-4601, F, F, H, cyclohexylmethyl, Br), (M-4602, F, F, H, cyclohexylmethyl, CH₃), (M-4603, F, F, F, H, H), (M-4604, F, F, F, H, Cl), (M-4605, F, F, F, H, F), (M-4606, F, F, F, H, CF₃), (M-4607, F, F, F, H, Br), (M-4608, F, F, F, H, CH₃), (M-4609, F, F, F, F, H), (M-4610, F, F, F, F, Cl), (M-4611, F, F, F, F, F), (M-4612, F, F, F, F, CF₃), (M-4613, F, F, F, F, Br), (M-4614, F, F, F, F, CH₃), (M-4615, F, F, F, Cl, H), (M-4616, F, F, F, Cl, Cl), (M-4617, F, F, F, Cl, F), (M-4618, F, F, F, Cl, CF₃), (M-4619, F, F, F, Cl, Br), (M-4620, F, F, F, Cl, CH₃), (M-4621, F, F, F, CH₃, H), (M-4622, F, F, F, CH₃, Cl), (M-4623, F, F, F, CH₃, F), (M-4624, F, F, F, CH₃, CF₃), (M-4625, F, F, F, CH₃, Br), (M-4626, F, F, F, CH₃, CH₃), (M-4627, F, F, F, Et, H), (M-4628, F, F, F, Et, Cl), (M-4629, F, F, F, Et, F), (M-4630, F, F, F, Et, CF₃), (M-4631, F, F, F, Et, Br), (M-4632, F, F, F, Et, CH₃), (M-4633, F, F, F, n-Pr, H), (M-4634, F, F, F, n-Pr, Cl), (M-4635, F, F, F, n-Pr, F), (M-4636, F, F, F, n-Pr, CF₃), (M-4637, F, F, F, n-Pr, Br), (M-4638, F, F, F, n-Pr, CH₃), (M-4639, F, F, F, c-Pr, H), (M-4640, F, F, F, c-Pr, Cl), (M-4641, F, F, F, c-Pr, F), (M-4642, F, F, F, c-Pr, CF₃), (M-4643, F, F, F, c-Pr, Br), (M-4644, F, F, F, c-Pr, CH₃), (M-4645, F, F, F, i-Pr, H), (M-4646, F, F, F, i-Pr, Cl), (M-4647, F, F, F, i-Pr, F), (M-4648, F, F, F, i-Pr, CF₃), (M-4649, F, F, F, i-Pr, Br), (M-4650, F, F, F, i-Pr, CH₃), (M-4651, F, F, F, n-Bu, H), (M-4652, F, F, F, n-Bu, Cl), (M-4653, F, F, F, n-Bu, F), (M-4654, F, F, F, n-Bu, CF₃), (M-4655, F, F, F, n-Bu, Br), (M-4656, F, F, F, n-Bu, CH₃), (M-4657, F, F, F, i-Bu, H), (M-4658, F, F, F, i-Bu, Cl), (M-4659, F, F, F, i-Bu, F), (M-4660, F, F, F, i-Bu, CF₃), (M-4661, F, F, F, i-Bu, Br), (M-4662, F, F, F, i-Bu, CH₃), (M-4663, F, F, F, sec-Bu, H), (M-4664, F, F, F, sec-Bu, Cl), (M-4665, F, F, F, sec-Bu, F), (M-4666, F, F, F, sec-Bu, CF₃), (M-4667, F, F, F, sec-Bu, Br), (M-4668, F, F, F, sec-Bu, CH₃), (M-4669, F, F, F, n-Pen, H), (M-4670, F, F, F, n-Pen, Cl), (M-4671, F, F, F, n-Pen, F), (M-4672, F, F, F, n-Pen, CF₃), (M-4673, F, F, F, n-Pen, Br), (M-4674, F, F, F, n-Pen, CH₃), (M-4675, F, F, F, c-Pen, H), (M-4676, F, F, F, c-Pen, Cl), (M-4677, F, F, F, c-Pen, F), (M-4678, F, F, F, c-Pen, CF₃), (M-4679, F, F, F, c-Pen, Br), (M-4680, F, F, F, c-Pen, CH₃), (M-4681, F, F, F, n-Hex, H), (M-4682, F, F, F, n-Hex, Cl), (M-4683, F, F, F, n-Hex, F), (M-4684, F, F, F, n-Hex, CF₃), (M-4685, F, F, F, n-Hex, Br), (M-4686, F, F, F, n-Hex, CH₃), (M-4687, F, F, F, c-Hex, H), (M-4688, F, F, F, c-Hex, Cl), (M-4689, F, F, F, c-Hex, F), (M-4690, F, F, F, c-Hex, CF₃), (M-4691, F, F, F, c-Hex, Br), (M-4692, F, F, F, c-Hex, CH₃), (M-4693, F, F, F, OH, H), (M-4694, F, F, F, OH, Cl), (M-4695, F, F, F, OH, F), (M-4696, F, F, F, OH, CF₃), (M-4697, F, F, F, OH, Br), (M-4698, F, F, F, OH, CH₃), (M-4699, F, F, F, EtO, H), (M-4700, F, F, F, EtO, Cl), (M-4701, F, F, F, EtO, F), (M-4702, F, F, F, EtO, CF₃), (M-4703, F, F, F, EtO, Br), (M-4704, F, F, F, EtO, CH₃), (M-4705, F, F, F, n-PrO, H), (M-4706, F, F, F, n-PrO, Cl), (M-4707, F, F, F, n-PrO, F), (M-4708, F, F, F, n-PrO, CF₃), (M-4709, F, F, F, n-PrO, Br), (M-4710, F, F, F, n-PrO, CH₃), (M-4711, F, F, F, PhO, H), (M-4712, F, F, F, PhO, Cl), (M-4713, F, F, F, PhO, F), (M-4714, F, F, F, PhO, CF₃), (M-4715, F, F, F, PhO, Br), (M-4716, F, F, F, PhO, CH₃), (M-4717, F, F, F, BnO, H), (M-4718, F, F, F, BnO, Cl), (M-4719, F, F, F, BnO, F), (M-4720, F, F, F, BnO, CF₃), (M-4721, F, F, F, BnO, Br), (M-4722, F, F, F, BnO, CH₃), (M-4723, F, F, F, PhCH₂CH₂O, H), (M-4724, F, F, F, PhCH₂CH₂O, Cl), (M-4725, F, F, F, PhCH₂CH₂O, F), (M-4726, F, F, F, PhCH₂CH₂O, CF₃), (M-4727, F, F, F, PhCH₂CH₂O, Br), (M-4728, F, F, F, PhCH₂CH₂O, CH₃), (M-4729, F, F, F, CF₃O, H), (M-4730, F, F, F, CF₃O, Cl), (M-4731, F, F, F, CF₃O, F), (M-4732, F, F, F, CF₃O, CF₃), (M-4733, F, F, F, CF₃O, Br), (M-4734, F, F, F, CF₃O, CH₃), (M-4735, F, F, F, Ph, H), (M-4736, F, F, F, Ph, Cl), (M-4737, F, F, F, Ph, F), (M-4738, F, F, F, Ph, CF₃), (M-4739, F, F, F, Ph, Br), (M-4740, F, F, F, Ph, CH₃), (M-4741, F, F, F, 4-F-Ph, H), (M-4742, F, F, F, 4-F-Ph, Cl), (M-4743, F, F, F, 4-F-Ph, F), (M-4744, F, F, F, 4-F-Ph, CF₃), (M-4745, F, F, F, 4-F-Ph, Br), (M-4746, F, F, F, 4-F-Ph, CH₃), (M-4747, F, F, F, 4-CF₃-Ph, H), (M-4748, F, F, F, 4-CF₃-Ph, Cl), (M-4749, F, F, F, 4-CF₃-Ph, F), (M-4750, F, F, F, 4-CF₃-Ph, CF₃), (M-4751, F, F, F, 4-CF₃-Ph, Br), (M-4752, F, F, F, 4-CF₃-Ph, CH₃), (M-4753, F, F, F, 4-(Me)₂N-Ph, H), (M-4754, F, F, F, 4-(Me)₂N-Ph, Cl), (M-4755, F, F, F, 4-(Me)₂N-Ph, F), (M-4756, F, F, F, 4-(Me)₂N-Ph, CF₃), (M-4757, F, F, F, 4-(Me)₂N-Ph, Br), (M-4758, F, F, F, 4-(Me)₂N-Ph, CH₃), (M-4759, F, F, F, 4-OH-Ph, H), (M-4760, F, F, F, 4-OH-Ph, Cl), (M-4761, F, F, F, 4-OH-Ph, F), (M-4762, F, F, F, 4-OH-Ph, CF₃), (M-4763, F, F, F, 4-OH-Ph, Br), (M-4764, F, F, F, 4-OH-Ph, CH₃), (M-4765, F, F, F, 3,4-di-F-Ph, H), (M-4766, F, F, F, 3,4-di-F-Ph, Cl), (M-4767, F, F, F, 3,4-di-F-Ph, F), (M-4768, F, F, F, 3,4-di-F-Ph, CF₃), (M-4769, F, F, F, 3,4-di-F-Ph, Br), (M-4770, F, F, F, 3,4-di-F-Ph, CH₃), (M-4771, F, F, F, 4-COOH-Ph, H), (M-4772, F, F, F, 4-COOH-Ph, Cl), (M-4773, F, F, F, 4-COOH-Ph, F), (M-4774, F, F, F, 4-COOH-Ph, CF₃), (M-4775, F, F, F, 4-COOH-Ph, Br), (M-4776, F, F, F, 4-COOH-Ph, CH₃), (M-4777, F, F, F, Bn, H), (M-4778, F, F, F, Bn, Cl), (M-4779, F, F, F, Bn, F), (M-4780, F, F, F, Bn, CF₃), (M-4781, F, F, F, Bn, Br), (M-4782, F, F, F, Bn, CH₃), (M-4783, F, F, F, 4-F-Bn, H), (M-4784, F, F, F, 4-F-Bn, Cl), (M-4785, F, F, F, 4-F-Bn, F), (M-4786, F, F, F, 4-F-Bn, CF₃), (M-4787, F, F, F, 4-F-Bn, Br), (M-4788, F, F, F, 4-F-Bn, CH₃), (M-4789, F, F, F, 2-Py, H), (M-4790, F, F, F, 2-Py, Cl), (M-4791, F, F, F, 2-Py, F), (M-4792, F, F, F, 2-Py, CF₃), (M-4793, F, F, F, 2-Py, Br), (M-4794, F, F, F, 2-Py, CH₃), (M-4795, F, F, F, 3-Py, H), (M-4796, F, F, F, 3-Py, Cl), (M-4797, F, F, F, 3-Py, F), (M-4798, F, F, F, 3-Py, CF₃), (M-4799, F, F, F, 3-Py, Br), (M-4800, F, F, F, 3
-Py, CH₃), (M-4801, F, F, F, 4-Py, H), (M-4802, F, F, F, 4-Py, Cl), (M-4803, F, F, F, 4-Py, F), (M-4804, F, F, F, 4-Py, CF₃), (M-4805, F, F, F, 4-Py, Br), (M-4806, F, F, F, 4-Py, CH₃), (M-4807, F, F, F, 2-Th, H), (M-4808, F, F, F, 2-Th, Cl), (M-4809, F, F, F, 2-Th, F), (M-4810, F, F, F, 2-Th, CF₃), (M-4811, F, F, F, 2-Th, Br), (M-4812, F, F, F, 2-Th, CH₃), (M-4813, F, F, F, 3-Th, H), (M-4814, F, F, F, 3-Th, Cl), (M-4815, F, F, F, 3-Th, F), (M-4816, F, F, F, 3-Th, CF₃), (M-4817, F, F, F, 3-Th, Br), (M-4818, F, F, F, 3-Th, CH₃), (M-4819, F, F, F, pyrazol-2-yl, H), (M-4820, F, F, F, pyrazol-2-yl, Cl), (M-4821, F, F, F, pyrazol-2-yl, F), (M-4822, F, F, F, pyrazol-2-yl, CF₃), (M-4823, F, F, F, pyrazol-2-yl, Br), (M-4824, F, F, F, pyrazol-2-yl, CH₃), (M-4825, F, F, F, pyrazol-3-yl, H), (M-4826, F, F, F, pyrazol-3-yl, Cl), (M-4827, F, F, F, pyrazol-3-yl, F), (M-4828, F, F, F, pyrazol-3-yl, CF₃), (M-4829, F, F, F, pyrazol-3-yl, Br), (M-4830, F, F, F, pyrazol-3-yl, CH₃), (M-4831, F, F, F, pyrimidin-2-yl, H), (M-4832, F, F, F, pyrimidin-2-yl, Cl), (M-4833, F, F, F, pyrimidin-2-yl, F), (M-4834, F, F, F, pyrimidin-2-yl, CF₃), (M-4835, F, F, F, pyrimidin-2-yl, Br), (M-4836, F, F, F, pyrimidin-2-yl, CH₃), (M-4837, F, F, F, pyrimidin-4-yl, H), (M-4838, F, F, F, pyrimidin-4-yl, Cl), (M-4839, F, F, F, pyrimidin-4-yl, F), (M-4840, F, F, F, pyrimidin-4-yl, CF₃), (M-4841, F, F, F, pyrimidin-4-yl, Br), (M-4842, F, F, F, pyrimidin-4-yl, CH₃), (M-4843, F, F, F, pyrimidin-5-yl, H), (M-4844, F, F, F, pyrimidin-5-yl, Cl), (M-4845, F, F, F, pyrimidin-5-yl, F), (M-4846, F, F, F, pyrimidin-5-yl, CF₃), (M-4847, F, F, F, pyrimidin-5-yl, Br), (M-4848, F, F, F, pyrimidin-5-yl, CH₃), (M-4849, F, F, F, HOOCCH₂CH₂CH₂, H), (M-4850, F, F, F, HOOCCH₂CH₂CH₂, Cl), (M-4851, F, F, F, HOOCCH₂CH₂CH₂, F), (M-4852, F, F, F, HOOCCH₂CH₂CH₂, CF₃), (M-4853, F, F, F, HOOCCH₂CH₂CH₂, Br), (M-4854, F, F, F, HOOCCH₂CH₂CH₂, CH₃), (M-4855, F, F, F, HOOCCH₂CH₂CH₂CH₂, H), (M-4856, F, F, F, HOOCCH₂CH₂CH₂CH₂, Cl), (M-4857, F, F, F, HOOCCH₂CH₂CH₂CH₂, F), (M-4858, F, F, F, HOOCCH₂CH₂CH₂CH₂, CF₃), (M-4859, F, F, F, HOOCCH₂CH₂CH₂CH₂, Br), (M-4860, F, F, F, HOOCCH₂CH₂CH₂CH₂, CH₃), (M-4861, F, F, F, (Me)₂NCOCH₂CH₂CH₂CH₂, H), (M-4862, F, F, F, (Me)₂NCOCH₂CH₂CH₂CH₂, Cl), (M-4863, F, F, F, (Me)₂NCOCH₂CH₂CH₂CH₂, F), (M-4864, F, F, F, (Me)₂NCOCH₂CH₂CH₂CH₂, CF₃), (M-4865, F, F, F, (Me)₂NCOCH₂CH₂CH₂CH₂, Br), (M-4866, F, F, F, (Me)₂NCOCH₂CH₂CH₂CH₂, CH₃), (M-4867, F, F, F, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, H), (M-4868, F, F, F, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, Cl), (M-4869, F, F, F, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, F), (M-4870, F, F, F, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, CF₃), (M-4871, F, F, F, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, Br), (M-4872, F, F, F, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, CH₃), (M-4873, F, F, F, MeOCH₂, H), (M-4874, F, F, F, MeOCH₂, Cl), (M-4875, F, F, F, MeOCH₂, F), (M-4876, F, F, F, MeOCH₂, CF₃), (M-4877, F, F, F, MeOCH₂, Br), (M-4878, F, F, F, MeOCH₂, CH₃), (M-4879, F, F, F, EtOCH₂, H), (M-4880, F, F, F, EtOCH₂, Cl), (M-4881, F, F, F, EtOCH₂, F), (M-4882, F, F, F, EtOCH₂, CF₃), (M-4883, F, F, F, EtOCH₂, Br), (M-4884, F, F, F, EtOCH₂, CH₃), (M-4885, F, F, F, EtOCH₂CH₂, H), (M-4886, F, F, F, EtOCH₂CH₂, Cl), (M-4887, F, F, F, EtOCH₂CH₂, F), (M-4888, F, F, F, EtOCH₂CH₂, CF₃), (M-4889, F, F, F, EtOCH₂CH₂, Br), (M-4890, F, F, F, EtOCH₂CH₂, CH₃), (M-4891, F, F, F, MeOCH₂CH₂OCH₂CH₂, H), (M-4892, F, F, F, MeOCH₂CH₂OCH₂CH₂, Cl), (M-4893, F, F, F, MeOCH₂CH₂OCH₂CH₂, F), (M-4894, F, F, F, MeOCH₂CH₂OCH₂CH₂, CF₃), (M-4895, F, F, F, MeOCH₂CH₂OCH₂CH₂, Br), (M-4896, F, F, F, MeOCH₂CH₂OCH₂CH₂, CH₃), (M-4897, F, F, F, MeOCH₂CH₂, H), (M-4898, F, F, F, MeOCH₂CH₂, Cl), (M-4899, F, F, F, MeOCH₂CH₂, F), (M-4900, F, F, F, MeOCH₂CH₂, CF₃), (M-4901, F, F, F, MeOCH₂CH₂, Br), (M-4902, F, F, F, MeOCH₂CH₂, CH₃), (M-4903, F, F, F, HOCH₂, H), (M-4904, F, F, F, HOCH₂, Cl), (M-4905, F, F, F, HOCH₂, F), (M-4906, F, F, F, HOCH₂, CF₃), (M-4907, F, F, F, HOCH₂, Br), (M-4908, F, F, F, HOCH₂, CH₃), (M-4909, F, F, F, HOCH₂CH₂, H), (M-4910, F, F, F, HOCH₂CH₂, Cl), (M-4911, F, F, F, HOCH₂CH₂, F), (M-4912, F, F, F, HOCH₂CH₂, CF₃), (M-4913, F, F, F, HOCH₂CH₂, Br), (M-4914, F, F, F, HOCH₂CH₂, CH₃), (M-4915, F, F, F, HOCH₂CH₂CH₂, H), (M-4916, F, F, F, HOCH₂CH₂CH₂, Cl), (M-4917, F, F, F, HOCH₂CH₂CH₂, F), (M-4918, F, F, F, HOCH₂CH₂CH₂, CF₃), (M-4919, F, F, F, HOCH₂CH₂CH₂, Br), (M-4920, F, F, F, HOCH₂CH₂CH₂, CH₃), (M-4921, F, F, F, HOCH₂CH₂CH₂CH₂, H), (M-4922, F, F, F, HOCH₂CH₂CH₂CH₂, Cl), (M-4923, F, F, F, HOCH₂CH₂CH₂CH₂, F), (M-4924, F, F, F, HOCH₂CH₂CH₂CH₂, CF₃), (M-4925, F, F, F, HOCH₂CH₂CH₂CH₂, Br), (M-4926, F, F, F, HOCH₂CH₂CH₂CH₂, CH₃), (M-4927, F, F, F, HOCH₂CH₂CH₂CH₂CH₂, H), (M-4928, F, F, F, HOCH₂CH₂CH₂CH₂CH₂, Cl), (M-4929, F, F, F, HOCH₂CH₂CH₂CH₂CH₂, F), (M-4930, F, F, F, HOCH₂CH₂CH₂CH₂CH₂, CF₃), (M-4931, F, F, F, HOCH₂CH₂CH₂CH₂CH₂, Br), (M-4932, F, F, F, HOCH₂CH₂CH₂CH₂CH₂, CH₃), (M-4933, F, F, F, HOCH₂CH₂OCH₂CH₂, H), (M-4934, F, F, F, HOCH₂CH₂OCH₂CH₂, Cl), (M-4935, F, F, F, HOCH₂CH₂OCH₂CH₂, F), (M-4936, F, F, F, HOCH₂CH₂OCH₂CH₂, CF₃), (M-4937, F, F, F, HOCH₂CH₂OCH₂CH₂, Br), (M-4938, F, F, F, HOCH₂CH₂OCH₂CH₂, CH₃), (M-4939, F, F, F, (Me)₂N, H), (M-4940, F, F, F, (Me)₂N, Cl), (M-4941, F, F, F, (Me)₂N, F), (M-4942, F, F, F, (Me)₂N, CF₃), (M-4943, F, F, F, (Me)₂N, Br), (M-4944, F, F, F, (Me)₂N, CH₃), (M-4945, F, F, F, piperidin-4-yl-methyl, H), (M-4946, F, F, F, piperidin-4-yl-methyl, Cl), (M-4947, F, F, F, piperidin-4-yl-methyl, F), (M-4948, F, F, F, piperidin-4-yl-methyl, CF₃), (M-4949, F, F, F, piperidin-4-yl-methyl, Br), (M-4950, F, F, F, piperidin-4-yl-methyl, CH₃), (M-4951, F, F, F, cyclohexylmethyl, H), (M-4952, F, F, F, cyclohexylmethyl, Cl), (M-4953, F, F, F, cyclohexylmethyl, F), (M-4954, F, F, F, cyclohexylmethyl, CF₃), (M-4955, F, F, F, cyclohexylmethyl, Br), (M-4956, F, F, F, cyclohexylmethyl, CH₃), (M-4957, F, F, Cl, H, H), (M-4958, F, F, Cl, H, Cl), (M-4959, F, F, Cl, H, F), (M-4960, F, F, Cl, H, CF₃), (M-4961, F, F, Cl, H, Br), (M-4962, F, F, Cl, H, CH₃), (M-4963, F, F, Cl, F, H), (M-4964, F, F, Cl, F, Cl), (M-4965, F, F, Cl, F, F), (M-4966, F, F, Cl, F, CF₃), (M-4967, F, F, Cl, F, Br), (M-4968, F, F, Cl, F, CH₃), (M-4969, F, F, Cl, Cl, H), (M-4970, F, F, Cl, Cl, Cl), (M-4971, F, F, Cl, Cl, F), (M-4972, F, F, Cl, Cl, CF₃), (M-4973, F, F, Cl, Cl, Br), (M-4974, F, F, Cl, Cl, CH₃), (M-4975, F, F, Cl, CH₃, H), (M-4976, F, F, Cl, CH₃, Cl), (M-4977, F, F, Cl, CH₃, F), (M-4978, F, F, Cl, CH₃, CF₃
), (M-4979, F, F, Cl, CH₃, Br), (M-4980, F, F, Cl, CH₃, CH₃), (M-4981, F, F, Cl, Et, H), (M-4982, F, F, Cl, Et, Cl), (M-4983, F, F, Cl, Et, F), (M-4984, F, F, Cl, Et, CF₃), (M-4985, F, F, Cl, Et, Br), (M-4986, F, F, Cl, Et, CH₃), (M-4987, F, F, Cl, n-Pr, H), (M-4988, F, F, Cl, n-Pr, Cl), (M-4989, F, F, Cl, n-Pr, F), (M-4990, F, F, Cl, n-Pr, CF₃), (M-4991, F, F, Cl, n-Pr, Br), (M-4992, F, F, Cl, n-Pr, CH₃), (M-4993, F, F, Cl, c-Pr, H), (M-4994, F, F, Cl, c-Pr, Cl), (M-4995, F, F, Cl, c-Pr, F), (M-4996, F, F, Cl, c-Pr, CF₃), (M-4997, F, F, Cl, c-Pr, Br), (M-4998, F, F, Cl, c-Pr, CH₃), (M-4999, F, F, Cl, i-Pr, H), (M-5000, F, F, Cl, i-Pr, Cl), (M-5001, F, F, Cl, i-Pr, F), (M-5002, F, F, Cl, i-Pr, CF₃), (M-5003, F, F, Cl, i-Pr, Br), (M-5004, F, F, Cl, i-Pr, CH₃), (M-5005, F, F, Cl, n-Bu, H), (M-5006, F, F, Cl, n-Bu, Cl), (M-5007, F, F, Cl, n-Bu, F), (M-5008, F, F, Cl, n-Bu, CF₃), (M-5009, F, F, Cl, n-Bu, Br), (M-5010, F, F, Cl, n-Bu, CH₃), (M-5011, F, F, Cl, i-Bu, H), (M-5012, F, F, Cl, i-Bu, Cl), (M-5013, F, F, Cl, i-Bu, F), (M-5014, F, F, Cl, i-Bu, CF₃), (M-5015, F, F, Cl, i-Bu, Br), (M-5016, F, F, Cl, i-Bu, CH₃), (M-5017, F, F, Cl, sec-Bu, H), (M-5018, F, F, Cl, sec-Bu, Cl), (M-5019, F, F, Cl, sec-Bu, F), (M-5020, F, F, Cl, sec-Bu, CF₃), (M-5021, F, F, Cl, sec-Bu, Br), (M-5022, F, F, Cl, sec-Bu, CH₃), (M-5023, F, F, Cl, n-Pen, H), (M-5024, F, F, Cl, n-Pen, Cl), (M-5025, F, F, Cl, n-Pen, F), (M-5026, F, F, Cl, n-Pen, CF₃), (M-5027, F, F, Cl, n-Pen, Br), (M-5028, F, F, Cl, n-Pen, CH₃), (M-5029, F, F, Cl, c-Pen, H), (M-5030, F, F, Cl, c-Pen, Cl), (M-5031, F, F, Cl, c-Pen, F), (M-5032, F, F, Cl, c-Pen, CF₃), (M-5033, F, F, Cl, c-Pen, Br), (M-5034, F, F, Cl, c-Pen, CH₃), (M-5035, F, F, Cl, n-Hex, H), (M-5036, F, F, Cl, n-Hex, Cl), (M-5037, F, F, Cl, n-Hex, F), (M-5038, F, F, Cl, n-Hex, CF₃), (M-5039, F, F, Cl, n-Hex, Br), (M-5040, F, F, Cl, n-Hex, CH₃), (M-5041, F, F, Cl, c-Hex, H), (M-5042, F, F, Cl, c-Hex, Cl), (M-5043, F, F, Cl, c-Hex, F), (M-5044, F, F, Cl, c-Hex, CF₃), (M-5045, F, F, Cl, c-Hex, Br), (M-5046, F, F, Cl, c-Hex, CH₃), (M-5047, F, F, Cl, OH, H), (M-5048, F, F, Cl, OH, Cl), (M-5049, F, F, Cl, OH, F), (M-5050, F, F, Cl, OH, CF₃), (M-5051, F, F, Cl, OH, Br), (M-5052, F, F, Cl, OH, CH₃), (M-5053, F, F, Cl, EtO, H), (M-5054, F, F, Cl, EtO, Cl), (M-5055, F, F, Cl, EtO, F), (M-5056, F, F, Cl, EtO, CF₃), (M-5057, F, F, Cl, EtO, Br), (M-5058, F, F, Cl, EtO, CH₃), (M-5059, F, F, Cl, n-PrO, H), (M-5060, F, F, Cl, n-PrO, Cl), (M-5061, F, F, Cl, n-PrO, F), (M-5062, F, F, Cl, n-PrO, CF₃), (M-5063, F, F, Cl, n-PrO, Br), (M-5064, F, F, Cl, n-PrO, CH₃), (M-5065, F, F, Cl, PhO, H), (M-5066, F, F, Cl, PhO, Cl), (M-5067, F, F, Cl, PhO, F), (M-5068, F, F, Cl, PhO, CF₃), (M-5069, F, F, Cl, PhO, Br), (M-5070, F, F, Cl, PhO, CH₃), (M-5071, F, F, Cl, BnO, H), (M-5072, F, F, Cl, BnO, Cl), (M-5073, F, F, Cl, BnO, F), (M-5074, F, F, Cl, BnO, CF₃), (M-5075, F, F, Cl, BnO, Br), (M-5076, F, F, Cl, BnO, CH₃), (M-5077, F, F, Cl, PhCH₂CH₂O, H), (M-5078, F, F, Cl, PhCH₂CH₂O, Cl), (M-5079, F, F, Cl, PhCH₂CH₂O, F), (M-5080, F, F, Cl, PhCH₂CH₂O, CF₃), (M-5081, F, F, Cl, PhCH₂CH₂O, Br), (M-5082, F, F, Cl, PhCH₂CH₂O, CH₃), (M-5083, F, F, Cl, CF₃O, H), (M-5084, F, F, Cl, CF₃O, Cl), (M-5085, F, F, Cl, CF₃O, F), (M-5086, F, F, Cl, CF₃O, CF₃), (M-5087, F, F, Cl, CF₃O, Br), (M-5088, F, F, Cl, CF₃O, CH₃), (M-5089, F, F, Cl, Ph, H), (M-5090, F, F, Cl, Ph, Cl), (M-5091, F, F, Cl, Ph, F), (M-5092, F, F, Cl, Ph, CF₃), (M-5093, F, F, Cl, Ph, Br), (M-5094, F, F, Cl, Ph, CH₃), (M-5095, F, F, Cl, 4-F-Ph, H), (M-5096, F, F, Cl, 4-F-Ph, Cl), (M-5097, F, F, Cl, 4-F-Ph, F), (M-5098, F, F, Cl, 4-F-Ph, CF₃), (M-5099, F, F, Cl, 4-F-Ph, Br), (M-5100, F, F, Cl, 4-F-Ph, CH₃), (M-5101, F, F, Cl, 4-CF₃-Ph, H), (M-5102, F, F, Cl, 4-CF₃-Ph, Cl), (M-5103, F, F, Cl, 4-CF₃-Ph, F), (M-5104, F, F, Cl, 4-CF₃-Ph, CF₃), (M-5105, F, F, Cl, 4-CF₃-Ph, Br), (M-5106, F, F, Cl, 4-CF₃-Ph, CH₃), (M-5107, F, F, Cl, 4-(Me)₂N-Ph, H), (M-5108, F, F, Cl, 4-(Me)₂N-Ph, Cl), (M-5109, F, F, Cl, 4-(Me)₂N-Ph, F), (M-5110, F, F, Cl, 4-(Me)₂N-Ph, CF₃), (M-5111, F, F, Cl, 4-(Me)₂N-Ph, Br), (M-5112, F, F, Cl, 4-(Me)₂N-Ph, CH₃), (M-5113, F, F, Cl, 4-OH-Ph, H), (M-5114, F, F, Cl, 4-OH-Ph, Cl), (M-5115, F, F, Cl, 4-OH-Ph, F), (M-5116, F, F, Cl, 4-OH-Ph, CF₃), (M-5117, F, F, Cl, 4-OH-Ph, Br), (M-5118, F, F, Cl, 4-OH-Ph, CH₃), (M-5119, F, F, Cl, 3,4-di-F-Ph, H), (M-5120, F, F, Cl, 3,4-di-F-Ph, Cl), (M-5121, F, F, Cl, 3,4-di-F-Ph, F), (M-5122, F, F, Cl, 3,4-di-F-Ph, CF₃), (M-5123, F, F, Cl, 3,4-di-F-Ph, Br), (M-5124, F, F, Cl, 3,4-di-F-Ph, CH₃), (M-5125, F, F, Cl, 4-COOH-Ph, H), (M-5126, F, F, Cl, 4-COOH-Ph, Cl), (M-5127, F, F, Cl, 4-COOH-Ph, F), (M-5128, F, F, Cl, 4-COOH-Ph, CF₃), (M-5129, F, F, Cl, 4-COOH-Ph, Br), (M-5130, F, F, Cl, 4-COOH-Ph, CH₃), (M-5131, F, F, Cl, Bn, H), (M-5132, F, F, Cl, Bn, Cl), (M-5133, F, F, Cl, Bn, F), (M-5134, F, F, Cl, Bn, CF₃), (M-5135, F, F, Cl, Bn, Br), (M-5136, F, F, Cl, Bn, CH₃), (M-5137, F, F, Cl, 4-F-Bn, H), (M-5138, F, F, Cl, 4-F-Bn, Cl), (M-5139, F, F, Cl, 4-F-Bn, F), (M-5140, F, F, Cl, 4-F-Bn, CF₃), (M-5141, F, F, Cl, 4-F-Bn, Br), (M-5142, F, F, Cl, 4-F-Bn, CH₃), (M-5143, F, F, Cl, 2-Py, H), (M-5144, F, F, Cl, 2-Py, Cl), (M-5145, F, F, Cl, 2-Py, F), (M-5146, F, F, Cl, 2-Py, CF₃), (M-5147, F, F, Cl, 2-Py, Br), (M-5148, F, F, Cl, 2-Py, CH₃), (M-5149, F, F, Cl, 3-Py, H), (M-5150, F, F, Cl, 3-Py, Cl), (M-5151, F, F, Cl, 3-Py, F), (M-5152, F, F, Cl, 3-Py, CF₃), (M-5153, F, F, Cl, 3-Py, Br), (M-5154, F, F, Cl, 3-Py, CH₃), (M-5155, F, F, Cl, 4-Py, H), (M-5156, F, F, Cl, 4-Py, Cl), (M-5157, F, F, Cl, 4-Py, F), (M-5158, F, F, Cl, 4-Py, CF₃), (M-5159, F, F, Cl, 4-Py, Br), (M-5160, F, F, Cl, 4-Py, CH₃), (M-5161, F, F, Cl, 2-Th, H), (M-5162, F, F, Cl, 2-Th, Cl), (M-5163, F, F, Cl, 2-Th, F), (M-5164, F, F, Cl, 2-Th, CF₃), (M-5165, F, F, Cl, 2-Th, Br), (M-5166, F, F, Cl, 2-Th, CH₃), (M-5167, F, F, Cl, 3-Th, H), (M-5168, F, F, Cl, 3-Th, Cl), (M-5169, F, F, Cl, 3-Th, F), (M-5170, F, F, Cl, 3-Th, CF₃), (M-5171, F, F, Cl, 3-Th, Br), (M-5172, F, F, Cl, 3-Th, CH₃), (M-5173, F, F, Cl, pyrazol-2-yl, H), (M-5174, F, F, Cl, pyrazol-2-yl, Cl), (M-5175, F, F, Cl, pyrazol-2-yl, F), (M-5176, F, F, Cl, pyrazol-2-yl, CF₃), (M-5177, F, F, Cl, pyrazol-2-yl, Br), (M-5178, F, F, Cl, pyrazol-2-yl, CH₃), (M-5179, F, F, Cl, pyrazol-3-yl, H), (M-5180, F, F, Cl, pyrazol-3-yl, Cl), (M-5181, F, F, Cl, pyrazol-3-yl, F), (M-5182, F, F, Cl, pyrazol-3-yl, CF₃), (M-5183, F, F, Cl, pyrazol-3-yl, Br), (M-5184, F, F, Cl, pyrazol-3-yl, CH₃), (M-5185, F, F, Cl, pyrimidin-2-yl, H), (M-5186, F, F, Cl, pyrimidin-2-yl, Cl), (M-5187, F, F, Cl, pyrimidin-2-yl, F), (M-5188, F, F, Cl, pyrimidin-2-yl, CF₃), (M-5189, F, F, Cl, pyrimidin-2-yl, Br), (M-5190, F, F, Cl, pyrimidin-2-yl, CH₃), (M-5191, F, F, Cl, pyrimidin-4-yl, H), (M-5192, F, F, Cl, pyrimidin-4-yl, Cl), (M-5193, F, F, Cl, pyrimidin-4-yl, F), (M-5194, F, F, Cl, pyrimidin-4-yl, CF₃), (M-5195, F, F, Cl, pyrimidin-4-yl, Br), (M-5196, F, F, Cl, pyrimidin-4-yl, CH₃), (M-5197, F, F, Cl, pyrimidin-5-yl, H), (M-5198, F, F, Cl, pyrimidin-5-yl, Cl), (M-5199, F, F, Cl, pyrimidin-5-yl, F), (M-5200, F, F, Cl, pyrimidin-5-yl, CF₃), (M-5201, F, F, Cl, pyrimidin-5-yl, Br), (M-5202, F, F, Cl, pyrimidin-5-yl, CH₃), (M-5203, F, F, Cl, HOOCCH₂CH₂CH₂, H), (M-5204, F, F, Cl, HOOCCH₂CH₂CH₂, Cl), (M-5205, F, F, Cl, HOOCCH₂CH₂CH₂, F), (M-5206, F, F, Cl, HOOCCH₂CH₂CH₂, CF₃), (M-5207, F, F, Cl, HOOCCH₂CH₂CH₂, Br), (M-5208, F, F, Cl, HOOCCH₂CH₂CH₂, CH₃), (M-5209, F, F, Cl, HOOCCH₂CH₂CH₂CH₂, H), (M-5210, F, F, Cl, HOOCCH₂CH₂CH₂CH₂, Cl), (M-5211, F, F, Cl, HOOCCH₂CH₂CH₂CH₂, F), (M-5212, F, F, Cl, HOOCCH₂CH₂CH₂CH₂, CF₃), (M-5213, F, F, Cl, HOOCCH₂CH₂CH₂CH₂, Br), (M-5214, F, F, Cl, HOOCCH₂CH₂CH₂CH₂, CH₃), (M-5215, F, F, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂, H), (M-5216, F, F, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂, Cl), (M-5217, F, F, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂, F), (M-5218, F, F, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂, CF₃), (M-5219, F, F, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂, Br), (M-5220, F, F, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂, CH₃), (M-5221, F, F, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, H), (M-5222, F, F, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, Cl), (M-5223, F, F, Cl, (Me)₂
NCOCH₂CH₂CH₂CH₂CH₂, F), (M-5224, F, F, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, CF₃), (M-5225, F, F, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, Br), (M-5226, F, F, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, CH₃), (M-5227, F, F, Cl, MeOCH₂, H), (M-5228, F, F, Cl, MeOCH₂, Cl), (M-5229, F, F, Cl, MeOCH₂, F), (M-5230, F, F, Cl, MeOCH₂, CF₃), (M-5231, F, F, Cl, MeOCH₂, Br), (M-5232, F, F, Cl, MeOCH₂, CH₃), (M-5233, F, F, Cl, EtOCH₂, H), (M-5234, F, F, Cl, EtOCH₂, Cl), (M-5235, F, F, Cl, EtOCH₂, F), (M-5236, F, F, Cl, EtOCH₂, CF₃), (M-5237, F, F, Cl, EtOCH₂, Br), (M-5238, F, F, Cl, EtOCH₂, CH₃), (M-5239, F, F, Cl, EtOCH₂CH₂, H), (M-5240, F, F, Cl, EtOCH₂CH₂, Cl), (M-5241, F, F, Cl, EtOCH₂CH₂, F), (M-5242, F, F, Cl, EtOCH₂CH₂, CF₃), (M-5243, F, F, Cl, EtOCH₂CH₂, Br), (M-5244, F, F, Cl, EtOCH₂CH₂, CH₃), (M-5245, F, F, Cl, MeOCH₂CH₂OCH₂CH₂, H), (M-5246, F, F, Cl, MeOCH₂CH₂OCH₂CH₂, Cl), (M-5247, F, F, Cl, MeOCH₂CH₂OCH₂CH₂, F), (M-5248, F, F, Cl, MeOCH₂CH₂OCH₂CH₂, CF₃), (M-5249, F, F, Cl, MeOCH₂CH₂OCH₂CH₂, Br), (M-5250, F, F, Cl, MeOCH₂CH₂OCH₂CH₂, CH₃), (M-5251, F, F, Cl, MeOCH₂CH₂, H), (M-5252, F, F, Cl, MeOCH₂CH₂, Cl), (M-5253, F, F, Cl, MeOCH₂CH₂, F), (M-5254, F, F, Cl, MeOCH₂CH₂, CF₃), (M-5255, F, F, Cl, MeOCH₂CH₂, Br), (M-5256, F, F, Cl, MeOCH₂CH₂, CH₃), (M-5257, F, F, Cl, HOCH₂, H), (M-5258, F, F, Cl, HOCH₂, Cl), (M-5259, F, F, Cl, HOCH₂, F), (M-5260, F, F, Cl, HOCH₂, CF₃), (M-5261, F, F, Cl, HOCH₂, Br), (M-5262, F, F, Cl, HOCH₂, CH₃), (M-5263, F, F, Cl, HOCH₂CH₂, H), (M-5264, F, F, Cl, HOCH₂CH₂, Cl), (M-5265, F, F, Cl, HOCH₂CH₂, F), (M-5266, F, F, Cl, HOCH₂CH₂, CF₃), (M-5267, F, F, Cl, HOCH₂CH₂, Br), (M-5268, F, F, Cl, HOCH₂CH₂, CH₃), (M-5269, F, F, Cl, HOCH₂CH₂CH₂, H), (M-5270, F, F, Cl, HOCH₂CH₂CH₂, Cl), (M-5271, F, F, Cl, HOCH₂CH₂CH₂, F), (M-5272, F, F, Cl, HOCH₂CH₂CH₂, CF₃), (M-5273, F, F, Cl, HOCH₂CH₂CH₂, Br), (M-5274, F, F, Cl, HOCH₂CH₂CH₂, CH₃), (M-5275, F, F, Cl, HOCH₂CH₂CH₂CH₂, H), (M-5276, F, F, Cl, HOCH₂CH₂CH₂CH₂, Cl), (M-5277, F, F, Cl, HOCH₂CH₂CH₂CH₂, F), (M-5278, F, F, Cl, HOCH₂CH₂CH₂CH₂, CF₃), (M-5279, F, F, Cl, HOCH₂CH₂CH₂CH₂, Br), (M-5280, F, F, Cl, HOCH₂CH₂CH₂CH₂, CH₃), (M-5281, F, F, Cl, HOCH₂CH₂CH₂CH₂CH₂, H), (M-5282, F, F, Cl, HOCH₂CH₂CH₂CH₂CH₂, Cl), (M-5283, F, F, Cl, HOCH₂CH₂CH₂CH₂CH₂, F), (M-5284, F, F, Cl, HOCH₂CH₂CH₂CH₂CH₂, CF₃), (M-5285, F, F, Cl, HOCH₂CH₂CH₂CH₂CH₂, Br), (M-5286, F, F, Cl, HOCH₂CH₂CH₂CH₂CH₂, CH₃), (M-5287, F, F, Cl, HOCH₂CH₂OCH₂CH₂, H), (M-5288, F, F, Cl, HOCH₂CH₂OCH₂CH₂, Cl), (M-5289, F, F, Cl, HOCH₂CH₂OCH₂CH₂, F), (M-5290, F, F, Cl, HOCH₂CH₂OCH₂CH₂, CF₃), (M-5291, F, F, Cl, HOCH₂CH₂OCH₂CH₂, Br), (M-5292, F, F, Cl, HOCH₂CH₂OCH₂CH₂, CH₃), (M-5293, F, F, Cl, (Me)₂N, H), (M-5294, F, F, Cl, (Me)₂N, Cl), (M-5295, F, F, Cl, (Me)₂N, F), (M-5296, F, F, Cl, (Me)₂N, CF₃), (M-5297, F, F, Cl, (Me)₂N, Br), (M-5298, F, F, Cl, (Me)₂N, CH₃), (M-5299, F, F, Cl, piperidin-4-yl-methyl, H), (M-5300, F, F, Cl, piperidin-4-yl-methyl, Cl), (M-5301, F, F, Cl, piperidin-4-yl-methyl, F), (M-5302, F, F, Cl, piperidin-4-yl-methyl, CF₃), (M-5303, F, F, Cl, piperidin-4-yl-methyl, Br), (M-5304, F, F, Cl, piperidin-4-yl-methyl, CH₃), (M-5305, F, F, Cl, cyclohexylmethyl, H), (M-5306, F, F, Cl, cyclohexylmethyl, Cl), (M-5307, F, F, Cl, cyclohexylmethyl, F), (M-5308, F, F, Cl, cyclohexylmethyl, CF₃), (M-5309, F, F, Cl, cyclohexylmethyl, Br), (M-5310, F, F, Cl, cyclohexylmethyl, CH₃), (M-5311, F, CH₃, H, H, H), (M-5312, F, CH₃, H, H, Cl), (M-5313, F, CH₃, H, H, F), (M-5314, F, CH₃, H, H, CF₃), (M-5315, F, CH₃, H, H, Br), (M-5316, F, CH₃, H, H, CH₃), (M-5317, F, CH₃, H, F, H), (M-5318, F, CH₃, H, F, Cl), (M-5319, F, CH₃, H, F, F), (M-5320, F, CH₃, H, F, CF₃), (M-5321, F, CH₃, H, F, Br), (M-5322, F, CH₃, H, F, CH₃), (M-5323, F, CH₃, H, Cl, H), (M-5324, F, CH₃, H, Cl, Cl), (M-5325, F, CH₃, H, Cl, F), (M-5326, F, CH₃, H, Cl, CF₃), (M-5327, F, CH₃, H, Cl, Br), (M-5328, F, CH₃, H, Cl, CH₃), (M-5329, F, CH₃, H, CH₃, H), (M-5330, F, CH₃, H, CH₃, Cl), (M-5331, F, CH₃, H, CH₃, F), (M-5332, F, CH₃, H, CH₃, CF₃), (M-5333, F, CH₃, H, CH₃, Br), (M-5334, F, CH₃, H, CH₃, CH₃), (M-5335, F, CH₃, H, Et, H), (M-5336, F, CH₃, H, Et, Cl), (M-5337, F, CH₃, H, Et, F), (M-5338, F, CH₃, H, Et, CF₃), (M-5339, F, CH₃, H, Et, Br), (M-5340, F, CH₃, H, Et, CH₃), (M-5341, F, CH₃, H, n-Pr, H), (M-5342, F, CH₃, H, n-Pr, Cl), (M-5343, F, CH₃, H, n-Pr, F), (M-5344, F, CH₃, H, n-Pr, CF₃), (M-5345, F, CH₃, H, n-Pr, Br), (M-5346, F, CH₃, H, n-Pr, CH₃), (M-5347, F, CH₃, H, c-Pr, H), (M-5348, F, CH₃, H, c-Pr, Cl), (M-5349, F, CH₃, H, c-Pr, F), (M-5350, F, CH₃, H, c-Pr, CF₃), (M-5351, F, CH₃, H, c-Pr, Br), (M-5352, F, CH₃, H, c-Pr, CH₃), (M-5353, F, CH₃, H, i-Pr, H), (M-5354, F, CH₃, H, i-Pr, Cl), (M-5355, F, CH₃, H, i-Pr, F), (M-5356, F, CH₃, H, i-Pr, CF₃), (M-5357, F, CH₃, H, i-Pr, Br), (M-5358, F, CH₃, H, i-Pr, CH₃), (M-5359, F, CH₃, H, n-Bu, H), (M-5360, F, CH₃, H, n-Bu, Cl), (M-5361, F, CH₃, H, n-Bu, F), (M-5362, F, CH₃, H, n-Bu, CF₃), (M-5363, F, CH₃, H, n-Bu, Br), (M-5364, F, CH₃, H, n-Bu, CH₃), (M-5365, F, CH₃, H, i-Bu, H), (M-5366, F, CH₃, H, i-Bu, Cl), (M-5367, F, CH₃, H, i-Bu, F), (M-5368, F, CH₃, H, i-Bu, CF₃), (M-5369, F, CH₃, H, i-Bu, Br), (M-5370, F, CH₃, H, i-Bu, CH₃), (M-5371, F, CH₃, H, sec-Bu, H), (M-5372, F, CH₃, H, sec-Bu, Cl), (M-5373, F, CH₃, H, sec-Bu, F), (M-5374, F, CH₃, H, sec-Bu, CF₃), (M-5375, F, CH₃, H, sec-Bu, Br), (M-5376, F, CH₃, H, sec-Bu, CH₃), (M-5377, F, CH₃, H, n-Pen, H), (M-5378, F, CH₃, H, n-Pen, Cl), (M-5379, F, CH₃, H, n-Pen, F), (M-5380, F, CH₃, H, n-Pen, CF₃), (M-5381, F, CH₃, H, n-Pen, Br), (M-5382, F, CH₃, H, n-Pen, CH₃), (M-5383, F, CH₃, H, c-Pen, H), (M-5384, F, CH₃, H, c-Pen, Cl), (M-5385, F, CH₃, H, c-Pen, F), (M-5386, F, CH₃, H, c-Pen, CF₃), (M-5387, F, CH₃, H, c-Pen, Br), (M-5388, F, CH₃, H, c-Pen, CH₃), (M-5389, F, CH₃, H, n-Hex, H), (M-5390, F, CH₃, H, n-Hex, Cl), (M-5391, F, CH₃, H, n-Hex, F), (M-5392, F, CH₃, H, n-Hex, CF₃), (M-5393, F, CH₃, H, n-Hex, Br), (M-5394, F, CH₃, H, n-Hex, CH₃), (M-5395, F, CH₃, H, c-Hex, H), (M-5396, F, CH₃, H, c-Hex, Cl), (M-5397, F, CH₃, H, c-Hex, F), (M-5398, F, CH₃, H, c-Hex, CF₃), (M-5399, F, CH₃, H, c-Hex, Br), (M-5400, F, CH₃, H, c-Hex, CH₃), (M-5401, F, CH₃, H, OH, H), (M-5402, F, CH₃, H, OH, Cl), (M-5403, F, CH₃, H, OH, F), (M-5404, F, CH₃, H, OH, CF₃), (M-5405, F, CH₃, H, OH, Br), (M-5406, F,
CH₃, H, OH, CH₃), (M-5407, F, CH₃, H, EtO, H), (M-5408, F, CH₃, H, EtO, Cl), (M-5409, F, CH₃, H, EtO, F), (M-5410, F, CH₃, H, EtO, CF₃), (M-5411, F, CH₃, H, EtO, Br), (M-5412, F, CH₃, H, EtO, CH₃), (M-5413, F, CH₃, H, n-PrO, H), (M-5414, F, CH₃, H, n-PrO, Cl), (M-5415, F, CH₃, H, n-PrO, F), (M-5416, F, CH₃, H, n-PrO, CF₃), (M-5417, F, CH₃, H, n-PrO, Br), (M-5418, F, CH₃, H, n-PrO, CH₃), (M-5419, F, CH₃, H, PhO, H), (M-5420, F, CH₃, H, PhO, Cl), (M-5421, F, CH₃, H, PhO, F), (M-5422, F, CH₃, H, PhO, CF₃), (M-5423, F, CH₃, H, PhO, Br), (M-5424, F, CH₃, H, PhO, CH₃), (M-5425, F, CH₃, H, BnO, H), (M-5426, F, CH₃, H, BnO, Cl), (M-5427, F, CH₃, H, BnO, F), (M-5428, F, CH₃, H, BnO, CF₃), (M-5429, F, CH₃, H, BnO, Br), (M-5430, F, CH₃, H, BnO, CH₃), (M-5431, F, CH₃, H, PhCH₂CH₂O, H), (M-5432, F, CH₃, H, PhCH₂CH₂O, Cl), (M-5433, F, CH₃, H, PhCH₂CH₂O, F), (M-5434, F, CH₃, H, PhCH₂CH₂O, CF₃), (M-5435, F, CH₃, H, PhCH₂CH₂O, Br), (M-5436, F, CH₃, H, PhCH₂CH₂O, CH₃), (M-5437, F, CH₃, H, CF₃O, H), (M-5438, F, CH₃, H, CF₃O, Cl), (M-5439, F, CH₃, H, CF₃O, F), (M-5440, F, CH₃, H, CF₃O, CF₃), (M-5441, F, CH₃, H, CF₃O, Br), (M-5442, F, CH₃, H, CF₃O, CH₃), (M-5443, F, CH₃, H, Ph, H), (M-5444, F, CH₃, H, Ph, Cl), (M-5445, F, CH₃, H, Ph, F), (M-5446, F, CH₃, H, Ph, CF₃), (M-5447, F, CH₃, H, Ph, Br), (M-5448, F, CH₃, H, Ph, CH₃), (M-5449, F, CH₃, H, 4-F-Ph, H), (M-5450, F, CH₃, H, 4-F-Ph, Cl), (M-5451, F, CH₃, H, 4-F-Ph, F), (M-5452, F, CH₃, H, 4-F-Ph, CF₃), (M-5453, F, CH₃, H, 4-F-Ph, Br), (M-5454, F, CH₃, H, 4-F-Ph, CH₃), (M-5455, F, CH₃, H, 4-CF₃-Ph, H), (M-5456, F, CH₃, H, 4-CF₃-Ph, Cl), (M-5457, F, CH₃, H, 4-CF₃-Ph, F), (M-5458, F, CH₃, H, 4-CF₃-Ph, CF₃), (M-5459, F, CH₃, H, 4-CF₃-Ph, Br), (M-5460, F, CH₃, H, 4-CF₃-Ph, CH₃), (M-5461, F, CH₃, H, 4-(Me)₂N-Ph, H), (M-5462, F, CH₃, H, 4-(Me)₂N-Ph, Cl), (M-5463, F, CH₃, H, 4-(Me)₂N-Ph, F), (M-5464, F, CH₃, H, 4-(Me)₂N-Ph, CF₃), (M-5465, F, CH₃, H, 4-(Me)₂N-Ph, Br), (M-5466, F, CH₃, H, 4-(Me)₂N-Ph, CH₃), (M-5467, F, CH₃, H, 4-OH-Ph, H), (M-5468, F, CH₃, H, 4-OH-Ph, Cl), (M-5469, F, CH₃, H, 4-OH-Ph, F), (M-5470, F, CH₃, H, 4-OH-Ph, CF₃), (M-5471, F, CH₃, H, 4-OH-Ph, Br), (M-5472, F, CH₃, H, 4-OH-Ph, CH₃), (M-5473, F, CH₃, H, 3,4-di-F-Ph, H), (M-5474, F, CH₃, H, 3,4-di-F-Ph, Cl), (M-5475, F, CH₃, H, 3,4-di-F-Ph, F), (M-5476, F, CH₃, H, 3,4-di-F-Ph, CF₃), (M-5477, F, CH₃, H, 3,4-di-F-Ph, Br), (M-5478, F, CH₃, H, 3,4-di-F-Ph, CH₃), (M-5479, F, CH₃, H, 4-COOH-Ph, H), (M-5480, F, CH₃, H, 4-COOH-Ph, Cl), (M-5481, F, CH₃, H, 4-COOH-Ph, F), (M-5482, F, CH₃, H, 4-COOH-Ph, CF₃), (M-5483, F, CH₃, H, 4-COOH-Ph, Br), (M-5484, F, CH₃, H, 4-COOH-Ph, CH₃), (M-5485, F, CH₃, H, Bn, H), (M-5486, F, CH₃, H, Bn, Cl), (M-5487, F, CH₃, H, Bn, F), (M-5488, F, CH₃, H, Bn, CF₃), (M-5489, F, CH₃, H, Bn, Br), (M-5490, F, CH₃, H, Bn, CH₃), (M-5491, F, CH₃, H, 4-F-Bn, H), (M-5492, F, CH₃, H, 4-F-Bn, Cl), (M-5493, F, CH₃, H, 4-F-Bn, F), (M-5494, F, CH₃, H, 4-F-Bn, CF₃), (M-5495, F, CH₃, H, 4-F-Bn, Br), (M-5496, F, CH₃, H, 4-F-Bn, CH₃), (M-5497, F, CH₃, H, 2-Py, H), (M-5498, F, CH₃, H, 2-Py, Cl), (M-5499, F, CH₃, H, 2-Py, F), (M-5500, F, CH₃, H, 2-Py, CF₃), (M-5501, F, CH₃, H, 2-Py, Br), (M-5502, F, CH₃, H, 2-Py, CH₃), (M-5503, F, CH₃, H, 3-Py, H), (M-5504, F, CH₃, H, 3-Py, Cl), (M-5505, F, CH₃, H, 3-Py, F), (M-5506, F, CH₃, H, 3-Py, CF₃), (M-5507, F, CH₃, H, 3-Py, Br), (M-5508, F, CH₃, H, 3-Py, CH₃), (M-5509, F, CH₃, H, 4-Py, H), (M-5510, F, CH₃, H, 4-Py, Cl), (M-5511, F, CH₃, H, 4-Py, F), (M-5512, F, CH₃, H, 4-Py, CF₃), (M-5513, F, CH₃, H, 4-Py, Br), (M-5514, F, CH₃, H, 4-Py, CH₃), (M-5515, F, CH₃, H, 2-Th, H), (M-5516, F, CH₃, H, 2-Th, Cl), (M-5517, F, CH₃, H, 2-Th, F), (M-5518, F, CH₃, H, 2-Th, CF₃), (M-5519, F, CH₃, H, 2-Th, Br), (M-5520, F, CH₃, H, 2-Th, CH₃), (M-5521, F, CH₃, H, 3-Th, H), (M-5522, F, CH₃, H, 3-Th, Cl), (M-5523, F, CH₃, H, 3-Th, F), (M-5524, F, CH₃, H, 3-Th, CF₃), (M-5525, F, CH₃, H, 3-Th, Br), (M-5526, F, CH₃, H, 3-Th, CH₃), (M-5527, F, CH₃, H, pyrazol-2-yl, H), (M-5528, F, CH₃, H, pyrazol-2-yl, Cl), (M-5529, F, CH₃, H, pyrazol-2-yl, F), (M-5530, F, CH₃, H, pyrazol-2-yl, CF₃), (M-5531, F, CH₃, H, pyrazol-2-yl, Br), (M-5532, F, CH₃, H, pyrazol-2-yl, CH₃), (M-5533, F, CH₃, H, pyrazol-3-yl, H), (M-5534, F, CH₃, H, pyrazol-3-yl, Cl), (M-5535, F, CH₃, H, pyrazol-3-yl, F), (M-5536, F, CH₃, H, pyrazol-3-yl, CF₃), (M-5537, F, CH₃, H, pyrazol-3-yl, Br), (M-5538, F, CH₃, H, pyrazol-3-yl, CH₃), (M-5539, F, CH₃, H, pyrimidin-2-yl, H), (M-5540, F, CH₃, H, pyrimidin-2-yl, Cl), (M-5541, F, CH₃, H, pyrimidin-2-yl, F), (M-5542, F, CH₃, H, pyrimidin-2-yl, CF₃), (M-5543, F, CH₃, H, pyrimidin-2-yl, Br), (M-5544, F, CH₃, H, pyrimidin-2-yl, CH₃), (M-5545, F, CH₃, H, pyrimidin-4-yl, H), (M-5546, F, CH₃, H, pyrimidin-4-yl, Cl), (M-5547, F, CH₃, H, pyrimidin-4-yl, F), (M-5548, F, CH₃, H, pyrimidin-4-yl, CF₃), (M-5549, F, CH₃, H, pyrimidin-4-yl, Br), (M-5550, F, CH₃, H, pyrimidin-4-yl, CH₃), (M-5551, F, CH₃, H, pyrimidin-5-yl, H), (M-5552, F, CH₃, H, pyrimidin-5-yl, Cl), (M-5553, F, CH₃, H, pyrimidin-5-yl, F), (M-5554, F, CH₃, H, pyrimidin-5-yl, CF₃), (M-5555, F, CH₃, H, pyrimidin-5-yl, Br), (M-5556, F, CH₃, H, pyrimidin-5-yl, CH₃), (M-5557, F, CH₃, H, HOOCCH₂CH₂CH₂, H), (M-5558, F, CH₃, H, HOOCCH₂CH₂CH₂, Cl), (M-5559, F, CH₃, H, HOOCCH₂CH₂CH₂, F), (M-5560, F, CH₃, H, HOOCCH₂CH₂CH₂, CF₃), (M-5561, F, CH₃, H, HOOCCH₂CH₂CH₂, Br), (M-5562, F, CH₃, H, HOOCCH₂CH₂CH₂, CH₃), (M-5563, F, CH₃, H, HOOCCH₂CH₂CH₂CH₂, H), (M-5564, F, CH₃, H, HOOCCH₂CH₂CH₂CH₂, Cl), (M-5565, F, CH₃, H, HOOCCH₂CH₂CH₂CH₂, F), (M-5566, F, CH₃, H, HOOCCH₂CH₂CH₂CH₂, CF₃), (M-5567, F, CH₃, H, HOOCCH₂CH₂CH₂CH₂, Br), (M-5568, F, CH₃, H, HOOCCH₂CH₂CH₂CH₂, CH₃), (M-5569, F, CH₃, H, (Me)₂NCOCH₂CH₂CH₂CH₂, H), (M-5570, F, CH₃, H, (Me)₂NCOCH₂CH₂CH₂CH₂, Cl), (M-5571, F, CH₃, H, (Me)₂NCOCH₂CH₂CH₂CH₂, F), (M-5572, F, CH₃, H, (Me)₂NCOCH₂CH₂CH₂CH₂, CF₃), (M-5573, F, CH₃, H, (Me)₂NCOCH₂CH₂CH₂CH₂, Br), (M-5574, F, CH₃, H, (Me)₂NCOCH₂CH₂CH₂CH₂, CH₃), (M-5575, F, CH₃, H, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, H), (M-5576, F, CH₃, H, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, Cl), (M-5577, F, CH₃, H, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, F), (M-5578, F, CH₃, H, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, CF₃), (M-5579, F, CH₃, H, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, Br), (M-5580, F, CH₃, H, (Me)₂NCOCH₂CH₂CH₂
CH₂CH₂, CH₃), (M-5581, F, CH₃, H, MeOCH₂, H), (M-5582, F, CH₃, H, MeOCH₂, Cl), (M-5583, F, CH₃, H, MeOCH₂, F), (M-5584, F, CH₃, H, MeOCH₂, CF₃), (M-5585, F, CH₃, H, MeOCH₂, Br), (M-5586, F, CH₃, H, MeOCH₂, CH₃), (M-5587, F, CH₃, H, EtOCH₂, H), (M-5588, F, CH₃, H, EtOCH₂, Cl), (M-5589, F, CH₃, H, EtOCH₂, F), (M-5590, F, CH₃, H, EtOCH₂, CF₃), (M-5591, F, CH₃, H, EtOCH₂, Br), (M-5592, F, CH₃, H, EtOCH₂, CH₃), (M-5593, F, CH₃, H, EtOCH₂CH₂, H), (M-5594, F, CH₃, H, EtOCH₂CH₂, Cl), (M-5595, F, CH₃, H, EtOCH₂CH₂, F), (M-5596, F, CH₃, H, EtOCH₂CH₂, CF₃), (M-5597, F, CH₃, H, EtOCH₂CH₂, Br), (M-5598, F, CH₃, H, EtOCH₂CH₂, CH₃), (M-5599, F, CH₃, H, MeOCH₂CH₂OCH₂CH₂, H), (M-5600, F, CH₃, H, MeOCH₂CH₂OCH₂CH₂, Cl), (M-5601, F, CH₃, H, MeOCH₂CH₂OCH₂CH₂, F), (M-5602, F, CH₃, H, MeOCH₂CH₂OCH₂CH₂, CF₃), (M-5603, F, CH₃, H, MeOCH₂CH₂OCH₂CH₂, Br), (M-5604, F, CH₃, H, MeOCH₂CH₂OCH₂CH₂, CH₃), (M-5605, F, CH₃, H, MeOCH₂CH₂, H), (M-5606, F, CH₃, H, MeOCH₂CH₂, Cl), (M-5607, F, CH₃, H, MeOCH₂CH₂, F), (M-5608, F, CH₃, H, MeOCH₂CH₂, CF₃), (M-5609, F, CH₃, H, MeOCH₂CH₂, Br), (M-5610, F, CH₃, H, MeOCH₂CH₂, CH₃), (M-5611, F, CH₃, H, HOCH₂, H), (M-5612, F, CH₃, H, HOCH₂, Cl), (M-5613, F, CH₃, H, HOCH₂, F), (M-5614, F, CH₃, H, HOCH₂, CF₃), (M-5615, F, CH₃, H, HOCH₂, Br), (M-5616, F, CH₃, H, HOCH₂, CH₃), (M-5617, F, CH₃, H, HOCH₂CH₂, H), (M-5618, F, CH₃, H, HOCH₂CH₂, Cl), (M-5619, F, CH₃, H, HOCH₂CH₂, F), (M-5620, F, CH₃, H, HOCH₂CH₂, CF₃), (M-5621, F, CH₃, H, HOCH₂CH₂, Br), (M-5622, F, CH₃, H, HOCH₂CH₂, CH₃), (M-5623, F, CH₃, H, HOCH₂CH₂CH₂, H), (M-5624, F, CH₃, H, HOCH₂CH₂CH₂, Cl), (M-5625, F, CH₃, H, HOCH₂CH₂CH₂, F), (M-5626, F, CH₃, H, HOCH₂CH₂CH₂, CF₃), (M-5627, F, CH₃, H, HOCH₂CH₂CH₂, Br), (M-5628, F, CH₃, H, HOCH₂CH₂CH₂, CH₃), (M-5629, F, CH₃, H, HOCH₂CH₂CH₂CH₂, H), (M-5630, F, CH₃, H, HOCH₂CH₂CH₂CH₂, Cl), (M-5631, F, CH₃, H, HOCH₂CH₂CH₂CH₂, F), (M-5632, F, CH₃, H, HOCH₂CH₂CH₂CH₂, CF₃), (M-5633, F, CH₃, H, HOCH₂CH₂CH₂CH₂, Br), (M-5634, F, CH₃, H, HOCH₂CH₂CH₂CH₂, CH₃), (M-5635, F, CH₃, H, HOCH₂CH₂CH₂CH₂CH₂, H), (M-5636, F, CH₃, H, HOCH₂CH₂CH₂CH₂CH₂, Cl), (M-5637, F, CH₃, H, HOCH₂CH₂CH₂CH₂CH₂, F), (M-5638, F, CH₃, H, HOCH₂CH₂CH₂CH₂CH₂, CF₃), (M-5639, F, CH₃, H, HOCH₂CH₂CH₂CH₂CH₂, Br), (M-5640, F, CH₃, H, HOCH₂CH₂CH₂CH₂CH₂, CH₃), (M-5641, F, CH₃, H, HOCH₂CH₂OCH₂CH₂, H), (M-5642, F, CH₃, H, HOCH₂CH₂OCH₂CH₂, Cl), (M-5643, F, CH₃, H, HOCH₂CH₂OCH₂CH₂, F), (M-5644, F, CH₃, H, HOCH₂CH₂OCH₂CH₂, CF₃), (M-5645, F, CH₃, H, HOCH₂CH₂OCH₂CH₂, Br), (M-5646, F, CH₃, H, HOCH₂CH₂OCH₂CH₂, CH₃), (M-5647, F, CH₃, H, (Me)₂N, H), (M-5648, F, CH₃, H, (Me)₂N, Cl), (M-5649, F, CH₃, H, (Me)₂N, F), (M-5650, F, CH₃, H, (Me)₂N, CF₃), (M-5651, F, CH₃, H, (Me)₂N, Br), (M-5652, F, CH₃, H, (Me)₂N, CH₃), (M-5653, F, CH₃, H, piperidin-4-yl-methyl, H), (M-5654, F, CH₃, H, piperidin-4-yl-methyl, Cl), (M-5655, F, CH₃, H, piperidin-4-yl-methyl, F), (M-5656, F, CH₃, H, piperidin-4-yl-methyl, CF₃), (M-5657, F, CH₃, H, piperidin-4-yl-methyl, Br), (M-5658, F, CH₃, H, piperidin-4-yl-methyl, CH₃), (M-5659, F, CH₃, H, cyclohexylmethyl, H), (M-5660, F, CH₃, H, cyclohexylmethyl, Cl), (M-5661, F, CH₃, H, cyclohexylmethyl, F), (M-5662, F, CH₃, H, cyclohexylmethyl, CF₃), (M-5663, F, CH₃, H, cyclohexylmethyl, Br), (M-5664, F, CH₃, H, cyclohexylmethyl, CH₃), (M-5665, F, CH₃, F, H, H), (M-5666, F, CH₃, F, H, Cl), (M-5667, F, CH₃, F, H, F), (M-5668, F, CH₃, F, H, CF₃), (M-5669, F, CH₃, F, H, Br), (M-5670, F, CH₃, F, H, CH₃), (M-5671, F, CH₃, F, F, H), (M-5672, F, CH₃, F, F, Cl), (M-5673, F, CH₃, F, F, F), (M-5674, F, CH₃, F, F, CF₃), (M-5675, F, CH₃, F, F, Br), (M-5676, F, CH₃, F, F, CH₃), (M-5677, F, CH₃, F, Cl, H), (M-5678, F, CH₃, F, Cl, Cl), (M-5679, F, CH₃, F, Cl, F), (M-5680, F, CH₃, F, Cl, CF₃), (M-5681, F, CH₃, F, Cl, Br), (M-5682, F, CH₃, F, Cl, CH₃), (M-5683, F, CH₃, F, CH₃, H), (M-5684, F, CH₃, F, CH₃, Cl), (M-5685, F, CH₃, F, CH₃, F), (M-5686, F, CH₃, F, CH₃, CF₃), (M-5687, F, CH₃, F, CH₃, Br), (M-5688, F, CH₃, F, CH₃, CH₃), (M-5689, F, CH₃, F, Et, H), (M-5690, F, CH₃, F, Et, Cl), (M-5691, F, CH₃, F, Et, F), (M-5692, F, CH₃, F, Et, CF₃), (M-5693, F, CH₃, F, Et, Br), (M-5694, F, CH₃, F, Et, CH₃), (M-5695, F, CH₃, F, n-Pr, H), (M-5696, F, CH₃, F, n-Pr, Cl), (M-5697, F, CH₃, F, n-Pr, F), (M-5698, F, CH₃, F, n-Pr, CF₃), (M-5699, F, CH₃, F, n-Pr, Br), (M-5700, F, CH₃, F, n-Pr, CH₃), (M-5701, F, CH₃, F, c-Pr, H), (M-5702, F, CH₃, F, c-Pr, Cl), (M-5703, F, CH₃, F, c-Pr, F), (M-5704, F, CH₃, F, c-Pr, CF₃), (M-5705, F, CH₃, F, c-Pr, Br), (M-5706, F, CH₃, F, c-Pr, CH₃), (M-5707, F, CH₃, F, i-Pr, H), (M-5708, F, CH₃, F, i-Pr, Cl), (M-5709, F, CH₃, F, i-Pr, F), (M-5710, F, CH₃, F, i-Pr, CF₃), (M-5711, F, CH₃, F, i-Pr, Br), (M-5712, F, CH₃, F, i-Pr, CH₃), (M-5713, F, CH₃, F, n-Bu, H), (M-5714, F, CH₃, F, n-Bu, Cl), (M-5715, F, CH₃, F, n-Bu, F), (M-5716, F, CH₃, F, n-Bu, CF₃), (M-5717, F, CH₃, F, n-Bu, Br), (M-5718, F, CH₃, F, n-Bu, CH₃), (M-5719, F, CH₃, F, i-Bu, H), (M-5720, F, CH₃, F, i-Bu, Cl), (M-5721, F, CH₃, F, i-Bu, F), (M-5722, F, CH₃, F, i-Bu, CF₃), (M-5723, F, CH₃, F, i-Bu, Br), (M-5724, F, CH₃, F, i-Bu, CH₃), (M-5725, F, CH₃, F, sec-Bu, H), (M-5726, F, CH₃, F, sec-Bu, Cl), (M-5727, F, CH₃, F, sec-Bu, F), (M-5728, F, CH₃, F, sec-Bu, CF₃), (M-5729, F, CH₃, F, sec-Bu, Br), (M-5730, F, CH₃, F, sec-Bu, CH₃), (M-5731, F, CH₃, F, n-Pen, H), (M-5732, F, CH₃, F, n-Pen, Cl), (M-5733, F, CH₃, F, n-Pen, F), (M-5734, F, CH₃, F, n-Pen, CF₃), (M-5735, F, CH₃, F, n-Pen, Br), (M-5736, F, CH₃, F, n-Pen, CH₃), (M-5737, F, CH₃, F, c-Pen, H), (M-5738, F, CH₃, F, c-Pen, Cl), (M-5739, F, CH₃, F, c-Pen, F), (M-5740, F, CH₃, F, c-Pen, CF₃), (M-5741, F, CH₃, F, c-Pen, Br), (M-5742, F, CH₃, F, c-Pen, CH₃), (M-5743, F, CH₃, F, n-Hex, H), (M-5744, F, CH₃, F, n-Hex, Cl), (M-5745, F, CH₃, F, n-Hex, F), (M-5746, F, CH₃, F, n-Hex, CF₃
), (M-5747, F, CH₃, F, n-Hex, Br), (M-5748, F, CH₃, F, n-Hex, CH₃), (M-5749, F, CH₃, F, c-Hex, H), (M-5750, F, CH₃, F, c-Hex, Cl), (M-5751, F, CH₃, F, c-Hex, F), (M-5752, F, CH₃, F, c-Hex, CF₃), (M-5753, F, CH₃, F, c-Hex, Br), (M-5754, F, CH₃, F, c-Hex, CH₃), (M-5755, F, CH₃, F, OH, H), (M-5756, F, CH₃, F, OH, Cl), (M-5757, F, CH₃, F, OH, F), (M-5758, F, CH₃, F, OH, CF₃), (M-5759, F, CH₃, F, OH, Br), (M-5760, F, CH₃, F, OH, CH₃), (M-5761, F, CH₃, F, EtO, H), (M-5762, F, CH₃, F, EtO, Cl), (M-5763, F, CH₃, F, EtO, F), (M-5764, F, CH₃, F, EtO, CF₃), (M-5765, F, CH₃, F, EtO, Br), (M-5766, F, CH₃, F, EtO, CH₃), (M-5767, F, CH₃, F, n-PrO, H), (M-5768, F, CH₃, F, n-PrO, Cl), (M-5769, F, CH₃, F, n-PrO, F), (M-5770, F, CH₃, F, n-PrO, CF₃), (M-5771, F, CH₃, F, n-PrO, Br), (M-5772, F, CH₃, F, n-PrO, CH₃), (M-5773, F, CH₃, F, PhO, H), (M-5774, F, CH₃, F, PhO, Cl), (M-5775, F, CH₃, F, PhO, F), (M-5776, F, CH₃, F, PhO, CF₃), (M-5777, F, CH₃, F, PhO, Br), (M-5778, F, CH₃, F, PhO, CH₃), (M-5779, F, CH₃, F, BnO, H), (M-5780, F, CH₃, F, BnO, Cl), (M-5781, F, CH₃, F, BnO, F), (M-5782, F, CH₃, F, BnO, CF₃), (M-5783, F, CH₃, F, BnO, Br), (M-5784, F, CH₃, F, BnO, CH₃), (M-5785, F, CH₃, F, PhCH₂CH₂O, H), (M-5786, F, CH₃, F, PhCH₂CH₂O, Cl), (M-5787, F, CH₃, F, PhCH₂CH₂O, F), (M-5788, F, CH₃, F, PhCH₂CH₂O, CF₃), (M-5789, F, CH₃, F, PhCH₂CH₂O, Br), (M-5790, F, CH₃, F, PhCH₂CH₂O, CH₃), (M-5791, F, CH₃, F, CF₃O, H), (M-5792, F, CH₃, F, CF₃O, Cl), (M-5793, F, CH₃, F, CF₃O, F), (M-5794, F, CH₃, F, CF₃O, CF₃), (M-5795, F, CH₃, F, CF₃O, Br), (M-5796, F, CH₃, F, CF₃O, CH₃), (M-5797, F, CH₃, F, Ph, H), (M-5798, F, CH₃, F, Ph, Cl), (M-5799, F, CH₃, F, Ph, F), (M-5800, F, CH₃, F, Ph, CF₃), (M-5801, F, CH₃, F, Ph, Br), (M-5802, F, CH₃, F, Ph, CH₃), (M-5803, F, CH₃, F, 4-F-Ph, H), (M-5804, F, CH₃, F, 4-F-Ph, Cl), (M-5805, F, CH₃, F, 4-F-Ph, F), (M-5806, F, CH₃, F, 4-F-Ph, CF₃), (M-5807, F, CH₃, F, 4-F-Ph, Br), (M-5808, F, CH₃, F, 4-F-Ph, CH₃), (M-5809, F, CH₃, F, 4-CF₃-Ph, H), (M-5810, F, CH₃, F, 4-CF₃-Ph, Cl), (M-5811, F, CH₃, F, 4-CF₃-Ph, F), (M-5812, F, CH₃, F, 4-CF₃-Ph, CF₃), (M-5813, F, CH₃, F, 4-CF₃-Ph, Br), (M-5814, F, CH₃, F, 4-CF₃-Ph, CH₃), (M-5815, F, CH₃, F, 4-(Me)₂N-Ph, H), (M-5816, F, CH₃, F, 4-(Me)₂N-Ph, Cl), (M-5817, F, CH₃, F, 4-(Me)₂N-Ph, F), (M-5818, F, CH₃, F, 4-(Me)₂N-Ph, CF₃), (M-5819, F, CH₃, F, 4-(Me)₂N-Ph, Br), (M-5820, F, CH₃, F, 4-(Me)₂N-Ph, CH₃), (M-5821, F, CH₃, F, 4-OH-Ph, H), (M-5822, F, CH₃, F, 4-OH-Ph, Cl), (M-5823, F, CH₃, F, 4-OH-Ph, F), (M-5824, F, CH₃, F, 4-OH-Ph, CF₃), (M-5825, F, CH₃, F, 4-OH-Ph, Br), (M-5826, F, CH₃, F, 4-OH-Ph, CH₃), (M-5827, F, CH₃, F, 3,4-di-F-Ph, H), (M-5828, F, CH₃, F, 3,4-di-F-Ph, Cl), (M-5829, F, CH₃, F, 3,4-di-F-Ph, F), (M-5830, F, CH₃, F, 3,4-di-F-Ph, CF₃), (M-5831, F, CH₃, F, 3,4-di-F-Ph, Br), (M-5832, F, CH₃, F, 3,4-di-F-Ph, CH₃), (M-5833, F, CH₃, F, 4-COOH-Ph, H), (M-5834, F, CH₃, F, 4-COOH-Ph, Cl), (M-5835, F, CH₃, F, 4-COOH-Ph, F), (M-5836, F, CH₃, F, 4-COOH-Ph, CF₃), (M-5837, F, CH₃, F, 4-COOH-Ph, Br), (M-5838, F, CH₃, F, 4-COOH-Ph, CH₃), (M-5839, F, CH₃, F, Bn, H), (M-5840, F, CH₃, F, Bn, Cl), (M-5841, F, CH₃, F, Bn, F), (M-5842, F, CH₃, F, Bn, CF₃), (M-5843, F, CH₃, F, Bn, Br), (M-5844, F, CH₃, F, Bn, CH₃), (M-5845, F, CH₃, F, 4-F-Bn, H), (M-5846, F, CH₃, F, 4-F-Bn, Cl), (M-5847, F, CH₃, F, 4-F-Bn, F), (M-5848, F, CH₃, F, 4-F-Bn, CF₃), (M-5849, F, CH₃, F, 4-F-Bn, Br), (M-5850, F, CH₃, F, 4-F-Bn, CH₃), (M-5851, F, CH₃, F, 2-Py, H), (M-5852, F, CH₃, F, 2-Py, Cl), (M-5853, F, CH₃, F, 2-Py, F), (M-5854, F, CH₃, F, 2-Py, CF₃), (M-5855, F, CH₃, F, 2-Py, Br), (M-5856, F, CH₃, F, 2-Py, CH₃), (M-5857, F, CH₃, F, 3-Py, H), (M-5858, F, CH₃, F, 3-Py, Cl), (M-5859, F, CH₃, F, 3-Py, F), (M-5860, F, CH₃, F, 3-Py, CF₃), (M-5861, F, CH₃, F, 3-Py, Br), (M-5862, F, CH₃, F, 3-Py, CH₃), (M-5863, F, CH₃, F, 4-Py, H), (M-5864, F, CH₃, F, 4-Py, Cl), (M-5865, F, CH₃, F, 4-Py, F), (M-5866, F, CH₃, F, 4-Py, CF₃), (M-5867, F, CH₃, F, 4-Py, Br), (M-5868, F, CH₃, F, 4-Py, CH₃), (M-5869, F, CH₃, F, 2-Th, H), (M-5870, F, CH₃, F, 2-Th, Cl), (M-5871, F, CH₃, F, 2-Th, F), (M-5872, F, CH₃, F, 2-Th, CF₃), (M-5873, F, CH₃, F, 2-Th, Br), (M-5874, F, CH₃, F, 2-Th, CH₃), (M-5875, F, CH₃, F, 3-Th, H), (M-5876, F, CH₃, F, 3-Th, Cl), (M-5877, F, CH₃, F, 3-Th, F), (M-5878, F, CH₃, F, 3-Th, CF₃), (M-5879, F, CH₃, F, 3-Th, Br), (M-5880, F, CH₃, F, 3-Th, CH₃), (M-5881, F, CH₃, F, pyrazol-2-yl, H), (M-5882, F, CH₃, F, pyrazol-2-yl, Cl), (M-5883, F, CH₃, F, pyrazol-2-yl, F), (M-5884, F, CH₃, F, pyrazol-2-yl, CF₃), (M-5885, F, CH₃, F, pyrazol-2-yl, Br), (M-5886, F, CH₃, F, pyrazol-2-yl, CH₃), (M-5887, F, CH₃, F, pyrazol-3-yl, H), (M-5888, F, CH₃, F, pyrazol-3-yl, Cl), (M-5889, F, CH₃, F, pyrazol-3-yl, F), (M-5890, F, CH₃, F, pyrazol-3-yl, CF₃), (M-5891, F, CH₃, F, pyrazol-3-yl, Br), (M-5892, F, CH₃, F, pyrazol-3-yl, CH₃), (M-5893, F, CH₃, F, pyrimidin-2-yl, H), (M-5894, F, CH₃, F, pyrimidin-2-yl, Cl), (M-5895, F, CH₃, F, pyrimidin-2-yl, F), (M-5896, F, CH₃, F, pyrimidin-2-yl, CF₃), (M-5897, F, CH₃, F, pyrimidin-2-yl, Br), (M-5898, F, CH₃, F, pyrimidin-2-yl, CH₃), (M-5899, F, CH₃, F, pyrimidin-4-yl, H), (M-5900, F, CH₃, F, pyrimidin-4-yl, Cl), (M-5901, F, CH₃, F, pyrimidin-4-yl, F), (M-5902, F, CH₃, F, pyrimidin-4-yl, CF₃), (M-5903, F, CH₃, F, pyrimidin-4-yl, Br), (M-5904, F, CH₃, F, pyrimidin-4-yl, CH₃), (M-5905, F, CH₃, F, pyrimidin-5-yl, H), (M-5906, F, CH₃, F, pyrimidin-5-yl, Cl), (M-5907, F, CH₃, F, pyrimidin-5-yl, F), (M-5908, F, CH₃, F, pyrimidin-5-yl, CF₃), (M-5909, F, CH₃, F, pyrimidin-5-yl, Br), (M-5910, F, CH₃, F, pyrimidin-5-yl, CH₃), (M-5911, F, CH₃, F, HOOCCH₂CH₂CH₂, H), (M-5912, F, CH₃, F, HOOCCH₂CH₂CH₂, Cl), (M-5913, F, CH₃, F, HOOCCH₂CH₂CH₂, F), (M-5914, F, CH₃, F, HOOCCH₂CH₂CH₂, CF₃), (M-5915, F, CH₃, F, HOOCCH₂CH₂CH₂, Br), (M-5916, F, CH₃, F, HOOCCH₂CH₂CH₂, CH₃), (M-5917, F, CH₃, F, HOOCCH₂CH₂CH₂CH₂, H), (M-5918, F, CH₃, F, HOOCCH₂CH₂CH₂CH₂, Cl), (M-5919, F, CH₃, F, HOOCCH₂CH₂CH₂CH₂, F), (M-5920, F, CH₃, F, HOOCCH₂CH₂CH₂CH₂, CF₃), (M-5921, F, CH₃, F, HOOCCH₂CH₂CH₂CH₂, Br), (M-5922, F, CH₃, F, HOOCCH₂CH₂CH₂CH₂, CH₃), (M-5923, F, CH₃, F, (Me)₂NCOCH₂CH₂CH₂CH₂, H), (M-5924, F, CH₃, F, (Me)₂NCOCH₂CH₂CH₂CH₂, Cl), (M-5925, F, CH₃, F, (Me)₂NCOCH₂CH₂CH₂CH₂, F), (M-5926, F, CH₃, F, (Me)₂NCOCH₂CH₂CH₂CH₂, CF₃), (M-5927, F, CH₃, F, (Me)₂NCOCH₂CH₂CH₂CH₂, Br), (M-5928, F, CH₃, F, (Me)₂NCOCH₂CH₂CH₂CH₂, CH₃), (M-5929, F, CH₃, F, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, H), (M-593
0, F, CH₃, F, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, Cl), (M-5931, F, CH₃, F, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, F), (M-5932, F, CH₃, F, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, CF₃), (M-5933, F, CH₃, F, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, Br), (M-5934, F, CH₃, F, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, CH₃), (M-5935, F, CH₃, F, MeOCH₂, H), (M-5936, F, CH₃, F, MeOCH₂, Cl), (M-5937, F, CH₃, F, MeOCH₂, F), (M-5938, F, CH₃, F, MeOCH₂, CF₃), (M-5939, F, CH₃, F, MeOCH₂, Br), (M-5940, F, CH₃, F, MeOCH₂, CH₃), (M-5941, F, CH₃, F, EtOCH₂, H), (M-5942, F, CH₃, F, EtOCH₂, Cl), (M-5943, F, CH₃, F, EtOCH₂, F), (M-5944, F, CH₃, F, EtOCH₂, CF₃), (M-5945, F, CH₃, F, EtOCH₂, Br), (M-5946, F, CH₃, F, EtOCH₂, CH₃), (M-5947, F, CH₃, F, EtOCH₂CH₂, H), (M-5948, F, CH₃, F, EtOCH₂CH₂, Cl), (M-5949, F, CH₃, F, EtOCH₂CH₂, F), (M-5950, F, CH₃, F, EtOCH₂CH₂, CF₃), (M-5951, F, CH₃, F, EtOCH₂CH₂, Br), (M-5952, F, CH₃, F, EtOCH₂CH₂, CH₃), (M-5953, F, CH₃, F, MeOCH₂CH₂OCH₂CH₂, H), (M-5954, F, CH₃, F, MeOCH₂CH₂OCH₂CH₂, Cl), (M-5955, F, CH₃, F, MeOCH₂CH₂OCH₂CH₂, F), (M-5956, F, CH₃, F, MeOCH₂CH₂OCH₂CH₂, CF₃), (M-5957, F, CH₃, F, MeOCH₂CH₂OCH₂CH₂, Br), (M-5958, F, CH₃, F, MeOCH₂CH₂OCH₂CH₂, CH₃), (M-5959, F, CH₃, F, MeOCH₂CH₂, H), (M-5960, F, CH₃, F, MeOCH₂CH₂, Cl), (M-5961, F, CH₃, F, MeOCH₂CH₂, F), (M-5962, F, CH₃, F, MeOCH₂CH₂, CF₃), (M-5963, F, CH₃, F, MeOCH₂CH₂, Br), (M-5964, F, CH₃, F, MeOCH₂CH₂, CH₃), (M-5965, F, CH₃, F, HOCH₂, H), (M-5966, F, CH₃, F, HOCH₂, Cl), (M-5967, F, CH₃, F, HOCH₂, F), (M-5968, F, CH₃, F, HOCH₂, CF₃), (M-5969, F, CH₃, F, HOCH₂, Br), (M-5970, F, CH₃, F, HOCH₂, CH₃), (M-5971, F, CH₃, F, HOCH₂CH₂, H), (M-5972, F, CH₃, F, HOCH₂CH₂, Cl), (M-5973, F, CH₃, F, HOCH₂CH₂, F), (M-5974, F, CH₃, F, HOCH₂CH₂, CF₃), (M-5975, F, CH₃, F, HOCH₂CH₂, Br), (M-5976, F, CH₃, F, HOCH₂CH₂, CH₃), (M-5977, F, CH₃, F, HOCH₂CH₂CH₂, H), (M-5978, F, CH₃, F, HOCH₂CH₂CH₂, Cl), (M-5979, F, CH₃, F, HOCH₂CH₂CH₂, F), (M-5980, F, CH₃, F, HOCH₂CH₂CH₂, CF₃), (M-5981, F, CH₃, F, HOCH₂CH₂CH₂, Br), (M-5982, F, CH₃, F, HOCH₂CH₂CH₂, CH₃), (M-5983, F, CH₃, F, HOCH₂CH₂CH₂CH₂, H), (M-5984, F, CH₃, F, HOCH₂CH₂CH₂CH₂, Cl), (M-5985, F, CH₃, F, HOCH₂CH₂CH₂CH₂, F), (M-5986, F, CH₃, F, HOCH₂CH₂CH₂CH₂, CF₃), (M-5987, F, CH₃, F, HOCH₂CH₂CH₂CH₂, Br), (M-5988, F, CH₃, F, HOCH₂CH₂CH₂CH₂, CH₃), (M-5989, F, CH₃, F, HOCH₂CH₂CH₂CH₂CH₂, H), (M-5990, F, CH₃, F, HOCH₂CH₂CH₂CH₂CH₂, Cl), (M-5991, F, CH₃, F, HOCH₂CH₂CH₂CH₂CH₂, F), (M-5992, F, CH₃, F, HOCH₂CH₂CH₂CH₂CH₂, CF₃), (M-5993, F, CH₃, F, HOCH₂CH₂CH₂CH₂CH₂, Br), (M-5994, F, CH₃, F, HOCH₂CH₂CH₂CH₂CH₂, CH₃), (M-5995, F, CH₃, F, HOCH₂CH₂OCH₂CH₂, H), (M-5996, F, CH₃, F, HOCH₂CH₂OCH₂CH₂, Cl), (M-5997, F, CH₃, F, HOCH₂CH₂OCH₂CH₂, F), (M-5998, F, CH₃, F, HOCH₂CH₂OCH₂CH₂, CF₃), (M-5999, F, CH₃, F, HOCH₂CH₂OCH₂CH₂, Br), (M-6000, F, CH₃, F, HOCH₂CH₂OCH₂CH₂, CH₃), (M-6001, F, CH₃, F, (Me)₂N, H), (M-6002, F, CH₃, F, (Me)₂N, Cl), (M-6003, F, CH₃, F, (Me)₂N, F), (M-6004, F, CH₃, F, (Me)₂N, CF₃), (M-6005, F, CH₃, F, (Me)₂N, Br), (M-6006, F, CH₃, F, (Me)₂N, CH₃), (M-6007, F, CH₃, F, piperidin-4-yl-methyl, H), (M-6008, F, CH₃, F, piperidin-4-yl-methyl, Cl), (M-6009, F, CH₃, F, piperidin-4-yl-methyl, F), (M-6010, F, CH₃, F, piperidin-4-yl-methyl, CF₃), (M-6011, F, CH₃, F, piperidin-4-yl-methyl, Br), (M-6012, F, CH₃, F, piperidin-4-yl-methyl, CH₃), (M-6013, F, CH₃, F, cyclohexylmethyl, H), (M-6014, F, CH₃, F, cyclohexylmethyl, Cl), (M-6015, F, CH₃, F, cyclohexylmethyl, F), (M-6016, F, CH₃, F, cyclohexylmethyl, CF₃), (M-6017, F, CH₃, F, cyclohexylmethyl, Br), (M-6018, F, CH₃, F, cyclohexylmethyl, CH₃), (M-6019, F, CH₃, Cl, H, H), (M-6020, F, CH₃, Cl, H, Cl), (M-6021, F, CH₃, Cl, H, F), (M-6022, F, CH₃, Cl, H, CF₃), (M-6023, F, CH₃, Cl, H, Br), (M-6024, F, CH₃, Cl, H, CH₃), (M-6025, F, CH₃, Cl, F, H), (M-6026, F, CH₃, Cl, F, Cl), (M-6027, F, CH₃, Cl, F, F), (M-6028, F, CH₃, Cl, F, CF₃), (M-6029, F, CH₃, Cl, F, Br), (M-6030, F, CH₃, Cl, F, CH₃), (M-6031, F, CH₃, Cl, Cl, H), (M-6032, F, CH₃, Cl, Cl, Cl), (M-6033, F, CH₃, Cl, Cl, F), (M-6034, F, CH₃, Cl, Cl, CF₃), (M-6035, F, CH₃, Cl, Cl, Br), (M-6036, F, CH₃, Cl, Cl, CH₃), (M-6037, F, CH₃, Cl, CH₃, H), (M-6038, F, CH₃, Cl, CH₃, Cl), (M-6039, F, CH₃, Cl, CH₃, F), (M-6040, F, CH₃, Cl, CH₃, CF₃), (M-6041, F, CH₃, Cl, CH₃, Br), (M-6042, F, CH₃, Cl, CH₃, CH₃), (M-6043, F, CH₃, Cl, Et, H), (M-6044, F, CH₃, Cl, Et, Cl), (M-6045, F, CH₃, Cl, Et, F), (M-6046, F, CH₃, Cl, Et, CF₃), (M-6047, F, CH₃, Cl, Et, Br), (M-6048, F, CH₃, Cl, Et, CH₃), (M-6049, F, CH₃, Cl, n-Pr, H), (M-6050, F, CH₃, Cl, n-Pr, Cl), (M-6051, F, CH₃, Cl, n-Pr, F), (M-6052, F, CH₃, Cl, n-Pr, CF₃), (M-6053, F, CH₃, Cl, n-Pr, Br), (M-6054, F, CH₃, Cl, n-Pr, CH₃), (M-6055, F, CH₃, Cl, c-Pr, H), (M-6056, F, CH₃, Cl, c-Pr, Cl), (M-6057, F, CH₃, Cl, c-Pr, F), (M-6058, F, CH₃, Cl, c-Pr, CF₃), (M-6059, F, CH₃, Cl, c-Pr, Br), (M-6060, F, CH₃, Cl, c-Pr, CH₃), (M-6061, F, CH₃, Cl, i-Pr, H), (M-6062, F, CH₃, Cl, i-Pr, Cl), (M-6063, F, CH₃, Cl, i-Pr, F), (M-6064, F, CH₃, Cl, i-Pr, CF₃), (M-6065, F, CH₃, Cl, i-Pr, Br), (M-6066, F, CH₃, Cl, i-Pr, CH₃), (M-6067, F, CH₃, Cl, n-Bu, H), (M-6068, F, CH₃, Cl, n-Bu, Cl), (M-6069, F, CH₃, Cl, n-Bu, F), (M-6070, F, CH₃, Cl, n-Bu, CF₃), (M-6071, F, CH₃, Cl, n-Bu, Br), (M-6072, F, CH₃, Cl, n-Bu, CH₃), (M-6073, F, CH₃, Cl, i-Bu, H), (M-6074, F, CH₃, Cl, i-Bu, Cl), (M-6075, F, CH₃, Cl, i-Bu, F), (M-6076, F, CH₃, Cl, i-Bu, CF₃), (M-6077, F, CH₃, Cl, i-Bu, Br), (M-6078, F, CH₃, Cl, i-Bu, CH₃), (M-6079, F, CH₃, Cl, sec-Bu, H), (M-6080, F, CH₃, Cl, sec-Bu, Cl), (M-6081, F, CH₃, Cl, sec-Bu, F), (M-6082, F, CH₃, Cl, sec-Bu, CF₃), (M-6083, F, CH₃, Cl, sec-Bu, Br), (M-6084, F, CH₃, Cl, sec-Bu, CH₃), (M-6085, F, CH₃, Cl, n-Pen, H), (M-6086, F, CH₃
, Cl, n-Pen, Cl), (M-6087, F, CH₃, Cl, n-Pen, F), (M-6088, F, CH₃, Cl, n-Pen, CF₃), (M-6089, F, CH₃, Cl, n-Pen, Br), (M-6090, F, CH₃, Cl, n-Pen, CH₃), (M-6091, F, CH₃, Cl, c-Pen, H), (M-6092, F, CH₃, Cl, c-Pen, Cl), (M-6093, F, CH₃, Cl, c-Pen, F), (M-6094, F, CH₃, Cl, c-Pen, CF₃), (M-6095, F, CH₃, Cl, c-Pen, Br), (M-6096, F, CH₃, Cl, c-Pen, CH₃), (M-6097, F, CH₃, Cl, n-Hex, H), (M-6098, F, CH₃, Cl, n-Hex, Cl), (M-6099, F, CH₃, Cl, n-Hex, F), (M-6100, F, CH₃, Cl, n-Hex, CF₃), (M-6101, F, CH₃, Cl, n-Hex, Br), (M-6102, F, CH₃, Cl, n-Hex, CH₃), (M-6103, F, CH₃, Cl, c-Hex, H), (M-6104, F, CH₃, Cl, c-Hex, Cl), (M-6105, F, CH₃, Cl, c-Hex, F), (M-6106, F, CH₃, Cl, c-Hex, CF₃), (M-6107, F, CH₃, Cl, c-Hex, Br), (M-6108, F, CH₃, Cl, c-Hex, CH₃), (M-6109, F, CH₃, Cl, OH, H), (M-6110, F, CH₃, Cl, OH, Cl), (M-6111, F, CH₃, Cl, OH, F), (M-6112, F, CH₃, Cl, OH, CF₃), (M-6113, F, CH₃, Cl, OH, Br), (M-6114, F, CH₃, Cl, OH, CH₃), (M-6115, F, CH₃, Cl, EtO, H), (M-6116, F, CH₃, Cl, EtO, Cl), (M-6117, F, CH₃, Cl, EtO, F), (M-6118, F, CH₃, Cl, EtO, CF₃), (M-6119, F, CH₃, Cl, EtO, Br), (M-6120, F, CH₃, Cl, EtO, CH₃), (M-6121, F, CH₃, Cl, n-PrO, H), (M-6122, F, CH₃, Cl, n-PrO, Cl), (M-6123, F, CH₃, Cl, n-PrO, F), (M-6124, F, CH₃, Cl, n-PrO, CF₃), (M-6125, F, CH₃, Cl, n-PrO, Br), (M-6126, F, CH₃, Cl, n-PrO, CH₃), (M-6127, F, CH₃, Cl, PhO, H), (M-6128, F, CH₃, Cl, PhO, Cl), (M-6129, F, CH₃, Cl, PhO, F), (M-6130, F, CH₃, Cl, PhO, CF₃), (M-6131, F, CH₃, Cl, PhO, Br), (M-6132, F, CH₃, Cl, PhO, CH₃), (M-6133, F, CH₃, Cl, BnO, H), (M-6134, F, CH₃, Cl, BnO, Cl), (M-6135, F, CH₃, Cl, BnO, F), (M-6136, F, CH₃, Cl, BnO, CF₃), (M-6137, F, CH₃, Cl, BnO, Br), (M-6138, F, CH₃, Cl, BnO, CH₃), (M-6139, F, CH₃, Cl, PhCH₂CH₂O, H), (M-6140, F, CH₃, Cl, PhCH₂CH₂O, Cl), (M-6141, F, CH₃, Cl, PhCH₂CH₂O, F), (M-6142, F, CH₃, Cl, PhCH₂CH₂O, CF₃), (M-6143, F, CH₃, Cl, PhCH₂CH₂O, Br), (M-6144, F, CH₃, Cl, PhCH₂CH₂O, CH₃), (M-6145, F, CH₃, Cl, CF₃O, H), (M-6146, F, CH₃, Cl, CF₃O, Cl), (M-6147, F, CH₃, Cl, CF₃O, F), (M-6148, F, CH₃, Cl, CF₃O, CF₃), (M-6149, F, CH₃, Cl, CF₃O, Br), (M-6150, F, CH₃, Cl, CF₃O, CH₃), (M-6151, F, CH₃, Cl, Ph, H), (M-6152, F, CH₃, Cl, Ph, Cl), (M-6153, F, CH₃, Cl, Ph, F), (M-6154, F, CH₃, Cl, Ph, CF₃), (M-6155, F, CH₃, Cl, Ph, Br), (M-6156, F, CH₃, Cl, Ph, CH₃), (M-6157, F, CH₃, Cl, 4-F-Ph, H), (M-6158, F, CH₃, Cl, 4-F-Ph, Cl), (M-6159, F, CH₃, Cl, 4-F-Ph, F), (M-6160, F, CH₃, Cl, 4-F-Ph, CF₃), (M-6161, F, CH₃, Cl, 4-F-Ph, Br), (M-6162, F, CH₃, Cl, 4-F-Ph, CH₃), (M-6163, F, CH₃, Cl, 4-CF₃-Ph, H), (M-6164, F, CH₃, Cl, 4-CF₃-Ph, Cl), (M-6165, F, CH₃, Cl, 4-CF₃-Ph, F), (M-6166, F, CH₃, Cl, 4-CF₃-Ph, CF₃), (M-6167, F, CH₃, Cl, 4-CF₃-Ph, Br), (M-6168, F, CH₃, Cl, 4-CF₃-Ph, CH₃), (M-6169, F, CH₃, Cl, 4-(Me)₂N-Ph, H), (M-6170, F, CH₃, Cl, 4-(Me)₂N-Ph, Cl), (M-6171, F, CH₃, Cl, 4-(Me)₂N-Ph, F), (M-6172, F, CH₃, Cl, 4-(Me)₂N-Ph, CF₃), (M-6173, F, CH₃, Cl, 4-(Me)₂N-Ph, Br), (M-6174, F, CH₃, Cl, 4-(Me)₂N-Ph, CH₃), (M-6175, F, CH₃, Cl, 4-OH-Ph, H), (M-6176, F, CH₃, Cl, 4-OH-Ph, Cl), (M-6177, F, CH₃, Cl, 4-OH-Ph, F), (M-6178, F, CH₃, Cl, 4-OH-Ph, CF₃), (M-6179, F, CH₃, Cl, 4-OH-Ph, Br), (M-6180, F, CH₃, Cl, 4-OH-Ph, CH₃), (M-6181, F, CH₃, Cl, 3,4-di-F-Ph, H), (M-6182, F, CH₃, Cl, 3,4-di-F-Ph, Cl), (M-6183, F, CH₃, Cl, 3,4-di-F-Ph, F), (M-6184, F, CH₃, Cl, 3,4-di-F-Ph, CF₃), (M-6185, F, CH₃, Cl, 3,4-di-F-Ph, Br), (M-6186, F, CH₃, Cl, 3,4-di-F-Ph, CH₃), (M-6187, F, CH₃, Cl, 4-COOH-Ph, H), (M-6188, F, CH₃, Cl, 4-COOH-Ph, Cl), (M-6189, F, CH₃, Cl, 4-COOH-Ph, F), (M-6190, F, CH₃, Cl, 4-COOH-Ph, CF₃), (M-6191, F, CH₃, Cl, 4-COOH-Ph, Br), (M-6192, F, CH₃, Cl, 4-COOH-Ph, CH₃), (M-6193, F, CH₃, Cl, Bn, H), (M-6194, F, CH₃, Cl, Bn, Cl), (M-6195, F, CH₃, Cl, Bn, F), (M-6196, F, CH₃, Cl, Bn, CF₃), (M-6197, F, CH₃, Cl, Bn, Br), (M-6198, F, CH₃, Cl, Bn, CH₃), (M-6199, F, CH₃, Cl, 4-F-Bn, H), (M-6200, F, CH₃, Cl, 4-F-Bn, Cl), (M-6201, F, CH₃, Cl, 4-F-Bn, F), (M-6202, F, CH₃, Cl, 4-F-Bn, CF₃), (M-6203, F, CH₃, Cl, 4-F-Bn, Br), (M-6204, F, CH₃, Cl, 4-F-Bn, CH₃), (M-6205, F, CH₃, Cl, 2-Py, H), (M-6206, F, CH₃, Cl, 2-Py, Cl), (M-6207, F, CH₃, Cl, 2-Py, F), (M-6208, F, CH₃, Cl, 2-Py, CF₃), (M-6209, F, CH₃, Cl, 2-Py, Br), (M-6210, F, CH₃, Cl, 2-Py, CH₃), (M-6211, F, CH₃, Cl, 3-Py, H), (M-6212, F, CH₃, Cl, 3-Py, Cl), (M-6213, F, CH₃, Cl, 3-Py, F), (M-6214, F, CH₃, Cl, 3-Py, CF₃), (M-6215, F, CH₃, Cl, 3-Py, Br), (M-6216, F, CH₃, Cl, 3-Py, CH₃), (M-6217, F, CH₃, Cl, 4-Py, H), (M-6218, F, CH₃, Cl, 4-Py, Cl), (M-6219, F, CH₃, Cl, 4-Py, F), (M-6220, F, CH₃, Cl, 4-Py, CF₃), (M-6221, F, CH₃, Cl, 4-Py, Br), (M-6222, F, CH₃, Cl, 4-Py, CH₃), (M-6223, F, CH₃, Cl, 2-Th, H), (M-6224, F, CH₃, Cl, 2-Th, Cl), (M-6225, F, CH₃, Cl, 2-Th, F), (M-6226, F, CH₃, Cl, 2-Th, CF₃), (M-6227, F, CH₃, Cl, 2-Th, Br), (M-6228, F, CH₃, Cl, 2-Th, CH₃), (M-6229, F, CH₃, Cl, 3-Th, H), (M-6230, F, CH₃, Cl, 3-Th, Cl), (M-6231, F, CH₃, Cl, 3-Th, F), (M-6232, F, CH₃, Cl, 3-Th, CF₃), (M-6233, F, CH₃, Cl, 3-Th, Br), (M-6234, F, CH₃, Cl, 3-Th, CH₃), (M-6235, F, CH₃, Cl, pyrazol-2-yl, H), (M-6236, F, CH₃, Cl, pyrazol-2-yl, Cl), (M-6237, F, CH₃, Cl, pyrazol-2-yl, F), (M-6238, F, CH₃, Cl, pyrazol-2-yl, CF₃), (M-6239, F, CH₃, Cl, pyrazol-2-yl, Br), (M-6240, F, CH₃, Cl, pyrazol-2-yl, CH₃), (M-6241, F, CH₃, Cl, pyrazol-3-yl, H), (M-6242, F, CH₃, Cl, pyrazol-3-yl, Cl), (M-6243, F, CH₃, Cl, pyrazol-3-yl, F), (M-6244, F, CH₃, Cl, pyrazol-3-yl, CF₃), (M-6245, F, CH₃, Cl, pyrazol-3-yl, Br), (M-6246, F, CH₃, Cl, pyrazol-3-yl, CH₃), (M-6247, F, CH₃, Cl, pyrimidin-2-yl, H), (M-6248, F, CH₃, Cl, pyrimidin-2-yl, Cl), (M-6249, F, CH₃, Cl, pyrimidin-2-yl, F), (M-6250, F, CH₃, Cl, pyrimidin-2-yl, CF₃), (M-6251, F, CH₃, Cl, pyrimidin-2-yl, Br), (M-6252, F, CH₃, Cl, pyrimidin-2-yl, CH₃), (M-6253, F, CH₃, Cl, pyrimidin-4-yl, H), (M-6254, F, CH₃, Cl, pyrimidin-4-yl, Cl), (M-6255, F, CH₃, Cl, pyrimidin-4-yl, F), (M-6256, F, CH₃, Cl, pyrimidin-4-yl, CF₃), (M-6257, F, CH₃, Cl, pyrimidin-4-yl, Br), (M-6258, F, CH₃, Cl, pyrimidin-4-yl, CH₃), (M-6259, F, CH₃, Cl, pyrimidin-5-yl, H), (M-6260, F, CH₃, Cl, pyrimidin-5-yl, Cl), (M-6261, F, CH₃, Cl, pyrimidin-5-yl, F), (M-6262, F, CH₃, Cl, pyrimidin-5-yl, CF₃), (M-6263, F, CH₃, Cl, pyrimidin-5-yl, Br), (M-6264, F, CH₃, Cl, pyrimidin-5-yl, CH₃), (M-6265, F, CH₃, Cl, HOOCCH₂CH₂CH₂, H), (M-6266, F, CH₃, Cl, HOOCCH₂CH₂CH₂, Cl), (M-6267, F, CH₃, Cl, HOOCCH₂CH₂CH₂, F), (M-6268, F, CH₃, Cl, HOOCCH₂CH₂CH₂, CF₃), (M-6269, F, CH₃, Cl, HOOCCH₂CH₂CH₂, Br), (M-6270, F, CH₃, Cl, HOOCCH₂CH₂CH₂, CH₃), (M-6271, F, CH₃, Cl, HOOCCH₂CH₂CH₂CH₂, H), (M-6272, F, CH₃, Cl, HOOCCH₂CH₂CH₂CH₂, Cl), (M-6273, F, CH₃, Cl, HOOCCH₂CH₂CH₂CH₂, F), (M-6274, F, CH₃, Cl, HOOCCH₂CH₂CH₂CH₂, CF₃), (M-6275, F, CH₃, Cl, HOOCCH₂CH₂CH₂CH₂, Br), (M-6276, F, CH₃, Cl, HOOCCH₂CH₂CH₂
CH₂, CH₃), (M-6277, F, CH₃, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂, H), (M-6278, F, CH₃, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂, Cl), (M-6279, F, CH₃, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂, F), (M-6280, F, CH₃, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂, CF₃), (M-6281, F, CH₃, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂, Br), (M-6282, F, CH₃, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂, CH₃), (M-6283, F, CH₃, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, H), (M-6284, F, CH₃, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, Cl), (M-6285, F, CH₃, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, F), (M-6286, F, CH₃, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, CF₃), (M-6287, F, CH₃, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, Br), (M-6288, F, CH₃, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, CH₃), (M-6289, F, CH₃, Cl, MeOCH₂, H), (M-6290, F, CH₃, Cl, MeOCH₂, Cl), (M-6291, F, CH₃, Cl, MeOCH₂, F), (M-6292, F, CH₃, Cl, MeOCH₂, CF₃), (M-6293, F, CH₃, Cl, MeOCH₂, Br), (M-6294, F, CH₃, Cl, MeOCH₂, CH₃), (M-6295, F, CH₃, Cl, EtOCH₂, H), (M-6296, F, CH₃, Cl, EtOCH₂, Cl), (M-6297, F, CH₃, Cl, EtOCH₂, F), (M-6298, F, CH₃, Cl, EtOCH₂, CF₃), (M-6299, F, CH₃, Cl, EtOCH₂, Br), (M-6300, F, CH₃, Cl, EtOCH₂, CH₃), (M-6301, F, CH₃, Cl, EtOCH₂CH₂, H), (M-6302, F, CH₃, Cl, EtOCH₂CH₂, Cl), (M-6303, F, CH₃, Cl, EtOCH₂CH₂, F), (M-6304, F, CH₃, Cl, EtOCH₂CH₂, CF₃), (M-6305, F, CH₃, Cl, EtOCH₂CH₂, Br), (M-6306, F, CH₃, Cl, EtOCH₂CH₂, CH₃), (M-6307, F, CH₃, Cl, MeOCH₂CH₂OCH₂CH₂, H), (M-6308, F, CH₃, Cl, MeOCH₂CH₂OCH₂CH₂, Cl), (M-6309, F, CH₃, Cl, MeOCH₂CH₂OCH₂CH₂, F), (M-6310, F, CH₃, Cl, MeOCH₂CH₂OCH₂CH₂, CF₃), (M-6311, F, CH₃, Cl, MeOCH₂CH₂OCH₂CH₂, Br), (M-6312, F, CH₃, Cl, MeOCH₂CH₂OCH₂CH₂, CH₃), (M-6313, F, CH₃, Cl, MeOCH₂CH₂, H), (M-6314, F, CH₃, Cl, MeOCH₂CH₂, Cl), (M-6315, F, CH₃, Cl, MeOCH₂CH₂, F), (M-6316, F, CH₃, Cl, MeOCH₂CH₂, CF₃), (M-6317, F, CH₃, Cl, MeOCH₂CH₂, Br), (M-6318, F, CH₃, Cl, MeOCH₂CH₂, CH₃), (M-6319, F, CH₃, Cl, HOCH₂, H), (M-6320, F, CH₃, Cl, HOCH₂, Cl), (M-6321, F, CH₃, Cl, HOCH₂, F), (M-6322, F, CH₃, Cl, HOCH₂, CF₃), (M-6323, F, CH₃, Cl, HOCH₂, Br), (M-6324, F, CH₃, Cl, HOCH₂, CH₃), (M-6325, F, CH₃, Cl, HOCH₂CH₂, H), (M-6326, F, CH₃, Cl, HOCH₂CH₂, Cl), (M-6327, F, CH₃, Cl, HOCH₂CH₂, F), (M-6328, F, CH₃, Cl, HOCH₂CH₂, CF₃), (M-6329, F, CH₃, Cl, HOCH₂CH₂, Br), (M-6330, F, CH₃, Cl, HOCH₂CH₂, CH₃), (M-6331, F, CH₃, Cl, HOCH₂CH₂CH₂, H), (M-6332, F, CH₃, Cl, HOCH₂CH₂CH₂, Cl), (M-6333, F, CH₃, Cl, HOCH₂CH₂CH₂, F), (M-6334, F, CH₃, Cl, HOCH₂CH₂CH₂, CF₃), (M-6335, F, CH₃, Cl, HOCH₂CH₂CH₂, Br), (M-6336, F, CH₃, Cl, HOCH₂CH₂CH₂, CH₃), (M-6337, F, CH₃, Cl, HOCH₂CH₂CH₂CH₂, H), (M-6338, F, CH₃, Cl, HOCH₂CH₂CH₂CH₂, Cl), (M-6339, F, CH₃, Cl, HOCH₂CH₂CH₂CH₂, F), (M-6340, F, CH₃, Cl, HOCH₂CH₂CH₂CH₂, CF₃), (M-6341, F, CH₃, Cl, HOCH₂CH₂CH₂CH₂, Br), (M-6342, F, CH₃, Cl, HOCH₂CH₂CH₂CH₂, CH₃), (M-6343, F, CH₃, Cl, HOCH₂CH₂CH₂CH₂CH₂, H), (M-6344, F, CH₃, Cl, HOCH₂CH₂CH₂CH₂CH₂, Cl), (M-6345, F, CH₃, Cl, HOCH₂CH₂CH₂CH₂CH₂, F), (M-6346, F, CH₃, Cl, HOCH₂CH₂CH₂CH₂CH₂, CF₃), (M-6347, F, CH₃, Cl, HOCH₂CH₂CH₂CH₂CH₂, Br), (M-6348, F, CH₃, Cl, HOCH₂CH₂CH₂CH₂CH₂, CH₃), (M-6349, F, CH₃, Cl, HOCH₂CH₂OCH₂CH₂, H), (M-6350, F, CH₃, Cl, HOCH₂CH₂OCH₂CH₂, Cl), (M-6351, F, CH₃, Cl, HOCH₂CH₂OCH₂CH₂, F), (M-6352, F, CH₃, Cl, HOCH₂CH₂OCH₂CH₂, CF₃), (M-6353, F, CH₃, Cl, HOCH₂CH₂OCH₂CH₂, Br), (M-6354, F, CH₃, Cl, HOCH₂CH₂OCH₂CH₂, CH₃), (M-6355, F, CH₃, Cl, (Me)₂N, H), (M-6356, F, CH₃, Cl, (Me)₂N, Cl), (M-6357, F, CH₃, Cl, (Me)₂N, F), (M-6358, F, CH₃, Cl, (Me)₂N, CF₃), (M-6359, F, CH₃, Cl, (Me)₂N, Br), (M-6360, F, CH₃, Cl, (Me)₂N, CH₃), (M-6361, F, CH₃, Cl, piperidin-4-yl-methyl, H), (M-6362, F, CH₃, Cl, piperidin-4-yl-methyl, Cl), (M-6363, F, CH₃, Cl, piperidin-4-yl-methyl, F), (M-6364, F, CH₃, Cl, piperidin-4-yl-methyl, CF₃), (M-6365, F, CH₃, Cl, piperidin-4-yl-methyl, Br), (M-6366, F, CH₃, Cl, piperidin-4-yl-methyl, CH₃), (M-6367, F, CH₃, Cl, cyclohexylmethyl, H), (M-6368, F, CH₃, Cl, cyclohexylmethyl, Cl), (M-6369, F, CH₃, Cl, cyclohexylmethyl, F), (M-6370, F, CH₃, Cl, cyclohexylmethyl, CF₃), (M-6371, F, CH₃, Cl, cyclohexylmethyl, Br), (M-6372, F, CH₃, Cl, cyclohexylmethyl, CH₃), (M-6373, Cl, H, H, H, H), (M-6374, Cl, H, H, H, Cl), (M-6375, MeO, F, H, H, F), (M-6376, MeO, F, H, H, c-Pr), (M-6377, Cl, H, H, H, Br), (M-6378, Cl, H, H, H, CH₃), (M-6379, MeO, H, H, F, c-Pr), (M-6380, Cl, H, H, F, Cl), (M-6381, MeO, H, H, F, F), (M-6382, Cl, H, H, F, CF₃), (M-6383, Cl, H, H, F, Br), (M-6384, Cl, H, H, F, CH₃), (M-6385, Cl, H, H, Cl, H), (M-6386, MeO, F, H, H, Et), (M-6387, MeO, H, H, Cl, F), (M-6388, Cl, H, H, Cl, CF₃), (M-6389, Cl, H, H, Cl, Br), (M-6390, Cl, H, H, Cl, CH₃), (M-6391, Cl, H, H, CH₃, H), (M-6392, Cl, H, H, CH₃, Cl), (M-6393, Cl, H, H, CH₃, F), (M-6394, Cl, H, H, CH₃, CF₃), (M-6395, Cl, H, H, CH₃, Br), (M-6396, Cl, H, H, CH₃, CH₃), (M-6397, Cl, H, H, Et, H), (M-6398, Cl, H, H, Et, Cl), (M-6399, Cl, H, H, Et, F), (M-6400, Cl, H, H, Et, CF₃), (M-6401, Cl, H, H, Et, Br), (M-6402, Cl, H, H, Et, CH₃), (M-6403, Cl, H, H, n-Pr, H), (M-6404, Cl, H, H, n-Pr, Cl), (M-6405, Cl, H, H, n-Pr, F), (M-6406, Cl, H, H, n-Pr, CF₃), (M-6407, Cl, H, H, n-Pr, Br), (M-6408, Cl, H, H, n-Pr, CH₃), (M-6409, Cl, H, H, c-Pr, H), (M-6410, Cl, H, H, c-Pr, Cl), (M-6411, Cl, H, H, c-Pr, F), (M-6412, Cl, H, H, c-Pr, CF₃), (M-6413, Cl, H, H, c-Pr, Br), (M-6414, Cl, H, H, c-Pr, CH₃), (M-6415, Cl, H, H, i-Pr, H), (M-6416, Cl, H, H, i-Pr, Cl), (M-6417, Cl, H, H, i-Pr, F), (M-6418, Cl, H, H, i-Pr, CF₃), (M-6419, Cl, H, H, i-Pr, Br), (M-6420, Cl, H, H, i-Pr, CH₃), (M-6421, MeO, H, H, n-Bu, H), (M-6422, Cl, H, H, n-Bu, Cl), (M-6423, Cl, H, H, n-Bu, F), (M-6424, Cl, H, H, n-Bu, CF₃), (M-6425, Cl, H, H, n-Bu, Br), (M-6426, Cl, H, H, n-Bu, CH₃), (M-6427, Cl, H, H, i-Bu, H), (M-6428, Cl, H, H, i-Bu, Cl), (M-6429, Cl, H, H, i-Bu, F), (M-6430, Cl, H, H, i-Bu, CF₃), (M-6431, Cl, H, H, i-Bu, Br), (M-6432, Cl, H, H, i-Bu, CH₃), (M-6433, Cl, H, H, sec-Bu, H), (M-6434, Cl, H, H, sec-Bu, Cl), (M-6435, Cl, H, H, sec-Bu, F), (M-6436, Cl, H, H, sec-Bu, CF₃), (M-6437, Cl, H, H, sec-Bu, Br), (M-64
38, Cl, H, H, sec-Bu, CH₃), (M-6439, Cl, H, H, n-Pen, H), (M-6440, Cl, H, H, n-Pen, Cl), (M-6441, MeO, H, H, n-Pen, F), (M-6442, Cl, H, H, n-Pen, CF₃), (M-6443, Cl, H, H, n-Pen, Br), (M-6444, Cl, H, H, n-Pen, CH₃), (M-6445, Cl, H, H, c-Pen, H), (M-6446, Cl, H, H, c-Pen, Cl), (M-6447, Cl, H, H, c-Pen, F), (M-6448, Cl, H, H, c-Pen, CF₃), (M-6449, Cl, H, H, c-Pen, Br), (M-6450, Cl, H, H, c-Pen, CH₃), (M-6451, Cl, H, H, n-Hex, H), (M-6452, Cl, H, H, n-Hex, Cl), (M-6453, Cl, H, H, n-Hex, F), (M-6454, Cl, H, H, n-Hex, CF₃), (M-6455, Cl, H, H, n-Hex, Br), (M-6456, Cl, H, H, n-Hex, CH₃), (M-6457, Cl, H, H, c-Hex, H), (M-6458, Cl, H, H, c-Hex, Cl), (M-6459, Cl, H, H, c-Hex, F), (M-6460, Cl, H, H, c-Hex, CF₃), (M-6461, Cl, H, H, c-Hex, Br), (M-6462, Cl, H, H, c-Hex, CH₃), (M-6463, Cl, H, H, OH, H), (M-6464, Cl, H, H, OH, Cl), (M-6465, Cl, H, H, OH, F), (M-6466, Cl, H, H, OH, CF₃), (M-6467, Cl, H, H, OH, Br), (M-6468, Cl, H, H, OH, CH₃), (M-6469, Cl, H, H, EtO, H), (M-6470, Cl, H, H, EtO, Cl), (M-6471, Cl, H, H, EtO, F), (M-6472, Cl, H, H, EtO, CF₃), (M-6473, Cl, H, H, EtO, Br), (M-6474, Cl, H, H, EtO, CH₃), (M-6475, Cl, H, H, n-PrO, H), (M-6476, Cl, H, H, n-PrO, Cl), (M-6477, Cl, H, H, n-PrO, F), (M-6478, Cl, H, H, n-PrO, CF₃), (M-6479, Cl, H, H, n-PrO, Br), (M-6480, Cl, H, H, n-PrO, CH₃), (M-6481, Cl, H, H, PhO, H), (M-6482, Cl, H, H, PhO, Cl), (M-6483, Cl, H, H, PhO, F), (M-6484, Cl, H, H, PhO, CF₃), (M-6485, Cl, H, H, PhO, Br), (M-6486, Cl, H, H, PhO, CH₃), (M-6487, Cl, H, H, BnO, H), (M-6488, Cl, H, H, BnO, Cl), (M-6489, Cl, H, H, BnO, F), (M-6490, Cl, H, H, BnO, CF₃), (M-6491, Cl, H, H, BnO, Br), (M-6492, Cl, H, H, BnO, CH₃), (M-6493, Cl, H, H, PhCH₂CH₂O, H), (M-6494, Cl, H, H, PhCH₂CH₂O, Cl), (M-6495, Cl, H, H, PhCH₂CH₂O, F), (M-6496, Cl, H, H, PhCH₂CH₂O, CF₃), (M-6497, Cl, H, H, PhCH₂CH₂O, Br), (M-6498, Cl, H, H, PhCH₂CH₂O, CH₃), (M-6499, MeO, H, H, CF₃O, CF₃), (M-6500, Cl, H, H, CF₃O, Cl), (M-6501, Cl, H, H, CF₃O, F), (M-6502, Cl, H, H, CF₃O, CF₃), (M-6503, Cl, H, H, CF₃O, Br), (M-6504, Cl, H, H, CF₃O, CH₃), (M-6505, MeO, H, H, Ph, H), (M-6506, Cl, H, H, Ph, Cl), (M-6507, Cl, H, H, Ph, F), (M-6508, Cl, H, H, Ph, CF₃), (M-6509, Cl, H, H, Ph, Br), (M-6510, Cl, H, H, Ph, CH₃), (M-6511, Cl, H, H, 4-F-Ph, H), (M-6512, Cl, H, H, 4-F-Ph, Cl), (M-6513, Cl, H, H, 4-F-Ph, F), (M-6514, Cl, H, H, 4-F-Ph, CF₃), (M-6515, Cl, H, H, 4-F-Ph, Br), (M-6516, Cl, H, H, 4-F-Ph, CH₃), (M-6517, Cl, H, H, 4-CF₃-Ph, H), (M-6518, Cl, H, H, 4-CF₃-Ph, Cl), (M-6519, Cl, H, H, 4-CF₃-Ph, F), (M-6520, Cl, H, H, 4-CF₃-Ph, CF₃), (M-6521, Cl, H, H, 4-CF₃-Ph, Br), (M-6522, Cl, H, H, 4-CF₃-Ph, CH₃), (M-6523, Cl, H, H, 4-(Me)₂N-Ph, H), (M-6524, Cl, H, H, 4-(Me)₂N-Ph, Cl), (M-6525, Cl, H, H, 4-(Me)₂N-Ph, F), (M-6526, Cl, H, H, 4-(Me)₂N-Ph, CF₃), (M-6527, Cl, H, H, 4-(Me)₂N-Ph, Br), (M-6528, Cl, H, H, 4-(Me)₂N-Ph, CH₃), (M-6529, Cl, H, H, 4-OH-Ph, H), (M-6530, Cl, H, H, 4-OH-Ph, Cl), (M-6531, Cl, H, H, 4-OH-Ph, F), (M-6532, Cl, H, H, 4-OH-Ph, CF₃), (M-6533, Cl, H, H, 4-OH-Ph, Br), (M-6534, Cl, H, H, 4-OH-Ph, CH₃), (M-6535, Cl, H, H, 3,4-di-F-Ph, H), (M-6536, Cl, H, H, 3,4-di-F-Ph, Cl), (M-6537, Cl, H, H, 3,4-di-F-Ph, F), (M-6538, Cl, H, H, 3,4-di-F-Ph, CF₃), (M-6539, Cl, H, H, 3,4-di-F-Ph, Br), (M-6540, Cl, H, H, 3,4-di-F-Ph, CH₃), (M-6541, Cl, H, H, 4-COOH-Ph, H), (M-6542, Cl, H, H, 4-COOH-Ph, Cl), (M-6543, Cl, H, H, 4-COOH-Ph, F), (M-6544, Cl, H, H, 4-COOH-Ph, CF₃), (M-6545, Cl, H, H, 4-COOH-Ph, Br), (M-6546, Cl, H, H, 4-COOH-Ph, CH₃), (M-6547, Cl, H, H, Bn, H), (M-6548, Cl, H, H, Bn, Cl), (M-6549, Cl, H, H, Bn, F), (M-6550, Cl, H, H, Bn, CF₃), (M-6551, Cl, H, H, Bn, Br), (M-6552, Cl, H, H, Bn, CH₃), (M-6553, Cl, H, H, 4-F-Bn, H), (M-6554, Cl, H, H, 4-F-Bn, Cl), (M-6555, Cl, H, H, 4-F-Bn, F), (M-6556, Cl, H, H, 4-F-Bn, CF₃), (M-6557, Cl, H, H, 4-F-Bn, Br), (M-6558, Cl, H, H, 4-F-Bn, CH₃), (M-6559, Cl, H, H, 2-Py, H), (M-6560, Cl, H, H, 2-Py, Cl), (M-6561, Cl, H, H, 2-Py, F), (M-6562, Cl, H, H, 2-Py, CF₃), (M-6563, Cl, H, H, 2-Py, Br), (M-6564, Cl, H, H, 2-Py, CH₃), (M-6565, Cl, H, H, 3-Py, H), (M-6566, Cl, H, H, 3-Py, Cl), (M-6567, Cl, H, H, 3-Py, F), (M-6568, Cl, H, H, 3-Py, CF₃), (M-6569, Cl, H, H, 3-Py, Br), (M-6570, Cl, H, H, 3-Py, CH₃), (M-6571, Cl, H, H, 4-Py, H), (M-6572, Cl, H, H, 4-Py, Cl), (M-6573, Cl, H, H, 4-Py, F), (M-6574, Cl, H, H, 4-Py, CF₃), (M-6575, Cl, H, H, 4-Py, Br), (M-6576, Cl, H, H, 4-Py, CH₃), (M-6577, Cl, H, H, 2-Th, H), (M-6578, Cl, H, H, 2-Th, Cl), (M-6579, Cl, H, H, 2-Th, F), (M-6580, Cl, H, H, 2-Th, CF₃), (M-6581, Cl, H, H, 2-Th, Br), (M-6582, Cl, H, H, 2-Th, CH₃), (M-6583, Cl, H, H, 3-Th, H), (M-6584, Cl, H, H, 3-Th, Cl), (M-6585, Cl, H, H, 3-Th, F), (M-6586, Cl, H, H, 3-Th, CF₃), (M-6587, Cl, H, H, 3-Th, Br), (M-6588, Cl, H, H, 3-Th, CH₃), (M-6589, Cl, H, H, pyrazol-2-yl, H), (M-6590, Cl, H, H, pyrazol-2-yl, Cl), (M-6591, Cl, H, H, pyrazol-2-yl, F), (M-6592, Cl, H, H, pyrazol-2-yl, CF₃), (M-6593, Cl, H, H, pyrazol-2-yl, Br), (M-6594, Cl, H, H, pyrazol-2-yl, CH₃), (M-6595, Cl, H, H, pyrazol-3-yl, H), (M-6596, Cl, H, H, pyrazol-3-yl, Cl), (M-6597, Cl, H, H, pyrazol-3-yl, F), (M-6598, Cl, H, H, pyrazol-3-yl, CF₃), (M-6599, Cl, H, H, pyrazol-3-yl, Br), (M-6600, Cl, H, H, pyrazol-3-yl, CH₃), (M-6601, Cl, H, H, pyrimidin-2-yl, H), (M-6602, Cl, H, H, pyrimidin-2-yl, Cl), (M-6603, Cl, H, H, pyrimidin-2-yl, F), (M-6604, Cl, H, H, pyrimidin-2-yl, CF₃), (M-6605, Cl, H, H, pyrimidin-2-yl, Br), (M-6606, Cl, H, H, pyrimidin-2-yl, CH₃), (M-6607, Cl, H, H, pyrimidin-4-yl, H), (M-6608, Cl, H, H, pyrimidin-4-yl, Cl), (M-6609, Cl, H, H, pyrimidin-4-yl, F), (M-6610, Cl, H, H, pyrimidin-4-yl, CF₃), (M-6611, Cl, H, H, pyrimidin-4-yl, Br), (M-6612, Cl, H, H, pyrimidin-4-yl, CH₃), (M-6613, Cl, H, H, pyrimidin-5-yl, H), (M-6614, Cl, H, H, pyrimidin-5-yl, Cl), (M-6615, Cl, H, H, pyrimidin-5-yl, F), (M-6616, Cl, H, H, pyrimidin-5-yl, CF₃), (M-6617, Cl, H, H, pyrimidin-5-yl, Br), (M-6618, Cl, H, H, pyrimidin-5-yl, CH₃), (M-6619, Cl, H, H, HOOCCH₂CH₂CH₂, H), (M-6620, Cl, H, H, HOOCCH₂CH₂CH₂, Cl), (M-6621, Cl, H, H, HOOCCH₂CH₂CH₂, F), (M-6622, Cl, H, H, HOOCCH₂CH₂CH₂, CF₃), (M-6623, Cl, H, H, HOOCCH₂CH₂CH₂, Br), (M-6624, Cl, H, H, HOOCCH₂CH₂CH₂, CH₃), (M-6625, Cl, H, H, HOOCCH₂CH₂CH₂CH₂, H), (M-6626, Cl, H, H, HOOCCH₂CH₂CH₂CH₂, Cl), (M-6627, Cl, H, H, HOOCCH₂CH₂CH₂CH₂, F), (M-6628, Cl, H, H, HOOCCH₂CH₂CH₂CH₂, CF₃), (M-6629, Cl, H, H, HOOCCH₂CH₂CH₂CH₂, Br), (M-6630, Cl, H, H, HOOCCH₂CH₂CH₂CH₂, CH₃), (M-6631, Cl, H, H, (Me)₂NCOCH₂CH₂CH₂CH₂, H), (M-6632, Cl, H, H, (Me)₂NCOCH₂CH₂CH₂CH₂, Cl), (M-6633, Cl, H, H, (Me)₂NCOCH₂CH₂CH₂CH₂, F), (M-6634, Cl, H, H, (Me)₂NCOCH₂CH₂CH₂CH₂, CF₃), (M-6635, Cl, H, H, (Me)₂NCOCH₂CH₂CH₂CH₂, Br), (M-6636, Cl, H, H, (Me)₂NCOCH₂CH₂CH₂CH₂, CH₃), (M-6637, Cl, H, H, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, H), (M-6638, Cl, H, H, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, Cl), (M-6639, Cl, H, H, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, F), (M-6640, Cl, H, H, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, CF₃), (M-6641, Cl, H, H, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, Br), (M-6642, Cl, H, H, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, CH₃), (M-6643, Cl, H, H, MeOCH₂, H), (M-6644, Cl, H, H, MeOCH₂, Cl), (M-6645, Cl, H, H, MeOCH₂, F), (M-6646, Cl, H, H, MeOCH₂, CF₃), (M-6647, Cl, H, H, MeOCH₂, Br), (M-6648, Cl, H, H, MeOCH₂, CH₃), (M-6649, Cl, H, H, EtOCH₂, H), (M-6650, Cl, H, H, EtOCH₂, Cl), (M-6651, Cl, H, H, EtOCH₂, F), (M-6652, Cl, H, H, EtOCH₂, CF₃), (M-6653, Cl, H, H, EtOCH₂, Br), (M-6654, Cl, H, H, EtOCH₂, CH₃), (M-6655, Cl, H, H, EtOCH₂CH₂, H), (M-6656, Cl, H, H, EtOCH₂CH₂, Cl), (M-6657, Cl, H, H, EtOCH₂CH₂, F), (M-6658, Cl, H, H, EtOCH₂CH₂, CF₃), (M-6659, Cl, H, H, EtOCH₂CH₂, Br), (M-6660, Cl, H, H, EtOCH₂CH₂, CH₃), (M-6661, Cl, H, H, MeOCH₂CH₂OCH₂CH₂
, H), (M-6662, Cl, H, H, MeOCH₂CH₂OCH₂CH₂, Cl), (M-6663, Cl, H, H, MeOCH₂CH₂OCH₂CH₂, F), (M-6664, Cl, H, H, MeOCH₂CH₂OCH₂CH₂, CF₃), (M-6665, Cl, H, H, MeOCH₂CH₂OCH₂CH₂, Br), (M-6666, Cl, H, H, MeOCH₂CH₂OCH₂CH₂, CH₃), (M-6667, Cl, H, H, MeOCH₂CH₂, H), (M-6668, Cl, H, H, MeOCH₂CH₂, Cl), (M-6669, Cl, H, H, MeOCH₂CH₂, F), (M-6670, Cl, H, H, MeOCH₂CH₂, CF₃), (M-6671, Cl, H, H, MeOCH₂CH₂, Br), (M-6672, Cl, H, H, MeOCH₂CH₂, CH₃), (M-6673, Cl, H, H, HOCH₂, H), (M-6674, Cl, H, H, HOCH₂, Cl), (M-6675, Cl, H, H, HOCH₂, F), (M-6676, Cl, H, H, HOCH₂, CF₃), (M-6677, Cl, H, H, HOCH₂, Br), (M-6678, Cl, H, H, HOCH₂, CH₃), (M-6679, Cl, H, H, HOCH₂CH₂, H), (M-6680, Cl, H, H, HOCH₂CH₂, Cl), (M-6681, Cl, H, H, HOCH₂CH₂, F), (M-6682, Cl, H, H, HOCH₂CH₂, CF₃), (M-6683, Cl, H, H, HOCH₂CH₂, Br), (M-6684, Cl, H, H, HOCH₂CH₂, CH₃), (M-6685, Cl, H, H, HOCH₂CH₂CH₂, H), (M-6686, Cl, H, H, HOCH₂CH₂CH₂, Cl), (M-6687, Cl, H, H, HOCH₂CH₂CH₂, F), (M-6688, Cl, H, H, HOCH₂CH₂CH₂, CF₃), (M-6689, Cl, H, H, HOCH₂CH₂CH₂, Br), (M-6690, Cl, H, H, HOCH₂CH₂CH₂, CH₃), (M-6691, Cl, H, H, HOCH₂CH₂CH₂CH₂, H), (M-6692, Cl, H, H, HOCH₂CH₂CH₂CH₂, Cl), (M-6693, Cl, H, H, HOCH₂CH₂CH₂CH₂, F), (M-6694, Cl, H, H, HOCH₂CH₂CH₂CH₂, CF₃), (M-6695, Cl, H, H, HOCH₂CH₂CH₂CH₂, Br), (M-6696, Cl, H, H, HOCH₂CH₂CH₂CH₂, CH₃), (M-6697, Cl, H, H, HOCH₂CH₂CH₂CH₂CH₂, H), (M-6698, Cl, H, H, HOCH₂CH₂CH₂CH₂CH₂, Cl), (M-6699, Cl, H, H, HOCH₂CH₂CH₂CH₂CH₂, F), (M-6700, Cl, H, H, HOCH₂CH₂CH₂CH₂CH₂, CF₃), (M-6701, Cl, H, H, HOCH₂CH₂CH₂CH₂CH₂, Br), (M-6702, Cl, H, H, HOCH₂CH₂CH₂CH₂CH₂, CH₃), (M-6703, Cl, H, H, HOCH₂CH₂OCH₂CH₂, H), (M-6704, Cl, H, H, HOCH₂CH₂OCH₂CH₂, Cl), (M-6705, Cl, H, H, HOCH₂CH₂OCH₂CH₂, F), (M-6706, Cl, H, H, HOCH₂CH₂OCH₂CH₂, CF₃), (M-6707, Cl, H, H, HOCH₂CH₂OCH₂CH₂, Br), (M-6708, Cl, H, H, HOCH₂CH₂OCH₂CH₂, CH₃), (M-6709, Cl, H, H, (Me)₂N, H), (M-6710, Cl, H, H, (Me)₂N, Cl), (M-6711, Cl, H, H, (Me)₂N, F), (M-6712, Cl, H, H, (Me)₂N, CF₃), (M-6713, Cl, H, H, (Me)₂N, Br), (M-6714, Cl, H, H, (Me)₂N, CH₃), (M-6715, Cl, H, H, piperidin-4-yl-methyl, H), (M-6716, Cl, H, H, piperidin-4-yl-methyl, Cl), (M-6717, Cl, H, H, piperidin-4-yl-methyl, F), (M-6718, Cl, H, H, piperidin-4-yl-methyl, CF₃), (M-6719, Cl, H, H, piperidin-4-yl-methyl, Br), (M-6720, Cl, H, H, piperidin-4-yl-methyl, CH₃), (M-6721, Cl, H, H, cyclohexylmethyl, H), (M-6722, Cl, H, H, cyclohexylmethyl, Cl), (M-6723, Cl, H, H, cyclohexylmethyl, F), (M-6724, Cl, H, H, cyclohexylmethyl, CF₃), (M-6725, Cl, H, H, cyclohexylmethyl, Br), (M-6726, Cl, H, H, cyclohexylmethyl, CH₃), (M-6727, MeO, H, F, H, H), (M-6728, Cl, H, F, H, Cl), (M-6729, MeO, H, F, H, F), (M-6730, MeO, H, F, H, CF₃), (M-6731, MeO, H, F, H, Br), (M-6732, MeO, H, F, H, CH₃), (M-6733, MeO, H, F, F, H), (M-6734, Cl, H, F, F, Cl), (M-6735, Cl, H, F, F, F), (M-6736, Cl, H, F, F, CF₃), (M-6737, Cl, H, F, F, Br), (M-6738, Cl, H, F, F, CH₃), (M-6739, Cl, H, F, Cl, H), (M-6740, Cl, H, F, Cl, Cl), (M-6741, Cl, H, F, Cl, F), (M-6742, Cl, H, F, Cl, CF₃), (M-6743, Cl, H, F, Cl, Br), (M-6744, Cl, H, F, Cl, CH₃), (M-6745, MeO, H, F, CH₃, H), (M-6746, Cl, H, F, CH₃, Cl), (M-6747, Cl, H, F, CH₃, F), (M-6748, Cl, H, F, CH₃, CF₃), (M-6749, Cl, H, F, CH₃, Br), (M-6750, Cl, H, F, CH₃, CH₃), (M-6751, MeO, H, F, Et, H), (M-6752, Cl, H, F, Et, Cl), (M-6753, Cl, H, F, Et, F), (M-6754, Cl, H, F, Et, CF₃), (M-6755, Cl, H, F, Et, Br), (M-6756, Cl, H, F, Et, CH₃), (M-6757, MeO, H, F, n-Pr, H), (M-6758, Cl, H, F, n-Pr, Cl), (M-6759, Cl, H, F, n-Pr, F), (M-6760, Cl, H, F, n-Pr, CF₃), (M-6761, MeO, H, F, n-Pr, Br), (M-6762, Cl, H, F, n-Pr, CH₃), (M-6763, Cl, H, F, c-Pr, H), (M-6764, Cl, H, F, c-Pr, Cl), (M-6765, Cl, H, F, c-Pr, F), (M-6766, Cl, H, F, c-Pr, CF₃), (M-6767, Cl, H, F, c-Pr, Br), (M-6768, Cl, H, F, c-Pr, CH₃), (M-6769, Cl, H, F, i-Pr, H), (M-6770, Cl, H, F, i-Pr, Cl), (M-6771, Cl, H, F, i-Pr, F), (M-6772, Cl, H, F, i-Pr, CF₃), (M-6773, Cl, H, F, i-Pr, Br), (M-6774, Cl, H, F, i-Pr, CH₃), (M-6775, MeO, H, F, n-Bu, H), (M-6776, Cl, H, F, n-Bu, Cl), (M-6777, Cl, H, F, n-Bu, F), (M-6778, Cl, H, F, n-Bu, CF₃), (M-6779, Cl, H, F, n-Bu, Br), (M-6780, Cl, H, F, n-Bu, CH₃), (M-6781, Cl, H, F, i-Bu, H), (M-6782, Cl, H, F, i-Bu, Cl), (M-6783, Cl, H, F, i-Bu, F), (M-6784, Cl, H, F, i-Bu, CF₃), (M-6785, Cl, H, F, i-Bu, Br), (M-6786, Cl, H, F, i-Bu, CH₃), (M-6787, Cl, H, F, sec-Bu, H), (M-6788, Cl, H, F, sec-Bu, Cl), (M-6789, Cl, H, F, sec-Bu, F), (M-6790, Cl, H, F, sec-Bu, CF₃), (M-6791, Cl, H, F, sec-Bu, Br), (M-6792, Cl, H, F, sec-Bu, CH₃), (M-6793, MeO, H, F, n-Pen, H), (M-6794, Cl, H, F, n-Pen, Cl), (M-6795, MeO, H, F, n-Pen, F), (M-6796, Cl, H, F, n-Pen, CF₃), (M-6797, Cl, H, F, n-Pen, Br), (M-6798, Cl, H, F, n-Pen, CH₃), (M-6799, Cl, H, F, c-Pen, H), (M-6800, Cl, H, F, c-Pen, Cl), (M-6801, Cl, H, F, c-Pen, F), (M-6802, Cl, H, F, c-Pen, CF₃), (M-6803, Cl, H, F, c-Pen, Br), (M-6804, Cl, H, F, c-Pen, CH₃), (M-6805, MeO, H, F, n-Hex, H), (M-6806, Cl, H, F, n-Hex, Cl), (M-6807, Cl, H, F, n-Hex, F), (M-6808, Cl, H, F, n-Hex, CF₃), (M-6809, Cl, H, F, n-Hex, Br), (M-6810, Cl, H, F, n-Hex, CH₃), (M-6811, MeO, H, F, c-Hex, H), (M-6812, Cl, H, F, c-Hex, Cl), (M-6813, Cl, H, F, c-Hex, F), (M-6814, Cl, H, F, c-Hex, CF₃), (M-6815, Cl, H, F, c-Hex, Br), (M-6816, Cl, H, F, c-Hex, CH₃), (M-6817, Cl, H, F, OH, H), (M-6818, Cl, H, F, OH, Cl), (M-6819, Cl, H, F, OH, F), (M-6820, Cl, H, F, OH, CF₃), (M-6821, Cl, H, F, OH, Br), (M-6822, Cl, H, F, OH, CH₃), (M-6823, MeO, H, F, EtO, H), (M-6824, Cl, H, F, EtO, Cl), (M-6825, Cl, H, F, EtO, F), (M-6826, Cl, H, F, EtO, CF₃), (M-6827, Cl, H, F, EtO, Br), (M-6828, Cl, H, F, EtO, CH₃), (M-6829, Cl, H, F, n-PrO, H), (M-6830, Cl, H, F, n-PrO, Cl), (M-6831, Cl, H, F, n-PrO, F), (M-6832, Cl, H, F, n-PrO, CF₃), (M-6833, Cl, H, F, n-PrO, Br), (M-6834, Cl, H, F, n-PrO, CH₃), (M-6835, Cl, H, F, PhO, H), (M-6836, Cl, H, F, PhO, Cl), (M-6837, Cl, H, F, PhO, F), (M-6838, Cl, H, F, PhO, CF₃), (M-6839, Cl, H, F, PhO, Br), (M-6840, Cl, H, F, PhO, CH₃), (M-6841, Cl, H, F, BnO, H), (M-6842, Cl, H, F, BnO, Cl), (M-6843, Cl, H, F, BnO, F), (M-6844, Cl, H, F, BnO, CF₃), (M-6845, Cl, H, F, BnO, Br), (M-6846, Cl, H, F, BnO, CH₃), (M-6847, Cl, H, F, PhCH₂CH₂O, H), (M-6848, Cl, H, F, PhCH₂CH₂O, Cl), (M-6849, Cl, H, F, PhCH₂CH₂O, F), (M-6850, Cl, H, F, PhCH₂CH₂O, CF₃), (M-6851, Cl, H, F, PhCH₂CH₂O, Br), (M-6852, Cl, H, F, PhCH₂CH₂O, CH₃), (M-6853, Cl, H, F, CF₃O, H), (M-6854, Cl, H, F, CF₃O, Cl), (M-6855, Cl, H, F, CF₃O, F), (M-6856, Cl, H, F, CF₃O, CF₃), (M-6857, Cl, H, F, CF₃O, Br), (M-6858, Cl, H, F, CF₃O, CH₃), (M-6859, MeO, H, F, Ph, H), (M-6860, Cl, H, F, Ph, Cl), (M-6861, MeO, H, F, Ph, F), (M-6862, Cl, H, F, Ph, CF₃), (M-6863, Cl, H, F, Ph, Br), (M-6864, Cl, H, F, Ph, CH₃), (M-6865, MeO, H, F, 4-F-Ph, H), (M-6866, Cl, H, F, 4-F-Ph, Cl), (M-6867, Cl, H, F, 4-F-Ph, F), (M-6868, Cl, H, F, 4-F-Ph, CF₃), (M-6869, Cl, H, F, 4-F-Ph, Br), (M-6870, Cl, H, F, 4-F-Ph, CH₃), (M-6871, Cl, H, F, 4-CF₃-Ph, H), (M-6872, Cl, H, F, 4-CF₃-Ph, Cl), (M-6873, Cl, H, F, 4-CF₃-Ph, F), (M-6874, Cl, H, F, 4-CF₃-Ph, CF₃), (M-6875, Cl, H, F, 4-CF₃-Ph, Br), (M-6876, Cl, H, F, 4-CF₃-Ph, CH₃), (M-6877, Cl, H, F, 4-(Me)₂N-Ph, H), (M-6878, Cl, H, F, 4-(Me)₂N-Ph, Cl), (M-6879, Cl, H, F, 4-(Me)₂N-Ph, F), (M-6880, Cl, H, F, 4-(Me)₂N-Ph, CF₃), (M-6881, Cl, H, F, 4-(Me)₂N-Ph, Br), (M-6882, Cl, H, F, 4-(Me)₂N-Ph, CH₃), (M-6883, Cl, H, F, 4-OH-Ph, H), (M-6884, Cl, H, F, 4-OH-Ph, Cl), (M-6885, Cl, H, F, 4-OH-Ph, F), (M-6886, Cl,
H, F, 4-OH-Ph, CF₃), (M-6887, Cl, H, F, 4-OH-Ph, Br), (M-6888, Cl, H, F, 4-OH-Ph, CH₃), (M-6889, Cl, H, F, 3,4-di-F-Ph, H), (M-6890, Cl, H, F, 3,4-di-F-Ph, Cl), (M-6891, Cl, H, F, 3,4-di-F-Ph, F), (M-6892, Cl, H, F, 3,4-di-F-Ph, CF₃), (M-6893, Cl, H, F, 3,4-di-F-Ph, Br), (M-6894, Cl, H, F, 3,4-di-F-Ph, CH₃), (M-6895, Cl, H, F, 4-COOH-Ph, H), (M-6896, Cl, H, F, 4-COOH-Ph, Cl), (M-6897, Cl, H, F, 4-COOH-Ph, F), (M-6898, Cl, H, F, 4-COOH-Ph, CF₃), (M-6899, Cl, H, F, 4-COOH-Ph, Br), (M-6900, Cl, H, F, 4-COOH-Ph, CH₃), (M-6901, MeO, H, F, Bn, H), (M-6902, Cl, H, F, Bn, Cl), (M-6903, Cl, H, F, Bn, F), (M-6904, Cl, H, F, Bn, CF₃), (M-6905, Cl, H, F, Bn, Br), (M-6906, Cl, H, F, Bn, CH₃), (M-6907, Cl, H, F, 4-F-Bn, H), (M-6908, Cl, H, F, 4-F-Bn, Cl), (M-6909, Cl, H, F, 4-F-Bn, F), (M-6910, Cl, H, F, 4-F-Bn, CF₃), (M-6911, Cl, H, F, 4-F-Bn, Br), (M-6912, Cl, H, F, 4-F-Bn, CH₃), (M-6913, Cl, H, F, 2-Py, H), (M-6914, Cl, H, F, 2-Py, Cl), (M-6915, Cl, H, F, 2-Py, F), (M-6916, Cl, H, F, 2-Py, CF₃), (M-6917, Cl, H, F, 2-Py, Br), (M-6918, Cl, H, F, 2-Py, CH₃), (M-6919, MeO, H, F, 3-Py, H), (M-6920, Cl, H, F, 3-Py, Cl), (M-6921, Cl, H, F, 3-Py, F), (M-6922, Cl, H, F, 3-Py, CF₃), (M-6923, Cl, H, F, 3-Py, Br), (M-6924, Cl, H, F, 3-Py, CH₃), (M-6925, Cl, H, F, 4-Py, H), (M-6926, Cl, H, F, 4-Py, Cl), (M-6927, Cl, H, F, 4-Py, F), (M-6928, Cl, H, F, 4-Py, CF₃), (M-6929, Cl, H, F, 4-Py, Br), (M-6930, Cl, H, F, 4-Py, CH₃), (M-6931, Cl, H, F, 2-Th, H), (M-6932, Cl, H, F, 2-Th, Cl), (M-6933, Cl, H, F, 2-Th, F), (M-6934, Cl, H, F, 2-Th, CF₃), (M-6935, Cl, H, F, 2-Th, Br), (M-6936, Cl, H, F, 2-Th, CH₃), (M-6937, Cl, H, F, 3-Th, H), (M-6938, Cl, H, F, 3-Th, Cl), (M-6939, Cl, H, F, 3-Th, F), (M-6940, Cl, H, F, 3-Th, CF₃), (M-6941, Cl, H, F, 3-Th, Br), (M-6942, Cl, H, F, 3-Th, CH₃), (M-6943, Cl, H, F, pyrazol-2-yl, H), (M-6944, Cl, H, F, pyrazol-2-yl, Cl), (M-6945, Cl, H, F, pyrazol-2-yl, F), (M-6946, Cl, H, F, pyrazol-2-yl, CF₃), (M-6947, Cl, H, F, pyrazol-2-yl, Br), (M-6948, Cl, H, F, pyrazol-2-yl, CH₃), (M-6949, Cl, H, F, pyrazol-3-yl, H), (M-6950, Cl, H, F, pyrazol-3-yl, Cl), (M-6951, Cl, H, F, pyrazol-3-yl, F), (M-6952, Cl, H, F, pyrazol-3-yl, CF₃), (M-6953, Cl, H, F, pyrazol-3-yl, Br), (M-6954, Cl, H, F, pyrazol-3-yl, CH₃), (M-6955, Cl, H, F, pyrimidin-2-yl, H), (M-6956, Cl, H, F, pyrimidin-2-yl, Cl), (M-6957, Cl, H, F, pyrimidin-2-yl, F), (M-6958, Cl, H, F, pyrimidin-2-yl, CF₃), (M-6959, Cl, H, F, pyrimidin-2-yl, Br), (M-6960, Cl, H, F, pyrimidin-2-yl, CH₃), (M-6961, Cl, H, F, pyrimidin-4-yl, H), (M-6962, Cl, H, F, pyrimidin-4-yl, Cl), (M-6963, Cl, H, F, pyrimidin-4-yl, F), (M-6964, Cl, H, F, pyrimidin-4-yl, CF₃), (M-6965, Cl, H, F, pyrimidin-4-yl, Br), (M-6966, Cl, H, F, pyrimidin-4-yl, CH₃), (M-6967, Cl, H, F, pyrimidin-5-yl, H), (M-6968, Cl, H, F, pyrimidin-5-yl, Cl), (M-6969, Cl, H, F, pyrimidin-5-yl, F), (M-6970, Cl, H, F, pyrimidin-5-yl, CF₃), (M-6971, Cl, H, F, pyrimidin-5-yl, Br), (M-6972, Cl, H, F, pyrimidin-5-yl, CH₃), (M-6973, Cl, H, F, HOOCCH₂CH₂CH₂, H), (M-6974, Cl, H, F, HOOCCH₂CH₂CH₂, Cl), (M-6975, Cl, H, F, HOOCCH₂CH₂CH₂, F), (M-6976, Cl, H, F, HOOCCH₂CH₂CH₂, CF₃), (M-6977, Cl, H, F, HOOCCH₂CH₂CH₂, Br), (M-6978, Cl, H, F, HOOCCH₂CH₂CH₂, CH₃), (M-6979, Cl, H, F, HOOCCH₂CH₂CH₂CH₂, H), (M-6980, Cl, H, F, HOOCCH₂CH₂CH₂CH₂, Cl), (M-6981, Cl, H, F, HOOCCH₂CH₂CH₂CH₂, F), (M-6982, Cl, H, F, HOOCCH₂CH₂CH₂CH₂, CF₃), (M-6983, Cl, H, F, HOOCCH₂CH₂CH₂CH₂, Br), (M-6984, Cl, H, F, HOOCCH₂CH₂CH₂CH₂, CH₃), (M-6985, Cl, H, F, (Me)₂NCOCH₂CH₂CH₂CH₂, H), (M-6986, Cl, H, F, (Me)₂NCOCH₂CH₂CH₂CH₂, Cl), (M-6987, Cl, H, F, (Me)₂NCOCH₂CH₂CH₂CH₂, F), (M-6988, Cl, H, F, (Me)₂NCOCH₂CH₂CH₂CH₂, CF₃), (M-6989, Cl, H, F, (Me)₂NCOCH₂CH₂CH₂CH₂, Br), (M-6990, Cl, H, F, (Me)₂NCOCH₂CH₂CH₂CH₂, CH₃), (M-6991, Cl, H, F, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, H), (M-6992, Cl, H, F, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, Cl), (M-6993, Cl, H, F, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, F), (M-6994, Cl, H, F, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, CF₃), (M-6995, Cl, H, F, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, Br), (M-6996, Cl, H, F, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, CH₃), (M-6997, Cl, H, F, MeOCH₂, H), (M-6998, Cl, H, F, MeOCH₂, Cl), (M-6999, Cl, H, F, MeOCH₂, F), (M-7000, Cl, H, F, MeOCH₂, CF₃), (M-7001, Cl, H, F, MeOCH₂, Br), (M-7002, Cl, H, F, MeOCH₂, CH₃), (M-7003, Cl, H, F, EtOCH₂, H), (M-7004, Cl, H, F, EtOCH₂, Cl), (M-7005, Cl, H, F, EtOCH₂, F), (M-7006, Cl, H, F, EtOCH₂, CF₃), (M-7007, Cl, H, F, EtOCH₂, Br), (M-7008, Cl, H, F, EtOCH₂, CH₃), (M-7009, MeO, H, F, EtOCH₂CH₂, H), (M-7010, Cl, H, F, EtOCH₂CH₂, Cl), (M-7011, Cl, H, F, EtOCH₂CH₂, F), (M-7012, Cl, H, F, EtOCH₂CH₂, CF₃), (M-7013, Cl, H, F, EtOCH₂CH₂, Br), (M-7014, Cl, H, F, EtOCH₂CH₂, CH₃), (M-7015, Cl, H, F, MeOCH₂CH₂OCH₂CH₂, H), (M-7016, Cl, H, F, MeOCH₂CH₂OCH₂CH₂, Cl), (M-7017, Cl, H, F, MeOCH₂CH₂OCH₂CH₂, F), (M-7018, Cl, H, F, MeOCH₂CH₂OCH₂CH₂, CF₃), (M-7019, Cl, H, F, MeOCH₂CH₂OCH₂CH₂, Br), (M-7020, Cl, H, F, MeOCH₂CH₂OCH₂CH₂, CH₃), (M-7021, Cl, H, F, MeOCH₂CH₂, H), (M-7022, Cl, H, F, MeOCH₂CH₂, Cl), (M-7023, Cl, H, F, MeOCH₂CH₂, F), (M-7024, Cl, H, F, MeOCH₂CH₂, CF₃), (M-7025, Cl, H, F, MeOCH₂CH₂, Br), (M-7026, Cl, H, F, MeOCH₂CH₂, CH₃), (M-7027, Cl, H, F, HOCH₂, H), (M-7028, Cl, H, F, HOCH₂, Cl), (M-7029, Cl, H, F, HOCH₂, F), (M-7030, Cl, H, F, HOCH₂, CF₃), (M-7031, Cl, H, F, HOCH₂, Br), (M-7032, Cl, H, F, HOCH₂, CH₃), (M-7033, Cl, H, F, HOCH₂CH₂, H), (M-7034, Cl, H, F, HOCH₂CH₂, Cl), (M-7035, Cl, H, F, HOCH₂CH₂, F), (M-7036, Cl, H, F, HOCH₂CH₂, CF₃), (M-7037, Cl, H, F, HOCH₂CH₂, Br), (M-7038, Cl, H, F, HOCH₂CH₂, CH₃), (M-7039, Cl, H, F, HOCH₂CH₂CH₂, H), (M-7040, Cl, H, F, HOCH₂CH₂CH₂, Cl), (M-7041, Cl, H, F, HOCH₂CH₂CH₂, F), (M-7042, Cl, H, F, HOCH₂CH₂CH₂, CF₃), (M-7043, Cl, H, F, HOCH₂CH₂CH₂, Br), (M-7044, Cl, H, F, HOCH₂CH₂CH₂, CH₃), (M-7045, Cl, H, F, HOCH₂CH₂CH₂CH₂, H), (M-7046, Cl, H, F, HOCH₂CH₂CH₂CH₂, Cl), (M-7047, Cl, H, F, HOCH₂CH₂CH₂CH₂, F), (M-7048, Cl, H, F, HOCH₂CH₂CH₂CH₂, CF₃), (M-7049, Cl, H, F, HOCH₂CH₂CH₂CH₂, Br), (M-7050, Cl, H, F, HOCH₂CH₂CH₂CH₂, CH₃), (M-7051, Cl, H, F, HOCH₂CH₂CH₂CH₂CH₂, H), (M-7052, Cl, H, F, HOCH₂CH₂CH₂CH₂CH₂, Cl), (M-7053, Cl, H, F, HOCH₂CH₂CH₂CH₂CH₂, F), (M-7054, Cl, H, F, HOCH₂CH₂CH₂CH₂CH₂, CF₃), (M-7055, Cl, H, F, HOCH₂CH₂CH₂CH₂CH₂, Br), (M-7056, Cl, H, F, HOCH₂CH₂CH₂CH₂CH₂, CH₃), (M-7057, Cl, H, F, HOCH₂CH₂OCH₂CH₂, H), (M-7058, Cl, H, F, HOCH₂CH₂OCH₂CH₂, Cl), (M-7059, Cl, H, F, HOCH₂CH₂OCH₂CH₂, F), (M-7060, Cl, H, F, HOCH₂CH₂OCH₂CH₂, CF₃), (M-7061, Cl, H, F, HOCH₂CH₂OCH₂CH₂, Br), (M-7062, Cl, H, F, HOCH₂CH₂OCH₂CH₂, CH₃), (M-7063, Cl, H, F, (Me)₂N, H), (M-7064,
Cl, H, F, (Me)₂N, Cl), (M-7065, Cl, H, F, (Me)₂N, F), (M-7066, Cl, H, F, (Me)₂N, CF₃), (M-7067, Cl, H, F, (Me)₂N, Br), (M-7068, Cl, H, F, (Me)₂N, CH₃), (M-7069, Cl, H, F, piperidin-4-yl-methyl, H), (M-7070, Cl, H, F, piperidin-4-yl-methyl, Cl), (M-7071, Cl, H, F, piperidin-4-yl-methyl, F), (M-7072, Cl, H, F, piperidin-4-yl-methyl, CF₃), (M-7073, Cl, H, F, piperidin-4-yl-methyl, Br), (M-7074, Cl, H, F, piperidin-4-yl-methyl, CH₃), (M-7075, Cl, H, F, cyclohexylmethyl, H), (M-7076, Cl, H, F, cyclohexylmethyl, Cl), (M-7077, Cl, H, F, cyclohexylmethyl, F), (M-7078, Cl, H, F, cyclohexylmethyl, CF₃), (M-7079, Cl, H, F, cyclohexylmethyl, Br), (M-7080, Cl, H, F, cyclohexylmethyl, CH₃), (M-7081, Cl, H, Cl, H, H), (M-7082, Cl, H, Cl, H, Cl), (M-7083, Cl, H, Cl, H, F), (M-7084, Cl, H, Cl, H, CF₃), (M-7085, Cl, H, Cl, H, Br), (M-7086, Cl, H, Cl, H, CH₃), (M-7087, Cl, H, Cl, F, H), (M-7088, Cl, H, Cl, F, Cl), (M-7089, Cl, H, Cl, F, F), (M-7090, Cl, H, Cl, F, CF₃), (M-7091, Cl, H, Cl, F, Br), (M-7092, Cl, H, Cl, F, CH₃), (M-7093, MeO, H, Cl, Cl, H), (M-7094, Cl, H, Cl, Cl, Cl), (M-7095, Cl, H, Cl, Cl, F), (M-7096, Cl, H, Cl, Cl, CF₃), (M-7097, Cl, H, Cl, Cl, Br), (M-7098, Cl, H, Cl, Cl, CH₃), (M-7099, Cl, H, Cl, CH₃, H), (M-7100, Cl, H, Cl, CH₃, Cl), (M-7101, Cl, H, Cl, CH₃, F), (M-7102, Cl, H, Cl, CH₃, CF₃), (M-7103, Cl, H, Cl, CH₃, Br), (M-7104, Cl, H, Cl, CH₃, CH₃), (M-7105, Cl, H, Cl, Et, H), (M-7106, Cl, H, Cl, Et, Cl), (M-7107, Cl, H, Cl, Et, F), (M-7108, Cl, H, Cl, Et, CF₃), (M-7109, Cl, H, Cl, Et, Br), (M-7110, Cl, H, Cl, Et, CH₃), (M-7111, Cl, H, Cl, n-Pr, H), (M-7112, Cl, H, Cl, n-Pr, Cl), (M-7113, Cl, H, Cl, n-Pr, F), (M-7114, Cl, H, Cl, n-Pr, CF₃), (M-7115, Cl, H, Cl, n-Pr, Br), (M-7116, Cl, H, Cl, n-Pr, CH₃), (M-7117, Cl, H, Cl, c-Pr, H), (M-7118, Cl, H, Cl, c-Pr, Cl), (M-7119, Cl, H, Cl, c-Pr, F), (M-7120, Cl, H, Cl, c-Pr, CF₃), (M-7121, Cl, H, Cl, c-Pr, Br), (M-7122, Cl, H, Cl, c-Pr, CH₃), (M-7123, Cl, H, Cl, i-Pr, H), (M-7124, Cl, H, Cl, i-Pr, Cl), (M-7125, Cl, H, Cl, i-Pr, F), (M-7126, Cl, H, Cl, i-Pr, CF₃), (M-7127, Cl, H, Cl, i-Pr, Br), (M-7128, Cl, H, Cl, i-Pr, CH₃), (M-7129, Cl, H, Cl, n-Bu, H), (M-7130, Cl, H, Cl, n-Bu, Cl), (M-7131, Cl, H, Cl, n-Bu, F), (M-7132, Cl, H, Cl, n-Bu, CF₃), (M-7133, Cl, H, Cl, n-Bu, Br), (M-7134, Cl, H, Cl, n-Bu, CH₃), (M-7135, Cl, H, Cl, i-Bu, H), (M-7136, Cl, H, Cl, i-Bu, Cl), (M-7137, Cl, H, Cl, i-Bu, F), (M-7138, Cl, H, Cl, i-Bu, CF₃), (M-7139, Cl, H, Cl, i-Bu, Br), (M-7140, Cl, H, Cl, i-Bu, CH₃), (M-7141, Cl, H, Cl, sec-Bu, H), (M-7142, Cl, H, Cl, sec-Bu, Cl), (M-7143, Cl, H, Cl, sec-Bu, F), (M-7144, Cl, H, Cl, sec-Bu, CF₃), (M-7145, Cl, H, Cl, sec-Bu, Br), (M-7146, Cl, H, Cl, sec-Bu, CH₃), (M-7147, Cl, H, Cl, n-Pen, H), (M-7148, Cl, H, Cl, n-Pen, Cl), (M-7149, Cl, H, Cl, n-Pen, F), (M-7150, Cl, H, Cl, n-Pen, CF₃), (M-7151, Cl, H, Cl, n-Pen, Br), (M-7152, Cl, H, Cl, n-Pen, CH₃), (M-7153, Cl, H, Cl, c-Pen, H), (M-7154, Cl, H, Cl, c-Pen, Cl), (M-7155, Cl, H, Cl, c-Pen, F), (M-7156, Cl, H, Cl, c-Pen, CF₃), (M-7157, Cl, H, Cl, c-Pen, Br), (M-7158, Cl, H, Cl, c-Pen, CH₃), (M-7159, Cl, H, Cl, n-Hex, H), (M-7160, Cl, H, Cl, n-Hex, Cl), (M-7161, Cl, H, Cl, n-Hex, F), (M-7162, Cl, H, Cl, n-Hex, CF₃), (M-7163, Cl, H, Cl, n-Hex, Br), (M-7164, Cl, H, Cl, n-Hex, CH₃), (M-7165, Cl, H, Cl, c-Hex, H), (M-7166, Cl, H, Cl, c-Hex, Cl), (M-7167, Cl, H, Cl, c-Hex, F), (M-7168, Cl, H, Cl, c-Hex, CF₃), (M-7169, Cl, H, Cl, c-Hex, Br), (M-7170, Cl, H, Cl, c-Hex, CH₃), (M-7171, Cl, H, Cl, OH, H), (M-7172, Cl, H, Cl, OH, Cl), (M-7173, Cl, H, Cl, OH, F), (M-7174, Cl, H, Cl, OH, CF₃), (M-7175, Cl, H, Cl, OH, Br), (M-7176, Cl, H, Cl, OH, CH₃), (M-7177, Cl, H, Cl, EtO, H), (M-7178, Cl, H, Cl, EtO, Cl), (M-7179, Cl, H, Cl, EtO, F), (M-7180, Cl, H, Cl, EtO, CF₃), (M-7181, Cl, H, Cl, EtO, Br), (M-7182, Cl, H, Cl, EtO, CH₃), (M-7183, Cl, H, Cl, n-PrO, H), (M-7184, Cl, H, Cl, n-PrO, Cl), (M-7185, Cl, H, Cl, n-PrO, F), (M-7186, Cl, H, Cl, n-PrO, CF₃), (M-7187, Cl, H, Cl, n-PrO, Br), (M-7188, Cl, H, Cl, n-PrO, CH₃), (M-7189, Cl, H, Cl, PhO, H), (M-7190, Cl, H, Cl, PhO, Cl), (M-7191, Cl, H, Cl, PhO, F), (M-7192, Cl, H, Cl, PhO, CF₃), (M-7193, Cl, H, Cl, PhO, Br), (M-7194, Cl, H, Cl, PhO, CH₃), (M-7195, Cl, H, Cl, BnO, H), (M-7196, Cl, H, Cl, BnO, Cl), (M-7197, Cl, H, Cl, BnO, F), (M-7198, Cl, H, Cl, BnO, CF₃), (M-7199, Cl, H, Cl, BnO, Br), (M-7200, Cl, H, Cl, BnO, CH₃), (M-7201, Cl, H, Cl, PhCH₂CH₂O, H), (M-7202, Cl, H, Cl, PhCH₂CH₂O, Cl), (M-7203, Cl, H, Cl, PhCH₂CH₂O, F), (M-7204, Cl, H, Cl, PhCH₂CH₂O, CF₃), (M-7205, Cl, H, Cl, PhCH₂CH₂O, Br), (M-7206, Cl, H, Cl, PhCH₂CH₂O, CH₃), (M-7207, Cl, H, Cl, CF₃O, H), (M-7208, Cl, H, Cl, CF₃O, Cl), (M-7209, Cl, H, Cl, CF₃O, F), (M-7210, Cl, H, Cl, CF₃O, CF₃), (M-7211, Cl, H, Cl, CF₃O, Br), (M-7212, Cl, H, Cl, CF₃O, CH₃), (M-7213, Cl, H, Cl, Ph, H), (M-7214, Cl, H, Cl, Ph, Cl), (M-7215, Cl, H, Cl, Ph, F), (M-7216, Cl, H, Cl, Ph, CF₃), (M-7217, Cl, H, Cl, Ph, Br), (M-7218, Cl, H, Cl, Ph, CH₃), (M-7219, Cl, H, Cl, 4-F-Ph, H), (M-7220, Cl, H, Cl, 4-F-Ph, Cl), (M-7221, Cl, H, Cl, 4-F-Ph, F), (M-7222, Cl, H, Cl, 4-F-Ph, CF₃), (M-7223, Cl, H, Cl, 4-F-Ph, Br), (M-7224, Cl, H, Cl, 4-F-Ph, CH₃), (M-7225, Cl, H, Cl, 4-CF₃-Ph, H), (M-7226, Cl, H, Cl, 4-CF₃-Ph, Cl), (M-7227, Cl, H, Cl, 4-CF₃-Ph, F), (M-7228, Cl, H, Cl, 4-CF₃-Ph, CF₃), (M-7229, Cl, H, Cl, 4-CF₃-Ph, Br), (M-7230, Cl, H, Cl, 4-CF₃-Ph, CH₃), (M-7231, Cl, H, Cl, 4-(Me)₂N-Ph, H), (M-7232, Cl, H, Cl, 4-(Me)₂N-Ph, Cl), (M-7233, Cl, H, Cl, 4-(Me)₂N-Ph, F), (M-7234, Cl, H, Cl, 4-(Me)₂N-Ph, CF₃), (M-7235, Cl, H, Cl, 4-(Me)₂N-Ph, Br), (M-7236, Cl, H, Cl, 4-(Me)₂N-Ph, CH₃), (M-7237, Cl, H, Cl, 4-OH-Ph, H), (M-7238, Cl, H, Cl, 4-OH-Ph, Cl), (M-7239, Cl, H, Cl, 4-OH-Ph, F), (M-7240, Cl, H, Cl, 4-OH-Ph, CF₃), (M-7241, Cl, H, Cl, 4-OH-Ph, Br), (M-7242, Cl, H, Cl, 4-OH-Ph, CH₃), (M-7243, Cl, H, Cl, 3,4-di-F-Ph, H), (M-7244, Cl, H, Cl, 3,4-di-F-Ph, Cl), (M-7245, Cl, H, Cl, 3,4-di-F-Ph, F), (M-7246, Cl, H, Cl, 3,4-di-F-Ph, CF₃), (M-7247, Cl, H, Cl, 3,4-di-F-Ph, Br), (M-7248, Cl, H, Cl, 3,4-di-F-Ph, CH₃), (M-7249, Cl, H, Cl, 4-COOH-Ph, H), (M-7250, Cl, H, Cl, 4-COOH-Ph, Cl), (M-7251, Cl, H, Cl, 4-COOH-Ph, F), (M-7252, Cl, H, Cl, 4-COOH-Ph, CF₃), (M-7253, Cl, H, Cl, 4-COOH-Ph, Br), (M-7254, Cl, H, Cl, 4-COOH-Ph, CH₃), (M-7255, Cl, H, Cl, Bn, H), (M-7256, Cl, H, Cl, Bn, Cl), (M-7257, Cl, H, Cl, Bn, F), (M-7258, Cl, H, Cl, Bn, CF₃), (M-7259, Cl, H, Cl, Bn, Br), (M-7260, Cl, H, Cl, Bn, CH₃), (M-7261, Cl, H, Cl, 4-F-Bn, H), (M-7262, Cl, H, Cl, 4-F-Bn, Cl), (M-7263, Cl, H, Cl, 4-F-Bn, F), (M-7264, Cl, H, Cl, 4-F-Bn, CF₃), (M-7265, Cl, H, Cl, 4-F-Bn, Br), (M-7266, Cl, H, Cl, 4-F-Bn, CH₃), (M-7267, Cl, H, Cl, 2-Py, H), (M-7268, Cl, H, Cl, 2-Py, Cl), (M-7269, Cl, H, Cl, 2-Py, F), (M-7270, Cl, H, Cl, 2-Py, CF₃), (M-7271, Cl, H, Cl, 2-Py, Br), (M-7272, Cl, H, Cl, 2-Py, CH₃), (M-7273, Cl, H, Cl, 3-Py, H), (M-7274, Cl, H, Cl, 3-Py, Cl), (M-7275, Cl, H, Cl, 3-Py, F), (M-7276, Cl, H, Cl, 3-Py, CF₃), (M-7277, Cl, H, Cl, 3-Py, Br), (M-7278, Cl, H, Cl, 3-Py, CH₃), (M-7279, Cl, H, Cl, 4-Py, H), (M-7280, Cl, H, Cl, 4-Py, Cl), (M-7281, Cl, H, Cl, 4-Py, F), (M-7282, Cl, H, Cl, 4-Py, CF₃), (M-7283, Cl, H, Cl, 4-Py, Br), (M-7284, Cl, H, Cl, 4-Py, CH₃), (M-7285, Cl, H, Cl, 2-Th, H), (M-7286, Cl, H, Cl, 2-Th, Cl), (M-7287, Cl, H, Cl, 2-Th, F), (M-7288, Cl, H, Cl, 2-Th, CF₃), (M-7289, Cl, H, Cl, 2-Th, Br), (M-7290, Cl, H, Cl, 2-Th, CH₃), (M-7291, Cl, H, Cl, 3-Th, H), (M-7292, Cl, H, Cl, 3-Th, Cl), (M-7293, Cl, H, Cl, 3-Th, F), (M-7294, Cl, H, Cl, 3-Th, CF₃), (M-7295, Cl, H, Cl, 3-Th, Br), (M-7296, Cl, H, Cl, 3-Th, CH₃), (M-7297, Cl, H, Cl, pyrazol-2-yl, H), (M-7298, Cl, H, Cl, pyrazol-2-yl, Cl), (M-7299, Cl, H, Cl, pyrazol-2-yl, F), (M-7300, Cl, H, Cl, pyrazol-2-yl, CF₃), (M-7301, Cl, H, Cl, pyrazol-2-yl, Br), (M-7302, Cl, H, Cl, pyrazol-2-yl, CH₃), (M-7303, Cl, H, Cl, pyrazol-3-yl, H), (M-7304, Cl, H, Cl, pyrazol-3-yl, Cl), (M-7305, Cl, H, Cl, pyrazol-3-yl, F), (M-7306, Cl, H, Cl, pyrazol-3-yl, CF₃), (M-7307, Cl, H, Cl, pyrazol-3-yl, Br), (M-7308, Cl, H, Cl, pyrazol-3-yl, CH₃), (M-7309, Cl, H, Cl, pyrimidin-2-yl, H), (M-7310, Cl, H, Cl, pyrimidin-2-yl, Cl), (M-7311, Cl, H, Cl, pyrimidin-2-yl, F), (M-7312, Cl, H, Cl, pyrimidin-2-yl, CF₃), (M-7313, Cl, H, Cl, pyrimidin-2-yl, Br), (M-7314, Cl, H, Cl, pyrimidin-2-yl, CH₃), (M-7315, Cl, H, Cl, pyrimidin-4-yl, H), (M-7316, Cl, H, Cl, pyrimidin-4-yl, Cl), (M-7317, Cl, H, Cl, pyrimidin-4-yl, F), (M-7318, Cl, H, Cl, pyrimidin-4-yl, CF₃), (M-7319, Cl, H, Cl, pyrimidin-4-yl, Br), (M-7320, Cl, H, Cl, pyrimidin-4-yl, CH₃), (M-7321, Cl, H, Cl, pyrimidin-5-yl, H), (M-7322, Cl, H, Cl, pyrimidin-5-yl, Cl), (M-7323, Cl, H, Cl, pyrimidin-5-yl, F), (M-7324, Cl, H, Cl, pyrimidin-5-yl, CF₃), (M-7325, Cl, H, Cl, pyrimidin-5-yl, Br), (M-7326, Cl, H, Cl, pyrimidin-5-yl, CH₃), (M-7327, Cl, H, Cl, HOOCCH₂CH₂CH₂, H), (M-7328, Cl, H, Cl, HOOCCH
₂CH₂CH₂, Cl), (M-7329, Cl, H, Cl, HOOCCH₂CH₂CH₂, F), (M-7330, Cl, H, Cl, HOOCCH₂CH₂CH₂, CF₃), (M-7331, Cl, H, Cl, HOOCCH₂CH₂CH₂, Br), (M-7332, Cl, H, Cl, HOOCCH₂CH₂CH₂, CH₃), (M-7333, Cl, H, Cl, HOOCCH₂CH₂CH₂CH₂, H), (M-7334, Cl, H, Cl, HOOCCH₂CH₂CH₂CH₂, Cl), (M-7335, Cl, H, Cl, HOOCCH₂CH₂CH₂CH₂, F), (M-7336, Cl, H, Cl, HOOCCH₂CH₂CH₂CH₂, CF₃), (M-7337, Cl, H, Cl, HOOCCH₂CH₂CH₂CH₂, Br), (M-7338, Cl, H, Cl, HOOCCH₂CH₂CH₂CH₂, CH₃), (M-7339, Cl, H, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂, H), (M-7340, Cl, H, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂, Cl), (M-7341, Cl, H, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂, F), (M-7342, Cl, H, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂, CF₃), (M-7343, Cl, H, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂, Br), (M-7344, Cl, H, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂, CH₃), (M-7345, Cl, H, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, H), (M-7346, Cl, H, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, Cl), (M-7347, Cl, H, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, F), (M-7348, Cl, H, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, CF₃), (M-7349, Cl, H, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, Br), (M-7350, Cl, H, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, CH₃), (M-7351, Cl, H, Cl, MeOCH₂, H), (M-7352, Cl, H, Cl, MeOCH₂, Cl), (M-7353, Cl, H, Cl, MeOCH₂, F), (M-7354, Cl, H, Cl, MeOCH₂, CF₃), (M-7355, Cl, H, Cl, MeOCH₂, Br), (M-7356, Cl, H, Cl, MeOCH₂, CH₃), (M-7357, Cl, H, Cl, EtOCH₂, H), (M-7358, Cl, H, Cl, EtOCH₂, Cl), (M-7359, Cl, H, Cl, EtOCH₂, F), (M-7360, Cl, H, Cl, EtOCH₂, CF₃), (M-7361, Cl, H, Cl, EtOCH₂, Br), (M-7362, Cl, H, Cl, EtOCH₂, CH₃), (M-7363, Cl, H, Cl, EtOCH₂CH₂, H), (M-7364, Cl, H, Cl, EtOCH₂CH₂, Cl), (M-7365, Cl, H, Cl, EtOCH₂CH₂, F), (M-7366, Cl, H, Cl, EtOCH₂CH₂, CF₃), (M-7367, Cl, H, Cl, EtOCH₂CH₂, Br), (M-7368, Cl, H, Cl, EtOCH₂CH₂, CH₃), (M-7369, Cl, H, Cl, MeOCH₂CH₂OCH₂CH₂, H), (M-7370, Cl, H, Cl, MeOCH₂CH₂OCH₂CH₂, Cl), (M-7371, Cl, H, Cl, MeOCH₂CH₂OCH₂CH₂, F), (M-7372, Cl, H, Cl, MeOCH₂CH₂OCH₂CH₂, CF₃), (M-7373, Cl, H, Cl, MeOCH₂CH₂OCH₂CH₂, Br), (M-7374, Cl, H, Cl, MeOCH₂CH₂OCH₂CH₂, CH₃), (M-7375, Cl, H, Cl, MeOCH₂CH₂, H), (M-7376, Cl, H, Cl, MeOCH₂CH₂, Cl), (M-7377, Cl, H, Cl, MeOCH₂CH₂, F), (M-7378, Cl, H, Cl, MeOCH₂CH₂, CF₃), (M-7379, Cl, H, Cl, MeOCH₂CH₂, Br), (M-7380, Cl, H, Cl, MeOCH₂CH₂, CH₃), (M-7381, Cl, H, Cl, HOCH₂, H), (M-7382, Cl, H, Cl, HOCH₂, Cl), (M-7383, Cl, H, Cl, HOCH₂, F), (M-7384, Cl, H, Cl, HOCH₂, CF₃), (M-7385, Cl, H, Cl, HOCH₂, Br), (M-7386, Cl, H, Cl, HOCH₂, CH₃), (M-7387, Cl, H, Cl, HOCH₂CH₂, H), (M-7388, Cl, H, Cl, HOCH₂CH₂, Cl), (M-7389, Cl, H, Cl, HOCH₂CH₂, F), (M-7390, Cl, H, Cl, HOCH₂CH₂, CF₃), (M-7391, Cl, H, Cl, HOCH₂CH₂, Br), (M-7392, Cl, H, Cl, HOCH₂CH₂, CH₃), (M-7393, Cl, H, Cl, HOCH₂CH₂CH₂, H), (M-7394, Cl, H, Cl, HOCH₂CH₂CH₂, Cl), (M-7395, Cl, H, Cl, HOCH₂CH₂CH₂, F), (M-7396, Cl, H, Cl, HOCH₂CH₂CH₂, CF₃), (M-7397, Cl, H, Cl, HOCH₂CH₂CH₂, Br), (M-7398, Cl, H, Cl, HOCH₂CH₂CH₂, CH₃), (M-7399, Cl, H, Cl, HOCH₂CH₂CH₂CH₂, H), (M-7400, Cl, H, Cl, HOCH₂CH₂CH₂CH₂, Cl), (M-7401, Cl, H, Cl, HOCH₂CH₂CH₂CH₂, F), (M-7402, Cl, H, Cl, HOCH₂CH₂CH₂CH₂, CF₃), (M-7403, Cl, H, Cl, HOCH₂CH₂CH₂CH₂, Br), (M-7404, Cl, H, Cl, HOCH₂CH₂CH₂CH₂, CH₃), (M-7405, Cl, H, Cl, HOCH₂CH₂CH₂CH₂CH₂, H), (M-7406, Cl, H, Cl, HOCH₂CH₂CH₂CH₂CH₂, Cl), (M-7407, Cl, H, Cl, HOCH₂CH₂CH₂CH₂CH₂, F), (M-7408, Cl, H, Cl, HOCH₂CH₂CH₂CH₂CH₂, CF₃), (M-7409, Cl, H, Cl, HOCH₂CH₂CH₂CH₂CH₂, Br), (M-7410, Cl, H, Cl, HOCH₂CH₂CH₂CH₂CH₂, CH₃), (M-7411, Cl, H, Cl, HOCH₂CH₂OCH₂CH₂, H), (M-7412, Cl, H, Cl, HOCH₂CH₂OCH₂CH₂, Cl), (M-7413, Cl, H, Cl, HOCH₂CH₂OCH₂CH₂, F), (M-7414, Cl, H, Cl, HOCH₂CH₂OCH₂CH₂, CF₃), (M-7415, Cl, H, Cl, HOCH₂CH₂OCH₂CH₂, Br), (M-7416, Cl, H, Cl, HOCH₂CH₂OCH₂CH₂, CH₃), (M-7417, Cl, H, Cl, (Me)₂N, H), (M-7418, Cl, H, Cl, (Me)₂N, Cl), (M-7419, Cl, H, Cl, (Me)₂N, F), (M-7420, Cl, H, Cl, (Me)₂N, CF₃), (M-7421, Cl, H, Cl, (Me)₂N, Br), (M-7422, Cl, H, Cl, (Me)₂N, CH₃), (M-7423, Cl, H, Cl, piperidin-4-yl-methyl, H), (M-7424, Cl, H, Cl, piperidin-4-yl-methyl, Cl), (M-7425, Cl, H, Cl, piperidin-4-yl-methyl, F), (M-7426, Cl, H, Cl, piperidin-4-yl-methyl, CF₃), (M-7427, Cl, H, Cl, piperidin-4-yl-methyl, Br), (M-7428, Cl, H, Cl, piperidin-4-yl-methyl, CH₃), (M-7429, Cl, H, Cl, cyclohexylmethyl, H), (M-7430, Cl, H, Cl, cyclohexylmethyl, Cl), (M-7431, Cl, H, Cl, cyclohexylmethyl, F), (M-7432, Cl, H, Cl, cyclohexylmethyl, CF₃), (M-7433, Cl, H, Cl, cyclohexylmethyl, Br), (M-7434, Cl, H, Cl, cyclohexylmethyl, CH₃), (M-7435, Cl, F, H, H, H), (M-7436, Cl, F, H, H, Cl), (M-7437, Cl, F, H, H, F), (M-7438, Cl, F, H, H, CF₃), (M-7439, Cl, F, H, H, Br), (M-7440, Cl, F, H, H, CH₃), (M-7441, Cl, F, H, F, H), (M-7442, Cl, F, H, F, Cl), (M-7443, Cl, F, H, F, F), (M-7444, Cl, F, H, F, CF₃), (M-7445, Cl, F, H, F, Br), (M-7446, Cl, F, H, F, CH₃), (M-7447, Cl, F, H, Cl, H), (M-7448, Cl, F, H, Cl, Cl), (M-7449, Cl, F, H, Cl, F), (M-7450, Cl, F, H, Cl, CF₃), (M-7451, Cl, F, H, Cl, Br), (M-7452, Cl, F, H, Cl, CH₃), (M-7453, Cl, F, H, CH₃, H), (M-7454, Cl, F, H, CH₃, Cl), (M-7455, Cl, F, H, CH₃, F), (M-7456, Cl, F, H, CH₃, CF₃), (M-7457, Cl, F, H, CH₃, Br), (M-7458, Cl, F, H, CH₃, CH₃), (M-7459, Cl, F, H, Et, H), (M-7460, Cl, F, H, Et, Cl), (M-7461, Cl, F, H, Et, F), (M-7462, Cl, F, H, Et, CF₃), (M-7463, Cl, F, H, Et, Br), (M-7464, Cl, F, H, Et, CH₃), (M-7465, Cl, F, H, n-Pr, H), (M-7466, Cl, F, H, n-Pr, Cl), (M-7467, Cl, F, H, n-Pr, F), (M-7468, Cl, F, H, n-Pr, CF₃), (M-7469, Cl, F, H, n-Pr, Br), (M-7470, Cl, F, H, n-Pr, CH₃), (M-7471, Cl, F, H, c-Pr, H), (M-7472, Cl, F, H, c-Pr, Cl), (M-7473, Cl, F, H, c-Pr, F), (M-7474, Cl, F, H, c-Pr, CF₃), (M-7475, Cl, F, H, c-Pr, Br), (M-7476, Cl, F, H, c-Pr, CH₃), (M-7477, Cl, F, H, i-Pr, H), (M-7478, Cl, F, H, i-Pr, Cl), (M-7479, Cl, F, H, i-Pr, F), (M-7480, Cl, F, H, i-Pr, CF₃), (M-7481, Cl, F, H, i-Pr, Br), (M-7482, Cl, F, H, i-Pr, CH₃), (M-7483, MeO, F, H, n-Bu, H), (M-7484, Cl, F, H, n-Bu, Cl), (M-7485, Cl, F, H, n-Bu, F), (M-7486, Cl, F, H, n-Bu, CF₃), (M-7487, Cl, F, H, n-Bu, Br), (M-7488, Cl, F, H, n-Bu, CH₃), (M-7489, Cl, F, H, i-Bu, H), (M-7490, Cl, F, H, i-Bu, Cl), (M-7491, Cl, F, H, i-Bu, F), (M-7492, Cl, F, H, i-Bu, CF₃), (M-7493, Cl, F, H, i-Bu, Br), (M-7494, Cl, F, H, i-Bu, CH₃), (M-7495, Cl, F, H, sec-Bu, H), (M-7496, Cl, F, H, sec-Bu, Cl), (M-7497, Cl, F, H, sec-Bu, F), (M-7498, Cl, F, H, sec-Bu, CF₃), (M-7499, Cl, F, H, sec-Bu, Br), (M-7500, Cl, F, H, sec-Bu, CH₃), (M-7501, Cl, F, H, n-Pen, H), (M-7502, Cl, F, H, n-Pen, Cl), (M-7503, Cl, F, H, n-Pen, F), (M-7504, Cl, F, H, n-Pen, CF₃), (M-7505, Cl, F, H, n-Pen, Br), (M-7506, Cl, F, H, n-Pen, CH₃), (M-7507, Cl, F, H, c-Pen, H), (M-75
08, Cl, F, H, c-Pen, Cl), (M-7509, Cl, F, H, c-Pen, F), (M-7510, Cl, F, H, c-Pen, CF₃), (M-7511, Cl, F, H, c-Pen, Br), (M-7512, Cl, F, H, c-Pen, CH₃), (M-7513, Cl, F, H, n-Hex, H), (M-7514, Cl, F, H, n-Hex, Cl), (M-7515, Cl, F, H, n-Hex, F), (M-7516, Cl, F, H, n-Hex, CF₃), (M-7517, Cl, F, H, n-Hex, Br), (M-7518, Cl, F, H, n-Hex, CH₃), (M-7519, Cl, F, H, c-Hex, H), (M-7520, Cl, F, H, c-Hex, Cl), (M-7521, Cl, F, H, c-Hex, F), (M-7522, Cl, F, H, c-Hex, CF₃), (M-7523, Cl, F, H, c-Hex, Br), (M-7524, Cl, F, H, c-Hex, CH₃), (M-7525, Cl, F, H, OH, H), (M-7526, Cl, F, H, OH, Cl), (M-7527, Cl, F, H, OH, F), (M-7528, Cl, F, H, OH, CF₃), (M-7529, Cl, F, H, OH, Br), (M-7530, Cl, F, H, OH, CH₃), (M-7531, Cl, F, H, EtO, H), (M-7532, Cl, F, H, EtO, Cl), (M-7533, Cl, F, H, EtO, F), (M-7534, Cl, F, H, EtO, CF₃), (M-7535, Cl, F, H, EtO, Br), (M-7536, Cl, F, H, EtO, CH₃), (M-7537, Cl, F, H, n-PrO, H), (M-7538, Cl, F, H, n-PrO, Cl), (M-7539, Cl, F, H, n-PrO, F), (M-7540, Cl, F, H, n-PrO, CF₃), (M-7541, Cl, F, H, n-PrO, Br), (M-7542, Cl, F, H, n-PrO, CH₃), (M-7543, Cl, F, H, PhO, H), (M-7544, Cl, F, H, PhO, Cl), (M-7545, Cl, F, H, PhO, F), (M-7546, Cl, F, H, PhO, CF₃), (M-7547, Cl, F, H, PhO, Br), (M-7548, Cl, F, H, PhO, CH₃), (M-7549, Cl, F, H, BnO, H), (M-7550, Cl, F, H, BnO, Cl), (M-7551, Cl, F, H, BnO, F), (M-7552, Cl, F, H, BnO, CF₃), (M-7553, Cl, F, H, BnO, Br), (M-7554, Cl, F, H, BnO, CH₃), (M-7555, Cl, F, H, PhCH₂CH₂O, H), (M-7556, Cl, F, H, PhCH₂CH₂O, Cl), (M-7557, Cl, F, H, PhCH₂CH₂O, F), (M-7558, Cl, F, H, PhCH₂CH₂O, CF₃), (M-7559, Cl, F, H, PhCH₂CH₂O, Br), (M-7560, Cl, F, H, PhCH₂CH₂O, CH₃), (M-7561, Cl, F, H, CF₃O, H), (M-7562, Cl, F, H, CF₃O, Cl), (M-7563, Cl, F, H, CF₃O, F), (M-7564, Cl, F, H, CF₃O, CF₃), (M-7565, Cl, F, H, CF₃O, Br), (M-7566, Cl, F, H, CF₃O, CH₃), (M-7567, Cl, F, H, Ph, H), (M-7568, Cl, F, H, Ph, Cl), (M-7569, Cl, F, H, Ph, F), (M-7570, Cl, F, H, Ph, CF₃), (M-7571, Cl, F, H, Ph, Br), (M-7572, Cl, F, H, Ph, CH₃), (M-7573, Cl, F, H, 4-F-Ph, H), (M-7574, Cl, F, H, 4-F-Ph, Cl), (M-7575, Cl, F, H, 4-F-Ph, F), (M-7576, Cl, F, H, 4-F-Ph, CF₃), (M-7577, Cl, F, H, 4-F-Ph, Br), (M-7578, Cl, F, H, 4-F-Ph, CH₃), (M-7579, Cl, F, H, 4-CF₃-Ph, H), (M-7580, Cl, F, H, 4-CF₃-Ph, Cl), (M-7581, Cl, F, H, 4-CF₃-Ph, F), (M-7582, Cl, F, H, 4-CF₃-Ph, CF₃), (M-7583, Cl, F, H, 4-CF₃-Ph, Br), (M-7584, Cl, F, H, 4-CF₃-Ph, CH₃), (M-7585, Cl, F, H, 4-(Me)₂N-Ph, H), (M-7586, Cl, F, H, 4-(Me)₂N-Ph, Cl), (M-7587, Cl, F, H, 4-(Me)₂N-Ph, F), (M-7588, Cl, F, H, 4-(Me)₂N-Ph, CF₃), (M-7589, Cl, F, H, 4-(Me)₂N-Ph, Br), (M-7590, Cl, F, H, 4-(Me)₂N-Ph, CH₃), (M-7591, Cl, F, H, 4-OH-Ph, H), (M-7592, Cl, F, H, 4-OH-Ph, Cl), (M-7593, Cl, F, H, 4-OH-Ph, F), (M-7594, Cl, F, H, 4-OH-Ph, CF₃), (M-7595, Cl, F, H, 4-OH-Ph, Br), (M-7596, Cl, F, H, 4-OH-Ph, CH₃), (M-7597, Cl, F, H, 3,4-di-F-Ph, H), (M-7598, Cl, F, H, 3,4-di-F-Ph, Cl), (M-7599, Cl, F, H, 3,4-di-F-Ph, F), (M-7600, Cl, F, H, 3,4-di-F-Ph, CF₃), (M-7601, Cl, F, H, 3,4-di-F-Ph, Br), (M-7602, Cl, F, H, 3,4-di-F-Ph, CH₃), (M-7603, Cl, F, H, 4-COOH-Ph, H), (M-7604, Cl, F, H, 4-COOH-Ph, Cl), (M-7605, Cl, F, H, 4-COOH-Ph, F), (M-7606, Cl, F, H, 4-COOH-Ph, CF₃), (M-7607, Cl, F, H, 4-COOH-Ph, Br), (M-7608, Cl, F, H, 4-COOH-Ph, CH₃), (M-7609, Cl, F, H, Bn, H), (M-7610, Cl, F, H, Bn, Cl), (M-7611, Cl, F, H, Bn, F), (M-7612, Cl, F, H, Bn, CF₃), (M-7613, Cl, F, H, Bn, Br), (M-7614, Cl, F, H, Bn, CH₃), (M-7615, Cl, F, H, 4-F-Bn, H), (M-7616, Cl, F, H, 4-F-Bn, Cl), (M-7617, Cl, F, H, 4-F-Bn, F), (M-7618, Cl, F, H, 4-F-Bn, CF₃), (M-7619, Cl, F, H, 4-F-Bn, Br), (M-7620, Cl, F, H, 4-F-Bn, CH₃), (M-7621, Cl, F, H, 2-Py, H), (M-7622, Cl, F, H, 2-Py, Cl), (M-7623, Cl, F, H, 2-Py, F), (M-7624, Cl, F, H, 2-Py, CF₃), (M-7625, Cl, F, H, 2-Py, Br), (M-7626, Cl, F, H, 2-Py, CH₃), (M-7627, Cl, F, H, 3-Py, H), (M-7628, Cl, F, H, 3-Py, Cl), (M-7629, Cl, F, H, 3-Py, F), (M-7630, Cl, F, H, 3-Py, CF₃), (M-7631, Cl, F, H, 3-Py, Br), (M-7632, Cl, F, H, 3-Py, CH₃), (M-7633, Cl, F, H, 4-Py, H), (M-7634, Cl, F, H, 4-Py, Cl), (M-7635, Cl, F, H, 4-Py, F), (M-7636, Cl, F, H, 4-Py, CF₃), (M-7637, Cl, F, H, 4-Py, Br), (M-7638, Cl, F, H, 4-Py, CH₃), (M-7639, Cl, F, H, 2-Th, H), (M-7640, Cl, F, H, 2-Th, Cl), (M-7641, Cl, F, H, 2-Th, F), (M-7642, Cl, F, H, 2-Th, CF₃), (M-7643, Cl, F, H, 2-Th, Br), (M-7644, Cl, F, H, 2-Th, CH₃), (M-7645, Cl, F, H, 3-Th, H), (M-7646, Cl, F, H, 3-Th, Cl), (M-7647, Cl, F, H, 3-Th, F), (M-7648, Cl, F, H, 3-Th, CF₃), (M-7649, Cl, F, H, 3-Th, Br), (M-7650, Cl, F, H, 3-Th, CH₃), (M-7651, Cl, F, H, pyrazol-2-yl, H), (M-7652, Cl, F, H, pyrazol-2-yl, Cl), (M-7653, Cl, F, H, pyrazol-2-yl, F), (M-7654, Cl, F, H, pyrazol-2-yl, CF₃), (M-7655, Cl, F, H, pyrazol-2-yl, Br), (M-7656, Cl, F, H, pyrazol-2-yl, CH₃), (M-7657, Cl, F, H, pyrazol-3-yl, H), (M-7658, Cl, F, H, pyrazol-3-yl, Cl), (M-7659, Cl, F, H, pyrazol-3-yl, F), (M-7660, Cl, F, H, pyrazol-3-yl, CF₃), (M-7661, Cl, F, H, pyrazol-3-yl, Br), (M-7662, Cl, F, H, pyrazol-3-yl, CH₃), (M-7663, Cl, F, H, pyrimidin-2-yl, H), (M-7664, Cl, F, H, pyrimidin-2-yl, Cl), (M-7665, Cl, F, H, pyrimidin-2-yl, F), (M-7666, Cl, F, H, pyrimidin-2-yl, CF₃), (M-7667, Cl, F, H, pyrimidin-2-yl, Br), (M-7668, Cl, F, H, pyrimidin-2-yl, CH₃), (M-7669, Cl, F, H, pyrimidin-4-yl, H), (M-7670, Cl, F, H, pyrimidin-4-yl, Cl), (M-7671, Cl, F, H, pyrimidin-4-yl, F), (M-7672, Cl, F, H, pyrimidin-4-yl, CF₃), (M-7673, Cl, F, H, pyrimidin-4-yl, Br), (M-7674, Cl, F, H, pyrimidin-4-yl, CH₃), (M-7675, Cl, F, H, pyrimidin-5-yl, H), (M-7676, Cl, F, H, pyrimidin-5-yl, Cl), (M-7677, Cl, F, H, pyrimidin-5-yl, F), (M-7678, Cl, F, H, pyrimidin-5-yl, CF₃), (M-7679, Cl, F, H, pyrimidin-5-yl, Br), (M-7680, Cl, F, H, pyrimidin-5-yl, CH₃), (M-7681, Cl, F, H, HOOCCH₂CH₂CH₂, H), (M-7682, Cl, F, H, HOOCCH₂CH₂CH₂, Cl), (M-7683, Cl, F, H, HOOCCH₂CH₂CH₂, F), (M-7684, Cl, F, H, HOOCCH₂CH₂CH₂, CF₃), (M-7685, Cl, F, H, HOOCCH₂CH₂CH₂, Br), (M-7686, Cl, F, H, HOOCCH₂CH₂CH₂, CH₃), (M-7687, Cl, F, H, HOOCCH₂CH₂CH₂CH₂, H), (M-7688, Cl, F, H, HOOCCH₂CH₂CH₂CH₂, Cl), (M-7689, Cl, F, H, HOOCCH₂CH₂CH₂CH₂, F), (M-7690, Cl, F, H, HOOCCH₂CH₂CH₂CH₂, CF₃), (M-7691, Cl, F, H, HOOCCH₂CH₂CH₂CH₂, Br), (M-7692, Cl, F, H, HOOCCH₂CH₂CH₂CH₂, CH₃), (M-7693, Cl, F, H, (Me)₂NCOCH₂CH₂CH₂CH₂, H), (M-7694, Cl, F, H, (Me)₂NCOCH₂CH₂CH₂CH₂, Cl), (M-7695, Cl, F, H, (Me)₂NCOCH₂CH₂CH₂CH₂, F), (M-7696, Cl, F, H, (Me)₂NCOCH₂CH₂CH₂CH₂, CF₃), (M-7697, Cl, F, H, (Me)₂NCOCH₂CH₂CH₂CH₂, Br), (M-7698, Cl, F, H, (Me)₂NCOCH₂CH₂CH₂CH₂, CH₃), (M-7699, Cl, F, H, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, H), (M-7700, Cl, F, H, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, Cl), (M-7701, Cl, F, H, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, F), (M-7702, Cl, F, H, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, CF₃), (M-7703, Cl, F, H, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, Br), (M-7704, Cl, F, H, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, CH₃), (M-7705, Cl, F, H, MeOCH₂, H), (M-7706, Cl, F, H, MeOCH₂, Cl), (M-7707, Cl, F, H, MeOCH₂, F), (M-7708, Cl, F, H, MeOCH₂, CF₃), (M-7709, Cl, F, H, MeOCH₂, Br), (M-7710, Cl, F, H, MeOCH₂, CH₃), (M-7711, Cl, F, H, EtOCH₂, H), (M-7712, Cl, F, H, EtOCH₂, Cl), (M-7713, Cl, F, H, EtOCH₂, F), (M-7714, Cl, F, H, EtOCH₂, CF₃), (M-7715, Cl, F, H, EtOCH₂, Br), (M-7716, Cl, F, H, EtOCH₂, CH₃), (M-7717, Cl, F, H, EtOCH₂CH₂, H), (M-7718, Cl, F, H, EtOCH₂CH₂, Cl), (M-7719, Cl, F, H, EtOCH₂CH₂, F), (M-7720, Cl, F, H, EtOCH₂CH₂, CF₃), (M-7721, Cl, F, H, EtOCH₂CH₂, Br), (M-7722, Cl, F, H, EtOCH₂CH₂, CH₃), (M-7723, Cl, F, H, MeOCH₂CH₂OCH₂CH₂, H), (M-7724, Cl, F, H, MeOCH₂CH₂OCH₂CH₂, Cl), (M-7725, Cl, F, H, MeOCH₂CH₂OCH₂CH₂, F), (M-7726, Cl, F, H, MeOCH₂CH₂OCH₂CH₂, CF₃), (M-7727, Cl, F, H, MeO
CH₂CH₂OCH₂CH₂, Br), (M-7728, Cl, F, H, MeOCH₂CH₂OCH₂CH₂, CH₃), (M-7729, Cl, F, H, MeOCH₂CH₂, H), (M-7730, Cl, F, H, MeOCH₂CH₂, Cl), (M-7731, Cl, F, H, MeOCH₂CH₂, F), (M-7732, Cl, F, H, MeOCH₂CH₂, CF₃), (M-7733, Cl, F, H, MeOCH₂CH₂, Br), (M-7734, Cl, F, H, MeOCH₂CH₂, CH₃), (M-7735, Cl, F, H, HOCH₂, H), (M-7736, Cl, F, H, HOCH₂, Cl), (M-7737, Cl, F, H, HOCH₂, F), (M-7738, Cl, F, H, HOCH₂, CF₃), (M-7739, Cl, F, H, HOCH₂, Br), (M-7740, Cl, F, H, HOCH₂, CH₃), (M-7741, Cl, F, H, HOCH₂CH₂, H), (M-7742, Cl, F, H, HOCH₂CH₂, Cl), (M-7743, Cl, F, H, HOCH₂CH₂, F), (M-7744, Cl, F, H, HOCH₂CH₂, CF₃), (M-7745, Cl, F, H, HOCH₂CH₂, Br), (M-7746, Cl, F, H, HOCH₂CH₂, CH₃), (M-7747, Cl, F, H, HOCH₂CH₂CH₂, H), (M-7748, Cl, F, H, HOCH₂CH₂CH₂, Cl), (M-7749, Cl, F, H, HOCH₂CH₂CH₂, F), (M-7750, Cl, F, H, HOCH₂CH₂CH₂, CF₃), (M-7751, Cl, F, H, HOCH₂CH₂CH₂, Br), (M-7752, Cl, F, H, HOCH₂CH₂CH₂, CH₃), (M-7753, Cl, F, H, HOCH₂CH₂CH₂CH₂, H), (M-7754, Cl, F, H, HOCH₂CH₂CH₂CH₂, Cl), (M-7755, Cl, F, H, HOCH₂CH₂CH₂CH₂, F), (M-7756, Cl, F, H, HOCH₂CH₂CH₂CH₂, CF₃), (M-7757, Cl, F, H, HOCH₂CH₂CH₂CH₂, Br), (M-7758, Cl, F, H, HOCH₂CH₂CH₂CH₂, CH₃), (M-7759, Cl, F, H, HOCH₂CH₂CH₂CH₂CH₂, H), (M-7760, Cl, F, H, HOCH₂CH₂CH₂CH₂CH₂, Cl), (M-7761, Cl, F, H, HOCH₂CH₂CH₂CH₂CH₂, F), (M-7762, Cl, F, H, HOCH₂CH₂CH₂CH₂CH₂, CF₃), (M-7763, Cl, F, H, HOCH₂CH₂CH₂CH₂CH₂, Br), (M-7764, Cl, F, H, HOCH₂CH₂CH₂CH₂CH₂, CH₃), (M-7765, Cl, F, H, HOCH₂CH₂OCH₂CH₂, H), (M-7766, Cl, F, H, HOCH₂CH₂OCH₂CH₂, Cl), (M-7767, Cl, F, H, HOCH₂CH₂OCH₂CH₂, F), (M-7768, Cl, F, H, HOCH₂CH₂OCH₂CH₂, CF₃), (M-7769, Cl, F, H, HOCH₂CH₂OCH₂CH₂, Br), (M-7770, Cl, F, H, HOCH₂CH₂OCH₂CH₂, CH₃), (M-7771, Cl, F, H, (Me)₂N, H), (M-7772, Cl, F, H, (Me)₂N, Cl), (M-7773, Cl, F, H, (Me)₂N, F), (M-7774, Cl, F, H, (Me)₂N, CF₃), (M-7775, Cl, F, H, (Me)₂N, Br), (M-7776, Cl, F, H, (Me)₂N, CH₃), (M-7777, Cl, F, H, piperidin-4-yl-methyl, H), (M-7778, Cl, F, H, piperidin-4-yl-methyl, Cl), (M-7779, Cl, F, H, piperidin-4-yl-methyl, F), (M-7780, Cl, F, H, piperidin-4-yl-methyl, CF₃), (M-7781, Cl, F, H, piperidin-4-yl-methyl, Br), (M-7782, Cl, F, H, piperidin-4-yl-methyl, CH₃), (M-7783, Cl, F, H, cyclohexylmethyl, H), (M-7784, Cl, F, H, cyclohexylmethyl, Cl), (M-7785, Cl, F, H, cyclohexylmethyl, F), (M-7786, Cl, F, H, cyclohexylmethyl, CF₃), (M-7787, Cl, F, H, cyclohexylmethyl, Br), (M-7788, Cl, F, H, cyclohexylmethyl, CH₃), (M-7789, Cl, F, F, H, H), (M-7790, Cl, F, F, H, Cl), (M-7791, Cl, F, F, H, F), (M-7792, Cl, F, F, H, CF₃), (M-7793, Cl, F, F, H, Br), (M-7794, Cl, F, F, H, CH₃), (M-7795, Cl, F, F, F, H), (M-7796, Cl, F, F, F, Cl), (M-7797, Cl, F, F, F, F), (M-7798, Cl, F, F, F, CF₃), (M-7799, Cl, F, F, F, Br), (M-7800, Cl, F, F, F, CH₃), (M-7801, Cl, F, F, Cl, H), (M-7802, Cl, F, F, Cl, Cl), (M-7803, Cl, F, F, Cl, F), (M-7804, Cl, F, F, Cl, CF₃), (M-7805, Cl, F, F, Cl, Br), (M-7806, Cl, F, F, Cl, CH₃), (M-7807, Cl, F, F, CH₃, H), (M-7808, Cl, F, F, CH₃, Cl), (M-7809, Cl, F, F, CH₃, F), (M-7810, Cl, F, F, CH₃, CF₃), (M-7811, Cl, F, F, CH₃, Br), (M-7812, Cl, F, F, CH₃, CH₃), (M-7813, Cl, F, F, Et, H), (M-7814, Cl, F, F, Et, Cl), (M-7815, Cl, F, F, Et, F), (M-7816, Cl, F, F, Et, CF₃), (M-7817, Cl, F, F, Et, Br), (M-7818, Cl, F, F, Et, CH₃), (M-7819, Cl, F, F, n-Pr, H), (M-7820, Cl, F, F, n-Pr, Cl), (M-7821, Cl, F, F, n-Pr, F), (M-7822, Cl, F, F, n-Pr, CF₃), (M-7823, Cl, F, F, n-Pr, Br), (M-7824, Cl, F, F, n-Pr, CH₃), (M-7825, Cl, F, F, c-Pr, H), (M-7826, Cl, F, F, c-Pr, Cl), (M-7827, Cl, F, F, c-Pr, F), (M-7828, Cl, F, F, c-Pr, CF₃), (M-7829, Cl, F, F, c-Pr, Br), (M-7830, Cl, F, F, c-Pr, CH₃), (M-7831, Cl, F, F, i-Pr, H), (M-7832, Cl, F, F, i-Pr, Cl), (M-7833, Cl, F, F, i-Pr, F), (M-7834, Cl, F, F, i-Pr, CF₃), (M-7835, Cl, F, F, i-Pr, Br), (M-7836, Cl, F, F, i-Pr, CH₃), (M-7837, Cl, F, F, n-Bu, H), (M-7838, Cl, F, F, n-Bu, Cl), (M-7839, Cl, F, F, n-Bu, F), (M-7840, Cl, F, F, n-Bu, CF₃), (M-7841, Cl, F, F, n-Bu, Br), (M-7842, Cl, F, F, n-Bu, CH₃), (M-7843, Cl, F, F, i-Bu, H), (M-7844, Cl, F, F, i-Bu, Cl), (M-7845, Cl, F, F, i-Bu, F), (M-7846, Cl, F, F, i-Bu, CF₃), (M-7847, Cl, F, F, i-Bu, Br), (M-7848, Cl, F, F, i-Bu, CH₃), (M-7849, Cl, F, F, sec-Bu, H), (M-7850, Cl, F, F, sec-Bu, Cl), (M-7851, Cl, F, F, sec-Bu, F), (M-7852, Cl, F, F, sec-Bu, CF₃), (M-7853, Cl, F, F, sec-Bu, Br), (M-7854, Cl, F, F, sec-Bu, CH₃), (M-7855, Cl, F, F, n-Pen, H), (M-7856, Cl, F, F, n-Pen, Cl), (M-7857, Cl, F, F, n-Pen, F), (M-7858, Cl, F, F, n-Pen, CF₃), (M-7859, Cl, F, F, n-Pen, Br), (M-7860, Cl, F, F, n-Pen, CH₃), (M-7861, Cl, F, F, c-Pen, H), (M-7862, Cl, F, F, c-Pen, Cl), (M-7863, Cl, F, F, c-Pen, F), (M-7864, Cl, F, F, c-Pen, CF₃), (M-7865, Cl, F, F, c-Pen, Br), (M-7866, Cl, F, F, c-Pen, CH₃), (M-7867, Cl, F, F, n-Hex, H), (M-7868, Cl, F, F, n-Hex, Cl), (M-7869, Cl, F, F, n-Hex, F), (M-7870, Cl, F, F, n-Hex, CF₃), (M-7871, Cl, F, F, n-Hex, Br), (M-7872, Cl, F, F, n-Hex, CH₃), (M-7873, Cl, F, F, c-Hex, H), (M-7874, Cl, F, F, c-Hex, Cl), (M-7875, Cl, F, F, c-Hex, F), (M-7876, Cl, F, F, c-Hex, CF₃), (M-7877, Cl, F, F, c-Hex, Br), (M-7878, Cl, F, F, c-Hex, CH₃), (M-7879, Cl, F, F, OH, H), (M-7880, Cl, F, F, OH, Cl), (M-7881, Cl, F, F, OH, F), (M-7882, Cl, F, F, OH, CF₃), (M-7883, Cl, F, F, OH, Br), (M-7884, Cl, F, F, OH, CH₃), (M-7885, Cl, F, F, EtO, H), (M-7886, Cl, F, F, EtO, Cl), (M-7887, Cl, F, F, EtO, F), (M-7888, Cl, F, F, EtO, CF₃), (M-7889, Cl, F, F, EtO, Br), (M-7890, Cl, F, F, EtO, CH₃), (M-7891, Cl, F, F, n-PrO, H), (M-7892, Cl, F, F, n-PrO, Cl), (M-7893, Cl, F, F, n-PrO, F), (M-7894, Cl, F, F, n-PrO, CF₃), (M-7895, Cl, F, F, n-PrO, Br), (M-7896, Cl, F, F, n-PrO, CH₃), (M-7897, Cl, F, F, PhO, H), (M-7898, Cl, F, F, PhO, Cl), (M-7899, Cl, F, F, PhO, F), (M-7900, Cl, F, F, PhO, CF₃), (M-7901, Cl, F, F, PhO, Br), (M-7902, Cl, F, F, PhO, CH₃), (M-7903, Cl, F, F, BnO, H), (M-7904, Cl, F, F, BnO, Cl), (M-7905, Cl, F, F, BnO, F), (M-7906, Cl, F, F, BnO, CF₃), (M-7907, Cl, F, F, BnO, Br), (M-7908, Cl, F, F, BnO, CH₃), (M-7909, Cl, F, F, PhCH₂CH₂O, H), (M-7910, Cl, F, F, PhCH₂CH₂O, Cl), (M-7911, Cl, F, F, PhCH₂CH₂O, F), (M-7912, Cl, F, F, PhCH₂CH₂O, CF₃), (M-7913, Cl, F, F, PhCH₂CH₂O, Br), (M-7914, Cl, F, F, PhCH₂CH₂O, CH₃), (M-7915, Cl, F, F, CF₃O, H), (M-7916, Cl, F, F, CF₃O, Cl), (M-7917, Cl, F, F, CF₃O, F), (M-7918, Cl, F, F, CF₃O, CF₃), (M-7919, Cl, F, F, CF₃O, Br), (M-7920, Cl, F, F, CF₃O, CH₃), (M-7921, Cl, F, F, Ph, H), (M-7922, Cl, F, F, Ph, Cl), (M-7923, Cl, F, F, Ph, F), (M-7924, Cl, F, F, Ph, CF₃), (M-7925, Cl, F, F, Ph, Br), (M-7926, Cl, F, F, Ph, CH₃), (M-7927, Cl, F, F, 4-F-Ph, H), (M-7928, Cl, F, F, 4-F-Ph, Cl), (M-7929, Cl, F, F, 4-F-Ph, F), (M-7930, Cl, F, F, 4-F-Ph, CF₃), (M-7931, Cl, F, F, 4-F-Ph, Br), (M-7932, Cl, F, F, 4-F-Ph, CH₃), (M-7933, Cl, F, F, 4-CF₃-Ph, H), (M-7934, Cl, F, F, 4-CF₃-Ph, Cl), (M-7935, Cl, F, F, 4-CF₃-Ph, F), (M-7936, Cl, F, F, 4-CF₃-Ph, CF₃), (M-7937, Cl, F, F, 4-CF₃-Ph, Br), (M-7938, Cl, F, F, 4-CF₃-Ph, CH₃), (M-7939, Cl, F, F, 4-(Me)₂N-Ph, H), (M-7940, Cl, F, F, 4-(Me)₂N-Ph, Cl), (M-7941, Cl, F, F, 4-(Me)₂N-Ph, F), (M-7942, Cl, F, F, 4-(Me)₂N-Ph, CF₃), (M-7943, Cl, F, F, 4-(Me)₂N-Ph, Br), (M-7944, Cl, F, F, 4-(Me)₂N-Ph, CH₃), (M-7945, Cl, F, F, 4-OH-Ph, H), (M-7946, Cl, F, F, 4-OH-Ph, Cl), (M-7947, Cl, F, F, 4-OH-Ph, F), (M-7948, Cl, F, F, 4-OH-Ph, CF₃), (M-7949, Cl, F, F, 4-OH-Ph, Br), (M-7950, Cl, F, F, 4-OH-Ph, CH₃), (M-7951, Cl, F, F, 3,4-di-F-Ph, H), (M-7952, Cl, F, F, 3,4-di-F-Ph, Cl), (M-7953, Cl, F, F, 3,4-di-F-Ph, F), (M-7954, Cl, F, F, 3,4-di-F-Ph, CF₃), (M-7955, Cl, F, F, 3,4-di-F-Ph, Br), (M-7956, C
l, F, F, 3,4-di-F-Ph, CH₃), (M-7957, Cl, F, F, 4-COOH-Ph, H), (M-7958, Cl, F, F, 4-COOH-Ph, Cl), (M-7959, Cl, F, F, 4-COOH-Ph, F), (M-7960, Cl, F, F, 4-COOH-Ph, CF₃), (M-7961, Cl, F, F, 4-COOH-Ph, Br), (M-7962, Cl, F, F, 4-COOH-Ph, CH₃), (M-7963, Cl, F, F, Bn, H), (M-7964, Cl, F, F, Bn, Cl), (M-7965, Cl, F, F, Bn, F), (M-7966, Cl, F, F, Bn, CF₃), (M-7967, Cl, F, F, Bn, Br), (M-7968, Cl, F, F, Bn, CH₃), (M-7969, Cl, F, F, 4-F-Bn, H), (M-7970, Cl, F, F, 4-F-Bn, Cl), (M-7971, Cl, F, F, 4-F-Bn, F), (M-7972, Cl, F, F, 4-F-Bn, CF₃), (M-7973, Cl, F, F, 4-F-Bn, Br), (M-7974, Cl, F, F, 4-F-Bn, CH₃), (M-7975, Cl, F, F, 2-Py, H), (M-7976, Cl, F, F, 2-Py, Cl), (M-7977, Cl, F, F, 2-Py, F), (M-7978, Cl, F, F, 2-Py, CF₃), (M-7979, Cl, F, F, 2-Py, Br), (M-7980, Cl, F, F, 2-Py, CH₃), (M-7981, Cl, F, F, 3-Py, H), (M-7982, Cl, F, F, 3-Py, Cl), (M-7983, Cl, F, F, 3-Py, F), (M-7984, Cl, F, F, 3-Py, CF₃), (M-7985, Cl, F, F, 3-Py, Br), (M-7986, Cl, F, F, 3-Py, CH₃), (M-7987, Cl, F, F, 4-Py, H), (M-7988, Cl, F, F, 4-Py, Cl), (M-7989, Cl, F, F, 4-Py, F), (M-7990, Cl, F, F, 4-Py, CF₃), (M-7991, Cl, F, F, 4-Py, Br), (M-7992, Cl, F, F, 4-Py, CH₃), (M-7993, Cl, F, F, 2-Th, H), (M-7994, Cl, F, F, 2-Th, Cl), (M-7995, Cl, F, F, 2-Th, F), (M-7996, Cl, F, F, 2-Th, CF₃), (M-7997, Cl, F, F, 2-Th, Br), (M-7998, Cl, F, F, 2-Th, CH₃), (M-7999, Cl, F, F, 3-Th, H), (M-8000, Cl, F, F, 3-Th, Cl), (M-8001, Cl, F, F, 3-Th, F), (M-8002, Cl, F, F, 3-Th, CF₃), (M-8003, Cl, F, F, 3-Th, Br), (M-8004, Cl, F, F, 3-Th, CH₃), (M-8005, Cl, F, F, pyrazol-2-yl, H), (M-8006, Cl, F, F, pyrazol-2-yl, Cl), (M-8007, Cl, F, F, pyrazol-2-yl, F), (M-8008, Cl, F, F, pyrazol-2-yl, CF₃), (M-8009, Cl, F, F, pyrazol-2-yl, Br), (M-8010, Cl, F, F, pyrazol-2-yl, CH₃), (M-8011, Cl, F, F, pyrazol-3-yl, H), (M-8012, Cl, F, F, pyrazol-3-yl, Cl), (M-8013, Cl, F, F, pyrazol-3-yl, F), (M-8014, Cl, F, F, pyrazol-3-yl, CF₃), (M-8015, Cl, F, F, pyrazol-3-yl, Br), (M-8016, Cl, F, F, pyrazol-3-yl, CH₃), (M-8017, Cl, F, F, pyrimidin-2-yl, H), (M-8018, Cl, F, F, pyrimidin-2-yl, Cl), (M-8019, Cl, F, F, pyrimidin-2-yl, F), (M-8020, Cl, F, F, pyrimidin-2-yl, CF₃), (M-8021, Cl, F, F, pyrimidin-2-yl, Br), (M-8022, Cl, F, F, pyrimidin-2-yl, CH₃), (M-8023, Cl, F, F, pyrimidin-4-yl, H), (M-8024, Cl, F, F, pyrimidin-4-yl, Cl), (M-8025, Cl, F, F, pyrimidin-4-yl, F), (M-8026, Cl, F, F, pyrimidin-4-yl, CF₃), (M-8027, Cl, F, F, pyrimidin-4-yl, Br), (M-8028, Cl, F, F, pyrimidin-4-yl, CH₃), (M-8029, Cl, F, F, pyrimidin-5-yl, H), (M-8030, Cl, F, F, pyrimidin-5-yl, Cl), (M-8031, Cl, F, F, pyrimidin-5-yl, F), (M-8032, Cl, F, F, pyrimidin-5-yl, CF₃), (M-8033, Cl, F, F, pyrimidin-5-yl, Br), (M-8034, Cl, F, F, pyrimidin-5-yl, CH₃), (M-8035, Cl, F, F, HOOCCH₂CH₂CH₂, H), (M-8036, Cl, F, F, HOOCCH₂CH₂CH₂, Cl), (M-8037, Cl, F, F, HOOCCH₂CH₂CH₂, F), (M-8038, Cl, F, F, HOOCCH₂CH₂CH₂, CF₃), (M-8039, Cl, F, F, HOOCCH₂CH₂CH₂, Br), (M-8040, Cl, F, F, HOOCCH₂CH₂CH₂, CH₃), (M-8041, Cl, F, F, HOOCCH₂CH₂CH₂CH₂, H), (M-8042, Cl, F, F, HOOCCH₂CH₂CH₂CH₂, Cl), (M-8043, Cl, F, F, HOOCCH₂CH₂CH₂CH₂, F), (M-8044, Cl, F, F, HOOCCH₂CH₂CH₂CH₂, CF₃), (M-8045, Cl, F, F, HOOCCH₂CH₂CH₂CH₂, Br), (M-8046, Cl, F, F, HOOCCH₂CH₂CH₂CH₂, CH₃), (M-8047, Cl, F, F, (Me)₂NCOCH₂CH₂CH₂CH₂, H), (M-8048, Cl, F, F, (Me)₂NCOCH₂CH₂CH₂CH₂, Cl), (M-8049, Cl, F, F, (Me)₂NCOCH₂CH₂CH₂CH₂, F), (M-8050, Cl, F, F, (Me)₂NCOCH₂CH₂CH₂CH₂, CF₃), (M-8051, Cl, F, F, (Me)₂NCOCH₂CH₂CH₂CH₂, Br), (M-8052, Cl, F, F, (Me)₂NCOCH₂CH₂CH₂CH₂, CH₃), (M-8053, Cl, F, F, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, H), (M-8054, Cl, F, F, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, Cl), (M-8055, Cl, F, F, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, F), (M-8056, Cl, F, F, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, CF₃), (M-8057, Cl, F, F, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, Br), (M-8058, Cl, F, F, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, CH₃), (M-8059, Cl, F, F, MeOCH₂, H), (M-8060, Cl, F, F, MeOCH₂, Cl), (M-8061, Cl, F, F, MeOCH₂, F), (M-8062, Cl, F, F, MeOCH₂, CF₃), (M-8063, Cl, F, F, MeOCH₂, Br), (M-8064, Cl, F, F, MeOCH₂, CH₃), (M-8065, Cl, F, F, EtOCH₂, H), (M-8066, Cl, F, F, EtOCH₂, Cl), (M-8067, Cl, F, F, EtOCH₂, F), (M-8068, Cl, F, F, EtOCH₂, CF₃), (M-8069, Cl, F, F, EtOCH₂, Br), (M-8070, Cl, F, F, EtOCH₂, CH₃), (M-8071, Cl, F, F, EtOCH₂CH₂, H), (M-8072, Cl, F, F, EtOCH₂CH₂, Cl), (M-8073, Cl, F, F, EtOCH₂CH₂, F), (M-8074, Cl, F, F, EtOCH₂CH₂, CF₃), (M-8075, Cl, F, F, EtOCH₂CH₂, Br), (M-8076, Cl, F, F, EtOCH₂CH₂, CH₃), (M-8077, Cl, F, F, MeOCH₂CH₂OCH₂CH₂, H), (M-8078, Cl, F, F, MeOCH₂CH₂OCH₂CH₂, Cl), (M-8079, Cl, F, F, MeOCH₂CH₂OCH₂CH₂, F), (M-8080, Cl, F, F, MeOCH₂CH₂OCH₂CH₂, CF₃), (M-8081, Cl, F, F, MeOCH₂CH₂OCH₂CH₂, Br), (M-8082, Cl, F, F, MeOCH₂CH₂OCH₂CH₂, CH₃), (M-8083, Cl, F, F, MeOCH₂CH₂, H), (M-8084, Cl, F, F, MeOCH₂CH₂, Cl), (M-8085, Cl, F, F, MeOCH₂CH₂, F), (M-8086, Cl, F, F, MeOCH₂CH₂, CF₃), (M-8087, Cl, F, F, MeOCH₂CH₂, Br), (M-8088, Cl, F, F, MeOCH₂CH₂, CH₃), (M-8089, Cl, F, F, HOCH₂, H), (M-8090, Cl, F, F, HOCH₂, Cl), (M-8091, Cl, F, F, HOCH₂, F), (M-8092, Cl, F, F, HOCH₂, CF₃), (M-8093, Cl, F, F, HOCH₂, Br), (M-8094, Cl, F, F, HOCH₂, CH₃), (M-8095, Cl, F, F, HOCH₂CH₂, H), (M-8096, Cl, F, F, HOCH₂CH₂, Cl), (M-8097, Cl, F, F, HOCH₂CH₂, F), (M-8098, Cl, F, F, HOCH₂CH₂, CF₃), (M-8099, Cl, F, F, HOCH₂CH₂, Br), (M-8100, Cl, F, F, HOCH₂CH₂, CH₃), (M-8101, Cl, F, F, HOCH₂CH₂CH₂, H), (M-8102, Cl, F, F, HOCH₂CH₂CH₂, Cl), (M-8103, Cl, F, F, HOCH₂CH₂CH₂, F), (M-8104, Cl, F, F, HOCH₂CH₂CH₂, CF₃), (M-8105, Cl, F, F, HOCH₂CH₂CH₂, Br), (M-8106, Cl, F, F, HOCH₂CH₂CH₂, CH₃), (M-8107, Cl, F, F, HOCH₂CH₂CH₂CH₂, H), (M-8108, Cl, F, F, HOCH₂CH₂CH₂CH₂, Cl), (M-8109, Cl, F, F, HOCH₂CH₂CH₂CH₂, F), (M-8110, Cl, F, F, HOCH₂CH₂CH₂CH₂, CF₃), (M-8111, Cl, F, F, HOCH₂CH₂CH₂CH₂, Br), (M-8112, Cl, F, F, HOCH₂CH₂CH₂CH₂, CH₃), (M-8113, Cl, F, F, HOCH₂CH₂CH₂CH₂CH₂, H), (M-8114, Cl, F, F, HOCH₂CH₂CH₂CH₂CH₂, Cl), (M-8115, Cl, F, F, HOCH₂CH₂CH₂CH₂CH₂, F), (M-8116, Cl, F, F, HOCH₂CH₂CH₂CH₂CH₂, CF₃), (M-8117, Cl, F, F, HOCH₂CH₂CH₂CH₂CH₂, Br), (M-8118, Cl, F, F, HOCH₂CH₂CH₂CH₂CH₂, CH₃), (M-8119, Cl, F, F, HOCH₂CH₂OCH₂CH₂, H), (M-8120, Cl, F, F, HOCH₂CH₂OCH₂CH₂, Cl), (M-8121, Cl, F, F, HOCH₂CH₂OCH₂CH₂, F), (M-8122, Cl, F, F, HOCH₂CH₂OCH₂CH₂, CF₃), (M-8123, Cl, F, F, HOCH₂CH₂OCH₂CH₂, Br), (M-8124, Cl, F, F, HOCH₂CH₂OCH₂CH₂, CH₃), (M-8125, Cl, F, F, (Me)₂N, H), (M-8126, Cl, F, F, (Me)₂N, Cl), (M-8127, Cl, F, F, (Me)₂N, F), (M-8128, Cl, F, F, (Me)₂N, CF₃), (M-8129, Cl, F, F, (Me)₂N, Br), (M-8130, Cl, F, F, (Me)₂N, CH₃), (M-8131, Cl, F, F, piperidin-4-yl-methyl, H), (M-8132, Cl, F, F, piperidin-4-yl-methyl, Cl
), (M-8133, Cl, F, F, piperidin-4-yl-methyl, F), (M-8134, Cl, F, F, piperidin-4-yl-methyl, CF₃), (M-8135, Cl, F, F, piperidin-4-yl-methyl, Br), (M-8136, Cl, F, F, piperidin-4-yl-methyl, CH₃), (M-8137, Cl, F, F, cyclohexylmethyl, H), (M-8138, Cl, F, F, cyclohexylmethyl, Cl), (M-8139, Cl, F, F, cyclohexylmethyl, F), (M-8140, Cl, F, F, cyclohexylmethyl, CF₃), (M-8141, Cl, F, F, cyclohexylmethyl, Br), (M-8142, Cl, F, F, cyclohexylmethyl, CH₃), (M-8143, Cl, F, Cl, H, H), (M-8144, Cl, F, Cl, H, Cl), (M-8145, Cl, F, Cl, H, F), (M-8146, Cl, F, Cl, H, CF₃), (M-8147, Cl, F, Cl, H, Br), (M-8148, Cl, F, Cl, H, CH₃), (M-8149, Cl, F, Cl, F, H), (M-8150, Cl, F, Cl, F, Cl), (M-8151, Cl, F, Cl, F, F), (M-8152, Cl, F, Cl, F, CF₃), (M-8153, Cl, F, Cl, F, Br), (M-8154, Cl, F, Cl, F, CH₃), (M-8155, Cl, F, Cl, Cl, H), (M-8156, Cl, F, Cl, Cl, Cl), (M-8157, Cl, F, Cl, Cl, F), (M-8158, Cl, F, Cl, Cl, CF₃), (M-8159, Cl, F, Cl, Cl, Br), (M-8160, Cl, F, Cl, Cl, CH₃), (M-8161, Cl, F, Cl, CH₃, H), (M-8162, Cl, F, Cl, CH₃, Cl), (M-8163, Cl, F, Cl, CH₃, F), (M-8164, Cl, F, Cl, CH₃, CF₃), (M-8165, Cl, F, Cl, CH₃, Br), (M-8166, Cl, F, Cl, CH₃, CH₃), (M-8167, Cl, F, Cl, Et, H), (M-8168, Cl, F, Cl, Et, Cl), (M-8169, Cl, F, Cl, Et, F), (M-8170, Cl, F, Cl, Et, CF₃), (M-8171, Cl, F, Cl, Et, Br), (M-8172, Cl, F, Cl, Et, CH₃), (M-8173, Cl, F, Cl, n-Pr, H), (M-8174, Cl, F, Cl, n-Pr, Cl), (M-8175, Cl, F, Cl, n-Pr, F), (M-8176, Cl, F, Cl, n-Pr, CF₃), (M-8177, Cl, F, Cl, n-Pr, Br), (M-8178, Cl, F, Cl, n-Pr, CH₃), (M-8179, Cl, F, Cl, c-Pr, H), (M-8180, Cl, F, Cl, c-Pr, Cl), (M-8181, Cl, F, Cl, c-Pr, F), (M-8182, Cl, F, Cl, c-Pr, CF₃), (M-8183, Cl, F, Cl, c-Pr, Br), (M-8184, Cl, F, Cl, c-Pr, CH₃), (M-8185, Cl, F, Cl, i-Pr, H), (M-8186, Cl, F, Cl, i-Pr, Cl), (M-8187, Cl, F, Cl, i-Pr, F), (M-8188, Cl, F, Cl, i-Pr, CF₃), (M-8189, Cl, F, Cl, i-Pr, Br), (M-8190, Cl, F, Cl, i-Pr, CH₃), (M-8191, Cl, F, Cl, n-Bu, H), (M-8192, Cl, F, Cl, n-Bu, Cl), (M-8193, Cl, F, Cl, n-Bu, F), (M-8194, Cl, F, Cl, n-Bu, CF₃), (M-8195, Cl, F, Cl, n-Bu, Br), (M-8196, Cl, F, Cl, n-Bu, CH₃), (M-8197, Cl, F, Cl, i-Bu, H), (M-8198, Cl, F, Cl, i-Bu, Cl), (M-8199, Cl, F, Cl, i-Bu, F), (M-8200, Cl, F, Cl, i-Bu, CF₃), (M-8201, Cl, F, Cl, i-Bu, Br), (M-8202, Cl, F, Cl, i-Bu, CH₃), (M-8203, Cl, F, Cl, sec-Bu, H), (M-8204, Cl, F, Cl, sec-Bu, Cl), (M-8205, Cl, F, Cl, sec-Bu, F), (M-8206, Cl, F, Cl, sec-Bu, CF₃), (M-8207, Cl, F, Cl, sec-Bu, Br), (M-8208, Cl, F, Cl, sec-Bu, CH₃), (M-8209, Cl, F, Cl, n-Pen, H), (M-8210, Cl, F, Cl, n-Pen, Cl), (M-8211, Cl, F, Cl, n-Pen, F), (M-8212, Cl, F, Cl, n-Pen, CF₃), (M-8213, Cl, F, Cl, n-Pen, Br), (M-8214, Cl, F, Cl, n-Pen, CH₃), (M-8215, Cl, F, Cl, c-Pen, H), (M-8216, Cl, F, Cl, c-Pen, Cl), (M-8217, Cl, F, Cl, c-Pen, F), (M-8218, Cl, F, Cl, c-Pen, CF₃), (M-8219, Cl, F, Cl, c-Pen, Br), (M-8220, Cl, F, Cl, c-Pen, CH₃), (M-8221, Cl, F, Cl, n-Hex, H), (M-8222, Cl, F, Cl, n-Hex, Cl), (M-8223, Cl, F, Cl, n-Hex, F), (M-8224, Cl, F, Cl, n-Hex, CF₃), (M-8225, Cl, F, Cl, n-Hex, Br), (M-8226, Cl, F, Cl, n-Hex, CH₃), (M-8227, Cl, F, Cl, c-Hex, H), (M-8228, Cl, F, Cl, c-Hex, Cl), (M-8229, Cl, F, Cl, c-Hex, F), (M-8230, Cl, F, Cl, c-Hex, CF₃), (M-8231, Cl, F, Cl, c-Hex, Br), (M-8232, Cl, F, Cl, c-Hex, CH₃), (M-8233, Cl, F, Cl, OH, H), (M-8234, Cl, F, Cl, OH, Cl), (M-8235, Cl, F, Cl, OH, F), (M-8236, Cl, F, Cl, OH, CF₃), (M-8237, Cl, F, Cl, OH, Br), (M-8238, Cl, F, Cl, OH, CH₃), (M-8239, Cl, F, Cl, EtO, H), (M-8240, Cl, F, Cl, EtO, Cl), (M-8241, Cl, F, Cl, EtO, F), (M-8242, Cl, F, Cl, EtO, CF₃), (M-8243, Cl, F, Cl, EtO, Br), (M-8244, Cl, F, Cl, EtO, CH₃), (M-8245, Cl, F, Cl, n-PrO, H), (M-8246, Cl, F, Cl, n-PrO, Cl), (M-8247, Cl, F, Cl, n-PrO, F), (M-8248, Cl, F, Cl, n-PrO, CF₃), (M-8249, Cl, F, Cl, n-PrO, Br), (M-8250, Cl, F, Cl, n-PrO, CH₃), (M-8251, Cl, F, Cl, PhO, H), (M-8252, Cl, F, Cl, PhO, Cl), (M-8253, Cl, F, Cl, PhO, F), (M-8254, Cl, F, Cl, PhO, CF₃), (M-8255, Cl, F, Cl, PhO, Br), (M-8256, Cl, F, Cl, PhO, CH₃), (M-8257, Cl, F, Cl, BnO, H), (M-8258, Cl, F, Cl, BnO, Cl), (M-8259, Cl, F, Cl, BnO, F), (M-8260, Cl, F, Cl, BnO, CF₃), (M-8261, Cl, F, Cl, BnO, Br), (M-8262, Cl, F, Cl, BnO, CH₃), (M-8263, Cl, F, Cl, PhCH₂CH₂O, H), (M-8264, Cl, F, Cl, PhCH₂CH₂O, Cl), (M-8265, Cl, F, Cl, PhCH₂CH₂O, F), (M-8266, Cl, F, Cl, PhCH₂CH₂O, CF₃), (M-8267, Cl, F, Cl, PhCH₂CH₂O, Br), (M-8268, Cl, F, Cl, PhCH₂CH₂O, CH₃), (M-8269, Cl, F, Cl, CF₃O, H), (M-8270, Cl, F, Cl, CF₃O, Cl), (M-8271, Cl, F, Cl, CF₃O, F), (M-8272, Cl, F, Cl, CF₃O, CF₃), (M-8273, Cl, F, Cl, CF₃O, Br), (M-8274, Cl, F, Cl, CF₃O, CH₃), (M-8275, Cl, F, Cl, Ph, H), (M-8276, Cl, F, Cl, Ph, Cl), (M-8277, Cl, F, Cl, Ph, F), (M-8278, Cl, F, Cl, Ph, CF₃), (M-8279, Cl, F, Cl, Ph, Br), (M-8280, Cl, F, Cl, Ph, CH₃), (M-8281, Cl, F, Cl, 4-F-Ph, H), (M-8282, Cl, F, Cl, 4-F-Ph, Cl), (M-8283, Cl, F, Cl, 4-F-Ph, F), (M-8284, Cl, F, Cl, 4-F-Ph, CF₃), (M-8285, Cl, F, Cl, 4-F-Ph, Br), (M-8286, Cl, F, Cl, 4-F-Ph, CH₃), (M-8287, Cl, F, Cl, 4-CF₃-Ph, H), (M-8288, Cl, F, Cl, 4-CF₃-Ph, Cl), (M-8289, Cl, F, Cl, 4-CF₃-Ph, F), (M-8290, Cl, F, Cl, 4-CF₃-Ph, CF₃), (M-8291, Cl, F, Cl, 4-CF₃-Ph, Br), (M-8292, Cl, F, Cl, 4-CF₃-Ph, CH₃), (M-8293, Cl, F, Cl, 4-(Me)₂N-Ph, H), (M-8294, Cl, F, Cl, 4-(Me)₂N-Ph, Cl), (M-8295, Cl, F, Cl, 4-(Me)₂N-Ph, F), (M-8296, Cl, F, Cl, 4-(Me)₂N-Ph, CF₃), (M-8297, Cl, F, Cl, 4-(Me)₂N-Ph, Br), (M-8298, Cl, F, Cl, 4-(Me)₂N-Ph, CH₃), (M-8299, Cl, F, Cl, 4-OH-Ph, H), (M-8300, Cl, F, Cl, 4-OH-Ph, Cl), (M-8301, Cl, F, Cl, 4-OH-Ph, F), (M-8302, Cl, F, Cl, 4-OH-Ph, CF₃), (M-8303, Cl, F, Cl, 4-OH-Ph, Br), (M-8304, Cl, F, Cl, 4-OH-Ph, CH₃), (M-8305, Cl, F, Cl, 3,4-di-F-Ph, H), (M-8306, Cl, F, Cl, 3,4-di-F-Ph, Cl), (M-8307, Cl, F, Cl, 3,4-di-F-Ph, F), (M-8308, Cl, F, Cl, 3,4-di-F-Ph, CF₃), (M-8309, Cl, F, Cl, 3,4-di-F-Ph, Br), (M-8310, Cl, F, Cl, 3,4-di-F-Ph, CH₃), (M-8311, Cl, F, Cl, 4-COOH-Ph, H), (M-8312, Cl, F, Cl, 4-COOH-Ph, Cl), (M-8313, Cl, F, Cl, 4-COOH-Ph, F), (M-8314, Cl, F, Cl, 4-COOH-Ph, CF₃), (M-8315, Cl, F, Cl, 4-COOH-Ph, Br), (M-8316, Cl, F, Cl, 4-COOH-Ph, CH₃), (M-8317, Cl, F, Cl, Bn, H), (M-8318, Cl, F, Cl, Bn, Cl), (M-8319, Cl, F, Cl, Bn, F), (M-8320, Cl, F, Cl, Bn, CF₃), (M-8321, Cl, F, Cl, Bn, Br), (M-8322, Cl, F, Cl, Bn, CH₃), (M-8323, Cl, F, Cl, 4-F-Bn, H), (M-8324, Cl, F, Cl, 4-F-Bn, Cl), (M-8325, Cl, F, Cl, 4-F-Bn, F), (M-8326, Cl, F, Cl, 4-F-Bn, CF₃), (M-8327, Cl, F, Cl, 4-F-Bn, Br), (M-8328, Cl, F, Cl, 4-F-Bn, CH₃), (M-8329, Cl, F, Cl, 2-Py, H), (M-8330, Cl, F, Cl, 2-Py, Cl), (M-8331, Cl, F, Cl, 2-Py, F), (M-8332, Cl, F, Cl, 2-Py, CF₃), (M-8333, Cl, F, Cl, 2-Py, Br), (M-8334, Cl, F, Cl, 2-Py, CH₃), (M-8335, Cl, F, Cl, 3-Py, H), (M-8336, Cl, F, Cl, 3-Py, Cl), (M-8337, Cl, F, Cl, 3-Py, F), (M-8338, Cl, F, Cl, 3-Py, CF₃), (M-8339, Cl, F, Cl, 3-Py, Br), (M-8340, Cl, F, Cl, 3-Py, CH₃), (M-8341, Cl, F, Cl, 4-Py, H), (M-8342, Cl, F, Cl, 4-Py, Cl), (M-8343, Cl, F, Cl, 4-Py, F), (M-8344, Cl, F, Cl, 4-Py, CF₃), (M-8345, Cl, F, Cl, 4-Py, Br), (M-8346, Cl, F, Cl, 4-Py, CH₃), (M-8347, Cl, F, Cl, 2-Th, H), (M-8348, Cl, F, Cl, 2-Th, Cl), (M-8349, Cl, F, Cl, 2-Th, F), (M-8350, Cl, F, Cl, 2-Th, CF₃), (M-8351, Cl, F, Cl, 2-Th, Br), (M-8352, Cl, F, Cl, 2-Th, CH₃), (M-8353, Cl, F, Cl, 3-Th, H), (M-8354, Cl, F, Cl, 3-Th, Cl), (M-8355, Cl, F, Cl, 3-Th, F), (M-8356, Cl, F, Cl, 3-Th, CF₃), (M-8357, Cl, F, Cl, 3-Th, Br), (M-8358, Cl, F, Cl, 3-Th, CH₃), (M-8359, Cl, F, Cl, pyrazol-2-yl, H), (M-8360, Cl, F, Cl, pyrazol-2-yl, Cl), (M-8361, Cl, F, Cl, pyrazol-2-yl, F), (M-8362, Cl, F, Cl, pyrazol-2-yl, CF₃), (M-8363, Cl, F, Cl, pyrazol-2-yl, Br), (M-8364, Cl, F, Cl, pyrazol-2-yl, CH₃), (M-8365, Cl, F, Cl, pyrazol-3-yl, H), (M-8366, Cl, F, Cl, pyrazol-3-yl, Cl), (M-8367, Cl, F, Cl, pyrazol-3-yl, F), (M-8368, Cl, F, Cl, pyrazol-3-yl, CF₃), (M-8369, Cl, F, Cl, pyrazol-3-yl, Br), (M-8370, Cl, F, Cl, pyrazol-3-yl, CH₃), (M-8371, Cl, F, Cl, pyrimidin-2-yl, H), (M-8372, Cl, F, Cl, pyrimidin-2-yl, Cl), (M-8373, Cl, F, Cl, pyrimidin-2-yl, F), (M-8374, Cl, F, Cl, pyrimidin-2-yl, CF₃), (M-8375, Cl, F, Cl, pyrimidin-2-yl, Br), (M-8376, Cl, F, Cl, pyrimidin-2-yl, CH₃), (M-8377, Cl, F, Cl, pyrimidin-4-yl, H), (M-8378, Cl, F, Cl, pyrimidin-4-yl, Cl), (M-8379, Cl, F, Cl, pyrimidin-4-yl, F), (M-8380, Cl, F, Cl, pyrimidin-4-yl, CF₃), (M-8381, Cl, F, Cl, pyrimidin-4-yl, Br), (M-8382, Cl, F, Cl, pyrimidin-4-yl, CH₃), (M-8383, Cl, F, Cl, pyrimidin-5-yl, H), (M-8384, Cl, F, Cl, pyrimidin-5-yl, Cl), (M-8385, Cl, F, Cl, pyrimidin-5-yl, F), (M-8386, Cl, F, Cl, pyrimidin-5-yl, CF₃), (M-8387, Cl, F, Cl, pyrimidin-5-yl, Br), (M-8388, Cl, F, Cl, pyrimidin-5-yl, CH₃), (M-8389, Cl, F, Cl, HOOCCH₂CH₂CH₂, H), (M-8390, Cl, F, Cl, HOOCCH₂CH₂CH₂, Cl), (M-8391, Cl, F, Cl, HOOCCH₂CH₂CH₂, F), (M-8392, Cl, F, Cl, HOOCCH₂CH₂CH₂, CF₃), (M-8393, Cl, F, Cl, HOOCCH₂CH₂CH₂, Br), (M-8394, Cl, F, Cl, HOOCCH₂CH₂
CH₂, CH₃), (M-8395, Cl, F, Cl, HOOCCH₂CH₂CH₂CH₂, H), (M-8396, Cl, F, Cl, HOOCCH₂CH₂CH₂CH₂, Cl), (M-8397, Cl, F, Cl, HOOCCH₂CH₂CH₂CH₂, F), (M-8398, Cl, F, Cl, HOOCCH₂CH₂CH₂CH₂, CF₃), (M-8399, Cl, F, Cl, HOOCCH₂CH₂CH₂CH₂, Br), (M-8400, Cl, F, Cl, HOOCCH₂CH₂CH₂CH₂, CH₃), (M-8401, Cl, F, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂, H), (M-8402, Cl, F, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂, Cl), (M-8403, Cl, F, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂, F), (M-8404, Cl, F, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂, CF₃), (M-8405, Cl, F, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂, Br), (M-8406, Cl, F, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂, CH₃), (M-8407, Cl, F, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, H), (M-8408, Cl, F, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, Cl), (M-8409, Cl, F, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, F), (M-8410, Cl, F, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, CF₃), (M-8411, Cl, F, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, Br), (M-8412, Cl, F, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, CH₃), (M-8413, Cl, F, Cl, MeOCH₂, H), (M-8414, Cl, F, Cl, MeOCH₂, Cl), (M-8415, Cl, F, Cl, MeOCH₂, F), (M-8416, Cl, F, Cl, MeOCH₂, CF₃), (M-8417, Cl, F, Cl, MeOCH₂, Br), (M-8418, Cl, F, Cl, MeOCH₂, CH₃), (M-8419, Cl, F, Cl, EtOCH₂, H), (M-8420, Cl, F, Cl, EtOCH₂, Cl), (M-8421, Cl, F, Cl, EtOCH₂, F), (M-8422, Cl, F, Cl, EtOCH₂, CF₃), (M-8423, Cl, F, Cl, EtOCH₂, Br), (M-8424, Cl, F, Cl, EtOCH₂, CH₃), (M-8425, Cl, F, Cl, EtOCH₂CH₂, H), (M-8426, Cl, F, Cl, EtOCH₂CH₂, Cl), (M-8427, Cl, F, Cl, EtOCH₂CH₂, F), (M-8428, Cl, F, Cl, EtOCH₂CH₂, CF₃), (M-8429, Cl, F, Cl, EtOCH₂CH₂, Br), (M-8430, Cl, F, Cl, EtOCH₂CH₂, CH₃), (M-8431, Cl, F, Cl, MeOCH₂CH₂OCH₂CH₂, H), (M-8432, Cl, F, Cl, MeOCH₂CH₂OCH₂CH₂, Cl), (M-8433, Cl, F, Cl, MeOCH₂CH₂OCH₂CH₂, F), (M-8434, Cl, F, Cl, MeOCH₂CH₂OCH₂CH₂, CF₃), (M-8435, Cl, F, Cl, MeOCH₂CH₂OCH₂CH₂, Br), (M-8436, Cl, F, Cl, MeOCH₂CH₂OCH₂CH₂, CH₃), (M-8437, Cl, F, Cl, MeOCH₂CH₂, H), (M-8438, Cl, F, Cl, MeOCH₂CH₂, Cl), (M-8439, Cl, F, Cl, MeOCH₂CH₂, F), (M-8440, Cl, F, Cl, MeOCH₂CH₂, CF₃), (M-8441, Cl, F, Cl, MeOCH₂CH₂, Br), (M-8442, Cl, F, Cl, MeOCH₂CH₂, CH₃), (M-8443, Cl, F, Cl, HOCH₂, H), (M-8444, Cl, F, Cl, HOCH₂, Cl), (M-8445, Cl, F, Cl, HOCH₂, F), (M-8446, Cl, F, Cl, HOCH₂, CF₃), (M-8447, Cl, F, Cl, HOCH₂, Br), (M-8448, Cl, F, Cl, HOCH₂, CH₃), (M-8449, Cl, F, Cl, HOCH₂CH₂, H), (M-8450, Cl, F, Cl, HOCH₂CH₂, Cl), (M-8451, Cl, F, Cl, HOCH₂CH₂, F), (M-8452, Cl, F, Cl, HOCH₂CH₂, CF₃), (M-8453, Cl, F, Cl, HOCH₂CH₂, Br), (M-8454, Cl, F, Cl, HOCH₂CH₂, CH₃), (M-8455, Cl, F, Cl, HOCH₂CH₂CH₂, H), (M-8456, Cl, F, Cl, HOCH₂CH₂CH₂, Cl), (M-8457, Cl, F, Cl, HOCH₂CH₂CH₂, F), (M-8458, Cl, F, Cl, HOCH₂CH₂CH₂, CF₃), (M-8459, Cl, F, Cl, HOCH₂CH₂CH₂, Br), (M-8460, Cl, F, Cl, HOCH₂CH₂CH₂, CH₃), (M-8461, Cl, F, Cl, HOCH₂CH₂CH₂CH₂, H), (M-8462, Cl, F, Cl, HOCH₂CH₂CH₂CH₂, Cl), (M-8463, Cl, F, Cl, HOCH₂CH₂CH₂CH₂, F), (M-8464, Cl, F, Cl, HOCH₂CH₂CH₂CH₂, CF₃), (M-8465, Cl, F, Cl, HOCH₂CH₂CH₂CH₂, Br), (M-8466, Cl, F, Cl, HOCH₂CH₂CH₂CH₂, CH₃), (M-8467, Cl, F, Cl, HOCH₂CH₂CH₂CH₂CH₂, H), (M-8468, Cl, F, Cl, HOCH₂CH₂CH₂CH₂CH₂, Cl), (M-8469, Cl, F, Cl, HOCH₂CH₂CH₂CH₂CH₂, F), (M-8470, Cl, F, Cl, HOCH₂CH₂CH₂CH₂CH₂, CF₃), (M-8471, Cl, F, Cl, HOCH₂CH₂CH₂CH₂CH₂, Br), (M-8472, Cl, F, Cl, HOCH₂CH₂CH₂CH₂CH₂, CH₃), (M-8473, Cl, F, Cl, HOCH₂CH₂OCH₂CH₂, H), (M-8474, Cl, F, Cl, HOCH₂CH₂OCH₂CH₂, Cl), (M-8475, Cl, F, Cl, HOCH₂CH₂OCH₂CH₂, F), (M-8476, Cl, F, Cl, HOCH₂CH₂OCH₂CH₂, CF₃), (M-8477, Cl, F, Cl, HOCH₂CH₂OCH₂CH₂, Br), (M-8478, Cl, F, Cl, HOCH₂CH₂OCH₂CH₂, CH₃), (M-8479, Cl, F, Cl, (Me)₂N, H), (M-8480, Cl, F, Cl, (Me)₂N, Cl), (M-8481, Cl, F, Cl, (Me)₂N, F), (M-8482, Cl, F, Cl, (Me)₂N, CF₃), (M-8483, Cl, F, Cl, (Me)₂N, Br), (M-8484, Cl, F, Cl, (Me)₂N, CH₃), (M-8485, Cl, F, Cl, piperidin-4-yl-methyl, H), (M-8486, Cl, F, Cl, piperidin-4-yl-methyl, Cl), (M-8487, Cl, F, Cl, piperidin-4-yl-methyl, F), (M-8488, Cl, F, Cl, piperidin-4-yl-methyl, CF₃), (M-8489, Cl, F, Cl, piperidin-4-yl-methyl, Br), (M-8490, Cl, F, Cl, piperidin-4-yl-methyl, CH₃), (M-8491, Cl, F, Cl, cyclohexylmethyl, H), (M-8492, Cl, F, Cl, cyclohexylmethyl, Cl), (M-8493, Cl, F, Cl, cyclohexylmethyl, F), (M-8494, Cl, F, Cl, cyclohexylmethyl, CF₃), (M-8495, Cl, F, Cl, cyclohexylmethyl, Br), (M-8496, Cl, F, Cl, cyclohexylmethyl, CH₃), (M-8497, Cl, CH₃, H, H, H), (M-8498, Cl, CH₃, H, H, Cl), (M-8499, Cl, CH₃, H, H, F), (M-8500, Cl, CH₃, H, H, CF₃), (M-8501, Cl, CH₃, H, H, Br), (M-8502, Cl, CH₃, H, H, CH₃), (M-8503, Cl, CH₃, H, F, H), (M-8504, Cl, CH₃, H, F, Cl), (M-8505, Cl, CH₃, H, F, F), (M-8506, Cl, CH₃, H, F, CF₃), (M-8507, Cl, CH₃, H, F, Br), (M-8508, Cl, CH₃, H, F, CH₃), (M-8509, Cl, CH₃, H, Cl, H), (M-8510, Cl, CH₃, H, Cl, Cl), (M-8511, Cl, CH₃, H, Cl, F), (M-8512, Cl, CH₃, H, Cl, CF₃), (M-8513, Cl, CH₃, H, Cl, Br), (M-8514, Cl, CH₃, H, Cl, CH₃), (M-8515, Cl, CH₃, H, CH₃, H), (M-8516, Cl, CH₃, H, CH₃, Cl), (M-8517, Cl, CH₃, H, CH₃, F), (M-8518, Cl, CH₃, H, CH₃, CF₃), (M-8519, Cl, CH₃, H, CH₃, Br), (M-8520, Cl, CH₃, H, CH₃, CH₃), (M-8521, Cl, CH₃, H, Et, H), (M-8522, Cl, CH₃, H, Et, Cl), (M-8523, Cl, CH₃, H, Et, F), (M-8524, Cl, CH₃, H, Et, CF₃), (M-8525, Cl, CH₃, H, Et, Br), (M-8526, Cl, CH₃, H, Et, CH₃), (M-8527, Cl, CH₃, H, n-Pr, H), (M-8528, Cl, CH₃, H, n-Pr, Cl), (M-8529, Cl, CH₃, H, n-Pr, F), (M-8530, Cl, CH₃, H, n-Pr, CF₃), (M-8531, Cl, CH₃, H, n-Pr, Br), (M-8532, Cl, CH₃, H, n-Pr, CH₃), (M-8533, Cl, CH₃, H, c-Pr, H), (M-8534, Cl, CH₃, H, c-Pr, Cl), (M-8535, Cl, CH₃, H, c-Pr, F), (M-8536, Cl, CH₃, H, c-Pr, CF₃), (M-8537, Cl, CH₃, H, c-Pr, Br), (M-8538, Cl, CH₃, H, c-Pr, CH₃), (M-8539, Cl, CH₃, H, i-Pr, H), (M-8540, Cl, CH₃, H, i-Pr, Cl), (M-8541, Cl, CH₃, H, i-Pr, F), (M-8542, Cl, CH₃, H, i-Pr, CF₃), (M-8543, Cl, CH₃, H, i-Pr, Br), (M-8544, Cl, CH₃, H, i-Pr, CH₃), (M-8545, Cl, CH₃, H, n-Bu, H), (M-8546, Cl, CH₃, H, n-Bu, Cl), (M-8547, Cl, CH₃, H, n-Bu, F), (M-8548, Cl, CH₃, H, n-Bu, CF₃), (M-8549, Cl, CH₃, H, n-Bu, Br), (M-8550, Cl, CH₃, H, n-Bu, CH₃), (M-8551, Cl, CH₃, H, i-Bu, H), (M-8552, Cl, CH₃, H, i-Bu, Cl), (M-8553, Cl, CH₃, H, i-Bu, F), (M-8554, Cl, CH₃, H, i-Bu, CF₃), (M-8555, Cl, CH₃, H, i-Bu, Br), (M-8556, Cl, CH₃, H, i-Bu, CH₃
), (M-8557, Cl, CH₃, H, sec-Bu, H), (M-8558, Cl, CH₃, H, sec-Bu, Cl), (M-8559, Cl, CH₃, H, sec-Bu, F), (M-8560, Cl, CH₃, H, sec-Bu, CF₃), (M-8561, Cl, CH₃, H, sec-Bu, Br), (M-8562, Cl, CH₃, H, sec-Bu, CH₃), (M-8563, Cl, CH₃, H, n-Pen, H), (M-8564, Cl, CH₃, H, n-Pen, Cl), (M-8565, Cl, CH₃, H, n-Pen, F), (M-8566, Cl, CH₃, H, n-Pen, CF₃), (M-8567, Cl, CH₃, H, n-Pen, Br), (M-8568, Cl, CH₃, H, n-Pen, CH₃), (M-8569, Cl, CH₃, H, c-Pen, H), (M-8570, Cl, CH₃, H, c-Pen, Cl), (M-8571, Cl, CH₃, H, c-Pen, F), (M-8572, Cl, CH₃, H, c-Pen, CF₃), (M-8573, Cl, CH₃, H, c-Pen, Br), (M-8574, Cl, CH₃, H, c-Pen, CH₃), (M-8575, Cl, CH₃, H, n-Hex, H), (M-8576, Cl, CH₃, H, n-Hex, Cl), (M-8577, Cl, CH₃, H, n-Hex, F), (M-8578, Cl, CH₃, H, n-Hex, CF₃), (M-8579, Cl, CH₃, H, n-Hex, Br), (M-8580, Cl, CH₃, H, n-Hex, CH₃), (M-8581, Cl, CH₃, H, c-Hex, H), (M-8582, Cl, CH₃, H, c-Hex, Cl), (M-8583, Cl, CH₃, H, c-Hex, F), (M-8584, Cl, CH₃, H, c-Hex, CF₃), (M-8585, Cl, CH₃, H, c-Hex, Br), (M-8586, Cl, CH₃, H, c-Hex, CH₃), (M-8587, Cl, CH₃, H, OH, H), (M-8588, Cl, CH₃, H, OH, Cl), (M-8589, Cl, CH₃, H, OH, F), (M-8590, Cl, CH₃, H, OH, CF₃), (M-8591, Cl, CH₃, H, OH, Br), (M-8592, Cl, CH₃, H, OH, CH₃), (M-8593, Cl, CH₃, H, EtO, H), (M-8594, Cl, CH₃, H, EtO, Cl), (M-8595, Cl, CH₃, H, EtO, F), (M-8596, Cl, CH₃, H, EtO, CF₃), (M-8597, Cl, CH₃, H, EtO, Br), (M-8598, Cl, CH₃, H, EtO, CH₃), (M-8599, Cl, CH₃, H, n-PrO, H), (M-8600, Cl, CH₃, H, n-PrO, Cl), (M-8601, Cl, CH₃, H, n-PrO, F), (M-8602, Cl, CH₃, H, n-PrO, CF₃), (M-8603, Cl, CH₃, H, n-PrO, Br), (M-8604, Cl, CH₃, H, n-PrO, CH₃), (M-8605, Cl, CH₃, H, PhO, H), (M-8606, Cl, CH₃, H, PhO, Cl), (M-8607, Cl, CH₃, H, PhO, F), (M-8608, Cl, CH₃, H, PhO, CF₃), (M-8609, Cl, CH₃, H, PhO, Br), (M-8610, Cl, CH₃, H, PhO, CH₃), (M-8611, Cl, CH₃, H, BnO, H), (M-8612, Cl, CH₃, H, BnO, Cl), (M-8613, Cl, CH₃, H, BnO, F), (M-8614, Cl, CH₃, H, BnO, CF₃), (M-8615, Cl, CH₃, H, BnO, Br), (M-8616, Cl, CH₃, H, BnO, CH₃), (M-8617, Cl, CH₃, H, PhCH₂CH₂O, H), (M-8618, Cl, CH₃, H, PhCH₂CH₂O, Cl), (M-8619, Cl, CH₃, H, PhCH₂CH₂O, F), (M-8620, Cl, CH₃, H, PhCH₂CH₂O, CF₃), (M-8621, Cl, CH₃, H, PhCH₂CH₂O, Br), (M-8622, Cl, CH₃, H, PhCH₂CH₂O, CH₃), (M-8623, Cl, CH₃, H, CF₃O, H), (M-8624, Cl, CH₃, H, CF₃O, Cl), (M-8625, Cl, CH₃, H, CF₃O, F), (M-8626, Cl, CH₃, H, CF₃O, CF₃), (M-8627, Cl, CH₃, H, CF₃O, Br), (M-8628, Cl, CH₃, H, CF₃O, CH₃), (M-8629, Cl, CH₃, H, Ph, H), (M-8630, Cl, CH₃, H, Ph, Cl), (M-8631, Cl, CH₃, H, Ph, F), (M-8632, Cl, CH₃, H, Ph, CF₃), (M-8633, Cl, CH₃, H, Ph, Br), (M-8634, Cl, CH₃, H, Ph, CH₃), (M-8635, Cl, CH₃, H, 4-F-Ph, H), (M-8636, Cl, CH₃, H, 4-F-Ph, Cl), (M-8637, Cl, CH₃, H, 4-F-Ph, F), (M-8638, Cl, CH₃, H, 4-F-Ph, CF₃), (M-8639, Cl, CH₃, H, 4-F-Ph, Br), (M-8640, Cl, CH₃, H, 4-F-Ph, CH₃), (M-8641, Cl, CH₃, H, 4-CF₃-Ph, H), (M-8642, Cl, CH₃, H, 4-CF₃-Ph, Cl), (M-8643, Cl, CH₃, H, 4-CF₃-Ph, F), (M-8644, Cl, CH₃, H, 4-CF₃-Ph, CF₃), (M-8645, Cl, CH₃, H, 4-CF₃-Ph, Br), (M-8646, Cl, CH₃, H, 4-CF₃-Ph, CH₃), (M-8647, Cl, CH₃, H, 4-(Me)₂N-Ph, H), (M-8648, Cl, CH₃, H, 4-(Me)₂N-Ph, Cl), (M-8649, Cl, CH₃, H, 4-(Me)₂N-Ph, F), (M-8650, Cl, CH₃, H, 4-(Me)₂N-Ph, CF₃), (M-8651, Cl, CH₃, H, 4-(Me)₂N-Ph, Br), (M-8652, Cl, CH₃, H, 4-(Me)₂N-Ph, CH₃), (M-8653, Cl, CH₃, H, 4-OH-Ph, H), (M-8654, Cl, CH₃, H, 4-OH-Ph, Cl), (M-8655, Cl, CH₃, H, 4-OH-Ph, F), (M-8656, Cl, CH₃, H, 4-OH-Ph, CF₃), (M-8657, Cl, CH₃, H, 4-OH-Ph, Br), (M-8658, Cl, CH₃, H, 4-OH-Ph, CH₃), (M-8659, Cl, CH₃, H, 3,4-di-F-Ph, H), (M-8660, Cl, CH₃, H, 3,4-di-F-Ph, Cl), (M-8661, Cl, CH₃, H, 3,4-di-F-Ph, F), (M-8662, Cl, CH₃, H, 3,4-di-F-Ph, CF₃), (M-8663, Cl, CH₃, H, 3,4-di-F-Ph, Br), (M-8664, Cl, CH₃, H, 3,4-di-F-Ph, CH₃), (M-8665, Cl, CH₃, H, 4-COOH-Ph, H), (M-8666, Cl, CH₃, H, 4-COOH-Ph, Cl), (M-8667, Cl, CH₃, H, 4-COOH-Ph, F), (M-8668, Cl, CH₃, H, 4-COOH-Ph, CF₃), (M-8669, Cl, CH₃, H, 4-COOH-Ph, Br), (M-8670, Cl, CH₃, H, 4-COOH-Ph, CH₃), (M-8671, Cl, CH₃, H, Bn, H), (M-8672, Cl, CH₃, H, Bn, Cl), (M-8673, Cl, CH₃, H, Bn, F), (M-8674, Cl, CH₃, H, Bn, CF₃), (M-8675, Cl, CH₃, H, Bn, Br), (M-8676, Cl, CH₃, H, Bn, CH₃), (M-8677, Cl, CH₃, H, 4-F-Bn, H), (M-8678, Cl, CH₃, H, 4-F-Bn, Cl), (M-8679, Cl, CH₃, H, 4-F-Bn, F), (M-8680, Cl, CH₃, H, 4-F-Bn, CF₃), (M-8681, Cl, CH₃, H, 4-F-Bn, Br), (M-8682, Cl, CH₃, H, 4-F-Bn, CH₃), (M-8683, Cl, CH₃, H, 2-Py, H), (M-8684, Cl, CH₃, H, 2-Py, Cl), (M-8685, Cl, CH₃, H, 2-Py, F), (M-8686, Cl, CH₃, H, 2-Py, CF₃), (M-8687, Cl, CH₃, H, 2-Py, Br), (M-8688, Cl, CH₃, H, 2-Py, CH₃), (M-8689, Cl, CH₃, H, 3-Py, H), (M-8690, Cl, CH₃, H, 3-Py, Cl), (M-8691, Cl, CH₃, H, 3-Py, F), (M-8692, Cl, CH₃, H, 3-Py, CF₃), (M-8693, Cl, CH₃, H, 3-Py, Br), (M-8694, Cl, CH₃, H, 3-Py, CH₃), (M-8695, Cl, CH₃, H, 4-Py, H), (M-8696, Cl, CH₃, H, 4-Py, Cl), (M-8697, Cl, CH₃, H, 4-Py, F), (M-8698, Cl, CH₃, H, 4-Py, CF₃), (M-8699, Cl, CH₃, H, 4-Py, Br), (M-8700, Cl, CH₃, H, 4-Py, CH₃), (M-8701, Cl, CH₃, H, 2-Th, H), (M-8702, Cl, CH₃, H, 2-Th, Cl), (M-8703, Cl, CH₃, H, 2-Th, F), (M-8704, Cl, CH₃, H, 2-Th, CF₃), (M-8705, Cl, CH₃, H, 2-Th, Br), (M-8706, Cl, CH₃, H, 2-Th, CH₃), (M-8707, Cl, CH₃, H, 3-Th, H), (M-8708, Cl, CH₃, H, 3-Th, Cl), (M-8709, Cl, CH₃, H, 3-Th, F), (M-8710, Cl, CH₃, H, 3-Th, CF₃), (M-8711, Cl, CH₃, H, 3-Th, Br), (M-8712, Cl, CH₃, H, 3-Th, CH₃), (M-8713, Cl, CH₃, H, pyrazol-2-yl, H), (M-8714, Cl, CH₃, H, pyrazol-2-yl, Cl), (M-8715, Cl, CH₃, H, pyrazol-2-yl, F), (M-8716, Cl, CH₃, H, pyrazol-2-yl, CF₃), (M-8717, Cl, CH₃, H, pyrazol-2-yl, Br), (M-8718, Cl, CH₃, H, pyrazol-2-yl, CH₃), (M-8719, Cl, CH₃, H, pyrazol-3-yl, H), (M-8720, Cl, CH₃, H, pyrazol-3-yl, Cl), (M-8721, Cl, CH₃, H, pyrazol-3-yl, F), (M-8722, Cl, CH₃, H, pyrazol-3-yl, CF₃), (M-8723, Cl, CH₃, H, pyrazol-3-yl, Br), (M-8724, Cl, CH₃, H, pyrazol-3-yl, CH₃), (M-8725, Cl, CH₃, H, pyrimidin-2-yl, H), (M-8726, Cl, CH₃, H, pyrimidin-2-yl, Cl), (M-8727, Cl, CH₃, H, pyrimidin-2-yl, F), (M-8728, Cl, CH₃, H, pyrimidin-2-yl, CF₃), (M-8729, Cl, CH₃, H, pyrimidin-2-yl, Br), (M-8730, Cl, CH₃, H, pyrimidin-2-yl, CH₃), (M-8731, Cl, CH₃, H, pyrimidin-4-yl, H), (M-8732, Cl, CH₃, H, pyrimidin-4-yl, Cl), (M-8733, Cl, CH₃, H, pyrimidin-4-yl, F), (M-8734, Cl, CH₃, H, pyrimidin-4-yl, CF₃), (M-8735, Cl, CH₃, H, pyrimidin-4-yl, Br), (M-8736, Cl, CH₃, H, pyrimidin-4-yl, CH₃), (M-8737, Cl, CH₃, H, pyrimidin-5-yl, H), (M-8738, Cl, CH₃, H, pyrimidin-5-yl, Cl), (M-8739, Cl, CH₃, H, pyrimidin-5-yl, F), (M-8740, Cl, CH₃, H, pyrimidin-5-yl, CF₃), (M-8741, Cl, CH₃, H, pyrimidin-5-yl, Br), (M-8742, Cl, CH₃, H, pyrimidin-5-yl, CH₃), (M-8743, Cl, CH₃, H, HOOCCH₂CH₂CH₂, H), (M-8744, Cl, CH₃, H, HOOCCH₂CH₂CH₂, Cl), (M-8745, Cl, CH₃, H, HOOCCH₂CH₂CH₂, F), (M-8746, Cl, CH₃, H, HOOCCH₂CH₂CH₂, CF₃), (M-8747, Cl, CH₃, H, HOOCCH₂CH₂CH₂, Br), (M-8748, Cl, CH₃, H, HOOCCH₂CH₂CH₂, CH₃), (M-8749, Cl, CH₃, H, HOOCCH₂CH₂CH₂CH₂, H), (M-8750, Cl, CH₃, H, HOOCCH₂CH₂CH₂CH₂, Cl), (M-8751, Cl, CH₃
, H, HOOCCH₂CH₂CH₂CH₂, F), (M-8752, Cl, CH₃, H, HOOCCH₂CH₂CH₂CH₂, CF₃), (M-8753, Cl, CH₃, H, HOOCCH₂CH₂CH₂CH₂, Br), (M-8754, Cl, CH₃, H, HOOCCH₂CH₂CH₂CH₂, CH₃), (M-8755, Cl, CH₃, H, (Me)₂NCOCH₂CH₂CH₂CH₂, H), (M-8756, Cl, CH₃, H, (Me)₂NCOCH₂CH₂CH₂CH₂, Cl), (M-8757, Cl, CH₃, H, (Me)₂NCOCH₂CH₂CH₂CH₂, F), (M-8758, Cl, CH₃, H, (Me)₂NCOCH₂CH₂CH₂CH₂, CF₃), (M-8759, Cl, CH₃, H, (Me)₂NCOCH₂CH₂CH₂CH₂, Br), (M-8760, Cl, CH₃, H, (Me)₂NCOCH₂CH₂CH₂CH₂, CH₃), (M-8761, Cl, CH₃, H, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, H), (M-8762, Cl, CH₃, H, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, Cl), (M-8763, Cl, CH₃, H, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, F), (M-8764, Cl, CH₃, H, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, CF₃), (M-8765, Cl, CH₃, H, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, Br), (M-8766, Cl, CH₃, H, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, CH₃), (M-8767, Cl, CH₃, H, MeOCH₂, H), (M-8768, Cl, CH₃, H, MeOCH₂, Cl), (M-8769, Cl, CH₃, H, MeOCH₂, F), (M-8770, Cl, CH₃, H, MeOCH₂, CF₃), (M-8771, Cl, CH₃, H, MeOCH₂, Br), (M-8772, Cl, CH₃, H, MeOCH₂, CH₃), (M-8773, Cl, CH₃, H, EtOCH₂, H), (M-8774, Cl, CH₃, H, EtOCH₂, Cl), (M-8775, Cl, CH₃, H, EtOCH₂, F), (M-8776, Cl, CH₃, H, EtOCH₂, CF₃), (M-8777, Cl, CH₃, H, EtOCH₂, Br), (M-8778, Cl, CH₃, H, EtOCH₂, CH₃), (M-8779, Cl, CH₃, H, EtOCH₂CH₂, H), (M-8780, Cl, CH₃, H, EtOCH₂CH₂, Cl), (M-8781, Cl, CH₃, H, EtOCH₂CH₂, F), (M-8782, Cl, CH₃, H, EtOCH₂CH₂, CF₃), (M-8783, Cl, CH₃, H, EtOCH₂CH₂, Br), (M-8784, Cl, CH₃, H, EtOCH₂CH₂, CH₃), (M-8785, Cl, CH₃, H, MeOCH₂CH₂OCH₂CH₂, H), (M-8786, Cl, CH₃, H, MeOCH₂CH₂OCH₂CH₂, Cl), (M-8787, Cl, CH₃, H, MeOCH₂CH₂OCH₂CH₂, F), (M-8788, Cl, CH₃, H, MeOCH₂CH₂OCH₂CH₂, CF₃), (M-8789, Cl, CH₃, H, MeOCH₂CH₂OCH₂CH₂, Br), (M-8790, Cl, CH₃, H, MeOCH₂CH₂OCH₂CH₂, CH₃), (M-8791, Cl, CH₃, H, MeOCH₂CH₂, H), (M-8792, Cl, CH₃, H, MeOCH₂CH₂, Cl), (M-8793, Cl, CH₃, H, MeOCH₂CH₂, F), (M-8794, Cl, CH₃, H, MeOCH₂CH₂, CF₃), (M-8795, Cl, CH₃, H, MeOCH₂CH₂, Br), (M-8796, Cl, CH₃, H, MeOCH₂CH₂, CH₃), (M-8797, Cl, CH₃, H, HOCH₂, H), (M-8798, Cl, CH₃, H, HOCH₂, Cl), (M-8799, Cl, CH₃, H, HOCH₂, F), (M-8800, Cl, CH₃, H, HOCH₂, CF₃), (M-8801, Cl, CH₃, H, HOCH₂, Br), (M-8802, Cl, CH₃, H, HOCH₂, CH₃), (M-8803, Cl, CH₃, H, HOCH₂CH₂, H), (M-8804, Cl, CH₃, H, HOCH₂CH₂, Cl), (M-8805, Cl, CH₃, H, HOCH₂CH₂, F), (M-8806, Cl, CH₃, H, HOCH₂CH₂, CF₃), (M-8807, Cl, CH₃, H, HOCH₂CH₂, Br), (M-8808, Cl, CH₃, H, HOCH₂CH₂, CH₃), (M-8809, Cl, CH₃, H, HOCH₂CH₂CH₂, H), (M-8810, Cl, CH₃, H, HOCH₂CH₂CH₂, Cl), (M-8811, Cl, CH₃, H, HOCH₂CH₂CH₂, F), (M-8812, Cl, CH₃, H, HOCH₂CH₂CH₂, CF₃), (M-8813, Cl, CH₃, H, HOCH₂CH₂CH₂, Br), (M-8814, Cl, CH₃, H, HOCH₂CH₂CH₂, CH₃), (M-8815, Cl, CH₃, H, HOCH₂CH₂CH₂CH₂, H), (M-8816, Cl, CH₃, H, HOCH₂CH₂CH₂CH₂, Cl), (M-8817, Cl, CH₃, H, HOCH₂CH₂CH₂CH₂, F), (M-8818, Cl, CH₃, H, HOCH₂CH₂CH₂CH₂, CF₃), (M-8819, Cl, CH₃, H, HOCH₂CH₂CH₂CH₂, Br), (M-8820, Cl, CH₃, H, HOCH₂CH₂CH₂CH₂, CH₃), (M-8821, Cl, CH₃, H, HOCH₂CH₂CH₂CH₂CH₂, H), (M-8822, Cl, CH₃, H, HOCH₂CH₂CH₂CH₂CH₂, Cl), (M-8823, Cl, CH₃, H, HOCH₂CH₂CH₂CH₂CH₂, F), (M-8824, Cl, CH₃, H, HOCH₂CH₂CH₂CH₂CH₂, CF₃), (M-8825, Cl, CH₃, H, HOCH₂CH₂CH₂CH₂CH₂, Br), (M-8826, Cl, CH₃, H, HOCH₂CH₂CH₂CH₂CH₂, CH₃), (M-8827, Cl, CH₃, H, HOCH₂CH₂OCH₂CH₂, H), (M-8828, Cl, CH₃, H, HOCH₂CH₂OCH₂CH₂, Cl), (M-8829, Cl, CH₃, H, HOCH₂CH₂OCH₂CH₂, F), (M-8830, Cl, CH₃, H, HOCH₂CH₂OCH₂CH₂, CF₃), (M-8831, Cl, CH₃, H, HOCH₂CH₂OCH₂CH₂, Br), (M-8832, Cl, CH₃, H, HOCH₂CH₂OCH₂CH₂, CH₃), (M-8833, Cl, CH₃, H, (Me)₂N, H), (M-8834, Cl, CH₃, H, (Me)₂N, Cl), (M-8835, Cl, CH₃, H, (Me)₂N, F), (M-8836, Cl, CH₃, H, (Me)₂N, CF₃), (M-8837, Cl, CH₃, H, (Me)₂N, Br), (M-8838, Cl, CH₃, H, (Me)₂N, CH₃), (M-8839, Cl, CH₃, H, piperidin-4-yl-methyl, H), (M-8840, Cl, CH₃, H, piperidin-4-yl-methyl, Cl), (M-8841, Cl, CH₃, H, piperidin-4-yl-methyl, F), (M-8842, Cl, CH₃, H, piperidin-4-yl-methyl, CF₃), (M-8843, Cl, CH₃, H, piperidin-4-yl-methyl, Br), (M-8844, Cl, CH₃, H, piperidin-4-yl-methyl, CH₃), (M-8845, Cl, CH₃, H, cyclohexylmethyl, H), (M-8846, Cl, CH₃, H, cyclohexylmethyl, Cl), (M-8847, Cl, CH₃, H, cyclohexylmethyl, F), (M-8848, Cl, CH₃, H, cyclohexylmethyl, CF₃), (M-8849, Cl, CH₃, H, cyclohexylmethyl, Br), (M-8850, Cl, CH₃, H, cyclohexylmethyl, CH₃), (M-8851, Cl, CH₃, F, H, H), (M-8852, Cl, CH₃, F, H, Cl), (M-8853, MeO, CH₃, F, H, F), (M-8854, Cl, CH₃, F, H, CF₃), (M-8855, Cl, CH₃, F, H, Br), (M-8856, Cl, CH₃, F, H, CH₃), (M-8857, Cl, CH₃, F, F, H), (M-8858, Cl, CH₃, F, F, Cl), (M-8859, Cl, CH₃, F, F, F), (M-8860, Cl, CH₃, F, F, CF₃), (M-8861, Cl, CH₃, F, F, Br), (M-8862, Cl, CH₃, F, F, CH₃), (M-8863, Cl, CH₃, F, Cl, H), (M-8864, Cl, CH₃, F, Cl, Cl), (M-8865, Cl, CH₃, F, Cl, F), (M-8866, Cl, CH₃, F, Cl, CF₃), (M-8867, Cl, CH₃, F, Cl, Br), (M-8868, Cl, CH₃, F, Cl, CH₃), (M-8869, Cl, CH₃, F, CH₃, H), (M-8870, Cl, CH₃, F, CH₃, Cl), (M-8871, Cl, CH₃, F, CH₃, F), (M-8872, Cl, CH₃, F, CH₃, CF₃), (M-8873, Cl, CH₃, F, CH₃, Br), (M-8874, Cl, CH₃, F, CH₃, CH₃), (M-8875, Cl, CH₃, F, Et, H), (M-8876, Cl, CH₃, F, Et, Cl), (M-8877, Cl, CH₃, F, Et, F), (M-8878, Cl, CH₃, F, Et, CF₃), (M-8879, Cl, CH₃, F, Et, Br), (M-8880, Cl, CH₃, F, Et, CH₃), (M-8881, Cl, CH₃, F, n-Pr, H), (M-8882, Cl, CH₃, F, n-Pr, Cl), (M-8883, Cl, CH₃, F, n-Pr, F), (M-8884, Cl, CH₃, F, n-Pr, CF₃), (M-8885, Cl, CH₃, F, n-Pr, Br), (M-8886, Cl, CH₃, F, n-Pr, CH₃), (M-8887, Cl, CH₃, F, c-Pr, H), (M-8888, Cl, CH₃, F, c-Pr, Cl), (M-8889, Cl, CH₃, F, c-Pr, F), (M-8890, Cl, CH₃
, F, c-Pr, CF₃), (M-8891, Cl, CH₃, F, c-Pr, Br), (M-8892, Cl, CH₃, F, c-Pr, CH₃), (M-8893, Cl, CH₃, F, i-Pr, H), (M-8894, Cl, CH₃, F, i-Pr, Cl), (M-8895, Cl, CH₃, F, i-Pr, F), (M-8896, Cl, CH₃, F, i-Pr, CF₃), (M-8897, Cl, CH₃, F, i-Pr, Br), (M-8898, Cl, CH₃, F, i-Pr, CH₃), (M-8899, Cl, CH₃, F, n-Bu, H), (M-8900, Cl, CH₃, F, n-Bu, Cl), (M-8901, Cl, CH₃, F, n-Bu, F), (M-8902, Cl, CH₃, F, n-Bu, CF₃), (M-8903, Cl, CH₃, F, n-Bu, Br), (M-8904, Cl, CH₃, F, n-Bu, CH₃), (M-8905, Cl, CH₃, F, i-Bu, H), (M-8906, Cl, CH₃, F, i-Bu, Cl), (M-8907, Cl, CH₃, F, i-Bu, F), (M-8908, Cl, CH₃, F, i-Bu, CF₃), (M-8909, Cl, CH₃, F, i-Bu, Br), (M-8910, Cl, CH₃, F, i-Bu, CH₃), (M-8911, Cl, CH₃, F, sec-Bu, H), (M-8912, Cl, CH₃, F, sec-Bu, Cl), (M-8913, Cl, CH₃, F, sec-Bu, F), (M-8914, Cl, CH₃, F, sec-Bu, CF₃), (M-8915, Cl, CH₃, F, sec-Bu, Br), (M-8916, Cl, CH₃, F, sec-Bu, CH₃), (M-8917, Cl, CH₃, F, n-Pen, H), (M-8918, Cl, CH₃, F, n-Pen, Cl), (M-8919, Cl, CH₃, F, n-Pen, F), (M-8920, Cl, CH₃, F, n-Pen, CF₃), (M-8921, Cl, CH₃, F, n-Pen, Br), (M-8922, Cl, CH₃, F, n-Pen, CH₃), (M-8923, Cl, CH₃, F, c-Pen, H), (M-8924, Cl, CH₃, F, c-Pen, Cl), (M-8925, Cl, CH₃, F, c-Pen, F), (M-8926, Cl, CH₃, F, c-Pen, CF₃), (M-8927, Cl, CH₃, F, c-Pen, Br), (M-8928, Cl, CH₃, F, c-Pen, CH₃), (M-8929, Cl, CH₃, F, n-Hex, H), (M-8930, Cl, CH₃, F, n-Hex, Cl), (M-8931, Cl, CH₃, F, n-Hex, F), (M-8932, Cl, CH₃, F, n-Hex, CF₃), (M-8933, Cl, CH₃, F, n-Hex, Br), (M-8934, Cl, CH₃, F, n-Hex, CH₃), (M-8935, Cl, CH₃, F, c-Hex, H), (M-8936, Cl, CH₃, F, c-Hex, Cl), (M-8937, Cl, CH₃, F, c-Hex, F), (M-8938, Cl, CH₃, F, c-Hex, CF₃), (M-8939, Cl, CH₃, F, c-Hex, Br), (M-8940, Cl, CH₃, F, c-Hex, CH₃), (M-8941, Cl, CH₃, F, OH, H), (M-8942, Cl, CH₃, F, OH, Cl), (M-8943, Cl, CH₃, F, OH, F), (M-8944, Cl, CH₃, F, OH, CF₃), (M-8945, Cl, CH₃, F, OH, Br), (M-8946, Cl, CH₃, F, OH, CH₃), (M-8947, Cl, CH₃, F, EtO, H), (M-8948, Cl, CH₃, F, EtO, Cl), (M-8949, Cl, CH₃, F, EtO, F), (M-8950, Cl, CH₃, F, EtO, CF₃), (M-8951, Cl, CH₃, F, EtO, Br), (M-8952, Cl, CH₃, F, EtO, CH₃), (M-8953, Cl, CH₃, F, n-PrO, H), (M-8954, Cl, CH₃, F, n-PrO, Cl), (M-8955, Cl, CH₃, F, n-PrO, F), (M-8956, Cl, CH₃, F, n-PrO, CF₃), (M-8957, Cl, CH₃, F, n-PrO, Br), (M-8958, Cl, CH₃, F, n-PrO, CH₃), (M-8959, Cl, CH₃, F, PhO, H), (M-8960, Cl, CH₃, F, PhO, Cl), (M-8961, Cl, CH₃, F, PhO, F), (M-8962, Cl, CH₃, F, PhO, CF₃), (M-8963, Cl, CH₃, F, PhO, Br), (M-8964, Cl, CH₃, F, PhO, CH₃), (M-8965, Cl, CH₃, F, BnO, H), (M-8966, Cl, CH₃, F, BnO, Cl), (M-8967, Cl, CH₃, F, BnO, F), (M-8968, Cl, CH₃, F, BnO, CF₃), (M-8969, Cl, CH₃, F, BnO, Br), (M-8970, Cl, CH₃, F, BnO, CH₃), (M-8971, Cl, CH₃, F, PhCH₂CH₂O, H), (M-8972, Cl, CH₃, F, PhCH₂CH₂O, Cl), (M-8973, Cl, CH₃, F, PhCH₂CH₂O, F), (M-8974, Cl, CH₃, F, PhCH₂CH₂O, CF₃), (M-8975, Cl, CH₃, F, PhCH₂CH₂O, Br), (M-8976, Cl, CH₃, F, PhCH₂CH₂O, CH₃), (M-8977, Cl, CH₃, F, CF₃O, H), (M-8978, Cl, CH₃, F, CF₃O, Cl), (M-8979, Cl, CH₃, F, CF₃O, F), (M-8980, Cl, CH₃, F, CF₃O, CF₃), (M-8981, Cl, CH₃, F, CF₃O, Br), (M-8982, Cl, CH₃, F, CF₃O, CH₃), (M-8983, Cl, CH₃, F, Ph, H), (M-8984, Cl, CH₃, F, Ph, Cl), (M-8985, Cl, CH₃, F, Ph, F), (M-8986, Cl, CH₃, F, Ph, CF₃), (M-8987, Cl, CH₃, F, Ph, Br), (M-8988, Cl, CH₃, F, Ph, CH₃), (M-8989, Cl, CH₃, F, 4-F-Ph, H), (M-8990, Cl, CH₃, F, 4-F-Ph, Cl), (M-8991, Cl, CH₃, F, 4-F-Ph, F), (M-8992, Cl, CH₃, F, 4-F-Ph, CF₃), (M-8993, Cl, CH₃, F, 4-F-Ph, Br), (M-8994, Cl, CH₃, F, 4-F-Ph, CH₃), (M-8995, Cl, CH₃, F, 4-CF₃-Ph, H), (M-8996, Cl, CH₃, F, 4-CF₃-Ph, Cl), (M-8997, Cl, CH₃, F, 4-CF₃-Ph, F), (M-8998, Cl, CH₃, F, 4-CF₃-Ph, CF₃), (M-8999, Cl, CH₃, F, 4-CF₃-Ph, Br), (M-9000, Cl, CH₃, F, 4-CF₃-Ph, CH₃), (M-9001, Cl, CH₃, F, 4-(Me)₂N-Ph, H), (M-9002, Cl, CH₃, F, 4-(Me)₂N-Ph, Cl), (M-9003, Cl, CH₃, F, 4-(Me)₂N-Ph, F), (M-9004, Cl, CH₃, F, 4-(Me)₂N-Ph, CF₃), (M-9005, Cl, CH₃, F, 4-(Me)₂N-Ph, Br), (M-9006, Cl, CH₃, F, 4-(Me)₂N-Ph, CH₃), (M-9007, Cl, CH₃, F, 4-OH-Ph, H), (M-9008, Cl, CH₃, F, 4-OH-Ph, Cl), (M-9009, Cl, CH₃, F, 4-OH-Ph, F), (M-9010, Cl, CH₃, F, 4-OH-Ph, CF₃), (M-9011, Cl, CH₃, F, 4-OH-Ph, Br), (M-9012, Cl, CH₃, F, 4-OH-Ph, CH₃), (M-9013, Cl, CH₃, F, 3,4-di-F-Ph, H), (M-9014, Cl, CH₃, F, 3,4-di-F-Ph, Cl), (M-9015, Cl, CH₃, F, 3,4-di-F-Ph, F), (M-9016, Cl, CH₃, F, 3,4-di-F-Ph, CF₃), (M-9017, Cl, CH₃, F, 3,4-di-F-Ph, Br), (M-9018, Cl, CH₃, F, 3,4-di-F-Ph, CH₃), (M-9019, Cl, CH₃, F, 4-COOH-Ph, H), (M-9020, Cl, CH₃, F, 4-COOH-Ph, Cl), (M-9021, Cl, CH₃, F, 4-COOH-Ph, F), (M-9022, Cl, CH₃, F, 4-COOH-Ph, CF₃), (M-9023, Cl, CH₃, F, 4-COOH-Ph, Br), (M-9024, Cl, CH₃, F, 4-COOH-Ph, CH₃), (M-9025, Cl, CH₃, F, Bn, H), (M-9026, Cl, CH₃, F, Bn, Cl), (M-9027, Cl, CH₃, F, Bn, F), (M-9028, Cl, CH₃, F, Bn, CF₃), (M-9029, Cl, CH₃, F, Bn, Br), (M-9030, Cl, CH₃, F, Bn, CH₃), (M-9031, Cl, CH₃, F, 4-F-Bn, H), (M-9032, Cl, CH₃, F, 4-F-Bn, Cl), (M-9033, Cl, CH₃, F, 4-F-Bn, F), (M-9034, Cl, CH₃, F, 4-F-Bn, CF₃), (M-9035, Cl, CH₃, F, 4-F-Bn, Br), (M-9036, Cl, CH₃, F, 4-F-Bn, CH₃), (M-9037, Cl, CH₃, F, 2-Py, H), (M-9038, Cl, CH₃, F, 2-Py, Cl), (M-9039, Cl, CH₃, F, 2-Py, F), (M-9040, Cl, CH₃, F, 2-Py, CF₃), (M-9041, Cl, CH₃, F, 2-Py, Br), (M-9042, Cl, CH₃, F, 2-Py, CH₃), (M-9043, Cl, CH₃, F, 3-Py, H), (M-9044, Cl, CH₃, F, 3-Py, Cl), (M-9045, Cl, CH₃, F, 3-Py, F), (M-9046, Cl, CH₃, F, 3-Py, CF₃), (M-9047, Cl, CH₃, F, 3-Py, Br), (M-9048, Cl, CH₃, F, 3-Py, CH₃), (M-9049, Cl, CH₃, F, 4-Py, H), (M-9050, Cl, CH₃, F, 4-Py, Cl), (M-9051, Cl, CH₃, F, 4-Py, F), (M-9052, Cl, CH₃, F, 4-Py, CF₃), (M-9053, Cl, CH₃, F, 4-Py, Br), (M-9054, Cl, CH₃, F, 4-Py, CH₃), (M-9055, Cl, CH₃, F, 2-Th, H), (M-9056, Cl, CH₃, F, 2-Th, Cl), (M-9057, Cl, CH₃, F, 2-Th, F), (M-9058, Cl, CH₃, F, 2-Th, CF₃), (M-9059, Cl, CH₃, F, 2-Th, Br), (M-9060, Cl, CH₃, F, 2-Th, CH₃), (M-9061, Cl, CH₃, F, 3-Th, H), (M-9062, Cl, CH₃, F, 3-Th, Cl), (M-9063, Cl, CH₃, F, 3-Th, F), (M-9064, Cl, CH₃, F, 3-Th, CF₃), (M-9065, Cl, CH₃, F, 3-Th, Br), (M-9066, Cl, CH₃, F, 3-Th, CH₃), (M-9067, Cl, CH₃, F, pyrazol-2-yl, H), (M-9068, Cl, CH₃, F, pyrazol-2-yl, Cl), (M-9069, Cl, CH₃, F, pyrazol-2-yl, F), (M-9070, Cl, CH₃, F, pyrazol-2-yl, CF₃), (M-9071, Cl, CH₃, F, pyrazol-2-yl, Br), (M-9072, Cl, CH₃, F, pyrazol-2-yl, CH₃), (M-9073, Cl, CH₃, F, pyrazol-3-yl, H), (M-9074, Cl, CH₃, F, pyrazol-3-yl, Cl), (M-9075, Cl, CH₃, F, pyrazol-3-yl, F), (M-9076, Cl, CH₃, F, pyrazol-3-yl, CF₃), (M-9077, Cl, CH₃, F, pyrazol-3-yl, Br), (M-9078, Cl, CH₃, F, pyrazol-3-yl, CH₃), (M-9079, Cl, CH₃, F, pyrimidin-2-yl, H), (M-9080, Cl, CH₃, F, pyrimidin-2-yl, Cl), (M-9081, Cl, CH₃, F, pyrimidin-2-yl, F), (M-9082, Cl, CH₃, F, pyrimidin-2-yl, CF₃), (M-9083, Cl, CH₃, F, pyrimidin-2-yl, Br), (M-9084, Cl, CH₃, F, pyrimidin-2-yl, CH₃), (M-9085, Cl, CH₃, F, pyrimidin-4-yl, H), (M-9086, Cl, CH₃, F, pyrimidin-4-yl, Cl), (M-9087, Cl, CH₃, F, pyrimidin-4-yl, F), (M-9088, Cl, CH₃, F, pyrimidin-4-yl, CF₃), (M-9089, Cl, CH₃, F, pyrimidin-4-yl, Br), (M-9090, Cl, CH₃, F, pyrimidin-4-yl, CH₃), (M-9091, Cl, CH₃, F, pyrimidin-5-yl, H), (M-9092, Cl, CH₃, F, pyrimidin-5-yl, Cl), (M-9093, Cl, CH₃
, F, pyrimidin-5-yl, F), (M-9094, Cl, CH₃, F, pyrimidin-5-yl, CF₃), (M-9095, Cl, CH₃, F, pyrimidin-5-yl, Br), (M-9096, Cl, CH₃, F, pyrimidin-5-yl, CH₃), (M-9097, Cl, CH₃, F, HOOCCH₂CH₂CH₂, H), (M-9098, Cl, CH₃, F, HOOCCH₂CH₂CH₂, Cl), (M-9099, Cl, CH₃, F, HOOCCH₂CH₂CH₂, F), (M-9100, Cl, CH₃, F, HOOCCH₂CH₂CH₂, CF₃), (M-9101, Cl, CH₃, F, HOOCCH₂CH₂CH₂, Br), (M-9102, Cl, CH₃, F, HOOCCH₂CH₂CH₂, CH₃), (M-9103, Cl, CH₃, F, HOOCCH₂CH₂CH₂CH₂, H), (M-9104, Cl, CH₃, F, HOOCCH₂CH₂CH₂CH₂, Cl), (M-9105, Cl, CH₃, F, HOOCCH₂CH₂CH₂CH₂, F), (M-9106, Cl, CH₃, F, HOOCCH₂CH₂CH₂CH₂, CF₃), (M-9107, Cl, CH₃, F, HOOCCH₂CH₂CH₂CH₂, Br), (M-9108, Cl, CH₃, F, HOOCCH₂CH₂CH₂CH₂, CH₃), (M-9109, Cl, CH₃, F, (Me)₂NCOCH₂CH₂CH₂CH₂, H), (M-9110, Cl, CH₃, F, (Me)₂NCOCH₂CH₂CH₂CH₂, Cl), (M-9111, Cl, CH₃, F, (Me)₂NCOCH₂CH₂CH₂CH₂, F), (M-9112, Cl, CH₃, F, (Me)₂NCOCH₂CH₂CH₂CH₂, CF₃), (M-9113, Cl, CH₃, F, (Me)₂NCOCH₂CH₂CH₂CH₂, Br), (M-9114, Cl, CH₃, F, (Me)₂NCOCH₂CH₂CH₂CH₂, CH₃), (M-9115, Cl, CH₃, F, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, H), (M-9116, Cl, CH₃, F, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, Cl), (M-9117, Cl, CH₃, F, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, F), (M-9118, Cl, CH₃, F, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, CF₃), (M-9119, Cl, CH₃, F, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, Br), (M-9120, Cl, CH₃, F, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, CH₃), (M-9121, Cl, CH₃, F, MeOCH₂, H), (M-9122, Cl, CH₃, F, MeOCH₂, Cl), (M-9123, Cl, CH₃, F, MeOCH₂, F), (M-9124, Cl, CH₃, F, MeOCH₂, CF₃), (M-9125, Cl, CH₃, F, MeOCH₂, Br), (M-9126, Cl, CH₃, F, MeOCH₂, CH₃), (M-9127, Cl, CH₃, F, EtOCH₂, H), (M-9128, Cl, CH₃, F, EtOCH₂, Cl), (M-9129, Cl, CH₃, F, EtOCH₂, F), (M-9130, Cl, CH₃, F, EtOCH₂, CF₃), (M-9131, Cl, CH₃, F, EtOCH₂, Br), (M-9132, Cl, CH₃, F, EtOCH₂, CH₃), (M-9133, Cl, CH₃, F, EtOCH₂CH₂, H), (M-9134, Cl, CH₃, F, EtOCH₂CH₂, Cl), (M-9135, Cl, CH₃, F, EtOCH₂CH₂, F), (M-9136, Cl, CH₃, F, EtOCH₂CH₂, CF₃), (M-9137, Cl, CH₃, F, EtOCH₂CH₂, Br), (M-9138, Cl, CH₃, F, EtOCH₂CH₂, CH₃), (M-9139, Cl, CH₃, F, MeOCH₂CH₂OCH₂CH₂, H), (M-9140, Cl, CH₃, F, MeOCH₂CH₂OCH₂CH₂, Cl), (M-9141, Cl, CH₃, F, MeOCH₂CH₂OCH₂CH₂, F), (M-9142, Cl, CH₃, F, MeOCH₂CH₂OCH₂CH₂, CF₃), (M-9143, Cl, CH₃, F, MeOCH₂CH₂OCH₂CH₂, Br), (M-9144, Cl, CH₃, F, MeOCH₂CH₂OCH₂CH₂, CH₃), (M-9145, Cl, CH₃, F, MeOCH₂CH₂, H), (M-9146, Cl, CH₃, F, MeOCH₂CH₂, Cl), (M-9147, Cl, CH₃, F, MeOCH₂CH₂, F), (M-9148, Cl, CH₃, F, MeOCH₂CH₂, CF₃), (M-9149, Cl, CH₃, F, MeOCH₂CH₂, Br), (M-9150, Cl, CH₃, F, MeOCH₂CH₂, CH₃), (M-9151, Cl, CH₃, F, HOCH₂, H), (M-9152, Cl, CH₃, F, HOCH₂, Cl), (M-9153, Cl, CH₃, F, HOCH₂, F), (M-9154, Cl, CH₃, F, HOCH₂, CF₃), (M-9155, Cl, CH₃, F, HOCH₂, Br), (M-9156, Cl, CH₃, F, HOCH₂, CH₃), (M-9157, Cl, CH₃, F, HOCH₂CH₂, H), (M-9158, Cl, CH₃, F, HOCH₂CH₂, Cl), (M-9159, Cl, CH₃, F, HOCH₂CH₂, F), (M-9160, Cl, CH₃, F, HOCH₂CH₂, CF₃), (M-9161, Cl, CH₃, F, HOCH₂CH₂, Br), (M-9162, Cl, CH₃, F, HOCH₂CH₂, CH₃), (M-9163, Cl, CH₃, F, HOCH₂CH₂CH₂, H), (M-9164, Cl, CH₃, F, HOCH₂CH₂CH₂, Cl), (M-9165, Cl, CH₃, F, HOCH₂CH₂CH₂, F), (M-9166, Cl, CH₃, F, HOCH₂CH₂CH₂, CF₃), (M-9167, Cl, CH₃, F, HOCH₂CH₂CH₂, Br), (M-9168, Cl, CH₃, F, HOCH₂CH₂CH₂, CH₃), (M-9169, Cl, CH₃, F, HOCH₂CH₂CH₂CH₂, H), (M-9170, Cl, CH₃, F, HOCH₂CH₂CH₂CH₂, Cl), (M-9171, Cl, CH₃, F, HOCH₂CH₂CH₂CH₂, F), (M-9172, Cl, CH₃, F, HOCH₂CH₂CH₂CH₂, CF₃), (M-9173, Cl, CH₃, F, HOCH₂CH₂CH₂CH₂, Br), (M-9174, Cl, CH₃, F, HOCH₂CH₂CH₂CH₂, CH₃), (M-9175, Cl, CH₃, F, HOCH₂CH₂CH₂CH₂CH₂, H), (M-9176, Cl, CH₃, F, HOCH₂CH₂CH₂CH₂CH₂, Cl), (M-9177, Cl, CH₃, F, HOCH₂CH₂CH₂CH₂CH₂, F), (M-9178, Cl, CH₃, F, HOCH₂CH₂CH₂CH₂CH₂, CF₃), (M-9179, Cl, CH₃, F, HOCH₂CH₂CH₂CH₂CH₂, Br), (M-9180, Cl, CH₃, F, HOCH₂CH₂CH₂CH₂CH₂, CH₃), (M-9181, Cl, CH₃, F, HOCH₂CH₂OCH₂CH₂, H), (M-9182, Cl, CH₃, F, HOCH₂CH₂OCH₂CH₂, Cl), (M-9183, Cl, CH₃, F, HOCH₂CH₂OCH₂CH₂, F), (M-9184, Cl, CH₃, F, HOCH₂CH₂OCH₂CH₂, CF₃), (M-9185, Cl, CH₃, F, HOCH₂CH₂OCH₂CH₂, Br), (M-9186, Cl, CH₃, F, HOCH₂CH₂OCH₂CH₂, CH₃), (M-9187, Cl, CH₃, F, (Me)₂N, H), (M-9188, Cl, CH₃, F, (Me)₂N, Cl), (M-9189, Cl, CH₃, F, (Me)₂N, F), (M-9190, Cl, CH₃, F, (Me)₂N, CF₃), (M-9191, Cl, CH₃, F, (Me)₂N, Br), (M-9192, Cl, CH₃, F, (Me)₂N, CH₃), (M-9193, Cl, CH₃, F, piperidin-4-yl-methyl, H), (M-9194, Cl, CH₃, F, piperidin-4-yl-methyl, Cl), (M-9195, Cl, CH₃, F, piperidin-4-yl-methyl, F), (M-9196, Cl, CH₃, F, piperidin-4-yl-methyl, CF₃), (M-9197, Cl, CH₃, F, piperidin-4-yl-methyl, Br), (M-9198, Cl, CH₃, F, piperidin-4-yl-methyl, CH₃), (M-9199, Cl, CH₃, F, cyclohexylmethyl, H), (M-9200, Cl, CH₃, F, cyclohexylmethyl, Cl), (M-9201, Cl, CH₃, F, cyclohexylmethyl, F), (M-9202, Cl, CH₃, F, cyclohexylmethyl, CF₃), (M-9203, Cl, CH₃, F, cyclohexylmethyl, Br), (M-9204, Cl, CH₃, F, cyclohexylmethyl, CH₃), (M-9205, Cl, CH₃, Cl, H, H), (M-9206, Cl, CH₃, Cl, H, Cl), (M-9207, Cl, CH₃, Cl, H, F), (M-9208, Cl, CH₃, Cl, H, CF₃), (M-9209, Cl, CH₃, Cl, H, Br), (M-9210, Cl, CH₃, Cl, H, CH₃), (M-9211, Cl, CH₃, Cl, F, H), (M-9212, Cl, CH₃, Cl, F, Cl), (M-9213, Cl, CH₃, Cl, F, F), (M-9214, Cl, CH₃, Cl, F, CF₃), (M-9215, Cl, CH₃, Cl, F, Br), (M-9216, Cl, CH₃, Cl, F, CH₃), (M-9217, Cl, CH₃, Cl, Cl, H), (M-9218, Cl, CH₃, Cl, Cl, Cl), (M-9219, Cl, CH₃, Cl, Cl, F), (M-9220, Cl, CH₃, Cl, Cl, CF₃), (M-9221, Cl, CH₃, Cl, Cl, Br), (M-9222, Cl, CH₃, Cl, Cl, CH₃), (M-9223, Cl, CH₃, Cl, CH₃, H), (M-9224,
Cl, CH₃, Cl, CH₃, Cl), (M-9225, Cl, CH₃, Cl, CH₃, F), (M-9226, Cl, CH₃, Cl, CH₃, CF₃), (M-9227, Cl, CH₃, Cl, CH₃, Br), (M-9228, Cl, CH₃, Cl, CH₃, CH₃), (M-9229, Cl, CH₃, Cl, Et, H), (M-9230, Cl, CH₃, Cl, Et, Cl), (M-9231, Cl, CH₃, Cl, Et, F), (M-9232, Cl, CH₃, Cl, Et, CF₃), (M-9233, Cl, CH₃, Cl, Et, Br), (M-9234, Cl, CH₃, Cl, Et, CH₃), (M-9235, Cl, CH₃, Cl, n-Pr, H), (M-9236, Cl, CH₃, Cl, n-Pr, Cl), (M-9237, Cl, CH₃, Cl, n-Pr, F), (M-9238, Cl, CH₃, Cl, n-Pr, CF₃), (M-9239, Cl, CH₃, Cl, n-Pr, Br), (M-9240, Cl, CH₃, Cl, n-Pr, CH₃), (M-9241, Cl, CH₃, Cl, c-Pr, H), (M-9242, Cl, CH₃, Cl, c-Pr, Cl), (M-9243, Cl, CH₃, Cl, c-Pr, F), (M-9244, Cl, CH₃, Cl, c-Pr, CF₃), (M-9245, Cl, CH₃, Cl, c-Pr, Br), (M-9246, Cl, CH₃, Cl, c-Pr, CH₃), (M-9247, Cl, CH₃, Cl, i-Pr, H), (M-9248, Cl, CH₃, Cl, i-Pr, Cl), (M-9249, Cl, CH₃, Cl, i-Pr, F), (M-9250, Cl, CH₃, Cl, i-Pr, CF₃), (M-9251, Cl, CH₃, Cl, i-Pr, Br), (M-9252, Cl, CH₃, Cl, i-Pr, CH₃), (M-9253, Cl, CH₃, Cl, n-Bu, H), (M-9254, Cl, CH₃, Cl, n-Bu, Cl), (M-9255, Cl, CH₃, Cl, n-Bu, F), (M-9256, Cl, CH₃, Cl, n-Bu, CF₃), (M-9257, Cl, CH₃, Cl, n-Bu, Br), (M-9258, Cl, CH₃, Cl, n-Bu, CH₃), (M-9259, Cl, CH₃, Cl, i-Bu, H), (M-9260, Cl, CH₃, Cl, i-Bu, Cl), (M-9261, Cl, CH₃, Cl, i-Bu, F), (M-9262, Cl, CH₃, Cl, i-Bu, CF₃), (M-9263, Cl, CH₃, Cl, i-Bu, Br), (M-9264, Cl, CH₃, Cl, i-Bu, CH₃), (M-9265, Cl, CH₃, Cl, sec-Bu, H), (M-9266, Cl, CH₃, Cl, sec-Bu, Cl), (M-9267, Cl, CH₃, Cl, sec-Bu, F), (M-9268, Cl, CH₃, Cl, sec-Bu, CF₃), (M-9269, Cl, CH₃, Cl, sec-Bu, Br), (M-9270, Cl, CH₃, Cl, sec-Bu, CH₃), (M-9271, Cl, CH₃, Cl, n-Pen, H), (M-9272, Cl, CH₃, Cl, n-Pen, Cl), (M-9273, Cl, CH₃, Cl, n-Pen, F), (M-9274, Cl, CH₃, Cl, n-Pen, CF₃), (M-9275, Cl, CH₃, Cl, n-Pen, Br), (M-9276, Cl, CH₃, Cl, n-Pen, CH₃), (M-9277, Cl, CH₃, Cl, c-Pen, H), (M-9278, Cl, CH₃, Cl, c-Pen, Cl), (M-9279, Cl, CH₃, Cl, c-Pen, F), (M-9280, Cl, CH₃, Cl, c-Pen, CF₃), (M-9281, Cl, CH₃, Cl, c-Pen, Br), (M-9282, Cl, CH₃, Cl, c-Pen, CH₃), (M-9283, Cl, CH₃, Cl, n-Hex, H), (M-9284, Cl, CH₃, Cl, n-Hex, Cl), (M-9285, Cl, CH₃, Cl, n-Hex, F), (M-9286, Cl, CH₃, Cl, n-Hex, CF₃), (M-9287, Cl, CH₃, Cl, n-Hex, Br), (M-9288, Cl, CH₃, Cl, n-Hex, CH₃), (M-9289, Cl, CH₃, Cl, c-Hex, H), (M-9290, Cl, CH₃, Cl, c-Hex, Cl), (M-9291, Cl, CH₃, Cl, c-Hex, F), (M-9292, Cl, CH₃, Cl, c-Hex, CF₃), (M-9293, Cl, CH₃, Cl, c-Hex, Br), (M-9294, Cl, CH₃, Cl, c-Hex, CH₃), (M-9295, Cl, CH₃, Cl, OH, H), (M-9296, Cl, CH₃, Cl, OH, Cl), (M-9297, Cl, CH₃, Cl, OH, F), (M-9298, Cl, CH₃, Cl, OH, CF₃), (M-9299, Cl, CH₃, Cl, OH, Br), (M-9300, Cl, CH₃, Cl, OH, CH₃), (M-9301, Cl, CH₃, Cl, EtO, H), (M-9302, Cl, CH₃, Cl, EtO, Cl), (M-9303, Cl, CH₃, Cl, EtO, F), (M-9304, Cl, CH₃, Cl, EtO, CF₃), (M-9305, Cl, CH₃, Cl, EtO, Br), (M-9306, Cl, CH₃, Cl, EtO, CH₃), (M-9307, Cl, CH₃, Cl, n-PrO, H), (M-9308, Cl, CH₃, Cl, n-PrO, Cl), (M-9309, Cl, CH₃, Cl, n-PrO, F), (M-9310, Cl, CH₃, Cl, n-PrO, CF₃), (M-9311, Cl, CH₃, Cl, n-PrO, Br), (M-9312, Cl, CH₃, Cl, n-PrO, CH₃), (M-9313, Cl, CH₃, Cl, PhO, H), (M-9314, Cl, CH₃, Cl, PhO, Cl), (M-9315, Cl, CH₃, Cl, PhO, F), (M-9316, Cl, CH₃, Cl, PhO, CF₃), (M-9317, Cl, CH₃, Cl, PhO, Br), (M-9318, Cl, CH₃, Cl, PhO, CH₃), (M-9319, Cl, CH₃, Cl, BnO, H), (M-9320, Cl, CH₃, Cl, BnO, Cl), (M-9321, Cl, CH₃, Cl, BnO, F), (M-9322, Cl, CH₃, Cl, BnO, CF₃), (M-9323, Cl, CH₃, Cl, BnO, Br), (M-9324, Cl, CH₃, Cl, BnO, CH₃), (M-9325, Cl, CH₃, Cl, PhCH₂CH₂O, H), (M-9326, Cl, CH₃, Cl, PhCH₂CH₂O, Cl), (M-9327, Cl, CH₃, Cl, PhCH₂CH₂O, F), (M-9328, Cl, CH₃, Cl, PhCH₂CH₂O, CF₃), (M-9329, Cl, CH₃, Cl, PhCH₂CH₂O, Br), (M-9330, Cl, CH₃, Cl, PhCH₂CH₂O, CH₃), (M-9331, Cl, CH₃, Cl, CF₃O, H), (M-9332, Cl, CH₃, Cl, CF₃O, Cl), (M-9333, Cl, CH₃, Cl, CF₃O, F), (M-9334, Cl, CH₃, Cl, CF₃O, CF₃), (M-9335, Cl, CH₃, Cl, CF₃O, Br), (M-9336, Cl, CH₃, Cl, CF₃O, CH₃), (M-9337, Cl, CH₃, Cl, Ph, H), (M-9338, Cl, CH₃, Cl, Ph, Cl), (M-9339, Cl, CH₃, Cl, Ph, F), (M-9340, Cl, CH₃, Cl, Ph, CF₃), (M-9341, Cl, CH₃, Cl, Ph, Br), (M-9342, Cl, CH₃, Cl, Ph, CH₃), (M-9343, Cl, CH₃, Cl, 4-F-Ph, H), (M-9344, Cl, CH₃, Cl, 4-F-Ph, Cl), (M-9345, Cl, CH₃, Cl, 4-F-Ph, F), (M-9346, Cl, CH₃, Cl, 4-F-Ph, CF₃), (M-9347, Cl, CH₃, Cl, 4-F-Ph, Br), (M-9348, Cl, CH₃, Cl, 4-F-Ph, CH₃), (M-9349, Cl, CH₃, Cl, 4-CF₃-Ph, H), (M-9350, Cl, CH₃, Cl, 4-CF₃-Ph, Cl), (M-9351, Cl, CH₃, Cl, 4-CF₃-Ph, F), (M-9352, Cl, CH₃, Cl, 4-CF₃-Ph, CF₃), (M-9353, Cl, CH₃, Cl, 4-CF₃-Ph, Br), (M-9354, Cl, CH₃, Cl, 4-CF₃-Ph, CH₃), (M-9355, Cl, CH₃, Cl, 4-(Me)₂N-Ph, H), (M-9356, Cl, CH₃, Cl, 4-(Me)₂N-Ph, Cl), (M-9357, Cl, CH₃, Cl, 4-(Me)₂N-Ph, F), (M-9358, Cl, CH₃, Cl, 4-(Me)₂N-Ph, CF₃), (M-9359, Cl, CH₃, Cl, 4-(Me)₂N-Ph, Br), (M-9360, Cl, CH₃, Cl, 4-(Me)₂N-Ph, CH₃), (M-9361, Cl, CH₃, Cl, 4-OH-Ph, H), (M-9362, Cl, CH₃, Cl, 4-OH-Ph, Cl), (M-9363, Cl, CH₃, Cl, 4-OH-Ph, F), (M-9364, Cl, CH₃, Cl, 4-OH-Ph, CF₃), (M-9365, Cl, CH₃, Cl, 4-OH-Ph, Br), (M-9366, Cl, CH₃, Cl, 4-OH-Ph, CH₃), (M-9367, Cl, CH₃, Cl, 3,4-di-F-Ph, H), (M-9368, Cl, CH₃, Cl, 3,4-di-F-Ph, Cl), (M-9369, Cl, CH₃, Cl, 3,4-di-F-Ph, F), (M-9370, Cl, CH₃, Cl, 3,4-di-F-Ph, CF₃), (M-9371, Cl, CH₃, Cl, 3,4-di-F-Ph, Br), (M-9372, Cl, CH₃, Cl, 3,4-di-F-Ph, CH₃), (M-9373, Cl, CH₃, Cl, 4-COOH-Ph, H), (M-9374, Cl, CH₃, Cl, 4-COOH-Ph, Cl), (M-9375, Cl, CH₃, Cl, 4-COOH-Ph, F), (M-9376, Cl, CH₃, Cl, 4-COOH-Ph, CF₃), (M-9377, Cl, CH₃, Cl, 4-COOH-Ph, Br), (M-9378, Cl, CH₃, Cl, 4-COOH-Ph, CH₃), (M-9379, Cl, CH₃, Cl, Bn, H), (M-9380, Cl, CH₃, Cl, Bn, Cl), (M-9381, Cl, CH₃, Cl, Bn, F), (M-9382, Cl, CH₃, Cl, Bn, CF₃), (M-9383, Cl, CH₃, Cl, Bn, Br), (M-9384, Cl, CH₃, Cl, Bn, CH₃), (M-9385, Cl, CH₃, Cl, 4-F-Bn, H), (M-9386, Cl, CH₃, Cl, 4-F-Bn, Cl), (M-9387, Cl, CH₃, Cl, 4-F-Bn, F), (M-9388, Cl, CH₃, Cl, 4-F-Bn, CF₃), (M-9389, Cl, CH₃, Cl, 4-F-Bn, Br), (M-9390, Cl, CH₃, Cl, 4-F-Bn, CH₃), (M-9391, Cl, CH₃, Cl, 2-Py, H), (M-9392, Cl, CH₃, Cl, 2-Py, Cl), (M-9393, Cl, CH₃, Cl, 2-Py, F), (M-9394, Cl, CH₃, Cl, 2-Py, CF₃), (M-9395, Cl, CH₃, Cl, 2-Py, Br), (M-9396, Cl, CH₃, Cl, 2-Py, CH₃), (M-9397, Cl, CH₃, Cl, 3-Py, H), (M-9398, Cl, CH₃, Cl, 3-Py, Cl), (M-9399, Cl, CH₃, Cl, 3-Py, F), (M-9400, Cl, CH₃, Cl, 3-Py, CF₃), (M-9401, Cl, CH₃, Cl, 3-Py, Br), (M-9402, Cl, CH₃, Cl, 3-Py, CH₃), (M-9403, Cl, CH₃, Cl, 4-Py, H), (M-9404, Cl, CH₃, Cl, 4-Py, Cl), (M-9405, Cl, CH₃, Cl, 4-Py, F), (M-9406, Cl, CH₃, Cl, 4-Py, CF₃), (M-9407, Cl, CH₃, Cl, 4-Py, Br), (M-9408, Cl, CH₃, Cl, 4-Py, CH₃), (M-9409, Cl, CH₃, Cl, 2-Th, H), (M-9410, Cl, CH₃, Cl, 2-Th, Cl), (M-9411, Cl, CH₃, Cl, 2-Th, F), (M-9412, Cl, CH₃, Cl, 2-Th, CF₃), (M-9413, Cl, CH₃, Cl, 2-Th, Br), (M-9414, Cl, CH₃, Cl, 2-Th, CH₃), (M-9415, Cl, CH₃, Cl, 3-Th, H), (M-9416, Cl, CH₃, Cl, 3-Th, Cl), (M-9417, Cl, CH₃, Cl, 3-Th, F), (M-9418, Cl, CH₃, Cl, 3-Th, CF₃), (M-9419, Cl, CH₃, Cl, 3-Th, Br), (M-9420, Cl, CH₃, Cl, 3-Th, CH₃), (M-9421, Cl, CH₃, Cl, pyrazol-2-yl, H), (M-9422, Cl, CH₃, Cl, pyrazol-2-yl, Cl), (M-9423, Cl, CH₃, Cl, pyrazol-2-yl, F), (M-9424, Cl, CH₃, Cl, pyrazol-2-yl, CF₃), (M-9425, Cl, CH₃, Cl, pyrazol-2-yl, Br), (M-9426, Cl, CH
₃, Cl, pyrazol-2-yl, CH₃), (M-9427, Cl, CH₃, Cl, pyrazol-3-yl, H), (M-9428, Cl, CH₃, Cl, pyrazol-3-yl, Cl), (M-9429, Cl, CH₃, Cl, pyrazol-3-yl, F), (M-9430, Cl, CH₃, Cl, pyrazol-3-yl, CF₃), (M-9431, Cl, CH₃, Cl, pyrazol-3-yl, Br), (M-9432, Cl, CH₃, Cl, pyrazol-3-yl, CH₃), (M-9433, Cl, CH₃, Cl, pyrimidin-2-yl, H), (M-9434, Cl, CH₃, Cl, pyrimidin-2-yl, Cl), (M-9435, Cl, CH₃, Cl, pyrimidin-2-yl, F), (M-9436, Cl, CH₃, Cl, pyrimidin-2-yl, CF₃), (M-9437, Cl, CH₃, Cl, pyrimidin-2-yl, Br), (M-9438, Cl, CH₃, Cl, pyrimidin-2-yl, CH₃), (M-9439, Cl, CH₃, Cl, pyrimidin-4-yl, H), (M-9440, Cl, CH₃, Cl, pyrimidin-4-yl, Cl), (M-9441, Cl, CH₃, Cl, pyrimidin-4-yl, F), (M-9442, Cl, CH₃, Cl, pyrimidin-4-yl, CF₃), (M-9443, Cl, CH₃, Cl, pyrimidin-4-yl, Br), (M-9444, Cl, CH₃, Cl, pyrimidin-4-yl, CH₃), (M-9445, Cl, CH₃, Cl, pyrimidin-5-yl, H), (M-9446, Cl, CH₃, Cl, pyrimidin-5-yl, Cl), (M-9447, Cl, CH₃, Cl, pyrimidin-5-yl, F), (M-9448, Cl, CH₃, Cl, pyrimidin-5-yl, CF₃), (M-9449, Cl, CH₃, Cl, pyrimidin-5-yl, Br), (M-9450, Cl, CH₃, Cl, pyrimidin-5-yl, CH₃), (M-9451, Cl, CH₃, Cl, HOOCCH₂CH₂CH₂, H), (M-9452, Cl, CH₃, Cl, HOOCCH₂CH₂CH₂, Cl), (M-9453, Cl, CH₃, Cl, HOOCCH₂CH₂CH₂, F), (M-9454, Cl, CH₃, Cl, HOOCCH₂CH₂CH₂, CF₃), (M-9455, Cl, CH₃, Cl, HOOCCH₂CH₂CH₂, Br), (M-9456, Cl, CH₃, Cl, HOOCCH₂CH₂CH₂, CH₃), (M-9457, Cl, CH₃, Cl, HOOCCH₂CH₂CH₂CH₂, H), (M-9458, Cl, CH₃, Cl, HOOCCH₂CH₂CH₂CH₂, Cl), (M-9459, Cl, CH₃, Cl, HOOCCH₂CH₂CH₂CH₂, F), (M-9460, Cl, CH₃, Cl, HOOCCH₂CH₂CH₂CH₂, CF₃), (M-9461, Cl, CH₃, Cl, HOOCCH₂CH₂CH₂CH₂, Br), (M-9462, Cl, CH₃, Cl, HOOCCH₂CH₂CH₂CH₂, CH₃), (M-9463, Cl, CH₃, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂, H), (M-9464, Cl, CH₃, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂, Cl), (M-9465, Cl, CH₃, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂, F), (M-9466, Cl, CH₃, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂, CF₃), (M-9467, Cl, CH₃, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂, Br), (M-9468, Cl, CH₃, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂, CH₃), (M-9469, Cl, CH₃, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, H), (M-9470, Cl, CH₃, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, Cl), (M-9471, Cl, CH₃, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, F), (M-9472, Cl, CH₃, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, CF₃), (M-9473, Cl, CH₃, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, Br), (M-9474, Cl, CH₃, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, CH₃), (M-9475, Cl, CH₃, Cl, MeOCH₂, H), (M-9476, Cl, CH₃, Cl, MeOCH₂, Cl), (M-9477, Cl, CH₃, Cl, MeOCH₂, F), (M-9478, Cl, CH₃, Cl, MeOCH₂, CF₃), (M-9479, Cl, CH₃, Cl, MeOCH₂, Br), (M-9480, Cl, CH₃, Cl, MeOCH₂, CH₃), (M-9481, Cl, CH₃, Cl, EtOCH₂, H), (M-9482, Cl, CH₃, Cl, EtOCH₂, Cl), (M-9483, Cl, CH₃, Cl, EtOCH₂, F), (M-9484, Cl, CH₃, Cl, EtOCH₂, CF₃), (M-9485, Cl, CH₃, Cl, EtOCH₂, Br), (M-9486, Cl, CH₃, Cl, EtOCH₂, CH₃), (M-9487, Cl, CH₃, Cl, EtOCH₂CH₂, H), (M-9488, Cl, CH₃, Cl, EtOCH₂CH₂, Cl), (M-9489, Cl, CH₃, Cl, EtOCH₂CH₂, F), (M-9490, Cl, CH₃, Cl, EtOCH₂CH₂, CF₃), (M-9491, Cl, CH₃, Cl, EtOCH₂CH₂, Br), (M-9492, Cl, CH₃, Cl, EtOCH₂CH₂, CH₃), (M-9493, Cl, CH₃, Cl, MeOCH₂CH₂OCH₂CH₂, H), (M-9494, Cl, CH₃, Cl, MeOCH₂CH₂OCH₂CH₂, Cl), (M-9495, Cl, CH₃, Cl, MeOCH₂CH₂OCH₂CH₂, F), (M-9496, Cl, CH₃, Cl, MeOCH₂CH₂OCH₂CH₂, CF₃), (M-9497, Cl, CH₃, Cl, MeOCH₂CH₂OCH₂CH₂, Br), (M-9498, Cl, CH₃, Cl, MeOCH₂CH₂OCH₂CH₂, CH₃), (M-9499, Cl, CH₃, Cl, MeOCH₂CH₂, H), (M-9500, Cl, CH₃, Cl, MeOCH₂CH₂, Cl), (M-9501, Cl, CH₃, Cl, MeOCH₂CH₂, F), (M-9502, Cl, CH₃, Cl, MeOCH₂CH₂, CF₃), (M-9503, Cl, CH₃, Cl, MeOCH₂CH₂, Br), (M-9504, Cl, CH₃, Cl, MeOCH₂CH₂, CH₃), (M-9505, Cl, CH₃, Cl, HOCH₂, H), (M-9506, Cl, CH₃, Cl, HOCH₂, Cl), (M-9507, Cl, CH₃, Cl, HOCH₂, F), (M-9508, Cl, CH₃, Cl, HOCH₂, CF₃), (M-9509, Cl, CH₃, Cl, HOCH₂, Br), (M-9510, Cl, CH₃, Cl, HOCH₂, CH₃), (M-9511, Cl, CH₃, Cl, HOCH₂CH₂, H), (M-9512, Cl, CH₃, Cl, HOCH₂CH₂, Cl), (M-9513, Cl, CH₃, Cl, HOCH₂CH₂, F), (M-9514, Cl, CH₃, Cl, HOCH₂CH₂, CF₃), (M-9515, Cl, CH₃, Cl, HOCH₂CH₂, Br), (M-9516, Cl, CH₃, Cl, HOCH₂CH₂, CH₃), (M-9517, Cl, CH₃, Cl, HOCH₂CH₂CH₂, H), (M-9518, Cl, CH₃, Cl, HOCH₂CH₂CH₂, Cl), (M-9519, Cl, CH₃, Cl, HOCH₂CH₂CH₂, F), (M-9520, Cl, CH₃, Cl, HOCH₂CH₂CH₂, CF₃), (M-9521, Cl, CH₃, Cl, HOCH₂CH₂CH₂, Br), (M-9522, Cl, CH₃, Cl, HOCH₂CH₂CH₂, CH₃), (M-9523, Cl, CH₃, Cl, HOCH₂CH₂CH₂CH₂, H), (M-9524, Cl, CH₃, Cl, HOCH₂CH₂CH₂CH₂, Cl), (M-9525, Cl, CH₃, Cl, HOCH₂CH₂CH₂CH₂, F), (M-9526, Cl, CH₃, Cl, HOCH₂CH₂CH₂CH₂, CF₃), (M-9527, Cl, CH₃, Cl, HOCH₂CH₂CH₂CH₂, Br), (M-9528, Cl, CH₃, Cl, HOCH₂CH₂CH₂CH₂, CH₃), (M-9529, Cl, CH₃, Cl, HOCH₂CH₂CH₂CH₂CH₂, H), (M-9530, Cl, CH₃, Cl, HOCH₂CH₂CH₂CH₂CH₂, Cl), (M-9531, Cl, CH₃, Cl, HOCH₂CH₂CH₂CH₂CH₂, F), (M-9532, Cl, CH₃, Cl, HOCH₂CH₂CH₂CH₂CH₂, CF₃), (M-9533, Cl, CH₃, Cl, HOCH₂CH₂CH₂CH₂CH₂, Br), (M-9534, Cl, CH₃, Cl, HOCH₂CH₂CH₂CH₂CH₂, CH₃), (M-9535, Cl, CH₃, Cl, HOCH₂CH₂OCH₂CH₂, H), (M-9536, Cl, CH₃, Cl, HOCH₂CH₂OCH₂CH₂, Cl), (M-9537, Cl, CH₃, Cl, HOCH₂CH₂OCH₂CH₂, F), (M-9538, Cl, CH₃, Cl, HOCH₂CH₂OCH₂CH₂, CF₃), (M-9539, Cl, CH₃, Cl, HOCH₂CH₂OCH₂CH₂, Br), (M-9540, Cl, CH₃, Cl, HOCH₂CH₂OCH₂CH₂, CH₃), (M-9541, Cl, CH₃, Cl, (Me)₂N, H), (M-9542, Cl, CH₃, Cl, (Me)₂N, Cl), (M-9543, Cl, CH₃, Cl, (Me)₂N, F), (M-9544, Cl, CH₃, Cl, (Me)₂N, CF₃), (M-9545, Cl, CH₃, Cl, (Me)₂N, Br), (M-9546, Cl, CH₃, Cl, (Me)₂N, CH₃), (M-9547, Cl, CH₃, Cl, piperidin-4-yl-methyl, H), (M-9548, Cl, CH₃, Cl, piperidin-4-yl-methyl, Cl), (M-9549, Cl, CH₃, Cl, piperidin-4-yl-methyl, F), (M-9550, Cl, CH₃, Cl, piperidin-4-yl-methyl, CF₃), (M-9551, Cl, CH₃, Cl, piperidin-4-yl
-methyl, Br), (M-9552, Cl, CH₃, Cl, piperidin-4-yl-methyl, CH₃), (M-9553, Cl, CH₃, Cl, cyclohexylmethyl, H), (M-9554, Cl, CH₃, Cl, cyclohexylmethyl, Cl), (M-9555, Cl, CH₃, Cl, cyclohexylmethyl, F), (M-9556, Cl, CH₃, Cl, cyclohexylmethyl, CF₃), (M-9557, Cl, CH₃, Cl, cyclohexylmethyl, Br), (M-9558, Cl, CH₃, Cl, cyclohexylmethyl, CH₃), (M-9559, CH₃, H, H, H, H), (M-9560, CH₃, H, H, H, Cl), (M-9561, MeO, H, H, H, F), (M-9562, MeO, H, H, H, CF₃), (M-9563, CH₃, H, H, H, Br), (M-9564, CH₃, H, H, H, CH₃), (M-9565, MeO, H, H, F, H), (M-9566, CH₃, H, H, F, Cl), (M-9567, MeO, F, H, F, F), (M-9568, CH₃, H, H, F, CF₃), (M-9569, CH₃, H, H, F, Br), (M-9570, CH₃, H, H, F, CH₃), (M-9571, CH₃, H, H, Cl, H), (M-9572, MeO, F, H, H, i-Pr), (M-9573, CH₃, H, H, Cl, F), (M-9574, CH₃, H, H, Cl, CF₃), (M-9575, CH₃, H, H, Cl, Br), (M-9576, CH₃, H, H, Cl, CH₃), (M-9577, CH₃, H, H, CH₃, H), (M-9578, CH₃, H, H, CH₃, Cl), (M-9579, CH₃, H, H, CH₃, F), (M-9580, CH₃, H, H, CH₃, CF₃), (M-9581, CH₃, H, H, CH₃, Br), (M-9582, CH₃, H, H, CH₃, CH₃), (M-9583, CH₃, H, H, Et, H), (M-9584, CH₃, H, H, Et, Cl), (M-9585, CH₃, H, H, Et, F), (M-9586, CH₃, H, H, Et, CF₃), (M-9587, CH₃, H, H, Et, Br), (M-9588, CH₃, H, H, Et, CH₃), (M-9589, CH₃, H, H, n-Pr, H), (M-9590, CH₃, H, H, n-Pr, Cl), (M-9591, CH₃, H, H, n-Pr, F), (M-9592, CH₃, H, H, n-Pr, CF₃), (M-9593, CH₃, H, H, n-Pr, Br), (M-9594, CH₃, H, H, n-Pr, CH₃), (M-9595, CH₃, H, H, c-Pr, H), (M-9596, CH₃, H, H, c-Pr, Cl), (M-9597, CH₃, H, H, c-Pr, F), (M-9598, CH₃, H, H, c-Pr, CF₃), (M-9599, CH₃, H, H, c-Pr, Br), (M-9600, CH₃, H, H, c-Pr, CH₃), (M-9601, CH₃, H, H, i-Pr, H), (M-9602, CH₃, H, H, i-Pr, Cl), (M-9603, CH₃, H, H, i-Pr, F), (M-9604, CH₃, H, H, i-Pr, CF₃), (M-9605, CH₃, H, H, i-Pr, Br), (M-9606, CH₃, H, H, i-Pr, CH₃), (M-9607, CH₃, H, H, n-Bu, H), (M-9608, CH₃, H, H, n-Bu, Cl), (M-9609, CH₃, H, H, n-Bu, F), (M-9610, CH₃, H, H, n-Bu, CF₃), (M-9611, CH₃, H, H, n-Bu, Br), (M-9612, CH₃, H, H, n-Bu, CH₃), (M-9613, CH₃, H, H, i-Bu, H), (M-9614, CH₃, H, H, i-Bu, Cl), (M-9615, CH₃, H, H, i-Bu, F), (M-9616, CH₃, H, H, i-Bu, CF₃), (M-9617, CH₃, H, H, i-Bu, Br), (M-9618, CH₃, H, H, i-Bu, CH₃), (M-9619, CH₃, H, H, sec-Bu, H), (M-9620, CH₃, H, H, sec-Bu, Cl), (M-9621, CH₃, H, H, sec-Bu, F), (M-9622, CH₃, H, H, sec-Bu, CF₃), (M-9623, CH₃, H, H, sec-Bu, Br), (M-9624, CH₃, H, H, sec-Bu, CH₃), (M-9625, CH₃, H, H, n-Pen, H), (M-9626, CH₃, H, H, n-Pen, Cl), (M-9627, CH₃, H, H, n-Pen, F), (M-9628, CH₃, H, H, n-Pen, CF₃), (M-9629, CH₃, H, H, n-Pen, Br), (M-9630, CH₃, H, H, n-Pen, CH₃), (M-9631, CH₃, H, H, c-Pen, H), (M-9632, CH₃, H, H, c-Pen, Cl), (M-9633, CH₃, H, H, c-Pen, F), (M-9634, CH₃, H, H, c-Pen, CF₃), (M-9635, CH₃, H, H, c-Pen, Br), (M-9636, CH₃, H, H, c-Pen, CH₃), (M-9637, CH₃, H, H, n-Hex, H), (M-9638, CH₃, H, H, n-Hex, Cl), (M-9639, CH₃, H, H, n-Hex, F), (M-9640, CH₃, H, H, n-Hex, CF₃), (M-9641, CH₃, H, H, n-Hex, Br), (M-9642, CH₃, H, H, n-Hex, CH₃), (M-9643, CH₃, H, H, c-Hex, H), (M-9644, CH₃, H, H, c-Hex, Cl), (M-9645, CH₃, H, H, c-Hex, F), (M-9646, CH₃, H, H, c-Hex, CF₃), (M-9647, CH₃, H, H, c-Hex, Br), (M-9648, CH₃, H, H, c-Hex, CH₃), (M-9649, CH₃, H, H, OH, H), (M-9650, CH₃, H, H, OH, Cl), (M-9651, CH₃, H, H, OH, F), (M-9652, CH₃, H, H, OH, CF₃), (M-9653, CH₃, H, H, OH, Br), (M-9654, CH₃, H, H, OH, CH₃), (M-9655, CH₃, H, H, EtO, H), (M-9656, CH₃, H, H, EtO, Cl), (M-9657, CH₃, H, H, EtO, F), (M-9658, CH₃, H, H, EtO, CF₃), (M-9659, CH₃, H, H, EtO, Br), (M-9660, CH₃, H, H, EtO, CH₃), (M-9661, CH₃, H, H, n-PrO, H), (M-9662, CH₃, H, H, n-PrO, Cl), (M-9663, CH₃, H, H, n-PrO, F), (M-9664, CH₃, H, H, n-PrO, CF₃), (M-9665, CH₃, H, H, n-PrO, Br), (M-9666, CH₃, H, H, n-PrO, CH₃), (M-9667, CH₃, H, H, PhO, H), (M-9668, CH₃, H, H, PhO, Cl), (M-9669, CH₃, H, H, PhO, F), (M-9670, CH₃, H, H, PhO, CF₃), (M-9671, CH₃, H, H, PhO, Br), (M-9672, CH₃, H, H, PhO, CH₃), (M-9673, CH₃, H, H, BnO, H), (M-9674, CH₃, H, H, BnO, Cl), (M-9675, CH₃, H, H, BnO, F), (M-9676, CH₃, H, H, BnO, CF₃), (M-9677, CH₃, H, H, BnO, Br), (M-9678, CH₃, H, H, BnO, CH₃), (M-9679, CH₃, H, H, PhCH₂CH₂O, H), (M-9680, CH₃, H, H, PhCH₂CH₂O, Cl), (M-9681, CH₃, H, H, PhCH₂CH₂O, F), (M-9682, CH₃, H, H, PhCH₂CH₂O, CF₃), (M-9683, CH₃, H, H, PhCH₂CH₂O, Br), (M-9684, CH₃, H, H, PhCH₂CH₂O, CH₃), (M-9685, MeO, H, H, CF₃O, H), (M-9686, CH₃, H, H, CF₃O, Cl), (M-9687, CH₃, H, H, CF₃O, F), (M-9688, CH₃, H, H, CF₃O, CF₃), (M-9689, CH₃, H, H, CF₃O, Br), (M-9690, CH₃, H, H, CF₃O, CH₃), (M-9691, CH₃, H, H, Ph, H), (M-9692, CH₃, H, H, Ph, Cl), (M-9693, CH₃, H, H, Ph, F), (M-9694, CH₃, H, H, Ph, CF₃), (M-9695, CH₃, H, H, Ph, Br), (M-9696, CH₃, H, H, Ph, CH₃), (M-9697, CH₃, H, H, 4-F-Ph, H), (M-9698, CH₃, H, H, 4-F-Ph, Cl), (M-9699, CH₃, H, H, 4-F-Ph, F), (M-9700, CH₃, H, H, 4-F-Ph, CF₃), (M-9701, CH₃, H, H, 4-F-Ph, Br), (M-9702, CH₃, H, H, 4-F-Ph, CH₃), (M-9703, CH₃, H, H, 4-CF₃-Ph, H), (M-9704, CH₃, H, H, 4-CF₃-Ph, Cl), (M-9705, CH₃, H, H, 4-CF₃-Ph, F), (M-9706, CH₃, H, H, 4-CF₃-Ph, CF₃), (M-9707, CH₃, H, H, 4-CF₃-Ph, Br), (M-9708, CH₃, H, H, 4-CF₃-Ph, CH₃), (M-9709, CH₃, H, H, 4-(Me)₂N-Ph, H), (M-9710, CH₃, H, H, 4-(Me)₂N-Ph, Cl), (M-9711, CH₃, H, H, 4-(Me)₂N-Ph, F), (M-9712, CH₃, H, H, 4-(Me)₂N-Ph, CF₃), (M-9713, CH₃, H, H, 4-(Me)₂N-Ph, Br), (M-9714, CH₃, H, H, 4-(Me)₂N-Ph, CH₃), (M-9715, CH₃, H, H, 4-OH-Ph, H), (M-9716, CH₃, H, H, 4-OH-Ph, Cl), (M-9717, CH₃, H, H, 4-OH-Ph, F), (M-9718, CH₃, H, H, 4-OH-Ph, CF₃), (M-9719, CH₃, H, H, 4-OH-Ph, Br), (M-9720, CH₃, H, H, 4-OH-Ph, CH₃), (M-9721, CH₃, H, H, 3,4-di-F-Ph, H), (M-9722, CH₃, H, H, 3,4-di-F-Ph, Cl), (M-9723, CH₃, H, H, 3,4-di-F-Ph, F), (M-9724, CH₃, H, H, 3,4-di-F-Ph, CF₃), (M-9725, CH₃, H, H, 3,4-di-F-Ph, Br), (M-9726, CH₃, H, H, 3,4-di-F-Ph, CH₃), (M-9727, CH₃, H, H, 4-COOH-Ph, H), (M-9728, CH₃, H, H, 4-COOH-Ph, Cl), (M-9729, CH₃, H, H, 4-COOH-Ph, F), (M-9730, CH₃, H, H, 4-COOH-Ph, CF₃), (M-9731, CH₃, H, H, 4-COOH-Ph, Br), (M-9732, CH₃, H, H, 4-COOH-Ph, CH₃), (M-9733, CH₃, H, H, Bn, H), (M-9734, CH₃, H, H, Bn, Cl), (M-9735, CH₃, H, H, Bn, F), (M-9736, CH₃, H, H, Bn, CF₃), (M-9737, CH₃, H, H, Bn, Br), (M-9738, CH₃, H, H, Bn, CH₃), (M-9739, CH₃, H, H, 4-F-Bn, H), (M-9740, CH₃, H, H, 4-F-Bn, Cl), (M-9741, CH₃, H, H, 4-F-Bn, F), (M-9742, CH₃, H, H, 4-F-Bn, CF₃), (M-9743, CH₃, H, H, 4-F-Bn, Br), (M-9744, CH₃, H, H, 4-F-Bn, CH₃), (M-9745, CH₃, H, H, 2-Py, H), (M-9746, CH₃, H, H, 2-Py, Cl), (M-9747, CH₃, H, H, 2-Py, F), (M-9748, CH₃, H, H, 2-Py, CF₃), (M-9749, CH₃, H, H, 2-Py, Br), (M-9750, CH₃, H, H, 2-Py, CH₃), (M-9751, CH₃, H, H, 3-Py, H), (M-9752, CH₃, H, H, 3-Py, Cl), (M-9753, CH₃, H, H, 3-Py, F), (M-9754, CH₃, H, H, 3-Py, CF₃), (M-9755, CH₃, H, H, 3-Py, Br), (M-9756, CH₃, H, H, 3-Py, CH₃), (M-9757, CH₃, H, H, 4-Py, H), (M-9758, CH₃, H, H, 4-Py, Cl), (M-9759, CH₃, H, H, 4-Py, F), (M-9760, CH₃, H, H, 4-Py, CF₃), (M-9761, CH₃, H, H, 4-Py, Br), (M-9762, CH₃, H, H, 4-Py, CH₃), (M-9763, CH₃
, H, H, 2-Th, H), (M-9764, CH₃, H, H, 2-Th, Cl), (M-9765, CH₃, H, H, 2-Th, F), (M-9766, CH₃, H, H, 2-Th, CF₃), (M-9767, CH₃, H, H, 2-Th, Br), (M-9768, CH₃, H, H, 2-Th, CH₃), (M-9769, CH₃, H, H, 3-Th, H), (M-9770, CH₃, H, H, 3-Th, Cl), (M-9771, CH₃, H, H, 3-Th, F), (M-9772, CH₃, H, H, 3-Th, CF₃), (M-9773, CH₃, H, H, 3-Th, Br), (M-9774, CH₃, H, H, 3-Th, CH₃), (M-9775, CH₃, H, H, pyrazol-2-yl, H), (M-9776, CH₃, H, H, pyrazol-2-yl, Cl), (M-9777, CH₃, H, H, pyrazol-2-yl, F), (M-9778, CH₃, H, H, pyrazol-2-yl, CF₃), (M-9779, CH₃, H, H, pyrazol-2-yl, Br), (M-9780, CH₃, H, H, pyrazol-2-yl, CH₃), (M-9781, CH₃, H, H, pyrazol-3-yl, H), (M-9782, CH₃, H, H, pyrazol-3-yl, Cl), (M-9783, CH₃, H, H, pyrazol-3-yl, F), (M-9784, CH₃, H, H, pyrazol-3-yl, CF₃), (M-9785, CH₃, H, H, pyrazol-3-yl, Br), (M-9786, CH₃, H, H, pyrazol-3-yl, CH₃), (M-9787, CH₃, H, H, pyrimidin-2-yl, H), (M-9788, CH₃, H, H, pyrimidin-2-yl, Cl), (M-9789, CH₃, H, H, pyrimidin-2-yl, F), (M-9790, CH₃, H, H, pyrimidin-2-yl, CF₃), (M-9791, CH₃, H, H, pyrimidin-2-yl, Br), (M-9792, CH₃, H, H, pyrimidin-2-yl, CH₃), (M-9793, CH₃, H, H, pyrimidin-4-yl, H), (M-9794, CH₃, H, H, pyrimidin-4-yl, Cl), (M-9795, CH₃, H, H, pyrimidin-4-yl, F), (M-9796, CH₃, H, H, pyrimidin-4-yl, CF₃), (M-9797, CH₃, H, H, pyrimidin-4-yl, Br), (M-9798, CH₃, H, H, pyrimidin-4-yl, CH₃), (M-9799, CH₃, H, H, pyrimidin-5-yl, H), (M-9800, CH₃, H, H, pyrimidin-5-yl, Cl), (M-9801, CH₃, H, H, pyrimidin-5-yl, F), (M-9802, CH₃, H, H, pyrimidin-5-yl, CF₃), (M-9803, CH₃, H, H, pyrimidin-5-yl, Br), (M-9804, CH₃, H, H, pyrimidin-5-yl, CH₃), (M-9805, CH₃, H, H, HOOCCH₂CH₂CH₂, H), (M-9806, CH₃, H, H, HOOCCH₂CH₂CH₂, Cl), (M-9807, CH₃, H, H, HOOCCH₂CH₂CH₂, F), (M-9808, CH₃, H, H, HOOCCH₂CH₂CH₂, CF₃), (M-9809, CH₃, H, H, HOOCCH₂CH₂CH₂, Br), (M-9810, CH₃, H, H, HOOCCH₂CH₂CH₂, CH₃), (M-9811, CH₃, H, H, HOOCCH₂CH₂CH₂CH₂, H), (M-9812, CH₃, H, H, HOOCCH₂CH₂CH₂CH₂, Cl), (M-9813, CH₃, H, H, HOOCCH₂CH₂CH₂CH₂, F), (M-9814, CH₃, H, H, HOOCCH₂CH₂CH₂CH₂, CF₃), (M-9815, CH₃, H, H, HOOCCH₂CH₂CH₂CH₂, Br), (M-9816, CH₃, H, H, HOOCCH₂CH₂CH₂CH₂, CH₃), (M-9817, CH₃, H, H, (Me)₂NCOCH₂CH₂CH₂CH₂, H), (M-9818, CH₃, H, H, (Me)₂NCOCH₂CH₂CH₂CH₂, Cl), (M-9819, CH₃, H, H, (Me)₂NCOCH₂CH₂CH₂CH₂, F), (M-9820, CH₃, H, H, (Me)₂NCOCH₂CH₂CH₂CH₂, CF₃), (M-9821, CH₃, H, H, (Me)₂NCOCH₂CH₂CH₂CH₂, Br), (M-9822, CH₃, H, H, (Me)₂NCOCH₂CH₂CH₂CH₂, CH₃), (M-9823, CH₃, H, H, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, H), (M-9824, CH₃, H, H, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, Cl), (M-9825, CH₃, H, H, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, F), (M-9826, CH₃, H, H, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, CF₃), (M-9827, CH₃, H, H, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, Br), (M-9828, CH₃, H, H, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, CH₃), (M-9829, CH₃, H, H, MeOCH₂, H), (M-9830, CH₃, H, H, MeOCH₂, Cl), (M-9831, CH₃, H, H, MeOCH₂, F), (M-9832, CH₃, H, H, MeOCH₂, CF₃), (M-9833, CH₃, H, H, MeOCH₂, Br), (M-9834, CH₃, H, H, MeOCH₂, CH₃), (M-9835, CH₃, H, H, EtOCH₂, H), (M-9836, CH₃, H, H, EtOCH₂, Cl), (M-9837, CH₃, H, H, EtOCH₂, F), (M-9838, CH₃, H, H, EtOCH₂, CF₃), (M-9839, CH₃, H, H, EtOCH₂, Br), (M-9840, CH₃, H, H, EtOCH₂, CH₃), (M-9841, CH₃, H, H, EtOCH₂CH₂, H), (M-9842, CH₃, H, H, EtOCH₂CH₂, Cl), (M-9843, CH₃, H, H, EtOCH₂CH₂, F), (M-9844, CH₃, H, H, EtOCH₂CH₂, CF₃), (M-9845, CH₃, H, H, EtOCH₂CH₂, Br), (M-9846, CH₃, H, H, EtOCH₂CH₂, CH₃), (M-9847, CH₃, H, H, MeOCH₂CH₂OCH₂CH₂, H), (M-9848, CH₃, H, H, MeOCH₂CH₂OCH₂CH₂, Cl), (M-9849, CH₃, H, H, MeOCH₂CH₂OCH₂CH₂, F), (M-9850, CH₃, H, H, MeOCH₂CH₂OCH₂CH₂, CF₃), (M-9851, CH₃, H, H, MeOCH₂CH₂OCH₂CH₂, Br), (M-9852, CH₃, H, H, MeOCH₂CH₂OCH₂CH₂, CH₃), (M-9853, CH₃, H, H, MeOCH₂CH₂, H), (M-9854, CH₃, H, H, MeOCH₂CH₂, Cl), (M-9855, CH₃, H, H, MeOCH₂CH₂, F), (M-9856, CH₃, H, H, MeOCH₂CH₂, CF₃), (M-9857, CH₃, H, H, MeOCH₂CH₂, Br), (M-9858, CH₃, H, H, MeOCH₂CH₂, CH₃), (M-9859, CH₃, H, H, HOCH₂, H), (M-9860, CH₃, H, H, HOCH₂, Cl), (M-9861, CH₃, H, H, HOCH₂, F), (M-9862, CH₃, H, H, HOCH₂, CF₃), (M-9863, CH₃, H, H, HOCH₂, Br), (M-9864, CH₃, H, H, HOCH₂, CH₃), (M-9865, CH₃, H, H, HOCH₂CH₂, H), (M-9866, CH₃, H, H, HOCH₂CH₂, Cl), (M-9867, CH₃, H, H, HOCH₂CH₂, F), (M-9868, CH₃, H, H, HOCH₂CH₂, CF₃), (M-9869, CH₃, H, H, HOCH₂CH₂, Br), (M-9870, CH₃, H, H, HOCH₂CH₂, CH₃), (M-9871, CH₃, H, H, HOCH₂CH₂CH₂, H), (M-9872, CH₃, H, H, HOCH₂CH₂CH₂, Cl), (M-9873, CH₃, H, H, HOCH₂CH₂CH₂, F), (M-9874, CH₃, H, H, HOCH₂CH₂CH₂, CF₃), (M-9875, CH₃, H, H, HOCH₂CH₂CH₂, Br), (M-9876, CH₃, H, H, HOCH₂CH₂CH₂, CH₃), (M-9877, CH₃, H, H, HOCH₂CH₂CH₂CH₂, H), (M-9878, CH₃, H, H, HOCH₂CH₂CH₂CH₂, Cl), (M-9879, CH₃, H, H, HOCH₂CH₂CH₂CH₂, F), (M-9880, CH₃, H, H, HOCH₂CH₂CH₂CH₂, CF₃), (M-9881, CH₃, H, H, HOCH₂CH₂CH₂CH₂, Br), (M-9882, CH₃, H, H, HOCH₂CH₂CH₂CH₂, CH₃), (M-9883, CH₃, H, H, HOCH₂CH₂CH₂CH₂CH₂, H), (M-9884, CH₃, H, H, HOCH₂CH₂CH₂CH₂CH₂, Cl), (M-9885, CH₃, H, H, HOCH₂CH₂CH₂CH₂CH₂, F), (M-9886, CH₃, H, H, HOCH₂CH₂CH₂CH₂CH₂, CF₃), (M-9887, CH₃, H, H, HOCH₂CH₂CH₂CH₂CH₂, Br), (M-9888, CH₃, H, H, HOCH₂CH₂CH₂CH₂CH₂, CH₃), (M-9889, CH₃, H, H, HOCH₂CH₂OCH₂CH₂, H), (M-9890, CH₃, H, H, HOCH₂CH₂OCH₂CH₂, Cl), (M-9891, CH₃, H, H, HOCH₂CH₂OCH₂CH₂, F), (M-9892, CH₃, H, H, HOCH₂CH₂OCH₂CH₂, CF₃), (M-9893, CH₃, H, H, HOCH₂CH₂OCH₂CH₂, Br), (M-9894, CH₃, H, H, HOCH₂CH₂OCH₂CH₂, CH₃), (M-9895, CH₃, H, H, (Me)₂N, H), (M-9896, CH₃, H, H,
(Me)₂N, Cl), (M-9897, CH₃, H, H, (Me)₂N, F), (M-9898, CH₃, H, H, (Me)₂N, CF₃), (M-9899, CH₃, H, H, (Me)₂N, Br), (M-9900, CH₃, H, H, (Me)₂N, CH₃), (M-9901, CH₃, H, H, piperidin-4-yl-methyl, H), (M-9902, CH₃, H, H, piperidin-4-yl-methyl, Cl), (M-9903, CH₃, H, H, piperidin-4-yl-methyl, F), (M-9904, CH₃, H, H, piperidin-4-yl-methyl, CF₃), (M-9905, CH₃, H, H, piperidin-4-yl-methyl, Br), (M-9906, CH₃, H, H, piperidin-4-yl-methyl, CH₃), (M-9907, CH₃, H, H, cyclohexylmethyl, H), (M-9908, CH₃, H, H, cyclohexylmethyl, Cl), (M-9909, CH₃, H, H, cyclohexylmethyl, F), (M-9910, CH₃, H, H, cyclohexylmethyl, CF₃), (M-9911, CH₃, H, H, cyclohexylmethyl, Br), (M-9912, CH₃, H, H, cyclohexylmethyl, CH₃), (M-9913, CH₃, H, F, H, H), (M-9914, CH₃, H, F, H, Cl), (M-9915, CH₃, H, F, H, F), (M-9916, CH₃, H, F, H, CF₃), (M-9917, CH₃, H, F, H, Br), (M-9918, CH₃, H, F, H, CH₃), (M-9919, CH₃, H, F, F, H), (M-9920, CH₃, H, F, F, Cl), (M-9921, CH₃, H, F, F, F), (M-9922, CH₃, H, F, F, CF₃), (M-9923, CH₃, H, F, F, Br), (M-9924, CH₃, H, F, F, CH₃), (M-9925, CH₃, H, F, Cl, H), (M-9926, CH₃, H, F, Cl, Cl), (M-9927, CH₃, H, F, Cl, F), (M-9928, CH₃, H, F, Cl, CF₃), (M-9929, CH₃, H, F, Cl, Br), (M-9930, CH₃, H, F, Cl, CH₃), (M-9931, CH₃, H, F, CH₃, H), (M-9932, CH₃, H, F, CH₃, Cl), (M-9933, CH₃, H, F, CH₃, F), (M-9934, CH₃, H, F, CH₃, CF₃), (M-9935, CH₃, H, F, CH₃, Br), (M-9936, CH₃, H, F, CH₃, CH₃), (M-9937, CH₃, H, F, Et, H), (M-9938, CH₃, H, F, Et, Cl), (M-9939, CH₃, H, F, Et, F), (M-9940, CH₃, H, F, Et, CF₃), (M-9941, CH₃, H, F, Et, Br), (M-9942, CH₃, H, F, Et, CH₃), (M-9943, CH₃, H, F, n-Pr, H), (M-9944, CH₃, H, F, n-Pr, Cl), (M-9945, CH₃, H, F, n-Pr, F), (M-9946, CH₃, H, F, n-Pr, CF₃), (M-9947, CH₃, H, F, n-Pr, Br), (M-9948, CH₃, H, F, n-Pr, CH₃), (M-9949, CH₃, H, F, c-Pr, H), (M-9950, CH₃, H, F, c-Pr, Cl), (M-9951, CH₃, H, F, c-Pr, F), (M-9952, CH₃, H, F, c-Pr, CF₃), (M-9953, CH₃, H, F, c-Pr, Br), (M-9954, CH₃, H, F, c-Pr, CH₃), (M-9955, CH₃, H, F, i-Pr, H), (M-9956, CH₃, H, F, i-Pr, Cl), (M-9957, CH₃, H, F, i-Pr, F), (M-9958, CH₃, H, F, i-Pr, CF₃), (M-9959, CH₃, H, F, i-Pr, Br), (M-9960, CH₃, H, F, i-Pr, CH₃), (M-9961, CH₃, H, F, n-Bu, H), (M-9962, CH₃, H, F, n-Bu, Cl), (M-9963, CH₃, H, F, n-Bu, F), (M-9964, CH₃, H, F, n-Bu, CF₃), (M-9965, CH₃, H, F, n-Bu, Br), (M-9966, CH₃, H, F, n-Bu, CH₃), (M-9967, CH₃, H, F, i-Bu, H), (M-9968, CH₃, H, F, i-Bu, Cl), (M-9969, CH₃, H, F, i-Bu, F), (M-9970, CH₃, H, F, i-Bu, CF₃), (M-9971, CH₃, H, F, i-Bu, Br), (M-9972, CH₃, H, F, i-Bu, CH₃), (M-9973, CH₃, H, F, sec-Bu, H), (M-9974, CH₃, H, F, sec-Bu, Cl), (M-9975, CH₃, H, F, sec-Bu, F), (M-9976, CH₃, H, F, sec-Bu, CF₃), (M-9977, CH₃, H, F, sec-Bu, Br), (M-9978, CH₃, H, F, sec-Bu, CH₃), (M-9979, CH₃, H, F, n-Pen, H), (M-9980, CH₃, H, F, n-Pen, Cl), (M-9981, CH₃, H, F, n-Pen, F), (M-9982, CH₃, H, F, n-Pen, CF₃), (M-9983, CH₃, H, F, n-Pen, Br), (M-9984, CH₃, H, F, n-Pen, CH₃), (M-9985, CH₃, H, F, c-Pen, H), (M-9986, CH₃, H, F, c-Pen, Cl), (M-9987, CH₃, H, F, c-Pen, F), (M-9988, CH₃, H, F, c-Pen, CF₃), (M-9989, CH₃, H, F, c-Pen, Br), (M-9990, CH₃, H, F, c-Pen, CH₃), (M-9991, CH₃, H, F, n-Hex, H), (M-9992, CH₃, H, F, n-Hex, Cl), (M-9993, CH₃, H, F, n-Hex, F), (M-9994, CH₃, H, F, n-Hex, CF₃), (M-9995, CH₃, H, F, n-Hex, Br), (M-9996, CH₃, H, F, n-Hex, CH₃), (M-9997, CH₃, H, F, c-Hex, H), (M-9998, CH₃, H, F, c-Hex, Cl), (M-9999, CH₃, H, F, c-Hex, F), (M-10000, CH₃, H, F, c-Hex, CF₃), (M-10001, CH₃, H, F, c-Hex, Br), (M-10002, CH₃, H, F, c-Hex, CH₃), (M-10003, CH₃, H, F, OH, H), (M-10004, CH₃, H, F, OH, Cl), (M-10005, CH₃, H, F, OH, F), (M-10006, CH₃, H, F, OH, CF₃), (M-10007, CH₃, H, F, OH, Br), (M-10008, CH₃, H, F, OH, CH₃), (M-10009, CH₃, H, F, EtO, H), (M-10010, CH₃, H, F, EtO, Cl), (M-10011, CH₃, H, F, EtO, F), (M-10012, CH₃, H, F, EtO, CF₃), (M-10013, CH₃, H, F, EtO, Br), (M-10014, CH₃, H, F, EtO, CH₃), (M-10015, CH₃, H, F, n-PrO, H), (M-10016, CH₃, H, F, n-PrO, Cl), (M-10017, CH₃, H, F, n-PrO, F), (M-10018, CH₃, H, F, n-PrO, CF₃), (M-10019, CH₃, H, F, n-PrO, Br), (M-10020, CH₃, H, F, n-PrO, CH₃), (M-10021, CH₃, H, F, PhO, H), (M-10022, CH₃, H, F, PhO, Cl), (M-10023, CH₃, H, F, PhO, F), (M-10024, CH₃, H, F, PhO, CF₃), (M-10025, CH₃, H, F, PhO, Br), (M-10026, CH₃, H, F, PhO, CH₃), (M-10027, CH₃, H, F, BnO, H), (M-10028, CH₃, H, F, BnO, Cl), (M-10029, CH₃, H, F, BnO, F), (M-10030, CH₃, H, F, BnO, CF₃), (M-10031, CH₃, H, F, BnO, Br), (M-10032, CH₃, H, F, BnO, CH₃), (M-10033, CH₃, H, F, PhCH₂CH₂O, H), (M-10034, CH₃, H, F, PhCH₂CH₂O, Cl), (M-10035, CH₃, H, F, PhCH₂CH₂O, F), (M-10036, CH₃, H, F, PhCH₂CH₂O, CF₃), (M-10037, CH₃, H, F, PhCH₂CH₂O, Br), (M-10038, CH₃, H, F, PhCH₂CH₂O, CH₃), (M-10039, CH₃, H, F, CF₃O, H), (M-10040, CH₃, H, F, CF₃O, Cl), (M-10041, CH₃, H, F, CF₃O, F), (M-10042, CH₃, H, F, CF₃O, CF₃), (M-10043, CH₃, H, F, CF₃O, Br), (M-10044, CH₃, H, F, CF₃O, CH₃), (M-10045, CH₃, H, F, Ph, H), (M-10046, CH₃, H, F, Ph, Cl), (M-10047, CH₃, H, F, Ph, F), (M-10048, CH₃, H, F, Ph, CF₃), (M-10049, CH₃, H, F, Ph, Br), (M-10050, CH₃, H, F, Ph, CH₃), (M-10051, CH₃, H, F, 4-F-Ph, H), (M-10052, CH₃, H, F, 4-F-Ph, Cl), (M-10053, CH₃, H, F, 4-F-Ph, F), (M-10054, CH₃, H, F, 4-F-Ph, CF₃), (M-10055, CH₃, H, F, 4-F-Ph, Br), (M-10056, CH₃, H, F, 4-F-Ph, CH₃), (M-10057, CH₃, H, F, 4-CF₃-Ph, H), (M-10058, CH₃, H, F, 4-CF₃-Ph, Cl), (M-10059, CH₃, H, F, 4-CF₃-Ph, F), (M-10060, CH₃, H, F, 4-CF₃-Ph, CF₃), (M-10061, CH₃, H, F, 4-CF₃-Ph, Br), (M-10062, CH₃, H, F, 4-CF₃-Ph, CH₃), (M-10063, CH₃, H, F, 4-(Me)₂N-Ph, H), (M-10064, CH₃, H, F, 4-(Me)₂N-Ph, Cl), (M-10065, CH₃, H, F, 4-(Me)₂N-Ph, F), (M-10066, CH₃, H, F, 4-(Me)₂N-Ph, CF₃), (M-10067, CH₃, H, F, 4-(Me)₂N-Ph, Br), (M-10068, CH₃, H, F, 4-(Me)₂N-Ph, CH₃), (M-10069, CH₃, H, F, 4-OH-Ph, H), (M-10070, CH₃, H, F, 4-OH-Ph, Cl), (M-10071, CH₃, H, F, 4-OH-Ph, F), (M-10072, CH₃, H, F, 4-OH-Ph, CF₃), (M-10073, CH₃, H, F, 4-OH-Ph, Br), (M-10074, CH₃, H, F, 4-OH-Ph, CH₃), (M-10075, CH₃, H, F, 3,4-di-F-Ph, H), (M-10076, CH₃, H, F, 3,4-di-F-Ph, Cl), (M-10077, CH₃, H, F, 3,4-di-F-Ph, F), (M-10078, CH₃, H, F, 3,4-di-F-Ph, CF₃), (M-10079, CH₃, H, F, 3,4-di-F-Ph, Br), (M-10080, CH₃, H, F, 3,4-di-F-Ph, CH₃), (M-10081, CH₃, H, F, 4-COOH-Ph, H), (M-10082, CH₃, H, F, 4-COOH-Ph, Cl), (M-10083, CH₃, H, F, 4-COOH-Ph, F), (M-10084, CH₃, H, F, 4-COOH-Ph, CF₃), (M-10085, CH₃, H, F, 4-COOH-Ph, Br), (M-10086, CH₃, H, F, 4-COOH-Ph, CH₃), (M-10087, CH₃, H, F, Bn, H), (M-10088, CH₃, H, F, Bn, Cl), (M-10089, CH₃, H, F, Bn, F), (M-10090, CH₃, H, F, Bn, CF₃), (M-10091, CH₃, H, F, Bn, Br), (M-10092, CH₃, H, F, Bn, CH₃), (M-10093, CH₃, H, F, 4-F-Bn, H), (M-10094, CH₃, H, F, 4-F-Bn, Cl), (M-10095, CH₃, H, F, 4-F-Bn, F), (M-10096, CH₃, H, F, 4-F-Bn, CF₃), (M-10097, CH₃, H, F, 4-F-Bn, Br), (M-10098, CH₃, H, F, 4-F-Bn, CH₃), (M-10099, CH₃, H, F, 2-Py, H), (M-10100, CH₃, H, F, 2-Py, Cl), (M-10101, CH₃, H, F, 2-Py, F), (M-
10102, CH₃, H, F, 2-Py, CF₃), (M-10103, CH₃, H, F, 2-Py, Br), (M-10104, CH₃, H, F, 2-Py, CH₃), (M-10105, CH₃, H, F, 3-Py, H), (M-10106, CH₃, H, F, 3-Py, Cl), (M-10107, CH₃, H, F, 3-Py, F), (M-10108, CH₃, H, F, 3-Py, CF₃), (M-10109, CH₃, H, F, 3-Py, Br), (M-10110, CH₃, H, F, 3-Py, CH₃), (M-10111, CH₃, H, F, 4-Py, H), (M-10112, CH₃, H, F, 4-Py, Cl), (M-10113, CH₃, H, F, 4-Py, F), (M-10114, CH₃, H, F, 4-Py, CF₃), (M-10115, CH₃, H, F, 4-Py, Br), (M-10116, CH₃, H, F, 4-Py, CH₃), (M-10117, CH₃, H, F, 2-Th, H), (M-10118, CH₃, H, F, 2-Th, Cl), (M-10119, CH₃, H, F, 2-Th, F), (M-10120, CH₃, H, F, 2-Th, CF₃), (M-10121, CH₃, H, F, 2-Th, Br), (M-10122, CH₃, H, F, 2-Th, CH₃), (M-10123, CH₃, H, F, 3-Th, H), (M-10124, CH₃, H, F, 3-Th, Cl), (M-10125, CH₃, H, F, 3-Th, F), (M-10126, CH₃, H, F, 3-Th, CF₃), (M-10127, CH₃, H, F, 3-Th, Br), (M-10128, CH₃, H, F, 3-Th, CH₃), (M-10129, CH₃, H, F, pyrazol-2-yl, H), (M-10130, CH₃, H, F, pyrazol-2-yl, Cl), (M-10131, CH₃, H, F, pyrazol-2-yl, F), (M-10132, CH₃, H, F, pyrazol-2-yl, CF₃), (M-10133, CH₃, H, F, pyrazol-2-yl, Br), (M-10134, CH₃, H, F, pyrazol-2-yl, CH₃), (M-10135, CH₃, H, F, pyrazol-3-yl, H), (M-10136, CH₃, H, F, pyrazol-3-yl, Cl), (M-10137, CH₃, H, F, pyrazol-3-yl, F), (M-10138, CH₃, H, F, pyrazol-3-yl, CF₃), (M-10139, CH₃, H, F, pyrazol-3-yl, Br), (M-10140, CH₃, H, F, pyrazol-3-yl, CH₃), (M-10141, CH₃, H, F, pyrimidin-2-yl, H), (M-10142, CH₃, H, F, pyrimidin-2-yl, Cl), (M-10143, CH₃, H, F, pyrimidin-2-yl, F), (M-10144, CH₃, H, F, pyrimidin-2-yl, CF₃), (M-10145, CH₃, H, F, pyrimidin-2-yl, Br), (M-10146, CH₃, H, F, pyrimidin-2-yl, CH₃), (M-10147, CH₃, H, F, pyrimidin-4-yl, H), (M-10148, CH₃, H, F, pyrimidin-4-yl, Cl), (M-10149, CH₃, H, F, pyrimidin-4-yl, F), (M-10150, CH₃, H, F, pyrimidin-4-yl, CF₃), (M-10151, CH₃, H, F, pyrimidin-4-yl, Br), (M-10152, CH₃, H, F, pyrimidin-4-yl, CH₃), (M-10153, CH₃, H, F, pyrimidin-5-yl, H), (M-10154, CH₃, H, F, pyrimidin-5-yl, Cl), (M-10155, CH₃, H, F, pyrimidin-5-yl, F), (M-10156, CH₃, H, F, pyrimidin-5-yl, CF₃), (M-10157, CH₃, H, F, pyrimidin-5-yl, Br), (M-10158, CH₃, H, F, pyrimidin-5-yl, CH₃), (M-10159, CH₃, H, F, HOOCCH₂CH₂CH₂, H), (M-10160, CH₃, H, F, HOOCCH₂CH₂CH₂, Cl), (M-10161, CH₃, H, F, HOOCCH₂CH₂CH₂, F), (M-10162, CH₃, H, F, HOOCCH₂CH₂CH₂, CF₃), (M-10163, CH₃, H, F, HOOCCH₂CH₂CH₂, Br), (M-10164, CH₃, H, F, HOOCCH₂CH₂CH₂, CH₃), (M-10165, CH₃, H, F, HOOCCH₂CH₂CH₂CH₂, H), (M-10166, CH₃, H, F, HOOCCH₂CH₂CH₂CH₂, Cl), (M-10167, CH₃, H, F, HOOCCH₂CH₂CH₂CH₂, F), (M-10168, CH₃, H, F, HOOCCH₂CH₂CH₂CH₂, CF₃), (M-10169, CH₃, H, F, HOOCCH₂CH₂CH₂CH₂, Br), (M-10170, CH₃, H, F, HOOCCH₂CH₂CH₂CH₂, CH₃), (M-10171, CH₃, H, F, (Me)₂NCOCH₂CH₂CH₂CH₂, H), (M-10172, CH₃, H, F, (Me)₂NCOCH₂CH₂CH₂CH₂, Cl), (M-10173, CH₃, H, F, (Me)₂NCOCH₂CH₂CH₂CH₂, F), (M-10174, CH₃, H, F, (Me)₂NCOCH₂CH₂CH₂CH₂, CF₃), (M-10175, CH₃, H, F, (Me)₂NCOCH₂CH₂CH₂CH₂, Br), (M-10176, CH₃, H, F, (Me)₂NCOCH₂CH₂CH₂CH₂, CH₃), (M-10177, CH₃, H, F, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, H), (M-10178, CH₃, H, F, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, Cl), (M-10179, CH₃, H, F, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, F), (M-10180, CH₃, H, F, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, CF₃), (M-10181, CH₃, H, F, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, Br), (M-10182, CH₃, H, F, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, CH₃), (M-10183, CH₃, H, F, MeOCH₂, H), (M-10184, CH₃, H, F, MeOCH₂, Cl), (M-10185, CH₃, H, F, MeOCH₂, F), (M-10186, CH₃, H, F, MeOCH₂, CF₃), (M-10187, CH₃, H, F, MeOCH₂, Br), (M-10188, CH₃, H, F, MeOCH₂, CH₃), (M-10189, CH₃, H, F, EtOCH₂, H), (M-10190, CH₃, H, F, EtOCH₂, Cl), (M-10191, CH₃, H, F, EtOCH₂, F), (M-10192, CH₃, H, F, EtOCH₂, CF₃), (M-10193, CH₃, H, F, EtOCH₂, Br), (M-10194, CH₃, H, F, EtOCH₂, CH₃), (M-10195, CH₃, H, F, EtOCH₂CH₂, H), (M-10196, CH₃, H, F, EtOCH₂CH₂, Cl), (M-10197, CH₃, H, F, EtOCH₂CH₂, F), (M-10198, CH₃, H, F, EtOCH₂CH₂, CF₃), (M-10199, CH₃, H, F, EtOCH₂CH₂, Br), (M-10200, CH₃, H, F, EtOCH₂CH₂, CH₃), (M-10201, CH₃, H, F, MeOCH₂CH₂OCH₂CH₂, H), (M-10202, CH₃, H, F, MeOCH₂CH₂OCH₂CH₂, Cl), (M-10203, CH₃, H, F, MeOCH₂CH₂OCH₂CH₂, F), (M-10204, CH₃, H, F, MeOCH₂CH₂OCH₂CH₂, CF₃), (M-10205, CH₃, H, F, MeOCH₂CH₂OCH₂CH₂, Br), (M-10206, CH₃, H, F, MeOCH₂CH₂OCH₂CH₂, CH₃), (M-10207, CH₃, H, F, MeOCH₂CH₂, H), (M-10208, CH₃, H, F, MeOCH₂CH₂, Cl), (M-10209, CH₃, H, F, MeOCH₂CH₂, F), (M-10210, CH₃, H, F, MeOCH₂CH₂, CF₃), (M-10211, CH₃, H, F, MeOCH₂CH₂, Br), (M-10212, CH₃, H, F, MeOCH₂CH₂, CH₃), (M-10213, CH₃, H, F, HOCH₂, H), (M-10214, CH₃, H, F, HOCH₂, Cl), (M-10215, CH₃, H, F, HOCH₂, F), (M-10216, CH₃, H, F, HOCH₂, CF₃), (M-10217, CH₃, H, F, HOCH₂, Br), (M-10218, CH₃, H, F, HOCH₂, CH₃), (M-10219, CH₃, H, F, HOCH₂CH₂, H), (M-10220, CH₃, H, F, HOCH₂CH₂, Cl), (M-10221, CH₃, H, F, HOCH₂CH₂, F), (M-10222, CH₃, H, F, HOCH₂CH₂, CF₃), (M-10223, CH₃, H, F, HOCH₂CH₂, Br), (M-10224, CH₃, H, F, HOCH₂CH₂, CH₃), (M-10225, CH₃, H, F, HOCH₂CH₂CH₂, H), (M-10226, CH₃, H, F, HOCH₂CH₂CH₂, Cl), (M-10227, CH₃, H, F, HOCH₂CH₂CH₂, F), (M-10228, CH₃, H, F, HOCH₂CH₂CH₂, CF₃), (M-10229, CH₃, H, F, HOCH₂CH₂CH₂, Br), (M-10230, CH₃, H, F, HOCH₂CH₂CH₂, CH₃), (M-10231, CH₃, H, F, HOCH₂CH₂CH₂CH₂, H), (M-10232, CH₃, H, F, HOCH₂CH₂CH₂CH₂, Cl), (M-10233, CH₃, H, F, HOCH₂CH₂CH₂CH₂, F), (M-10234, CH₃, H, F, HOCH₂CH₂CH₂CH₂, CF₃), (M-10235, CH₃, H, F, HOCH₂CH₂CH₂CH₂, Br), (M-10236, CH₃, H, F, HOCH₂CH₂CH₂CH₂, CH₃), (M-10237, CH₃, H, F, HOCH₂CH₂CH₂CH₂CH₂, H), (M-10238, CH₃, H, F, HOCH₂CH₂CH₂CH₂CH₂, Cl), (M-10239, CH₃, H, F, HOCH₂CH₂CH₂CH₂CH₂, F), (M-10240, CH₃, H, F, HOCH₂CH₂CH₂CH₂CH₂, CF₃), (M-10241, CH₃, H, F, HOCH₂CH₂CH
₂CH₂CH₂, Br), (M-10242, CH₃, H, F, HOCH₂CH₂CH₂CH₂CH₂, CH₃), (M-10243, CH₃, H, F, HOCH₂CH₂OCH₂CH₂, H), (M-10244, CH₃, H, F, HOCH₂CH₂OCH₂CH₂, Cl), (M-10245, CH₃, H, F, HOCH₂CH₂OCH₂CH₂, F), (M-10246, CH₃, H, F, HOCH₂CH₂OCH₂CH₂, CF₃), (M-10247, CH₃, H, F, HOCH₂CH₂OCH₂CH₂, Br), (M-10248, CH₃, H, F, HOCH₂CH₂OCH₂CH₂, CH₃), (M-10249, CH₃, H, F, (Me)₂N, H), (M-10250, CH₃, H, F, (Me)₂N, Cl), (M-10251, CH₃, H, F, (Me)₂N, F), (M-10252, CH₃, H, F, (Me)₂N, CF₃), (M-10253, CH₃, H, F, (Me)₂N, Br), (M-10254, CH₃, H, F, (Me)₂N, CH₃), (M-10255, CH₃, H, F, piperidin-4-yl-methyl, H), (M-10256, CH₃, H, F, piperidin-4-yl-methyl, Cl), (M-10257, CH₃, H, F, piperidin-4-yl-methyl, F), (M-10258, CH₃, H, F, piperidin-4-yl-methyl, CF₃), (M-10259, CH₃, H, F, piperidin-4-yl-methyl, Br), (M-10260, CH₃, H, F, piperidin-4-yl-methyl, CH₃), (M-10261, CH₃, H, F, cyclohexylmethyl, H), (M-10262, CH₃, H, F, cyclohexylmethyl, Cl), (M-10263, CH₃, H, F, cyclohexylmethyl, F), (M-10264, CH₃, H, F, cyclohexylmethyl, CF₃), (M-10265, CH₃, H, F, cyclohexylmethyl, Br), (M-10266, CH₃, H, F, cyclohexylmethyl, CH₃), (M-10267, CH₃, H, Cl, H, H), (M-10268, CH₃, H, Cl, H, Cl), (M-10269, CH₃, H, Cl, H, F), (M-10270, CH₃, H, Cl, H, CF₃), (M-10271, CH₃, H, Cl, H, Br), (M-10272, CH₃, H, Cl, H, CH₃), (M-10273, CH₃, H, Cl, F, H), (M-10274, CH₃, H, Cl, F, Cl), (M-10275, CH₃, H, Cl, F, F), (M-10276, CH₃, H, Cl, F, CF₃), (M-10277, CH₃, H, Cl, F, Br), (M-10278, CH₃, H, Cl, F, CH₃), (M-10279, CH₃, H, Cl, Cl, H), (M-10280, CH₃, H, Cl, Cl, Cl), (M-10281, CH₃, H, Cl, Cl, F), (M-10282, CH₃, H, Cl, Cl, CF₃), (M-10283, CH₃, H, Cl, Cl, Br), (M-10284, CH₃, H, Cl, Cl, CH₃), (M-10285, CH₃, H, Cl, CH₃, H), (M-10286, CH₃, H, Cl, CH₃, Cl), (M-10287, CH₃, H, Cl, CH₃, F), (M-10288, CH₃, H, Cl, CH₃, CF₃), (M-10289, CH₃, H, Cl, CH₃, Br), (M-10290, CH₃, H, Cl, CH₃, CH₃), (M-10291, CH₃, H, Cl, Et, H), (M-10292, CH₃, H, Cl, Et, Cl), (M-10293, CH₃, H, Cl, Et, F), (M-10294, CH₃, H, Cl, Et, CF₃), (M-10295, CH₃, H, Cl, Et, Br), (M-10296, CH₃, H, Cl, Et, CH₃), (M-10297, CH₃, H, Cl, n-Pr, H), (M-10298, CH₃, H, Cl, n-Pr, Cl), (M-10299, CH₃, H, Cl, n-Pr, F), (M-10300, CH₃, H, Cl, n-Pr, CF₃), (M-10301, CH₃, H, Cl, n-Pr, Br), (M-10302, CH₃, H, Cl, n-Pr, CH₃), (M-10303, CH₃, H, Cl, c-Pr, H), (M-10304, CH₃, H, Cl, c-Pr, Cl), (M-10305, CH₃, H, Cl, c-Pr, F), (M-10306, CH₃, H, Cl, c-Pr, CF₃), (M-10307, CH₃, H, Cl, c-Pr, Br), (M-10308, CH₃, H, Cl, c-Pr, CH₃), (M-10309, CH₃, H, Cl, i-Pr, H), (M-10310, CH₃, H, Cl, i-Pr, Cl), (M-10311, CH₃, H, Cl, i-Pr, F), (M-10312, CH₃, H, Cl, i-Pr, CF₃), (M-10313, CH₃, H, Cl, i-Pr, Br), (M-10314, CH₃, H, Cl, i-Pr, CH₃), (M-10315, CH₃, H, Cl, n-Bu, H), (M-10316, CH₃, H, Cl, n-Bu, Cl), (M-10317, CH₃, H, Cl, n-Bu, F), (M-10318, CH₃, H, Cl, n-Bu, CF₃), (M-10319, CH₃, H, Cl, n-Bu, Br), (M-10320, CH₃, H, Cl, n-Bu, CH₃), (M-10321, CH₃, H, Cl, i-Bu, H), (M-10322, CH₃, H, Cl, i-Bu, Cl), (M-10323, CH₃, H, Cl, i-Bu, F), (M-10324, CH₃, H, Cl, i-Bu, CF₃), (M-10325, CH₃, H, Cl, i-Bu, Br), (M-10326, CH₃, H, Cl, i-Bu, CH₃), (M-10327, CH₃, H, Cl, sec-Bu, H), (M-10328, CH₃, H, Cl, sec-Bu, Cl), (M-10329, CH₃, H, Cl, sec-Bu, F), (M-10330, CH₃, H, Cl, sec-Bu, CF₃), (M-10331, CH₃, H, Cl, sec-Bu, Br), (M-10332, CH₃, H, Cl, sec-Bu, CH₃), (M-10333, CH₃, H, Cl, n-Pen, H), (M-10334, CH₃, H, Cl, n-Pen, Cl), (M-10335, CH₃, H, Cl, n-Pen, F), (M-10336, CH₃, H, Cl, n-Pen, CF₃), (M-10337, CH₃, H, Cl, n-Pen, Br), (M-10338, CH₃, H, Cl, n-Pen, CH₃), (M-10339, CH₃, H, Cl, c-Pen, H), (M-10340, CH₃, H, Cl, c-Pen, Cl), (M-10341, CH₃, H, Cl, c-Pen, F), (M-10342, CH₃, H, Cl, c-Pen, CF₃), (M-10343, CH₃, H, Cl, c-Pen, Br), (M-10344, CH₃, H, Cl, c-Pen, CH₃), (M-10345, CH₃, H, Cl, n-Hex, H), (M-10346, CH₃, H, Cl, n-Hex, Cl), (M-10347, CH₃, H, Cl, n-Hex, F), (M-10348, CH₃, H, Cl, n-Hex, CF₃), (M-10349, CH₃, H, Cl, n-Hex, Br), (M-10350, CH₃, H, Cl, n-Hex, CH₃), (M-10351, CH₃, H, Cl, c-Hex, H), (M-10352, CH₃, H, Cl, c-Hex, Cl), (M-10353, CH₃, H, Cl, c-Hex, F), (M-10354, CH₃, H, Cl, c-Hex, CF₃), (M-10355, CH₃, H, Cl, c-Hex, Br), (M-10356, CH₃, H, Cl, c-Hex, CH₃), (M-10357, CH₃, H, Cl, OH, H), (M-10358, CH₃, H, Cl, OH, Cl), (M-10359, CH₃, H, Cl, OH, F), (M-10360, CH₃, H, Cl, OH, CF₃), (M-10361, CH₃, H, Cl, OH, Br), (M-10362, CH₃, H, Cl, OH, CH₃), (M-10363, CH₃, H, Cl, EtO, H), (M-10364, CH₃, H, Cl, EtO, Cl), (M-10365, CH₃, H, Cl, EtO, F), (M-10366, CH₃, H, Cl, EtO, CF₃), (M-10367, CH₃, H, Cl, EtO, Br), (M-10368, CH₃, H, Cl, EtO, CH₃), (M-10369, CH₃, H, Cl, n-PrO, H), (M-10370, CH₃, H, Cl, n-PrO, Cl), (M-10371, CH₃, H, Cl, n-PrO, F), (M-10372, CH₃, H, Cl, n-PrO, CF₃), (M-10373, CH₃, H, Cl, n-PrO, Br), (M-10374, CH₃, H, Cl, n-PrO, CH₃), (M-10375, CH₃, H, Cl, PhO, H), (M-10376, CH₃, H, Cl, PhO, Cl), (M-10377, CH₃, H, Cl, PhO, F), (M-10378, CH₃, H, Cl, PhO, CF₃), (M-10379, CH₃, H, Cl, PhO, Br), (M-10380, CH₃, H, Cl, PhO, CH₃), (M-10381, CH₃, H, Cl, BnO, H), (M-10382, CH₃, H, Cl, BnO, Cl), (M-10383, CH₃, H, Cl, BnO, F), (M-10384, CH₃, H, Cl, BnO, CF₃), (M-10385, CH₃, H, Cl, BnO, Br), (M-10386, CH₃, H, Cl, BnO, CH₃), (M-10387, CH₃, H, Cl, PhCH₂CH₂O, H), (M-10388, CH₃, H, Cl, PhCH₂CH₂O, Cl), (M-10389, CH₃, H, Cl, PhCH₂CH₂O, F), (M-10390, CH₃, H, Cl, PhCH₂CH₂O, CF₃), (M-10391, CH₃, H, Cl, PhCH₂CH₂O, Br), (M-10392, CH₃, H, Cl, PhCH₂CH₂O, CH₃), (M-10393, CH₃, H, Cl, CF₃O, H), (M-10394, CH₃, H, Cl, CF₃O, Cl), (M-10395, CH₃, H, Cl, CF₃O, F), (M-10396, CH₃, H, Cl, CF₃O, CF₃), (M-10397, CH₃, H, Cl, CF₃O, Br), (M-10398, CH₃, H, Cl, CF₃O, CH₃), (M-10399, CH₃, H, Cl, Ph, H), (M-10400, CH₃, H, Cl, Ph, Cl), (M-10401, CH₃, H, Cl, Ph, F), (M-10402, CH₃, H, Cl, Ph, CF₃), (M-10403, CH₃, H, Cl, Ph, Br), (M-10404, CH₃, H, Cl, Ph, CH₃), (M-10405, CH₃, H, Cl, 4-F-Ph, H), (M-10406, CH₃, H, Cl, 4-F-Ph, Cl), (M-10407, CH₃, H, Cl, 4-F-Ph, F), (M-10408, CH₃, H, Cl, 4-F-Ph, CF₃), (M-10409, CH₃, H, Cl, 4-F-Ph, Br), (M-10410, CH₃, H, Cl, 4-F-Ph, CH₃), (M-10411, CH₃, H, Cl, 4-CF₃-Ph, H), (M-10412, CH₃, H, Cl, 4-CF₃-Ph, Cl), (M-10413, CH₃, H, Cl, 4-CF₃-Ph, F), (M-10414, CH₃, H, Cl, 4-CF₃-Ph, CF₃), (M-10415, CH₃, H, Cl, 4-CF₃-Ph, Br), (M-10416, CH₃, H, Cl, 4-CF₃-Ph, CH₃), (M-10417, CH₃, H, Cl, 4-(Me)₂N-Ph, H), (M-10418, CH₃, H, Cl, 4-(Me)₂N-Ph, Cl), (M-10419, CH₃, H, Cl, 4-(Me)₂N-Ph, F), (M-10420, CH₃, H, Cl, 4-(Me)₂N-Ph, CF₃), (M-10421, CH₃, H, Cl, 4-(Me)₂N-Ph, Br), (M-10422, CH₃, H, Cl, 4-(Me)₂N-Ph, CH₃), (M-10423, CH₃, H, Cl, 4-OH-Ph, H), (M-10424, CH₃, H, Cl, 4-OH-Ph, Cl), (M-10425, CH₃, H, Cl, 4-OH-Ph, F), (M-10426, CH₃, H, Cl, 4-OH-Ph, CF₃), (M-10427, CH₃, H, Cl, 4-OH-Ph, Br), (M-10428, CH₃, H, Cl, 4-OH-Ph, CH₃), (M-10429, CH₃, H, Cl, 3,4-di-F-Ph, H), (M-10430, CH₃, H, Cl, 3,4-di-F-Ph, Cl), (M-10431, CH₃, H, Cl, 3,4-di-F-Ph, F), (M-10432, CH₃, H, Cl, 3,4-di-F-Ph,
CF₃), (M-10433, CH₃, H, Cl, 3,4-di-F-Ph, Br), (M-10434, CH₃, H, Cl, 3,4-di-F-Ph, CH₃), (M-10435, CH₃, H, Cl, 4-COOH-Ph, H), (M-10436, CH₃, H, Cl, 4-COOH-Ph, Cl), (M-10437, CH₃, H, Cl, 4-COOH-Ph, F), (M-10438, CH₃, H, Cl, 4-COOH-Ph, CF₃), (M-10439, CH₃, H, Cl, 4-COOH-Ph, Br), (M-10440, CH₃, H, Cl, 4-COOH-Ph, CH₃), (M-10441, CH₃, H, Cl, Bn, H), (M-10442, CH₃, H, Cl, Bn, Cl), (M-10443, CH₃, H, Cl, Bn, F), (M-10444, CH₃, H, Cl, Bn, CF₃), (M-10445, CH₃, H, Cl, Bn, Br), (M-10446, CH₃, H, Cl, Bn, CH₃), (M-10447, CH₃, H, Cl, 4-F-Bn, H), (M-10448, CH₃, H, Cl, 4-F-Bn, Cl), (M-10449, CH₃, H, Cl, 4-F-Bn, F), (M-10450, CH₃, H, Cl, 4-F-Bn, CF₃), (M-10451, CH₃, H, Cl, 4-F-Bn, Br), (M-10452, CH₃, H, Cl, 4-F-Bn, CH₃), (M-10453, CH₃, H, Cl, 2-Py, H), (M-10454, CH₃, H, Cl, 2-Py, Cl), (M-10455, CH₃, H, Cl, 2-Py, F), (M-10456, CH₃, H, Cl, 2-Py, CF₃), (M-10457, CH₃, H, Cl, 2-Py, Br), (M-10458, CH₃, H, Cl, 2-Py, CH₃), (M-10459, CH₃, H, Cl, 3-Py, H), (M-10460, CH₃, H, Cl, 3-Py, Cl), (M-10461, CH₃, H, Cl, 3-Py, F), (M-10462, CH₃, H, Cl, 3-Py, CF₃), (M-10463, CH₃, H, Cl, 3-Py, Br), (M-10464, CH₃, H, Cl, 3-Py, CH₃), (M-10465, CH₃, H, Cl, 4-Py, H), (M-10466, CH₃, H, Cl, 4-Py, Cl), (M-10467, CH₃, H, Cl, 4-Py, F), (M-10468, CH₃, H, Cl, 4-Py, CF₃), (M-10469, CH₃, H, Cl, 4-Py, Br), (M-10470, CH₃, H, Cl, 4-Py, CH₃), (M-10471, CH₃, H, Cl, 2-Th, H), (M-10472, CH₃, H, Cl, 2-Th, Cl), (M-10473, CH₃, H, Cl, 2-Th, F), (M-10474, CH₃, H, Cl, 2-Th, CF₃), (M-10475, CH₃, H, Cl, 2-Th, Br), (M-10476, CH₃, H, Cl, 2-Th, CH₃), (M-10477, CH₃, H, Cl, 3-Th, H), (M-10478, CH₃, H, Cl, 3-Th, Cl), (M-10479, CH₃, H, Cl, 3-Th, F), (M-10480, CH₃, H, Cl, 3-Th, CF₃), (M-10481, CH₃, H, Cl, 3-Th, Br), (M-10482, CH₃, H, Cl, 3-Th, CH₃), (M-10483, CH₃, H, Cl, pyrazol-2-yl, H), (M-10484, CH₃, H, Cl, pyrazol-2-yl, Cl), (M-10485, CH₃, H, Cl, pyrazol-2-yl, F), (M-10486, CH₃, H, Cl, pyrazol-2-yl, CF₃), (M-10487, CH₃, H, Cl, pyrazol-2-yl, Br), (M-10488, CH₃, H, Cl, pyrazol-2-yl, CH₃), (M-10489, CH₃, H, Cl, pyrazol-3-yl, H), (M-10490, CH₃, H, Cl, pyrazol-3-yl, Cl), (M-10491, CH₃, H, Cl, pyrazol-3-yl, F), (M-10492, CH₃, H, Cl, pyrazol-3-yl, CF₃), (M-10493, CH₃, H, Cl, pyrazol-3-yl, Br), (M-10494, CH₃, H, Cl, pyrazol-3-yl, CH₃), (M-10495, CH₃, H, Cl, pyrimidin-2-yl, H), (M-10496, CH₃, H, Cl, pyrimidin-2-yl, Cl), (M-10497, CH₃, H, Cl, pyrimidin-2-yl, F), (M-10498, CH₃, H, Cl, pyrimidin-2-yl, CF₃), (M-10499, CH₃, H, Cl, pyrimidin-2-yl, Br), (M-10500, CH₃, H, Cl, pyrimidin-2-yl, CH₃), (M-10501, CH₃, H, Cl, pyrimidin-4-yl, H), (M-10502, CH₃, H, Cl, pyrimidin-4-yl, Cl), (M-10503, CH₃, H, Cl, pyrimidin-4-yl, F), (M-10504, CH₃, H, Cl, pyrimidin-4-yl, CF₃), (M-10505, CH₃, H, Cl, pyrimidin-4-yl, Br), (M-10506, CH₃, H, Cl, pyrimidin-4-yl, CH₃), (M-10507, CH₃, H, Cl, pyrimidin-5-yl, H), (M-10508, CH₃, H, Cl, pyrimidin-5-yl, Cl), (M-10509, CH₃, H, Cl, pyrimidin-5-yl, F), (M-10510, CH₃, H, Cl, pyrimidin-5-yl, CF₃), (M-10511, CH₃, H, Cl, pyrimidin-5-yl, Br), (M-10512, CH₃, H, Cl, pyrimidin-5-yl, CH₃), (M-10513, CH₃, H, Cl, HOOCCH₂CH₂CH₂, H), (M-10514, CH₃, H, Cl, HOOCCH₂CH₂CH₂, Cl), (M-10515, CH₃, H, Cl, HOOCCH₂CH₂CH₂, F), (M-10516, CH₃, H, Cl, HOOCCH₂CH₂CH₂, CF₃), (M-10517, CH₃, H, Cl, HOOCCH₂CH₂CH₂, Br), (M-10518, CH₃, H, Cl, HOOCCH₂CH₂CH₂, CH₃), (M-10519, CH₃, H, Cl, HOOCCH₂CH₂CH₂CH₂, H), (M-10520, CH₃, H, Cl, HOOCCH₂CH₂CH₂CH₂, Cl), (M-10521, CH₃, H, Cl, HOOCCH₂CH₂CH₂CH₂, F), (M-10522, CH₃, H, Cl, HOOCCH₂CH₂CH₂CH₂, CF₃), (M-10523, CH₃, H, Cl, HOOCCH₂CH₂CH₂CH₂, Br), (M-10524, CH₃, H, Cl, HOOCCH₂CH₂CH₂CH₂, CH₃), (M-10525, CH₃, H, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂, H), (M-10526, CH₃, H, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂, Cl), (M-10527, CH₃, H, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂, F), (M-10528, CH₃, H, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂, CF₃), (M-10529, CH₃, H, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂, Br), (M-10530, CH₃, H, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂, CH₃), (M-10531, CH₃, H, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, H), (M-10532, CH₃, H, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, Cl), (M-10533, CH₃, H, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, F), (M-10534, CH₃, H, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, CF₃), (M-10535, CH₃, H, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, Br), (M-10536, CH₃, H, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, CH₃), (M-10537, CH₃, H, Cl, MeOCH₂, H), (M-10538, CH₃, H, Cl, MeOCH₂, Cl), (M-10539, CH₃, H, Cl, MeOCH₂, F), (M-10540, CH₃, H, Cl, MeOCH₂, CF₃), (M-10541, CH₃, H, Cl, MeOCH₂, Br), (M-10542, CH₃, H, Cl, MeOCH₂, CH₃), (M-10543, CH₃, H, Cl, EtOCH₂, H), (M-10544, CH₃, H, Cl, EtOCH₂, Cl), (M-10545, CH₃, H, Cl, EtOCH₂, F), (M-10546, CH₃, H, Cl, EtOCH₂, CF₃), (M-10547, CH₃, H, Cl, EtOCH₂, Br), (M-10548, CH₃, H, Cl, EtOCH₂, CH₃), (M-10549, CH₃, H, Cl, EtOCH₂CH₂, H), (M-10550, CH₃, H, Cl, EtOCH₂CH₂, Cl), (M-10551, CH₃, H, Cl, EtOCH₂CH₂, F), (M-10552, CH₃, H, Cl, EtOCH₂CH₂, CF₃), (M-10553, CH₃, H, Cl, EtOCH₂CH₂, Br), (M-10554, CH₃, H, Cl, EtOCH₂CH₂, CH₃), (M-10555, CH₃, H, Cl, MeOCH₂CH₂OCH₂CH₂, H), (M-10556, CH₃, H, Cl, MeOCH₂CH₂OCH₂CH₂, Cl), (M-10557, CH₃, H, Cl, MeOCH₂CH₂OCH₂CH₂, F), (M-10558, CH₃, H, Cl, MeOCH₂CH₂OCH₂CH₂, CF₃), (M-10559, CH₃, H, Cl, MeOCH₂CH₂OCH₂CH₂, Br), (M-10560, CH₃, H, Cl, MeOCH₂CH₂OCH₂CH₂, CH₃), (M-10561, CH₃, H, Cl, MeOCH₂CH₂, H), (M-10562, CH₃, H, Cl, MeOCH₂CH₂, Cl), (M-10563, CH₃, H, Cl, MeOCH₂CH₂, F), (M-10564, CH₃, H, Cl, MeOCH₂CH₂, CF₃), (M-10565, CH₃, H, Cl, MeOCH₂CH₂, Br), (M-10566, CH₃, H, Cl, MeOCH₂CH₂, CH₃), (M-10567, CH₃, H, Cl, HOCH₂, H), (M-10568, CH₃, H, Cl, HOCH₂, Cl), (M-10569, CH₃, H, Cl, HOCH₂, F), (M-10570, CH₃, H, Cl, HOCH₂, CF₃), (M-10571, CH₃, H, Cl, HOCH₂, Br), (M-10572, CH₃, H, Cl, HOCH₂, CH₃), (M-10573, CH₃, H, Cl, HOCH₂CH₂, H), (M-10574, CH₃, H, Cl, HOCH₂CH₂, Cl), (M-10575, CH₃, H, Cl, HOCH₂CH₂, F), (M-10576, CH₃, H, Cl, HOCH₂CH₂, CF₃), (M-10577, CH₃, H, Cl, HOCH₂CH₂, Br), (M-10578, CH₃, H, Cl, HOCH₂CH₂, CH₃), (M-10579, CH₃, H, Cl, HOCH₂CH₂CH₂, H), (M-10580, CH₃, H, Cl, HOCH₂CH₂CH₂, Cl), (M-10581, CH₃, H, Cl, HOCH₂CH₂CH₂, F), (M-10582, CH₃, H, Cl, HOCH₂CH₂CH₂, CF₃), (M-10583, CH₃,
H, Cl, HOCH₂CH₂CH₂, Br), (M-10584, CH₃, H, Cl, HOCH₂CH₂CH₂, CH₃), (M-10585, CH₃, H, Cl, HOCH₂CH₂CH₂CH₂, H), (M-10586, CH₃, H, Cl, HOCH₂CH₂CH₂CH₂, Cl), (M-10587, CH₃, H, Cl, HOCH₂CH₂CH₂CH₂, F), (M-10588, CH₃, H, Cl, HOCH₂CH₂CH₂CH₂, CF₃), (M-10589, CH₃, H, Cl, HOCH₂CH₂CH₂CH₂, Br), (M-10590, CH₃, H, Cl, HOCH₂CH₂CH₂CH₂, CH₃), (M-10591, CH₃, H, Cl, HOCH₂CH₂CH₂CH₂CH₂, H), (M-10592, CH₃, H, Cl, HOCH₂CH₂CH₂CH₂CH₂, Cl), (M-10593, CH₃, H, Cl, HOCH₂CH₂CH₂CH₂CH₂, F), (M-10594, CH₃, H, Cl, HOCH₂CH₂CH₂CH₂CH₂, CF₃), (M-10595, CH₃, H, Cl, HOCH₂CH₂CH₂CH₂CH₂, Br), (M-10596, CH₃, H, Cl, HOCH₂CH₂CH₂CH₂CH₂, CH₃), (M-10597, CH₃, H, Cl, HOCH₂CH₂OCH₂CH₂, H), (M-10598, CH₃, H, Cl, HOCH₂CH₂OCH₂CH₂, Cl), (M-10599, CH₃, H, Cl, HOCH₂CH₂OCH₂CH₂, F), (M-10600, CH₃, H, Cl, HOCH₂CH₂OCH₂CH₂, CF₃), (M-10601, CH₃, H, Cl, HOCH₂CH₂OCH₂CH₂, Br), (M-10602, CH₃, H, Cl, HOCH₂CH₂OCH₂CH₂, CH₃), (M-10603, CH₃, H, Cl, (Me)₂N, H), (M-10604, CH₃, H, Cl, (Me)₂N, Cl), (M-10605, CH₃, H, Cl, (Me)₂N, F), (M-10606, CH₃, H, Cl, (Me)₂N, CF₃), (M-10607, CH₃, H, Cl, (Me)₂N, Br), (M-10608, CH₃, H, Cl, (Me)₂N, CH₃), (M-10609, CH₃, H, Cl, piperidin-4-yl-methyl, H), (M-10610, CH₃, H, Cl, piperidin-4-yl-methyl, Cl), (M-10611, CH₃, H, Cl, piperidin-4-yl-methyl, F), (M-10612, CH₃, H, Cl, piperidin-4-yl-methyl, CF₃), (M-10613, CH₃, H, Cl, piperidin-4-yl-methyl, Br), (M-10614, CH₃, H, Cl, piperidin-4-yl-methyl, CH₃), (M-10615, CH₃, H, Cl, cyclohexylmethyl, H), (M-10616, CH₃, H, Cl, cyclohexylmethyl, Cl), (M-10617, CH₃, H, Cl, cyclohexylmethyl, F), (M-10618, CH₃, H, Cl, cyclohexylmethyl, CF₃), (M-10619, CH₃, H, Cl, cyclohexylmethyl, Br), (M-10620, CH₃, H, Cl, cyclohexylmethyl, CH₃), (M-10621, CH₃, F, H, H, H), (M-10622, CH₃, F, H, H, Cl), (M-10623, CH₃, F, H, H, F), (M-10624, CH₃, F, H, H, CF₃), (M-10625, CH₃, F, H, H, Br), (M-10626, CH₃, F, H, H, CH₃), (M-10627, CH₃, F, H, F, H), (M-10628, CH₃, F, H, F, Cl), (M-10629, CH₃, F, H, F, F), (M-10630, CH₃, F, H, F, CF₃), (M-10631, CH₃, F, H, F, Br), (M-10632, CH₃, F, H, F, CH₃), (M-10633, CH₃, F, H, Cl, H), (M-10634, CH₃, F, H, Cl, Cl), (M-10635, CH₃, F, H, Cl, F), (M-10636, CH₃, F, H, Cl, CF₃), (M-10637, CH₃, F, H, Cl, Br), (M-10638, CH₃, F, H, Cl, CH₃), (M-10639, CH₃, F, H, CH₃, H), (M-10640, CH₃, F, H, CH₃, Cl), (M-10641, CH₃, F, H, CH₃, F), (M-10642, CH₃, F, H, CH₃, CF₃), (M-10643, CH₃, F, H, CH₃, Br), (M-10644, CH₃, F, H, CH₃, CH₃), (M-10645, CH₃, F, H, Et, H), (M-10646, CH₃, F, H, Et, Cl), (M-10647, CH₃, F, H, Et, F), (M-10648, CH₃, F, H, Et, CF₃), (M-10649, CH₃, F, H, Et, Br), (M-10650, CH₃, F, H, Et, CH₃), (M-10651, CH₃, F, H, n-Pr, H), (M-10652, CH₃, F, H, n-Pr, Cl), (M-10653, CH₃, F, H, n-Pr, F), (M-10654, CH₃, F, H, n-Pr, CF₃), (M-10655, CH₃, F, H, n-Pr, Br), (M-10656, CH₃, F, H, n-Pr, CH₃), (M-10657, CH₃, F, H, c-Pr, H), (M-10658, CH₃, F, H, c-Pr, Cl), (M-10659, CH₃, F, H, c-Pr, F), (M-10660, CH₃, F, H, c-Pr, CF₃), (M-10661, CH₃, F, H, c-Pr, Br), (M-10662, CH₃, F, H, c-Pr, CH₃), (M-10663, CH₃, F, H, i-Pr, H), (M-10664, CH₃, F, H, i-Pr, Cl), (M-10665, CH₃, F, H, i-Pr, F), (M-10666, CH₃, F, H, i-Pr, CF₃), (M-10667, CH₃, F, H, i-Pr, Br), (M-10668, CH₃, F, H, i-Pr, CH₃), (M-10669, CH₃, F, H, n-Bu, H), (M-10670, CH₃, F, H, n-Bu, Cl), (M-10671, CH₃, F, H, n-Bu, F), (M-10672, CH₃, F, H, n-Bu, CF₃), (M-10673, CH₃, F, H, n-Bu, Br), (M-10674, CH₃, F, H, n-Bu, CH₃), (M-10675, CH₃, F, H, i-Bu, H), (M-10676, CH₃, F, H, i-Bu, Cl), (M-10677, CH₃, F, H, i-Bu, F), (M-10678, CH₃, F, H, i-Bu, CF₃), (M-10679, CH₃, F, H, i-Bu, Br), (M-10680, CH₃, F, H, i-Bu, CH₃), (M-10681, CH₃, F, H, sec-Bu, H), (M-10682, CH₃, F, H, sec-Bu, Cl), (M-10683, CH₃, F, H, sec-Bu, F), (M-10684, CH₃, F, H, sec-Bu, CF₃), (M-10685, CH₃, F, H, sec-Bu, Br), (M-10686, CH₃, F, H, sec-Bu, CH₃), (M-10687, CH₃, F, H, n-Pen, H), (M-10688, CH₃, F, H, n-Pen, Cl), (M-10689, CH₃, F, H, n-Pen, F), (M-10690, CH₃, F, H, n-Pen, CF₃), (M-10691, CH₃, F, H, n-Pen, Br), (M-10692, CH₃, F, H, n-Pen, CH₃), (M-10693, CH₃, F, H, c-Pen, H), (M-10694, CH₃, F, H, c-Pen, Cl), (M-10695, CH₃, F, H, c-Pen, F), (M-10696, CH₃, F, H, c-Pen, CF₃), (M-10697, CH₃, F, H, c-Pen, Br), (M-10698, CH₃, F, H, c-Pen, CH₃), (M-10699, CH₃, F, H, n-Hex, H), (M-10700, CH₃, F, H, n-Hex, Cl), (M-10701, CH₃, F, H, n-Hex, F), (M-10702, CH₃, F, H, n-Hex, CF₃), (M-10703, CH₃, F, H, n-Hex, Br), (M-10704, CH₃, F, H, n-Hex, CH₃), (M-10705, CH₃, F, H, c-Hex, H), (M-10706, CH₃, F, H, c-Hex, Cl), (M-10707, CH₃, F, H, c-Hex, F), (M-10708, CH₃, F, H, c-Hex, CF₃), (M-10709, CH₃, F, H, c-Hex, Br), (M-10710, CH₃, F, H, c-Hex, CH₃), (M-10711, CH₃, F, H, OH, H), (M-10712, CH₃, F, H, OH, Cl), (M-10713, CH₃, F, H, OH, F), (M-10714, CH₃, F, H, OH, CF₃), (M-10715, CH₃, F, H, OH, Br), (M-10716, CH₃, F, H, OH, CH₃), (M-10717, CH₃, F, H, EtO, H), (M-10718, CH₃, F, H, EtO, Cl), (M-10719, CH₃, F, H, EtO, F), (M-10720, CH₃, F, H, EtO, CF₃), (M-10721, CH₃, F, H, EtO, Br), (M-10722, CH₃, F, H, EtO, CH₃), (M-10723, CH₃, F, H, n-PrO, H), (M-10724, CH₃, F, H, n-PrO, Cl), (M-10725, CH₃, F, H, n-PrO, F), (M-10726, CH₃, F, H, n-PrO, CF₃), (M-10727, CH₃, F, H, n-PrO, Br), (M-10728, CH₃, F, H, n-PrO, CH₃), (M-10729, CH₃, F, H, PhO, H), (M-10730, CH₃, F, H, PhO, Cl), (M-10731, CH₃, F, H, PhO, F), (M-10732, CH₃, F, H, PhO, CF₃), (M-10733, CH₃, F, H, PhO, Br), (M-10734, CH₃, F, H, PhO, CH₃), (M-10735, CH₃, F, H, BnO, H), (M-10736, CH₃, F, H, BnO, Cl), (M-10737, CH₃, F, H, BnO, F), (M-10738, CH₃, F, H, BnO, CF₃), (M-10739, CH₃, F, H, BnO, Br), (M-10740, CH₃, F, H, BnO, CH₃), (M-10741, CH₃, F, H, PhCH₂CH₂O, H), (M-10742, CH₃, F, H, PhCH₂CH₂O, Cl), (M-10743, CH₃, F, H, PhCH₂CH₂O, F), (M-10744, CH₃, F, H, PhCH₂CH₂O, CF₃), (M-10745, CH₃, F, H, PhCH₂CH₂O, Br), (M-10746, CH₃, F, H, PhCH₂CH₂O, CH₃), (M-10747, CH₃, F, H, CF₃O, H), (M-10748, CH₃, F, H, CF₃O, Cl), (M-10749, CH₃, F, H, CF₃O, F), (M-10750, CH₃, F, H, CF₃O, CF₃), (M-10751, CH₃, F, H, CF₃O, Br), (M-10752, CH₃, F, H, CF₃O, CH₃), (M-10753, CH₃, F, H, Ph, H), (M-10754, CH₃, F, H, Ph, Cl), (M-10755, CH₃, F, H, Ph, F), (M-10756, CH₃, F, H, Ph, CF₃), (M-10757, CH₃, F, H, Ph, Br), (M-10758, CH₃, F, H, Ph, CH₃), (M-10759, CH₃, F, H, 4-F-Ph, H), (M-10760, CH₃, F, H, 4-F-Ph, Cl), (M-10761, CH₃, F, H, 4-F-Ph, F), (M-10762, CH₃, F, H, 4-F-Ph, CF₃), (M-10763, CH₃, F, H, 4-F-Ph, Br), (M-10764, CH₃, F, H, 4-F-Ph, CH₃), (M-10765, CH₃, F, H, 4-CF₃-Ph, H), (M-10766, CH₃, F, H, 4-CF
₃-Ph, Cl), (M-10767, CH₃, F, H, 4-CF₃-Ph, F), (M-10768, CH₃, F, H, 4-CF₃-Ph, CF₃), (M-10769, CH₃, F, H, 4-CF₃-Ph, Br), (M-10770, CH₃, F, H, 4-CF₃-Ph, CH₃), (M-10771, CH₃, F, H, 4-(Me)₂N-Ph, H), (M-10772, CH₃, F, H, 4-(Me)₂N-Ph, Cl), (M-10773, CH₃, F, H, 4-(Me)₂N-Ph, F), (M-10774, CH₃, F, H, 4-(Me)₂N-Ph, CF₃), (M-10775, CH₃, F, H, 4-(Me)₂N-Ph, Br), (M-10776, CH₃, F, H, 4-(Me)₂N-Ph, CH₃), (M-10777, CH₃, F, H, 4-OH-Ph, H), (M-10778, CH₃, F, H, 4-OH-Ph, Cl), (M-10779, CH₃, F, H, 4-OH-Ph, F), (M-10780, CH₃, F, H, 4-OH-Ph, CF₃), (M-10781, CH₃, F, H, 4-OH-Ph, Br), (M-10782, CH₃, F, H, 4-OH-Ph, CH₃), (M-10783, CH₃, F, H, 3,4-di-F-Ph, H), (M-10784, CH₃, F, H, 3,4-di-F-Ph, Cl), (M-10785, CH₃, F, H, 3,4-di-F-Ph, F), (M-10786, CH₃, F, H, 3,4-di-F-Ph, CF₃), (M-10787, CH₃, F, H, 3,4-di-F-Ph, Br), (M-10788, CH₃, F, H, 3,4-di-F-Ph, CH₃), (M-10789, CH₃, F, H, 4-COOH-Ph, H), (M-10790, CH₃, F, H, 4-COOH-Ph, Cl), (M-10791, CH₃, F, H, 4-COOH-Ph, F), (M-10792, CH₃, F, H, 4-COOH-Ph, CF₃), (M-10793, CH₃, F, H, 4-COOH-Ph, Br), (M-10794, CH₃, F, H, 4-COOH-Ph, CH₃), (M-10795, CH₃, F, H, Bn, H), (M-10796, CH₃, F, H, Bn, Cl), (M-10797, CH₃, F, H, Bn, F), (M-10798, CH₃, F, H, Bn, CF₃), (M-10799, CH₃, F, H, Bn, Br), (M-10800, CH₃, F, H, Bn, CH₃), (M-10801, CH₃, F, H, 4-F-Bn, H), (M-10802, CH₃, F, H, 4-F-Bn, Cl), (M-10803, CH₃, F, H, 4-F-Bn, F), (M-10804, CH₃, F, H, 4-F-Bn, CF₃), (M-10805, CH₃, F, H, 4-F-Bn, Br), (M-10806, CH₃, F, H, 4-F-Bn, CH₃), (M-10807, CH₃, F, H, 2-Py, H), (M-10808, CH₃, F, H, 2-Py, Cl), (M-10809, CH₃, F, H, 2-Py, F), (M-10810, CH₃, F, H, 2-Py, CF₃), (M-10811, CH₃, F, H, 2-Py, Br), (M-10812, CH₃, F, H, 2-Py, CH₃), (M-10813, CH₃, F, H, 3-Py, H), (M-10814, CH₃, F, H, 3-Py, Cl), (M-10815, CH₃, F, H, 3-Py, F), (M-10816, CH₃, F, H, 3-Py, CF₃), (M-10817, CH₃, F, H, 3-Py, Br), (M-10818, CH₃, F, H, 3-Py, CH₃), (M-10819, CH₃, F, H, 4-Py, H), (M-10820, CH₃, F, H, 4-Py, Cl), (M-10821, CH₃, F, H, 4-Py, F), (M-10822, CH₃, F, H, 4-Py, CF₃), (M-10823, CH₃, F, H, 4-Py, Br), (M-10824, CH₃, F, H, 4-Py, CH₃), (M-10825, CH₃, F, H, 2-Th, H), (M-10826, CH₃, F, H, 2-Th, Cl), (M-10827, CH₃, F, H, 2-Th, F), (M-10828, CH₃, F, H, 2-Th, CF₃), (M-10829, CH₃, F, H, 2-Th, Br), (M-10830, CH₃, F, H, 2-Th, CH₃), (M-10831, CH₃, F, H, 3-Th, H), (M-10832, CH₃, F, H, 3-Th, Cl), (M-10833, CH₃, F, H, 3-Th, F), (M-10834, CH₃, F, H, 3-Th, CF₃), (M-10835, CH₃, F, H, 3-Th, Br), (M-10836, CH₃, F, H, 3-Th, CH₃), (M-10837, CH₃, F, H, pyrazol-2-yl, H), (M-10838, CH₃, F, H, pyrazol-2-yl, Cl), (M-10839, CH₃, F, H, pyrazol-2-yl, F), (M-10840, CH₃, F, H, pyrazol-2-yl, CF₃), (M-10841, CH₃, F, H, pyrazol-2-yl, Br), (M-10842, CH₃, F, H, pyrazol-2-yl, CH₃), (M-10843, CH₃, F, H, pyrazol-3-yl, H), (M-10844, CH₃, F, H, pyrazol-3-yl, Cl), (M-10845, CH₃, F, H, pyrazol-3-yl, F), (M-10846, CH₃, F, H, pyrazol-3-yl, CF₃), (M-10847, CH₃, F, H, pyrazol-3-yl, Br), (M-10848, CH₃, F, H, pyrazol-3-yl, CH₃), (M-10849, CH₃, F, H, pyrimidin-2-yl, H), (M-10850, CH₃, F, H, pyrimidin-2-yl, Cl), (M-10851, CH₃, F, H, pyrimidin-2-yl, F), (M-10852, CH₃, F, H, pyrimidin-2-yl, CF₃), (M-10853, CH₃, F, H, pyrimidin-2-yl, Br), (M-10854, CH₃, F, H, pyrimidin-2-yl, CH₃), (M-10855, CH₃, F, H, pyrimidin-4-yl, H), (M-10856, CH₃, F, H, pyrimidin-4-yl, Cl), (M-10857, CH₃, F, H, pyrimidin-4-yl, F), (M-10858, CH₃, F, H, pyrimidin-4-yl, CF₃), (M-10859, CH₃, F, H, pyrimidin-4-yl, Br), (M-10860, CH₃, F, H, pyrimidin-4-yl, CH₃), (M-10861, CH₃, F, H, pyrimidin-5-yl, H), (M-10862, CH₃, F, H, pyrimidin-5-yl, Cl), (M-10863, CH₃, F, H, pyrimidin-5-yl, F), (M-10864, CH₃, F, H, pyrimidin-5-yl, CF₃), (M-10865, CH₃, F, H, pyrimidin-5-yl, Br), (M-10866, CH₃, F, H, pyrimidin-5-yl, CH₃), (M-10867, CH₃, F, H, HOOCCH₂CH₂CH₂, H), (M-10868, CH₃, F, H, HOOCCH₂CH₂CH₂, Cl), (M-10869, CH₃, F, H, HOOCCH₂CH₂CH₂, F), (M-10870, CH₃, F, H, HOOCCH₂CH₂CH₂, CF₃), (M-10871, CH₃, F, H, HOOCCH₂CH₂CH₂, Br), (M-10872, CH₃, F, H, HOOCCH₂CH₂CH₂, CH₃), (M-10873, CH₃, F, H, HOOCCH₂CH₂CH₂CH₂, H), (M-10874, CH₃, F, H, HOOCCH₂CH₂CH₂CH₂, Cl), (M-10875, CH₃, F, H, HOOCCH₂CH₂CH₂CH₂, F), (M-10876, CH₃, F, H, HOOCCH₂CH₂CH₂CH₂, CF₃), (M-10877, CH₃, F, H, HOOCCH₂CH₂CH₂CH₂, Br), (M-10878, CH₃, F, H, HOOCCH₂CH₂CH₂CH₂, CH₃), (M-10879, CH₃, F, H, (Me)₂NCOCH₂CH₂CH₂CH₂, H), (M-10880, CH₃, F, H, (Me)₂NCOCH₂CH₂CH₂CH₂, Cl), (M-10881, CH₃, F, H, (Me)₂NCOCH₂CH₂CH₂CH₂, F), (M-10882, CH₃, F, H, (Me)₂NCOCH₂CH₂CH₂CH₂, CF₃), (M-10883, CH₃, F, H, (Me)₂NCOCH₂CH₂CH₂CH₂, Br), (M-10884, CH₃, F, H, (Me)₂NCOCH₂CH₂CH₂CH₂, CH₃), (M-10885, CH₃, F, H, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, H), (M-10886, CH₃, F, H, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, Cl), (M-10887, CH₃, F, H, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, F), (M-10888, CH₃, F, H, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, CF₃), (M-10889, CH₃, F, H, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, Br), (M-10890, CH₃, F, H, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, CH₃), (M-10891, CH₃, F, H, MeOCH₂, H), (M-10892, CH₃, F, H, MeOCH₂, Cl), (M-10893, CH₃, F, H, MeOCH₂, F), (M-10894, CH₃, F, H, MeOCH₂, CF₃), (M-10895, CH₃, F, H, MeOCH₂, Br), (M-10896, CH₃, F, H, MeOCH₂, CH₃), (M-10897, CH₃, F, H, EtOCH₂, H), (M-10898, CH₃, F, H, EtOCH₂, Cl), (M-10899, CH₃, F, H, EtOCH₂, F), (M-10900, CH₃, F, H, EtOCH₂, CF₃), (M-10901, CH₃, F, H, EtOCH₂, Br), (M-10902, CH₃, F, H, EtOCH₂, CH₃), (M-10903, CH₃, F, H, EtOCH₂CH₂, H), (M-10904, CH₃, F, H, EtOCH₂CH₂, Cl), (M-10905, CH₃, F, H, EtOCH₂CH₂, F), (M-10906, CH₃, F, H, EtOCH₂CH₂, CF₃), (M-10907, CH₃, F, H, EtOCH₂CH₂, Br), (M-10908, CH₃, F, H, EtOCH₂CH₂, CH₃), (M-10909, CH₃, F, H, MeOCH₂CH₂OCH₂CH₂, H), (M-10910, CH₃, F, H, MeOCH₂CH₂OCH₂CH₂, Cl), (M-10911, CH₃, F, H, MeOCH₂CH₂OCH₂CH₂, F), (M-10912, CH₃, F, H, MeOCH₂CH₂OCH₂CH₂, CF₃), (M-10913, CH₃, F, H, MeOCH₂CH₂OCH₂CH₂, Br), (M-10914, CH₃, F, H, MeOCH₂CH₂OCH₂CH₂, CH₃), (M-10915, CH₃, F, H, MeOCH₂CH₂, H), (M-10916, CH₃, F, H, MeOCH₂CH₂, Cl), (M-10917, CH₃, F, H, MeOCH₂CH₂, F), (M-10918, CH₃, F, H, MeOCH₂CH₂, CF₃), (M-10919, CH₃, F, H, MeOCH₂CH₂, Br), (M-10920, CH₃, F, H, MeOCH₂CH₂, CH₃), (M-10921, CH₃, F, H, HOCH₂, H), (M-10922, CH₃, F, H, HOCH₂, Cl), (M-10923, CH₃, F, H, HOCH₂
, F), (M-10924, CH₃, F, H, HOCH₂, CF₃), (M-10925, CH₃, F, H, HOCH₂, Br), (M-10926, CH₃, F, H, HOCH₂, CH₃), (M-10927, CH₃, F, H, HOCH₂CH₂, H), (M-10928, CH₃, F, H, HOCH₂CH₂, Cl), (M-10929, CH₃, F, H, HOCH₂CH₂, F), (M-10930, CH₃, F, H, HOCH₂CH₂, CF₃), (M-10931, CH₃, F, H, HOCH₂CH₂, Br), (M-10932, CH₃, F, H, HOCH₂CH₂, CH₃), (M-10933, CH₃, F, H, HOCH₂CH₂CH₂, H), (M-10934, CH₃, F, H, HOCH₂CH₂CH₂, Cl), (M-10935, CH₃, F, H, HOCH₂CH₂CH₂, F), (M-10936, CH₃, F, H, HOCH₂CH₂CH₂, CF₃), (M-10937, CH₃, F, H, HOCH₂CH₂CH₂, Br), (M-10938, CH₃, F, H, HOCH₂CH₂CH₂, CH₃), (M-10939, CH₃, F, H, HOCH₂CH₂CH₂CH₂, H), (M-10940, CH₃, F, H, HOCH₂CH₂CH₂CH₂, Cl), (M-10941, CH₃, F, H, HOCH₂CH₂CH₂CH₂, F), (M-10942, CH₃, F, H, HOCH₂CH₂CH₂CH₂, CF₃), (M-10943, CH₃, F, H, HOCH₂CH₂CH₂CH₂, Br), (M-10944, CH₃, F, H, HOCH₂CH₂CH₂CH₂, CH₃), (M-10945, CH₃, F, H, HOCH₂CH₂CH₂CH₂CH₂, H), (M-10946, CH₃, F, H, HOCH₂CH₂CH₂CH₂CH₂, Cl), (M-10947, CH₃, F, H, HOCH₂CH₂CH₂CH₂CH₂, F), (M-10948, CH₃, F, H, HOCH₂CH₂CH₂CH₂CH₂, CF₃), (M-10949, CH₃, F, H, HOCH₂CH₂CH₂CH₂CH₂, Br), (M-10950, CH₃, F, H, HOCH₂CH₂CH₂CH₂CH₂, CH₃), (M-10951, CH₃, F, H, HOCH₂CH₂OCH₂CH₂, H), (M-10952, CH₃, F, H, HOCH₂CH₂OCH₂CH₂, Cl), (M-10953, CH₃, F, H, HOCH₂CH₂OCH₂CH₂, F), (M-10954, CH₃, F, H, HOCH₂CH₂OCH₂CH₂, CF₃), (M-10955, CH₃, F, H, HOCH₂CH₂OCH₂CH₂, Br), (M-10956, CH₃, F, H, HOCH₂CH₂OCH₂CH₂, CH₃), (M-10957, CH₃, F, H, (Me)₂N, H), (M-10958, CH₃, F, H, (Me)₂N, Cl), (M-10959, CH₃, F, H, (Me)₂N, F), (M-10960, CH₃, F, H, (Me)₂N, CF₃), (M-10961, CH₃, F, H, (Me)₂N, Br), (M-10962, CH₃, F, H, (Me)₂N, CH₃), (M-10963, CH₃, F, H, piperidin-4-yl-methyl, H), (M-10964, CH₃, F, H, piperidin-4-yl-methyl, Cl), (M-10965, CH₃, F, H, piperidin-4-yl-methyl, F), (M-10966, CH₃, F, H, piperidin-4-yl-methyl, CF₃), (M-10967, CH₃, F, H, piperidin-4-yl-methyl, Br), (M-10968, CH₃, F, H, piperidin-4-yl-methyl, CH₃), (M-10969, CH₃, F, H, cyclohexylmethyl, H), (M-10970, CH₃, F, H, cyclohexylmethyl, Cl), (M-10971, CH₃, F, H, cyclohexylmethyl, F), (M-10972, CH₃, F, H, cyclohexylmethyl, CF₃), (M-10973, CH₃, F, H, cyclohexylmethyl, Br), (M-10974, CH₃, F, H, cyclohexylmethyl, CH₃), (M-10975, CH₃, F, F, H, H), (M-10976, CH₃, F, F, H, Cl), (M-10977, CH₃, F, F, H, F), (M-10978, CH₃, F, F, H, CF₃), (M-10979, CH₃, F, F, H, Br), (M-10980, CH₃, F, F, H, CH₃), (M-10981, CH₃, F, F, F, H), (M-10982, CH₃, F, F, F, Cl), (M-10983, CH₃, F, F, F, F), (M-10984, CH₃, F, F, F, CF₃), (M-10985, CH₃, F, F, F, Br), (M-10986, CH₃, F, F, F, CH₃), (M-10987, CH₃, F, F, Cl, H), (M-10988, CH₃, F, F, Cl, Cl), (M-10989, CH₃, F, F, Cl, F), (M-10990, CH₃, F, F, Cl, CF₃), (M-10991, CH₃, F, F, Cl, Br), (M-10992, CH₃, F, F, Cl, CH₃), (M-10993, CH₃, F, F, CH₃, H), (M-10994, CH₃, F, F, CH₃, Cl), (M-10995, CH₃, F, F, CH₃, F), (M-10996, CH₃, F, F, CH₃, CF₃), (M-10997, CH₃, F, F, CH₃, Br), (M-10998, CH₃, F, F, CH₃, CH₃), (M-10999, CH₃, F, F, Et, H), (M-11000, CH₃, F, F, Et, Cl), (M-11001, CH₃, F, F, Et, F), (M-11002, CH₃, F, F, Et, CF₃), (M-11003, CH₃, F, F, Et, Br), (M-11004, CH₃, F, F, Et, CH₃), (M-11005, CH₃, F, F, n-Pr, H), (M-11006, CH₃, F, F, n-Pr, Cl), (M-11007, CH₃, F, F, n-Pr, F), (M-11008, CH₃, F, F, n-Pr, CF₃), (M-11009, CH₃, F, F, n-Pr, Br), (M-11010, CH₃, F, F, n-Pr, CH₃), (M-11011, CH₃, F, F, c-Pr, H), (M-11012, CH₃, F, F, c-Pr, Cl), (M-11013, CH₃, F, F, c-Pr, F), (M-11014, CH₃, F, F, c-Pr, CF₃), (M-11015, CH₃, F, F, c-Pr, Br), (M-11016, CH₃, F, F, c-Pr, CH₃), (M-11017, CH₃, F, F, i-Pr, H), (M-11018, CH₃, F, F, i-Pr, Cl), (M-11019, CH₃, F, F, i-Pr, F), (M-11020, CH₃, F, F, i-Pr, CF₃), (M-11021, CH₃, F, F, i-Pr, Br), (M-11022, CH₃, F, F, i-Pr, CH₃), (M-11023, CH₃, F, F, n-Bu, H), (M-11024, CH₃, F, F, n-Bu, Cl), (M-11025, CH₃, F, F, n-Bu, F), (M-11026, CH₃, F, F, n-Bu, CF₃), (M-11027, CH₃, F, F, n-Bu, Br), (M-11028, CH₃, F, F, n-Bu, CH₃), (M-11029, CH₃, F, F, i-Bu, H), (M-11030, CH₃, F, F, i-Bu, Cl), (M-11031, CH₃, F, F, i-Bu, F), (M-11032, CH₃, F, F, i-Bu, CF₃), (M-11033, CH₃, F, F, i-Bu, Br), (M-11034, CH₃, F, F, i-Bu, CH₃), (M-11035, CH₃, F, F, sec-Bu, H), (M-11036, CH₃, F, F, sec-Bu, Cl), (M-11037, CH₃, F, F, sec-Bu, F), (M-11038, CH₃, F, F, sec-Bu, CF₃), (M-11039, CH₃, F, F, sec-Bu, Br), (M-11040, CH₃, F, F, sec-Bu, CH₃), (M-11041, CH₃, F, F, n-Pen, H), (M-11042, CH₃, F, F, n-Pen, Cl), (M-11043, CH₃, F, F, n-Pen, F), (M-11044, CH₃, F, F, n-Pen, CF₃), (M-11045, CH₃, F, F, n-Pen, Br), (M-11046, CH₃, F, F, n-Pen, CH₃), (M-11047, CH₃, F, F, c-Pen, H), (M-11048, CH₃, F, F, c-Pen, Cl), (M-11049, CH₃, F, F, c-Pen, F), (M-11050, CH₃, F, F, c-Pen, CF₃), (M-11051, CH₃, F, F, c-Pen, Br), (M-11052, CH₃, F, F, c-Pen, CH₃), (M-11053, CH₃, F, F, n-Hex, H), (M-11054, CH₃, F, F, n-Hex, Cl), (M-11055, CH₃, F, F, n-Hex, F), (M-11056, CH₃, F, F, n-Hex, CF₃), (M-11057, CH₃, F, F, n-Hex, Br), (M-11058, CH₃, F, F, n-Hex, CH₃), (M-11059, CH₃, F, F, c-Hex, H), (M-11060, CH₃, F, F, c-Hex, Cl), (M-11061, CH₃, F, F, c-Hex, F), (M-11062, CH₃, F, F, c-Hex, CF₃), (M-11063, CH₃, F, F, c-Hex, Br), (M-11064, CH₃, F, F, c-Hex, CH₃), (M-11065, CH₃, F, F, OH, H), (M-11066, CH₃, F, F, OH, Cl), (M-11067, CH₃, F, F, OH, F), (M-11068, CH₃, F, F, OH, CF₃), (M-11069, CH₃, F, F, OH, Br), (M-11070, CH₃, F, F, OH, CH₃), (M-11071, CH₃, F, F, EtO, H), (M-11072, CH₃, F, F, EtO, Cl), (M-11073, CH₃, F, F, EtO, F), (M-11074, CH₃, F, F, EtO, CF₃), (M-11075, CH₃, F, F, EtO, Br), (M-11076, CH₃, F, F, EtO, CH₃), (M-11077, CH₃, F, F, n-PrO, H), (M-11078, CH₃, F, F, n-PrO, Cl), (M-11079, CH₃, F, F, n-PrO, F), (M-11080, CH₃, F, F, n-PrO, CF₃), (M-11081, CH₃, F, F, n-PrO, Br), (M-11082, CH₃, F, F, n-PrO, CH₃), (M-11083, CH₃, F, F, PhO, H), (M-11084, CH₃, F, F, PhO, Cl), (M-11085, CH₃, F, F, PhO, F), (M-11086, CH₃, F, F, PhO, CF₃), (M-11087, CH₃, F, F, PhO, Br), (M-11088, CH₃, F, F, PhO, CH₃), (M-11089, CH₃, F, F, BnO, H), (M-11090, CH₃, F, F, BnO, Cl), (M-11091, CH₃, F, F, BnO, F), (M-11092, CH₃, F, F, BnO, CF₃), (M-11093, CH₃, F, F, BnO, Br), (M-11094, CH₃, F, F, BnO, CH₃), (M-11095, CH₃, F, F, PhCH₂CH₂O, H), (M-11096, CH₃, F, F, PhCH₂CH₂O, Cl), (M-11097, CH₃, F, F, PhCH₂CH₂O, F), (M-11098, CH₃, F, F, PhCH₂CH₂O, CF₃), (M-11099, CH₃, F, F, PhCH₂CH₂O, Br), (M-11100, CH₃, F, F, PhCH₂CH₂O, CH₃), (M-11101, CH₃, F, F, CF₃
O, H), (M-11102, CH₃, F, F, CF₃O, Cl), (M-11103, CH₃, F, F, CF₃O, F), (M-11104, CH₃, F, F, CF₃O, CF₃), (M-11105, CH₃, F, F, CF₃O, Br), (M-11106, CH₃, F, F, CF₃O, CH₃), (M-11107, CH₃, F, F, Ph, H), (M-11108, CH₃, F, F, Ph, Cl), (M-11109, CH₃, F, F, Ph, F), (M-11110, CH₃, F, F, Ph, CF₃), (M-11111, CH₃, F, F, Ph, Br), (M-11112, CH₃, F, F, Ph, CH₃), (M-11113, CH₃, F, F, 4-F-Ph, H), (M-11114, CH₃, F, F, 4-F-Ph, Cl), (M-11115, CH₃, F, F, 4-F-Ph, F), (M-11116, CH₃, F, F, 4-F-Ph, CF₃), (M-11117, CH₃, F, F, 4-F-Ph, Br), (M-11118, CH₃, F, F, 4-F-Ph, CH₃), (M-11119, CH₃, F, F, 4-CF₃-Ph, H), (M-11120, CH₃, F, F, 4-CF₃-Ph, Cl), (M-11121, CH₃, F, F, 4-CF₃-Ph, F), (M-11122, CH₃, F, F, 4-CF₃-Ph, CF₃), (M-11123, CH₃, F, F, 4-CF₃-Ph, Br), (M-11124, CH₃, F, F, 4-CF₃-Ph, CH₃), (M-11125, CH₃, F, F, 4-(Me)₂N-Ph, H), (M-11126, CH₃, F, F, 4-(Me)₂N-Ph, Cl), (M-11127, CH₃, F, F, 4-(Me)₂N-Ph, F), (M-11128, CH₃, F, F, 4-(Me)₂N-Ph, CF₃), (M-11129, CH₃, F, F, 4-(Me)₂N-Ph, Br), (M-11130, CH₃, F, F, 4-(Me)₂N-Ph, CH₃), (M-11131, CH₃, F, F, 4-OH-Ph, H), (M-11132, CH₃, F, F, 4-OH-Ph, Cl), (M-11133, CH₃, F, F, 4-OH-Ph, F), (M-11134, CH₃, F, F, 4-OH-Ph, CF₃), (M-11135, CH₃, F, F, 4-OH-Ph, Br), (M-11136, CH₃, F, F, 4-OH-Ph, CH₃), (M-11137, CH₃, F, F, 3,4-di-F-Ph, H), (M-11138, CH₃, F, F, 3,4-di-F-Ph, Cl), (M-11139, CH₃, F, F, 3,4-di-F-Ph, F), (M-11140, CH₃, F, F, 3,4-di-F-Ph, CF₃), (M-11141, CH₃, F, F, 3,4-di-F-Ph, Br), (M-11142, CH₃, F, F, 3,4-di-F-Ph, CH₃), (M-11143, CH₃, F, F, 4-COOH-Ph, H), (M-11144, CH₃, F, F, 4-COOH-Ph, Cl), (M-11145, CH₃, F, F, 4-COOH-Ph, F), (M-11146, CH₃, F, F, 4-COOH-Ph, CF₃), (M-11147, CH₃, F, F, 4-COOH-Ph, Br), (M-11148, CH₃, F, F, 4-COOH-Ph, CH₃), (M-11149, CH₃, F, F, Bn, H), (M-11150, CH₃, F, F, Bn, Cl), (M-11151, CH₃, F, F, Bn, F), (M-11152, CH₃, F, F, Bn, CF₃), (M-11153, CH₃, F, F, Bn, Br), (M-11154, CH₃, F, F, Bn, CH₃), (M-11155, CH₃, F, F, 4-F-Bn, H), (M-11156, CH₃, F, F, 4-F-Bn, Cl), (M-11157, CH₃, F, F, 4-F-Bn, F), (M-11158, CH₃, F, F, 4-F-Bn, CF₃), (M-11159, CH₃, F, F, 4-F-Bn, Br), (M-11160, CH₃, F, F, 4-F-Bn, CH₃), (M-11161, CH₃, F, F, 2-Py, H), (M-11162, CH₃, F, F, 2-Py, Cl), (M-11163, CH₃, F, F, 2-Py, F), (M-11164, CH₃, F, F, 2-Py, CF₃), (M-11165, CH₃, F, F, 2-Py, Br), (M-11166, CH₃, F, F, 2-Py, CH₃), (M-11167, CH₃, F, F, 3-Py, H), (M-11168, CH₃, F, F, 3-Py, Cl), (M-11169, CH₃, F, F, 3-Py, F), (M-11170, CH₃, F, F, 3-Py, CF₃), (M-11171, CH₃, F, F, 3-Py, Br), (M-11172, CH₃, F, F, 3-Py, CH₃), (M-11173, CH₃, F, F, 4-Py, H), (M-11174, CH₃, F, F, 4-Py, Cl), (M-11175, CH₃, F, F, 4-Py, F), (M-11176, CH₃, F, F, 4-Py, CF₃), (M-11177, CH₃, F, F, 4-Py, Br), (M-11178, CH₃, F, F, 4-Py, CH₃), (M-11179, CH₃, F, F, 2-Th, H), (M-11180, CH₃, F, F, 2-Th, Cl), (M-11181, CH₃, F, F, 2-Th, F), (M-11182, CH₃, F, F, 2-Th, CF₃), (M-11183, CH₃, F, F, 2-Th, Br), (M-11184, CH₃, F, F, 2-Th, CH₃), (M-11185, CH₃, F, F, 3-Th, H), (M-11186, CH₃, F, F, 3-Th, Cl), (M-11187, CH₃, F, F, 3-Th, F), (M-11188, CH₃, F, F, 3-Th, CF₃), (M-11189, CH₃, F, F, 3-Th, Br), (M-11190, CH₃, F, F, 3-Th, CH₃), (M-11191, CH₃, F, F, pyrazol-2-yl, H), (M-11192, CH₃, F, F, pyrazol-2-yl, Cl), (M-11193, CH₃, F, F, pyrazol-2-yl, F), (M-11194, CH₃, F, F, pyrazol-2-yl, CF₃), (M-11195, CH₃, F, F, pyrazol-2-yl, Br), (M-11196, CH₃, F, F, pyrazol-2-yl, CH₃), (M-11197, CH₃, F, F, pyrazol-3-yl, H), (M-11198, CH₃, F, F, pyrazol-3-yl, Cl), (M-11199, CH₃, F, F, pyrazol-3-yl, F), (M-11200, CH₃, F, F, pyrazol-3-yl, CF₃), (M-11201, CH₃, F, F, pyrazol-3-yl, Br), (M-11202, CH₃, F, F, pyrazol-3-yl, CH₃), (M-11203, CH₃, F, F, pyrimidin-2-yl, H), (M-11204, CH₃, F, F, pyrimidin-2-yl, Cl), (M-11205, CH₃, F, F, pyrimidin-2-yl, F), (M-11206, CH₃, F, F, pyrimidin-2-yl, CF₃), (M-11207, CH₃, F, F, pyrimidin-2-yl, Br), (M-11208, CH₃, F, F, pyrimidin-2-yl, CH₃), (M-11209, CH₃, F, F, pyrimidin-4-yl, H), (M-11210, CH₃, F, F, pyrimidin-4-yl, Cl), (M-11211, CH₃, F, F, pyrimidin-4-yl, F), (M-11212, CH₃, F, F, pyrimidin-4-yl, CF₃), (M-11213, CH₃, F, F, pyrimidin-4-yl, Br), (M-11214, CH₃, F, F, pyrimidin-4-yl, CH₃), (M-11215, CH₃, F, F, pyrimidin-5-yl, H), (M-11216, CH₃, F, F, pyrimidin-5-yl, Cl), (M-11217, CH₃, F, F, pyrimidin-5-yl, F), (M-11218, CH₃, F, F, pyrimidin-5-yl, CF₃), (M-11219, CH₃, F, F, pyrimidin-5-yl, Br), (M-11220, CH₃, F, F, pyrimidin-5-yl, CH₃), (M-11221, CH₃, F, F, HOOCCH₂CH₂CH₂, H), (M-11222, CH₃, F, F, HOOCCH₂CH₂CH₂, Cl), (M-11223, CH₃, F, F, HOOCCH₂CH₂CH₂, F), (M-11224, CH₃, F, F, HOOCCH₂CH₂CH₂, CF₃), (M-11225, CH₃, F, F, HOOCCH₂CH₂CH₂, Br), (M-11226, CH₃, F, F, HOOCCH₂CH₂CH₂, CH₃), (M-11227, CH₃, F, F, HOOCCH₂CH₂CH₂CH₂, H), (M-11228, CH₃, F, F, HOOCCH₂CH₂CH₂CH₂, Cl), (M-11229, CH₃, F, F, HOOCCH₂CH₂CH₂CH₂, F), (M-11230, CH₃, F, F, HOOCCH₂CH₂CH₂CH₂, CF₃), (M-11231, CH₃, F, F, HOOCCH₂CH₂CH₂CH₂, Br), (M-11232, CH₃, F, F, HOOCCH₂CH₂CH₂CH₂, CH₃), (M-11233, CH₃, F, F, (Me)₂NCOCH₂CH₂CH₂CH₂, H), (M-11234, CH₃, F, F, (Me)₂NCOCH₂CH₂CH₂CH₂, Cl), (M-11235, CH₃, F, F, (Me)₂NCOCH₂CH₂CH₂CH₂, F), (M-11236, CH₃, F, F, (Me)₂NCOCH₂CH₂CH₂CH₂, CF₃), (M-11237, CH₃, F, F, (Me)₂NCOCH₂CH₂CH₂CH₂, Br), (M-11238, CH₃, F, F, (Me)₂NCOCH₂CH₂CH₂CH₂, CH₃), (M-11239, CH₃, F, F, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, H), (M-11240, CH₃, F, F, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, Cl), (M-11241, CH₃, F, F, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, F), (M-11242, CH₃, F, F, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, CF₃), (M-11243, CH₃, F, F, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, Br), (M-11244, CH₃, F, F, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, CH₃), (M-11245, CH₃, F, F, MeOCH₂, H), (M-11246, CH₃, F, F, MeOCH₂, Cl), (M-11247, CH₃, F, F, MeOCH₂, F), (M-11248, CH₃, F, F, MeOCH₂, CF₃), (M-11249, CH₃, F, F, MeOCH₂, Br), (M-11250, CH₃, F, F, MeOCH₂, CH₃), (M-11251, CH₃, F, F, EtOCH₂, H), (M-11252, CH₃, F, F, EtOCH₂, Cl), (M-11253, CH₃, F, F, EtOCH₂, F), (M-11254, CH₃, F, F, EtOCH₂, CF₃), (M-11255, CH₃, F, F, EtOCH₂, Br), (M-11256, CH₃, F, F, EtOCH₂, CH₃), (M-11257, CH₃, F, F, EtOCH₂CH₂, H), (M-11258, CH₃, F, F, EtOCH₂CH₂, Cl), (M-11259, CH₃, F, F, EtOCH₂CH₂, F), (M-11260, CH₃, F, F, EtOCH₂CH₂, CF₃), (M-11261, CH₃, F, F, EtOCH₂CH₂, Br), (M-11262, CH₃, F, F, EtOCH₂CH₂, CH₃), (M-11263, CH₃, F, F, MeOCH₂CH₂OCH₂CH₂, H), (M-11264, CH₃, F, F, MeOCH₂CH₂OCH₂CH₂, Cl), (M-11265, CH₃, F, F, MeOCH₂CH₂
OCH₂CH₂, F), (M-11266, CH₃, F, F, MeOCH₂CH₂OCH₂CH₂, CF₃), (M-11267, CH₃, F, F, MeOCH₂CH₂OCH₂CH₂, Br), (M-11268, CH₃, F, F, MeOCH₂CH₂OCH₂CH₂, CH₃), (M-11269, CH₃, F, F, MeOCH₂CH₂, H), (M-11270, CH₃, F, F, MeOCH₂CH₂, Cl), (M-11271, CH₃, F, F, MeOCH₂CH₂, F), (M-11272, CH₃, F, F, MeOCH₂CH₂, CF₃), (M-11273, CH₃, F, F, MeOCH₂CH₂, Br), (M-11274, CH₃, F, F, MeOCH₂CH₂, CH₃), (M-11275, CH₃, F, F, HOCH₂, H), (M-11276, CH₃, F, F, HOCH₂, Cl), (M-11277, CH₃, F, F, HOCH₂, F), (M-11278, CH₃, F, F, HOCH₂, CF₃), (M-11279, CH₃, F, F, HOCH₂, Br), (M-11280, CH₃, F, F, HOCH₂, CH₃), (M-11281, CH₃, F, F, HOCH₂CH₂, H), (M-11282, CH₃, F, F, HOCH₂CH₂, Cl), (M-11283, CH₃, F, F, HOCH₂CH₂, F), (M-11284, CH₃, F, F, HOCH₂CH₂, CF₃), (M-11285, CH₃, F, F, HOCH₂CH₂, Br), (M-11286, CH₃, F, F, HOCH₂CH₂, CH₃), (M-11287, CH₃, F, F, HOCH₂CH₂CH₂, H), (M-11288, CH₃, F, F, HOCH₂CH₂CH₂, Cl), (M-11289, CH₃, F, F, HOCH₂CH₂CH₂, F), (M-11290, CH₃, F, F, HOCH₂CH₂CH₂, CF₃), (M-11291, CH₃, F, F, HOCH₂CH₂CH₂, Br), (M-11292, CH₃, F, F, HOCH₂CH₂CH₂, CH₃), (M-11293, CH₃, F, F, HOCH₂CH₂CH₂CH₂, H), (M-11294, CH₃, F, F, HOCH₂CH₂CH₂CH₂, Cl), (M-11295, CH₃, F, F, HOCH₂CH₂CH₂CH₂, F), (M-11296, CH₃, F, F, HOCH₂CH₂CH₂CH₂, CF₃), (M-11297, CH₃, F, F, HOCH₂CH₂CH₂CH₂, Br), (M-11298, CH₃, F, F, HOCH₂CH₂CH₂CH₂, CH₃), (M-11299, CH₃, F, F, HOCH₂CH₂CH₂CH₂CH₂, H), (M-11300, CH₃, F, F, HOCH₂CH₂CH₂CH₂CH₂, Cl), (M-11301, CH₃, F, F, HOCH₂CH₂CH₂CH₂CH₂, F), (M-11302, CH₃, F, F, HOCH₂CH₂CH₂CH₂CH₂, CF₃), (M-11303, CH₃, F, F, HOCH₂CH₂CH₂CH₂CH₂, Br), (M-11304, CH₃, F, F, HOCH₂CH₂CH₂CH₂CH₂, CH₃), (M-11305, CH₃, F, F, HOCH₂CH₂OCH₂CH₂, H), (M-11306, CH₃, F, F, HOCH₂CH₂OCH₂CH₂, Cl), (M-11307, CH₃, F, F, HOCH₂CH₂OCH₂CH₂, F), (M-11308, CH₃, F, F, HOCH₂CH₂OCH₂CH₂, CF₃), (M-11309, CH₃, F, F, HOCH₂CH₂OCH₂CH₂, Br), (M-11310, CH₃, F, F, HOCH₂CH₂OCH₂CH₂, CH₃), (M-11311, CH₃, F, F, (Me)₂N, H), (M-11312, CH₃, F, F, (Me)₂N, Cl), (M-11313, CH₃, F, F, (Me)₂N, F), (M-11314, CH₃, F, F, (Me)₂N, CF₃), (M-11315, CH₃, F, F, (Me)₂N, Br), (M-11316, CH₃, F, F, (Me)₂N, CH₃), (M-11317, CH₃, F, F, piperidin-4-yl-methyl, H), (M-11318, CH₃, F, F, piperidin-4-yl-methyl, Cl), (M-11319, CH₃, F, F, piperidin-4-yl-methyl, F), (M-11320, CH₃, F, F, piperidin-4-yl-methyl, CF₃), (M-11321, CH₃, F, F, piperidin-4-yl-methyl, Br), (M-11322, CH₃, F, F, piperidin-4-yl-methyl, CH₃), (M-11323, CH₃, F, F, cyclohexylmethyl, H), (M-11324, CH₃, F, F, cyclohexylmethyl, Cl), (M-11325, CH₃, F, F, cyclohexylmethyl, F), (M-11326, CH₃, F, F, cyclohexylmethyl, CF₃), (M-11327, CH₃, F, F, cyclohexylmethyl, Br), (M-11328, CH₃, F, F, cyclohexylmethyl, CH₃), (M-11329, CH₃, F, Cl, H, H), (M-11330, CH₃, F, Cl, H, Cl), (M-11331, CH₃, F, Cl, H, F), (M-11332, CH₃, F, Cl, H, CF₃), (M-11333, CH₃, F, Cl, H, Br), (M-11334, CH₃, F, Cl, H, CH₃), (M-11335, CH₃, F, Cl, F, H), (M-11336, CH₃, F, Cl, F, Cl), (M-11337, CH₃, F, Cl, F, F), (M-11338, CH₃, F, Cl, F, CF₃), (M-11339, CH₃, F, Cl, F, Br), (M-11340, CH₃, F, Cl, F, CH₃), (M-11341, CH₃, F, Cl, Cl, H), (M-11342, CH₃, F, Cl, Cl, Cl), (M-11343, CH₃, F, Cl, Cl, F), (M-11344, CH₃, F, Cl, Cl, CF₃), (M-11345, CH₃, F, Cl, Cl, Br), (M-11346, CH₃, F, Cl, Cl, CH₃), (M-11347, CH₃, F, Cl, CH₃, H), (M-11348, CH₃, F, Cl, CH₃, Cl), (M-11349, CH₃, F, Cl, CH₃, F), (M-11350, CH₃, F, Cl, CH₃, CF₃), (M-11351, CH₃, F, Cl, CH₃, Br), (M-11352, CH₃, F, Cl, CH₃, CH₃), (M-11353, CH₃, F, Cl, Et, H), (M-11354, CH₃, F, Cl, Et, Cl), (M-11355, CH₃, F, Cl, Et, F), (M-11356, CH₃, F, Cl, Et, CF₃), (M-11357, CH₃, F, Cl, Et, Br), (M-11358, CH₃, F, Cl, Et, CH₃), (M-11359, CH₃, F, Cl, n-Pr, H), (M-11360, CH₃, F, Cl, n-Pr, Cl), (M-11361, CH₃, F, Cl, n-Pr, F), (M-11362, CH₃, F, Cl, n-Pr, CF₃), (M-11363, CH₃, F, Cl, n-Pr, Br), (M-11364, CH₃, F, Cl, n-Pr, CH₃), (M-11365, CH₃, F, Cl, c-Pr, H), (M-11366, CH₃, F, Cl, c-Pr, Cl), (M-11367, CH₃, F, Cl, c-Pr, F), (M-11368, CH₃, F, Cl, c-Pr, CF₃), (M-11369, CH₃, F, Cl, c-Pr, Br), (M-11370, CH₃, F, Cl, c-Pr, CH₃), (M-11371, CH₃, F, Cl, i-Pr, H), (M-11372, CH₃, F, Cl, i-Pr, Cl), (M-11373, CH₃, F, Cl, i-Pr, F), (M-11374, CH₃, F, Cl, i-Pr, CF₃), (M-11375, CH₃, F, Cl, i-Pr, Br), (M-11376, CH₃, F, Cl, i-Pr, CH₃), (M-11377, CH₃, F, Cl, n-Bu, H), (M-11378, CH₃, F, Cl, n-Bu, Cl), (M-11379, CH₃, F, Cl, n-Bu, F), (M-11380, CH₃, F, Cl, n-Bu, CF₃), (M-11381, CH₃, F, Cl, n-Bu, Br), (M-11382, CH₃, F, Cl, n-Bu, CH₃), (M-11383, CH₃, F, Cl, i-Bu, H), (M-11384, CH₃, F, Cl, i-Bu, Cl), (M-11385, CH₃, F, Cl, i-Bu, F), (M-11386, CH₃, F, Cl, i-Bu, CF₃), (M-11387, CH₃, F, Cl, i-Bu, Br), (M-11388, CH₃, F, Cl, i-Bu, CH₃), (M-11389, CH₃, F, Cl, sec-Bu, H), (M-11390, CH₃, F, Cl, sec-Bu, Cl), (M-11391, CH₃, F, Cl, sec-Bu, F), (M-11392, CH₃, F, Cl, sec-Bu, CF₃), (M-11393, CH₃, F, Cl, sec-Bu, Br), (M-11394, CH₃, F, Cl, sec-Bu, CH₃), (M-11395, CH₃, F, Cl, n-Pen, H), (M-11396, CH₃, F, Cl, n-Pen, Cl), (M-11397, CH₃, F, Cl, n-Pen, F), (M-11398, CH₃, F, Cl, n-Pen, CF₃), (M-11399, CH₃, F, Cl, n-Pen, Br), (M-11400, CH₃, F, Cl, n-Pen, CH₃), (M-11401, CH₃, F, Cl, c-Pen, H), (M-11402, CH₃, F, Cl, c-Pen, Cl), (M-11403, CH₃, F, Cl, c-Pen, F), (M-11404, CH₃, F, Cl, c-Pen, CF₃), (M-11405, CH₃, F, Cl, c-Pen, Br), (M-11406, CH₃, F, Cl, c-Pen, CH₃), (M-11407, CH₃, F, Cl, n-Hex, H), (M-11408, CH₃, F, Cl, n-Hex, Cl), (M-11409, CH₃, F, Cl, n-Hex, F), (M-11410, CH₃, F, Cl, n-Hex, CF₃), (M-11411, CH₃, F, Cl, n-Hex, Br), (M-11412, CH₃, F, Cl, n-Hex, CH₃), (M-11413, CH₃, F, Cl, c-Hex, H), (M-11414, CH₃, F, Cl, c-Hex, Cl), (M-11415, CH₃, F, Cl, c-Hex, F), (M-11416, CH₃, F, Cl, c-Hex, CF₃), (M-11417, CH₃, F, Cl, c-Hex, Br), (M-11418, CH₃, F, Cl, c-Hex, CH₃), (M-11419, CH₃, F, Cl, OH, H), (M-11420, CH₃, F, Cl, OH, Cl), (M-11421, CH₃, F, Cl, OH, F), (M-11422, CH₃, F, Cl, OH, CF₃), (M-11423, CH₃, F, Cl, OH, Br), (M-11424, CH₃, F, Cl, OH, CH₃), (M-11425, CH₃, F, Cl, EtO, H), (M-11426, CH₃, F, Cl, EtO, Cl), (M-11427, CH₃, F, Cl, EtO, F), (M-11428, CH₃, F, Cl, EtO, CF₃), (M-11429, CH₃, F, Cl, EtO, Br), (M-11430, CH₃, F, Cl, EtO, CH₃), (M-11431, CH₃, F, Cl, n-PrO, H), (M-11432, CH₃, F, Cl, n-PrO, Cl), (M-11433, CH₃, F, Cl, n-PrO, F), (M-11434, CH₃, F, Cl, n-PrO, CF₃), (M-11435, CH₃, F, Cl, n-PrO, Br), (M-11436, CH₃,
F, Cl, n-PrO, CH₃), (M-11437, CH₃, F, Cl, PhO, H), (M-11438, CH₃, F, Cl, PhO, Cl), (M-11439, CH₃, F, Cl, PhO, F), (M-11440, CH₃, F, Cl, PhO, CF₃), (M-11441, CH₃, F, Cl, PhO, Br), (M-11442, CH₃, F, Cl, PhO, CH₃), (M-11443, CH₃, F, Cl, BnO, H), (M-11444, CH₃, F, Cl, BnO, Cl), (M-11445, CH₃, F, Cl, BnO, F), (M-11446, CH₃, F, Cl, BnO, CF₃), (M-11447, CH₃, F, Cl, BnO, Br), (M-11448, CH₃, F, Cl, BnO, CH₃), (M-11449, CH₃, F, Cl, PhCH₂CH₂O, H), (M-11450, CH₃, F, Cl, PhCH₂CH₂O, Cl), (M-11451, CH₃, F, Cl, PhCH₂CH₂O, F), (M-11452, CH₃, F, Cl, PhCH₂CH₂O, CF₃), (M-11453, CH₃, F, Cl, PhCH₂CH₂O, Br), (M-11454, CH₃, F, Cl, PhCH₂CH₂O, CH₃), (M-11455, CH₃, F, Cl, CF₃O, H), (M-11456, CH₃, F, Cl, CF₃O, Cl), (M-11457, CH₃, F, Cl, CF₃O, F), (M-11458, CH₃, F, Cl, CF₃O, CF₃), (M-11459, CH₃, F, Cl, CF₃O, Br), (M-11460, CH₃, F, Cl, CF₃O, CH₃), (M-11461, CH₃, F, Cl, Ph, H), (M-11462, CH₃, F, Cl, Ph, Cl), (M-11463, CH₃, F, Cl, Ph, F), (M-11464, CH₃, F, Cl, Ph, CF₃), (M-11465, CH₃, F, Cl, Ph, Br), (M-11466, CH₃, F, Cl, Ph, CH₃), (M-11467, CH₃, F, Cl, 4-F-Ph, H), (M-11468, CH₃, F, Cl, 4-F-Ph, Cl), (M-11469, CH₃, F, Cl, 4-F-Ph, F), (M-11470, CH₃, F, Cl, 4-F-Ph, CF₃), (M-11471, CH₃, F, Cl, 4-F-Ph, Br), (M-11472, CH₃, F, Cl, 4-F-Ph, CH₃), (M-11473, CH₃, F, Cl, 4-CF₃-Ph, H), (M-11474, CH₃, F, Cl, 4-CF₃-Ph, Cl), (M-11475, CH₃, F, Cl, 4-CF₃-Ph, F), (M-11476, CH₃, F, Cl, 4-CF₃-Ph, CF₃), (M-11477, CH₃, F, Cl, 4-CF₃-Ph, Br), (M-11478, CH₃, F, Cl, 4-CF₃-Ph, CH₃), (M-11479, CH₃, F, Cl, 4-(Me)₂N-Ph, H), (M-11480, CH₃, F, Cl, 4-(Me)₂N-Ph, Cl), (M-11481, CH₃, F, Cl, 4-(Me)₂N-Ph, F), (M-11482, CH₃, F, Cl, 4-(Me)₂N-Ph, CF₃), (M-11483, CH₃, F, Cl, 4-(Me)₂N-Ph, Br), (M-11484, CH₃, F, Cl, 4-(Me)₂N-Ph, CH₃), (M-11485, CH₃, F, Cl, 4-OH-Ph, H), (M-11486, CH₃, F, Cl, 4-OH-Ph, Cl), (M-11487, CH₃, F, Cl, 4-OH-Ph, F), (M-11488, CH₃, F, Cl, 4-OH-Ph, CF₃), (M-11489, CH₃, F, Cl, 4-OH-Ph, Br), (M-11490, CH₃, F, Cl, 4-OH-Ph, CH₃), (M-11491, CH₃, F, Cl, 3,4-di-F-Ph, H), (M-11492, CH₃, F, Cl, 3,4-di-F-Ph, Cl), (M-11493, CH₃, F, Cl, 3,4-di-F-Ph, F), (M-11494, CH₃, F, Cl, 3,4-di-F-Ph, CF₃), (M-11495, CH₃, F, Cl, 3,4-di-F-Ph, Br), (M-11496, CH₃, F, Cl, 3,4-di-F-Ph, CH₃), (M-11497, CH₃, F, Cl, 4-COOH-Ph, H), (M-11498, CH₃, F, Cl, 4-COOH-Ph, Cl), (M-11499, CH₃, F, Cl, 4-COOH-Ph, F), (M-11500, CH₃, F, Cl, 4-COOH-Ph, CF₃), (M-11501, CH₃, F, Cl, 4-COOH-Ph, Br), (M-11502, CH₃, F, Cl, 4-COOH-Ph, CH₃), (M-11503, CH₃, F, Cl, Bn, H), (M-11504, CH₃, F, Cl, Bn, Cl), (M-11505, CH₃, F, Cl, Bn, F), (M-11506, CH₃, F, Cl, Bn, CF₃), (M-11507, CH₃, F, Cl, Bn, Br), (M-11508, CH₃, F, Cl, Bn, CH₃), (M-11509, CH₃, F, Cl, 4-F-Bn, H), (M-11510, CH₃, F, Cl, 4-F-Bn, Cl), (M-11511, CH₃, F, Cl, 4-F-Bn, F), (M-11512, CH₃, F, Cl, 4-F-Bn, CF₃), (M-11513, CH₃, F, Cl, 4-F-Bn, Br), (M-11514, CH₃, F, Cl, 4-F-Bn, CH₃), (M-11515, CH₃, F, Cl, 2-Py, H), (M-11516, CH₃, F, Cl, 2-Py, Cl), (M-11517, CH₃, F, Cl, 2-Py, F), (M-11518, CH₃, F, Cl, 2-Py, CF₃), (M-11519, CH₃, F, Cl, 2-Py, Br), (M-11520, CH₃, F, Cl, 2-Py, CH₃), (M-11521, CH₃, F, Cl, 3-Py, H), (M-11522, CH₃, F, Cl, 3-Py, Cl), (M-11523, CH₃, F, Cl, 3-Py, F), (M-11524, CH₃, F, Cl, 3-Py, CF₃), (M-11525, CH₃, F, Cl, 3-Py, Br), (M-11526, CH₃, F, Cl, 3-Py, CH₃), (M-11527, CH₃, F, Cl, 4-Py, H), (M-11528, CH₃, F, Cl, 4-Py, Cl), (M-11529, CH₃, F, Cl, 4-Py, F), (M-11530, CH₃, F, Cl, 4-Py, CF₃), (M-11531, CH₃, F, Cl, 4-Py, Br), (M-11532, CH₃, F, Cl, 4-Py, CH₃), (M-11533, CH₃, F, Cl, 2-Th, H), (M-11534, CH₃, F, Cl, 2-Th, Cl), (M-11535, CH₃, F, Cl, 2-Th, F), (M-11536, CH₃, F, Cl, 2-Th, CF₃), (M-11537, CH₃, F, Cl, 2-Th, Br), (M-11538, CH₃, F, Cl, 2-Th, CH₃), (M-11539, CH₃, F, Cl, 3-Th, H), (M-11540, CH₃, F, Cl, 3-Th, Cl), (M-11541, CH₃, F, Cl, 3-Th, F), (M-11542, CH₃, F, Cl, 3-Th, CF₃), (M-11543, CH₃, F, Cl, 3-Th, Br), (M-11544, CH₃, F, Cl, 3-Th, CH₃), (M-11545, CH₃, F, Cl, pyrazol-2-yl, H), (M-11546, CH₃, F, Cl, pyrazol-2-yl, Cl), (M-11547, CH₃, F, Cl, pyrazol-2-yl, F), (M-11548, CH₃, F, Cl, pyrazol-2-yl, CF₃), (M-11549, CH₃, F, Cl, pyrazol-2-yl, Br), (M-11550, CH₃, F, Cl, pyrazol-2-yl, CH₃), (M-11551, CH₃, F, Cl, pyrazol-3-yl, H), (M-11552, CH₃, F, Cl, pyrazol-3-yl, Cl), (M-11553, CH₃, F, Cl, pyrazol-3-yl, F), (M-11554, CH₃, F, Cl, pyrazol-3-yl, CF₃), (M-11555, CH₃, F, Cl, pyrazol-3-yl, Br), (M-11556, CH₃, F, Cl, pyrazol-3-yl, CH₃), (M-11557, CH₃, F, Cl, pyrimidin-2-yl, H), (M-11558, CH₃, F, Cl, pyrimidin-2-yl, Cl), (M-11559, CH₃, F, Cl, pyrimidin-2-yl, F), (M-11560, CH₃, F, Cl, pyrimidin-2-yl, CF₃), (M-11561, CH₃, F, Cl, pyrimidin-2-yl, Br), (M-11562, CH₃, F, Cl, pyrimidin-2-yl, CH₃), (M-11563, CH₃, F, Cl, pyrimidin-4-yl, H), (M-11564, CH₃, F, Cl, pyrimidin-4-yl, Cl), (M-11565, CH₃, F, Cl, pyrimidin-4-yl, F), (M-11566, CH₃, F, Cl, pyrimidin-4-yl, CF₃), (M-11567, CH₃, F, Cl, pyrimidin-4-yl, Br), (M-11568, CH₃, F, Cl, pyrimidin-4-yl, CH₃), (M-11569, CH₃, F, Cl, pyrimidin-5-yl, H), (M-11570, CH₃, F, Cl, pyrimidin-5-yl, Cl), (M-11571, CH₃, F, Cl, pyrimidin-5-yl, F), (M-11572, CH₃, F, Cl, pyrimidin-5-yl, CF₃), (M-11573, CH₃, F, Cl, pyrimidin-5-yl, Br), (M-11574, CH₃, F, Cl, pyrimidin-5-yl, CH₃), (M-11575, CH₃, F, Cl, HOOCCH₂CH₂CH₂, H), (M-11576, CH₃, F, Cl, HOOCCH₂CH₂CH₂, Cl), (M-11577, CH₃, F, Cl, HOOCCH₂CH₂CH₂, F), (M-11578, CH₃, F, Cl, HOOCCH₂CH₂CH₂, CF₃), (M-11579, CH₃, F, Cl, HOOCCH₂CH₂CH₂, Br), (M-11580, CH₃, F, Cl, HOOCCH₂CH₂CH₂, CH₃), (M-11581, CH₃, F, Cl, HOOCCH₂CH₂CH₂CH₂, H), (M-11582, CH₃, F, Cl, HOOCCH₂CH₂CH₂CH₂, Cl), (M-11583, CH₃, F, Cl, HOOCCH₂CH₂CH₂CH₂, F), (M-11584, CH₃, F, Cl, HOOCCH₂CH₂CH₂CH₂, CF₃), (M-11585, CH₃, F, Cl, HOOCCH₂CH₂CH₂CH₂, Br), (M-11586, CH₃, F, Cl, HOOCCH₂CH₂CH₂CH₂, CH₃), (M-11587, CH₃, F, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂, H), (M-11588, CH₃, F, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂, Cl), (M-11589, CH₃, F, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂, F), (M-11590, CH₃, F, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂, CF₃), (M-11591, CH₃, F, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂, Br), (M-11592, CH₃, F, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂, CH₃), (M-11593, CH₃, F, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, H), (M-11594, CH₃, F, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, Cl), (M-11595, CH₃, F, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, F), (M-11596, CH₃, F, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, CF₃), (M-11597, CH₃, F, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, Br), (M-11598, CH₃, F, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, CH₃), (M-11599, CH₃, F, Cl, MeOCH₂, H), (M-11600, CH₃, F, Cl, MeOCH₂, Cl), (M-11601, CH₃, F, Cl, MeOCH₂, F), (M-11602, CH
₃, F, Cl, MeOCH₂, CF₃), (M-11603, CH₃, F, Cl, MeOCH₂, Br), (M-11604, CH₃, F, Cl, MeOCH₂, CH₃), (M-11605, CH₃, F, Cl, EtOCH₂, H), (M-11606, CH₃, F, Cl, EtOCH₂, Cl), (M-11607, CH₃, F, Cl, EtOCH₂, F), (M-11608, CH₃, F, Cl, EtOCH₂, CF₃), (M-11609, CH₃, F, Cl, EtOCH₂, Br), (M-11610, CH₃, F, Cl, EtOCH₂, CH₃), (M-11611, CH₃, F, Cl, EtOCH₂CH₂, H), (M-11612, CH₃, F, Cl, EtOCH₂CH₂, Cl), (M-11613, CH₃, F, Cl, EtOCH₂CH₂, F), (M-11614, CH₃, F, Cl, EtOCH₂CH₂, CF₃), (M-11615, CH₃, F, Cl, EtOCH₂CH₂, Br), (M-11616, CH₃, F, Cl, EtOCH₂CH₂, CH₃), (M-11617, CH₃, F, Cl, MeOCH₂CH₂OCH₂CH₂, H), (M-11618, CH₃, F, Cl, MeOCH₂CH₂OCH₂CH₂, Cl), (M-11619, CH₃, F, Cl, MeOCH₂CH₂OCH₂CH₂, F), (M-11620, CH₃, F, Cl, MeOCH₂CH₂OCH₂CH₂, CF₃), (M-11621, CH₃, F, Cl, MeOCH₂CH₂OCH₂CH₂, Br), (M-11622, CH₃, F, Cl, MeOCH₂CH₂OCH₂CH₂, CH₃), (M-11623, CH₃, F, Cl, MeOCH₂CH₂, H), (M-11624, CH₃, F, Cl, MeOCH₂CH₂, Cl), (M-11625, CH₃, F, Cl, MeOCH₂CH₂, F), (M-11626, CH₃, F, Cl, MeOCH₂CH₂, CF₃), (M-11627, CH₃, F, Cl, MeOCH₂CH₂, Br), (M-11628, CH₃, F, Cl, MeOCH₂CH₂, CH₃), (M-11629, CH₃, F, Cl, HOCH₂, H), (M-11630, CH₃, F, Cl, HOCH₂, Cl), (M-11631, CH₃, F, Cl, HOCH₂, F), (M-11632, CH₃, F, Cl, HOCH₂, CF₃), (M-11633, CH₃, F, Cl, HOCH₂, Br), (M-11634, CH₃, F, Cl, HOCH₂, CH₃), (M-11635, CH₃, F, Cl, HOCH₂CH₂, H), (M-11636, CH₃, F, Cl, HOCH₂CH₂, Cl), (M-11637, CH₃, F, Cl, HOCH₂CH₂, F), (M-11638, CH₃, F, Cl, HOCH₂CH₂, CF₃), (M-11639, CH₃, F, Cl, HOCH₂CH₂, Br), (M-11640, CH₃, F, Cl, HOCH₂CH₂, CH₃), (M-11641, CH₃, F, Cl, HOCH₂CH₂CH₂, H), (M-11642, CH₃, F, Cl, HOCH₂CH₂CH₂, Cl), (M-11643, CH₃, F, Cl, HOCH₂CH₂CH₂, F), (M-11644, CH₃, F, Cl, HOCH₂CH₂CH₂, CF₃), (M-11645, CH₃, F, Cl, HOCH₂CH₂CH₂, Br), (M-11646, CH₃, F, Cl, HOCH₂CH₂CH₂, CH₃), (M-11647, CH₃, F, Cl, HOCH₂CH₂CH₂CH₂, H), (M-11648, CH₃, F, Cl, HOCH₂CH₂CH₂CH₂, Cl), (M-11649, CH₃, F, Cl, HOCH₂CH₂CH₂CH₂, F), (M-11650, CH₃, F, Cl, HOCH₂CH₂CH₂CH₂, CF₃), (M-11651, CH₃, F, Cl, HOCH₂CH₂CH₂CH₂, Br), (M-11652, CH₃, F, Cl, HOCH₂CH₂CH₂CH₂, CH₃), (M-11653, CH₃, F, Cl, HOCH₂CH₂CH₂CH₂CH₂, H), (M-11654, CH₃, F, Cl, HOCH₂CH₂CH₂CH₂CH₂, Cl), (M-11655, CH₃, F, Cl, HOCH₂CH₂CH₂CH₂CH₂, F), (M-11656, CH₃, F, Cl, HOCH₂CH₂CH₂CH₂CH₂, CF₃), (M-11657, CH₃, F, Cl, HOCH₂CH₂CH₂CH₂CH₂, Br), (M-11658, CH₃, F, Cl, HOCH₂CH₂CH₂CH₂CH₂, CH₃), (M-11659, CH₃, F, Cl, HOCH₂CH₂OCH₂CH₂, H), (M-11660, CH₃, F, Cl, HOCH₂CH₂OCH₂CH₂, Cl), (M-11661, CH₃, F, Cl, HOCH₂CH₂OCH₂CH₂, F), (M-11662, CH₃, F, Cl, HOCH₂CH₂OCH₂CH₂, CF₃), (M-11663, CH₃, F, Cl, HOCH₂CH₂OCH₂CH₂, Br), (M-11664, CH₃, F, Cl, HOCH₂CH₂OCH₂CH₂, CH₃), (M-11665, CH₃, F, Cl, (Me)₂N, H), (M-11666, CH₃, F, Cl, (Me)₂N, Cl), (M-11667, CH₃, F, Cl, (Me)₂N, F), (M-11668, CH₃, F, Cl, (Me)₂N, CF₃), (M-11669, CH₃, F, Cl, (Me)₂N, Br), (M-11670, CH₃, F, Cl, (Me)₂N, CH₃), (M-11671, CH₃, F, Cl, piperidin-4-yl-methyl, H), (M-11672, CH₃, F, Cl, piperidin-4-yl-methyl, Cl), (M-11673, CH₃, F, Cl, piperidin-4-yl-methyl, F), (M-11674, CH₃, F, Cl, piperidin-4-yl-methyl, CF₃), (M-11675, CH₃, F, Cl, piperidin-4-yl-methyl, Br), (M-11676, CH₃, F, Cl, piperidin-4-yl-methyl, CH₃), (M-11677, CH₃, F, Cl, cyclohexylmethyl, H), (M-11678, CH₃, F, Cl, cyclohexylmethyl, Cl), (M-11679, CH₃, F, Cl, cyclohexylmethyl, F), (M-11680, CH₃, F, Cl, cyclohexylmethyl, CF₃), (M-11681, CH₃, F, Cl, cyclohexylmethyl, Br), (M-11682, CH₃, F, Cl, cyclohexylmethyl, CH₃), (M-11683, CH₃, CH₃, H, H, H), (M-11684, CH₃, CH₃, H, H, Cl), (M-11685, CH₃, CH₃, H, H, F), (M-11686, CH₃, CH₃, H, H, CF₃), (M-11687, CH₃, CH₃, H, H, Br), (M-11688, CH₃, CH₃, H, H, CH₃), (M-11689, CH₃, CH₃, H, F, H), (M-11690, CH₃, CH₃, H, F, Cl), (M-11691, CH₃, CH₃, H, F, F), (M-11692, CH₃, CH₃, H, F, CF₃), (M-11693, CH₃, CH₃, H, F, Br), (M-11694, CH₃, CH₃, H, F, CH₃), (M-11695, CH₃, CH₃, H, Cl, H), (M-11696, CH₃, CH₃, H, Cl, Cl), (M-11697, CH₃, CH₃, H, Cl, F), (M-11698, CH₃, CH₃, H, Cl, CF₃), (M-11699, CH₃, CH₃, H, Cl, Br), (M-11700, CH₃, CH₃, H, Cl, CH₃), (M-11701, CH₃, CH₃, H, CH₃, H), (M-11702, CH₃, CH₃, H, CH₃, Cl), (M-11703, CH₃, CH₃, H, CH₃, F), (M-11704, CH₃, CH₃, H, CH₃, CF₃), (M-11705, CH₃, CH₃, H, CH₃, Br), (M-11706, CH₃, CH₃, H, CH₃, CH₃), (M-11707, CH₃, CH₃, H, Et, H), (M-11708, CH₃, CH₃, H, Et, Cl), (M-11709, CH₃, CH₃, H, Et, F), (M-11710, CH₃, CH₃, H, Et, CF₃), (M-11711, CH₃, CH₃, H, Et, Br), (M-11712, CH₃, CH₃, H, Et, CH₃), (M-11713, CH₃, CH₃, H, n-Pr, H), (M-11714, CH₃, CH₃, H, n-Pr, Cl), (M-11715, CH₃, CH₃, H, n-Pr, F), (M-11716, CH₃, CH₃, H, n-Pr, CF₃), (M-11717, CH₃, CH₃, H, n-Pr, Br), (M-11718, CH₃, CH₃, H, n-Pr, CH₃), (M-11719, CH₃, CH₃, H, c-Pr, H), (M-11720, CH₃, CH₃, H, c-Pr, Cl), (M-11721, CH₃, CH₃, H, c-Pr, F), (M-11722, CH₃, CH₃, H, c-Pr, CF₃), (M-11723, CH₃, CH₃, H, c-Pr, Br), (M-11724, CH₃, CH₃, H, c-Pr, CH₃), (M-11725, CH₃, CH₃, H, i-Pr, H), (M-11726, CH₃, CH₃, H, i-Pr, Cl), (M-11727, CH₃, CH₃, H, i-Pr, F), (M-11728, CH₃, CH₃, H, i-Pr, CF₃), (M-11729, CH₃, CH₃, H, i-Pr, Br), (M-11730, CH₃, CH₃, H, i-Pr, CH₃), (M-11731, CH₃, CH₃, H, n-Bu, H), (M-11732, CH₃, CH₃, H, n-Bu, Cl), (M-11733, CH₃, CH₃, H, n-Bu, F), (M-11734, CH₃, CH₃, H, n-Bu, CF₃), (M-11735, CH₃, CH₃, H, n-Bu, Br), (M-11736, CH₃, CH₃, H, n-Bu, CH₃), (M-11737, CH₃, CH₃, H, i-Bu, H), (M-11738, CH₃, CH₃, H, i-Bu, Cl), (M-11739, CH₃, CH₃, H, i-Bu, F), (M-11740, CH₃, CH₃, H, i-Bu, CF₃), (M-11741, CH₃, CH₃, H, i-Bu, Br), (M-11742, CH₃, CH₃, H, i-Bu, CH₃), (M-11743, CH₃, CH₃, H, sec-Bu, H), (M-11744, CH₃, CH₃, H, sec-Bu, Cl), (M-11745, CH₃, CH₃, H, sec-Bu, F), (M-11746, CH₃, CH₃, H, sec-Bu, CF₃), (M-
11747, CH₃, CH₃, H, sec-Bu, Br), (M-11748, CH₃, CH₃, H, sec-Bu, CH₃), (M-11749, CH₃, CH₃, H, n-Pen, H), (M-11750, CH₃, CH₃, H, n-Pen, Cl), (M-11751, CH₃, CH₃, H, n-Pen, F), (M-11752, CH₃, CH₃, H, n-Pen, CF₃), (M-11753, CH₃, CH₃, H, n-Pen, Br), (M-11754, CH₃, CH₃, H, n-Pen, CH₃), (M-11755, CH₃, CH₃, H, c-Pen, H), (M-11756, CH₃, CH₃, H, c-Pen, Cl), (M-11757, CH₃, CH₃, H, c-Pen, F), (M-11758, CH₃, CH₃, H, c-Pen, CF₃), (M-11759, CH₃, CH₃, H, c-Pen, Br), (M-11760, CH₃, CH₃, H, c-Pen, CH₃), (M-11761, CH₃, CH₃, H, n-Hex, H), (M-11762, CH₃, CH₃, H, n-Hex, Cl), (M-11763, CH₃, CH₃, H, n-Hex, F), (M-11764, CH₃, CH₃, H, n-Hex, CF₃), (M-11765, CH₃, CH₃, H, n-Hex, Br), (M-11766, CH₃, CH₃, H, n-Hex, CH₃), (M-11767, CH₃, CH₃, H, c-Hex, H), (M-11768, CH₃, CH₃, H, c-Hex, Cl), (M-11769, CH₃, CH₃, H, c-Hex, F), (M-11770, CH₃, CH₃, H, c-Hex, CF₃), (M-11771, CH₃, CH₃, H, c-Hex, Br), (M-11772, CH₃, CH₃, H, c-Hex, CH₃), (M-11773, CH₃, CH₃, H, OH, H), (M-11774, CH₃, CH₃, H, OH, Cl), (M-11775, CH₃, CH₃, H, OH, F), (M-11776, CH₃, CH₃, H, OH, CF₃), (M-11777, CH₃, CH₃, H, OH, Br), (M-11778, CH₃, CH₃, H, OH, CH₃), (M-11779, CH₃, CH₃, H, EtO, H), (M-11780, CH₃, CH₃, H, EtO, Cl), (M-11781, CH₃, CH₃, H, EtO, F), (M-11782, CH₃, CH₃, H, EtO, CF₃), (M-11783, CH₃, CH₃, H, EtO, Br), (M-11784, CH₃, CH₃, H, EtO, CH₃), (M-11785, CH₃, CH₃, H, n-PrO, H), (M-11786, CH₃, CH₃, H, n-PrO, Cl), (M-11787, CH₃, CH₃, H, n-PrO, F), (M-11788, CH₃, CH₃, H, n-PrO, CF₃), (M-11789, CH₃, CH₃, H, n-PrO, Br), (M-11790, CH₃, CH₃, H, n-PrO, CH₃), (M-11791, CH₃, CH₃, H, PhO, H), (M-11792, CH₃, CH₃, H, PhO, Cl), (M-11793, CH₃, CH₃, H, PhO, F), (M-11794, CH₃, CH₃, H, PhO, CF₃), (M-11795, CH₃, CH₃, H, PhO, Br), (M-11796, CH₃, CH₃, H, PhO, CH₃), (M-11797, CH₃, CH₃, H, BnO, H), (M-11798, CH₃, CH₃, H, BnO, Cl), (M-11799, CH₃, CH₃, H, BnO, F), (M-11800, CH₃, CH₃, H, BnO, CF₃), (M-11801, CH₃, CH₃, H, BnO, Br), (M-11802, CH₃, CH₃, H, BnO, CH₃), (M-11803, CH₃, CH₃, H, PhCH₂CH₂O, H), (M-11804, CH₃, CH₃, H, PhCH₂CH₂O, Cl), (M-11805, CH₃, CH₃, H, PhCH₂CH₂O, F), (M-11806, CH₃, CH₃, H, PhCH₂CH₂O, CF₃), (M-11807, CH₃, CH₃, H, PhCH₂CH₂O, Br), (M-11808, CH₃, CH₃, H, PhCH₂CH₂O, CH₃), (M-11809, CH₃, CH₃, H, CF₃O, H), (M-11810, CH₃, CH₃, H, CF₃O, Cl), (M-11811, CH₃, CH₃, H, CF₃O, F), (M-11812, CH₃, CH₃, H, CF₃O, CF₃), (M-11813, CH₃, CH₃, H, CF₃O, Br), (M-11814, CH₃, CH₃, H, CF₃O, CH₃), (M-11815, CH₃, CH₃, H, Ph, H), (M-11816, CH₃, CH₃, H, Ph, Cl), (M-11817, CH₃, CH₃, H, Ph, F), (M-11818, CH₃, CH₃, H, Ph, CF₃), (M-11819, CH₃, CH₃, H, Ph, Br), (M-11820, CH₃, CH₃, H, Ph, CH₃), (M-11821, CH₃, CH₃, H, 4-F-Ph, H), (M-11822, CH₃, CH₃, H, 4-F-Ph, Cl), (M-11823, CH₃, CH₃, H, 4-F-Ph, F), (M-11824, CH₃, CH₃, H, 4-F-Ph, CF₃), (M-11825, CH₃, CH₃, H, 4-F-Ph, Br), (M-11826, CH₃, CH₃, H, 4-F-Ph, CH₃), (M-11827, CH₃, CH₃, H, 4-CF₃-Ph, H), (M-11828, CH₃, CH₃, H, 4-CF₃-Ph, Cl), (M-11829, CH₃, CH₃, H, 4-CF₃-Ph, F), (M-11830, CH₃, CH₃, H, 4-CF₃-Ph, CF₃), (M-11831, CH₃, CH₃, H, 4-CF₃-Ph, Br), (M-11832, CH₃, CH₃, H, 4-CF₃-Ph, CH₃), (M-11833, CH₃, CH₃, H, 4-(Me)₂N-Ph, H), (M-11834, CH₃, CH₃, H, 4-(Me)₂N-Ph, Cl), (M-11835, CH₃, CH₃, H, 4-(Me)₂N-Ph, F), (M-11836, CH₃, CH₃, H, 4-(Me)₂N-Ph, CF₃), (M-11837, CH₃, CH₃, H, 4-(Me)₂N-Ph, Br), (M-11838, CH₃, CH₃, H, 4-(Me)₂N-Ph, CH₃), (M-11839, CH₃, CH₃, H, 4-OH-Ph, H), (M-11840, CH₃, CH₃, H, 4-OH-Ph, Cl), (M-11841, CH₃, CH₃, H, 4-OH-Ph, F), (M-11842, CH₃, CH₃, H, 4-OH-Ph, CF₃), (M-11843, CH₃, CH₃, H, 4-OH-Ph, Br), (M-11844, CH₃, CH₃, H, 4-OH-Ph, CH₃), (M-11845, CH₃, CH₃, H, 3,4-di-F-Ph, H), (M-11846, CH₃, CH₃, H, 3,4-di-F-Ph, Cl), (M-11847, CH₃, CH₃, H, 3,4-di-F-Ph, F), (M-11848, CH₃, CH₃, H, 3,4-di-F-Ph, CF₃), (M-11849, CH₃, CH₃, H, 3,4-di-F-Ph, Br), (M-11850, CH₃, CH₃, H, 3,4-di-F-Ph, CH₃), (M-11851, CH₃, CH₃, H, 4-COOH-Ph, H), (M-11852, CH₃, CH₃, H, 4-COOH-Ph, Cl), (M-11853, CH₃, CH₃, H, 4-COOH-Ph, F), (M-11854, CH₃, CH₃, H, 4-COOH-Ph, CF₃), (M-11855, CH₃, CH₃, H, 4-COOH-Ph, Br), (M-11856, CH₃, CH₃, H, 4-COOH-Ph, CH₃), (M-11857, CH₃, CH₃, H, Bn, H), (M-11858, CH₃, CH₃, H, Bn, Cl), (M-11859, CH₃, CH₃, H, Bn, F), (M-11860, CH₃, CH₃, H, Bn, CF₃), (M-11861, CH₃, CH₃, H, Bn, Br), (M-11862, CH₃, CH₃, H, Bn, CH₃), (M-11863, CH₃, CH₃, H, 4-F-Bn, H), (M-11864, CH₃, CH₃, H, 4-F-Bn, Cl), (M-11865, CH₃, CH₃, H, 4-F-Bn, F), (M-11866, CH₃, CH₃, H, 4-F-Bn, CF₃), (M-11867, CH₃, CH₃, H, 4-F-Bn, Br), (M-11868, CH₃, CH₃, H, 4-F-Bn, CH₃), (M-11869, CH₃, CH₃, H, 2-Py, H), (M-11870, CH₃, CH₃, H, 2-Py, Cl), (M-11871, CH₃, CH₃, H, 2-Py, F), (M-11872, CH₃, CH₃, H, 2-Py, CF₃), (M-11873, CH₃, CH₃, H, 2-Py, Br), (M-11874, CH₃, CH₃, H, 2-Py, CH₃), (M-11875, CH₃, CH₃, H, 3-Py, H), (M-11876, CH₃, CH₃, H, 3-Py, Cl), (M-11877, CH₃, CH₃, H, 3-Py, F), (M-11878, CH₃, CH₃, H, 3-Py, CF₃), (M-11879, CH₃, CH₃, H, 3-Py, Br), (M-11880, CH₃, CH₃, H, 3-Py, CH₃), (M-11881, CH₃, CH₃, H, 4-Py, H), (M-11882, CH₃, CH₃, H, 4-Py, Cl), (M-11883, CH₃, CH₃, H, 4-Py, F), (M-11884, CH₃, CH₃, H, 4-Py, CF₃), (M-11885, CH₃, CH₃, H, 4-Py, Br), (M-11886, CH₃, CH₃, H, 4-Py, CH₃), (M-11887, CH₃, CH₃, H, 2-Th, H), (M-11888, CH₃, CH₃, H, 2-Th, Cl), (M-11889, CH₃, CH₃, H, 2-Th, F), (M-11890, CH₃, CH₃, H, 2-Th, CF₃), (M-11891, CH₃, CH₃, H, 2-Th, Br), (M-11892, CH₃, CH₃, H, 2-Th, CH₃), (M-11893, CH₃, CH₃, H, 3-Th, H), (M-11894, CH₃, CH₃, H, 3-Th, Cl), (M-11895, CH₃, CH₃, H, 3-Th, F), (M-11896, CH₃, CH₃, H, 3-Th, CF₃), (M-11897, CH₃, CH₃, H, 3-Th, Br), (M-11898, CH₃, CH₃, H, 3-Th, CH₃), (M-11899, CH₃, CH₃, H, pyrazol-2-yl, H), (M-11900, CH₃, CH₃, H, pyrazol-2-yl, Cl), (M-11901, CH₃, CH₃, H, pyrazol-2-yl, F), (M-11902, CH₃, CH₃, H, pyrazol-2-yl, CF₃), (M-11903, CH₃, CH₃, H, pyrazol-2-yl, Br), (M-11904, CH₃, CH₃, H, pyrazol-2-yl, CH₃), (M-11905, CH₃, CH₃, H, pyrazol-3-yl, H), (M-11906, CH₃, CH₃, H, pyrazol-3-yl, Cl), (M-11907, CH₃, CH₃, H, pyrazol-3-yl, F), (M-11908, CH₃, CH₃, H, pyrazol-3
-yl, CF₃), (M-11909, CH₃, CH₃, H, pyrazol-3-yl, Br), (M-11910, CH₃, CH₃, H, pyrazol-3-yl, CH₃), (M-11911, CH₃, CH₃, H, pyrimidin-2-yl, H), (M-11912, CH₃, CH₃, H, pyrimidin-2-yl, Cl), (M-11913, CH₃, CH₃, H, pyrimidin-2-yl, F), (M-11914, CH₃, CH₃, H, pyrimidin-2-yl, CF₃), (M-11915, CH₃, CH₃, H, pyrimidin-2-yl, Br), (M-11916, CH₃, CH₃, H, pyrimidin-2-yl, CH₃), (M-11917, CH₃, CH₃, H, pyrimidin-4-yl, H), (M-11918, CH₃, CH₃, H, pyrimidin-4-yl, Cl), (M-11919, CH₃, CH₃, H, pyrimidin-4-yl, F), (M-11920, CH₃, CH₃, H, pyrimidin-4-yl, CF₃), (M-11921, CH₃, CH₃, H, pyrimidin-4-yl, Br), (M-11922, CH₃, CH₃, H, pyrimidin-4-yl, CH₃), (M-11923, CH₃, CH₃, H, pyrimidin-5-yl, H), (M-11924, CH₃, CH₃, H, pyrimidin-5-yl, Cl), (M-11925, CH₃, CH₃, H, pyrimidin-5-yl, F), (M-11926, CH₃, CH₃, H, pyrimidin-5-yl, CF₃), (M-11927, CH₃, CH₃, H, pyrimidin-5-yl, Br), (M-11928, CH₃, CH₃, H, pyrimidin-5-yl, CH₃), (M-11929, CH₃, CH₃, H, HOOCCH₂CH₂CH₂, H), (M-11930, CH₃, CH₃, H, HOOCCH₂CH₂CH₂, Cl), (M-11931, CH₃, CH₃, H, HOOCCH₂CH₂CH₂, F), (M-11932, CH₃, CH₃, H, HOOCCH₂CH₂CH₂, CF₃), (M-11933, CH₃, CH₃, H, HOOCCH₂CH₂CH₂, Br), (M-11934, CH₃, CH₃, H, HOOCCH₂CH₂CH₂, CH₃), (M-11935, CH₃, CH₃, H, HOOCCH₂CH₂CH₂CH₂, H), (M-11936, CH₃, CH₃, H, HOOCCH₂CH₂CH₂CH₂, Cl), (M-11937, CH₃, CH₃, H, HOOCCH₂CH₂CH₂CH₂, F), (M-11938, CH₃, CH₃, H, HOOCCH₂CH₂CH₂CH₂, CF₃), (M-11939, CH₃, CH₃, H, HOOCCH₂CH₂CH₂CH₂, Br), (M-11940, CH₃, CH₃, H, HOOCCH₂CH₂CH₂CH₂, CH₃), (M-11941, CH₃, CH₃, H, (Me)₂NCOCH₂CH₂CH₂CH₂, H), (M-11942, CH₃, CH₃, H, (Me)₂NCOCH₂CH₂CH₂CH₂, Cl), (M-11943, CH₃, CH₃, H, (Me)₂NCOCH₂CH₂CH₂CH₂, F), (M-11944, CH₃, CH₃, H, (Me)₂NCOCH₂CH₂CH₂CH₂, CF₃), (M-11945, CH₃, CH₃, H, (Me)₂NCOCH₂CH₂CH₂CH₂, Br), (M-11946, CH₃, CH₃, H, (Me)₂NCOCH₂CH₂CH₂CH₂, CH₃), (M-11947, CH₃, CH₃, H, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, H), (M-11948, CH₃, CH₃, H, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, Cl), (M-11949, CH₃, CH₃, H, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, F), (M-11950, CH₃, CH₃, H, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, CF₃), (M-11951, CH₃, CH₃, H, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, Br), (M-11952, CH₃, CH₃, H, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, CH₃), (M-11953, CH₃, CH₃, H, MeOCH₂, H), (M-11954, CH₃, CH₃, H, MeOCH₂, Cl), (M-11955, CH₃, CH₃, H, MeOCH₂, F), (M-11956, CH₃, CH₃, H, MeOCH₂, CF₃), (M-11957, CH₃, CH₃, H, MeOCH₂, Br), (M-11958, CH₃, CH₃, H, MeOCH₂, CH₃), (M-11959, CH₃, CH₃, H, EtOCH₂, H), (M-11960, CH₃, CH₃, H, EtOCH₂, Cl), (M-11961, CH₃, CH₃, H, EtOCH₂, F), (M-11962, CH₃, CH₃, H, EtOCH₂, CF₃), (M-11963, CH₃, CH₃, H, EtOCH₂, Br), (M-11964, CH₃, CH₃, H, EtOCH₂, CH₃), (M-11965, CH₃, CH₃, H, EtOCH₂CH₂, H), (M-11966, CH₃, CH₃, H, EtOCH₂CH₂, Cl), (M-11967, CH₃, CH₃, H, EtOCH₂CH₂, F), (M-11968, CH₃, CH₃, H, EtOCH₂CH₂, CF₃), (M-11969, CH₃, CH₃, H, EtOCH₂CH₂, Br), (M-11970, CH₃, CH₃, H, EtOCH₂CH₂, CH₃), (M-11971, CH₃, CH₃, H, MeOCH₂CH₂OCH₂CH₂, H), (M-11972, CH₃, CH₃, H, MeOCH₂CH₂OCH₂CH₂, Cl), (M-11973, CH₃, CH₃, H, MeOCH₂CH₂OCH₂CH₂, F), (M-11974, CH₃, CH₃, H, MeOCH₂CH₂OCH₂CH₂, CF₃), (M-11975, CH₃, CH₃, H, MeOCH₂CH₂OCH₂CH₂, Br), (M-11976, CH₃, CH₃, H, MeOCH₂CH₂OCH₂CH₂, CH₃), (M-11977, CH₃, CH₃, H, MeOCH₂CH₂, H), (M-11978, CH₃, CH₃, H, MeOCH₂CH₂, Cl), (M-11979, CH₃, CH₃, H, MeOCH₂CH₂, F), (M-11980, CH₃, CH₃, H, MeOCH₂CH₂, CF₃), (M-11981, CH₃, CH₃, H, MeOCH₂CH₂, Br), (M-11982, CH₃, CH₃, H, MeOCH₂CH₂, CH₃), (M-11983, CH₃, CH₃, H, HOCH₂, H), (M-11984, CH₃, CH₃, H, HOCH₂, Cl), (M-11985, CH₃, CH₃, H, HOCH₂, F), (M-11986, CH₃, CH₃, H, HOCH₂, CF₃), (M-11987, CH₃, CH₃, H, HOCH₂, Br), (M-11988, CH₃, CH₃, H, HOCH₂, CH₃), (M-11989, CH₃, CH₃, H, HOCH₂CH₂, H), (M-11990, CH₃, CH₃, H, HOCH₂CH₂, Cl), (M-11991, CH₃, CH₃, H, HOCH₂CH₂, F), (M-11992, CH₃, CH₃, H, HOCH₂CH₂, CF₃), (M-11993, CH₃, CH₃, H, HOCH₂CH₂, Br), (M-11994, CH₃, CH₃, H, HOCH₂CH₂, CH₃), (M-11995, CH₃, CH₃, H, HOCH₂CH₂CH₂, H), (M-11996, CH₃, CH₃, H, HOCH₂CH₂CH₂, Cl), (M-11997, CH₃, CH₃, H, HOCH₂CH₂CH₂, F), (M-11998, CH₃, CH₃, H, HOCH₂CH₂CH₂, CF₃), (M-11999, CH₃, CH₃, H, HOCH₂CH₂CH₂, Br), (M-12000, CH₃, CH₃, H, HOCH₂CH₂CH₂, CH₃), (M-12001, CH₃, CH₃, H, HOCH₂CH₂CH₂CH₂, H), (M-12002, CH₃, CH₃, H, HOCH₂CH₂CH₂CH₂, Cl), (M-12003, CH₃, CH₃, H, HOCH₂CH₂CH₂CH₂, F), (M-12004, CH₃, CH₃, H, HOCH₂CH₂CH₂CH₂, CF₃), (M-12005, CH₃, CH₃, H, HOCH₂CH₂CH₂CH₂, Br), (M-12006, CH₃, CH₃, H, HOCH₂CH₂CH₂CH₂, CH₃), (M-12007, CH₃, CH₃, H, HOCH₂CH₂CH₂CH₂CH₂, H), (M-12008, CH₃, CH₃, H, HOCH₂CH₂CH₂CH₂CH₂, Cl), (M-12009, CH₃, CH₃, H, HOCH₂CH₂CH₂CH₂CH₂, F), (M-12010, CH₃, CH₃, H, HOCH₂CH₂CH₂CH₂CH₂, CF₃), (M-12011, CH₃, CH₃, H, HOCH₂CH₂CH₂CH₂CH₂, Br), (M-12012, CH₃, CH₃, H, HOCH₂CH₂CH₂CH₂CH₂, CH₃), (M-12013, CH₃, CH₃, H, HOCH₂CH₂OCH₂CH₂, H), (M-12014, CH₃, CH₃, H, HOCH₂CH₂OCH₂CH₂, Cl), (M-12015, CH₃, CH₃, H, HOCH
₂CH₂OCH₂CH₂, F), (M-12016, CH₃, CH₃, H, HOCH₂CH₂OCH₂CH₂, CF₃), (M-12017, CH₃, CH₃, H, HOCH₂CH₂OCH₂CH₂, Br), (M-12018, CH₃, CH₃, H, HOCH₂CH₂OCH₂CH₂, CH₃), (M-12019, CH₃, CH₃, H, (Me)₂N, H), (M-12020, CH₃, CH₃, H, (Me)₂N, Cl), (M-12021, CH₃, CH₃, H, (Me)₂N, F), (M-12022, CH₃, CH₃, H, (Me)₂N, CF₃), (M-12023, CH₃, CH₃, H, (Me)₂N, Br), (M-12024, CH₃, CH₃, H, (Me)₂N, CH₃), (M-12025, CH₃, CH₃, H, piperidin-4-yl-methyl, H), (M-12026, CH₃, CH₃, H, piperidin-4-yl-methyl, Cl), (M-12027, CH₃, CH₃, H, piperidin-4-yl-methyl, F), (M-12028, CH₃, CH₃, H, piperidin-4-yl-methyl, CF₃), (M-12029, CH₃, CH₃, H, piperidin-4-yl-methyl, Br), (M-12030, CH₃, CH₃, H, piperidin-4-yl-methyl, CH₃), (M-12031, CH₃, CH₃, H, cyclohexylmethyl, H), (M-12032, CH₃, CH₃, H, cyclohexylmethyl, Cl), (M-12033, CH₃, CH₃, H, cyclohexylmethyl, F), (M-12034, CH₃, CH₃, H, cyclohexylmethyl, CF₃), (M-12035, CH₃, CH₃, H, cyclohexylmethyl, Br), (M-12036, CH₃, CH₃, H, cyclohexylmethyl, CH₃), (M-12037, CH₃, CH₃, F, H, H), (M-12038, CH₃, CH₃, F, H, Cl), (M-12039, CH₃, CH₃, F, H, F), (M-12040, CH₃, CH₃, F, H, CF₃), (M-12041, CH₃, CH₃, F, H, Br), (M-12042, CH₃, CH₃, F, H, CH₃), (M-12043, CH₃, CH₃, F, F, H), (M-12044, CH₃, CH₃, F, F, Cl), (M-12045, CH₃, CH₃, F, F, F), (M-12046, CH₃, CH₃, F, F, CF₃), (M-12047, CH₃, CH₃, F, F, Br), (M-12048, CH₃, CH₃, F, F, CH₃), (M-12049, CH₃, CH₃, F, Cl, H), (M-12050, CH₃, CH₃, F, Cl, Cl), (M-12051, CH₃, CH₃, F, Cl, F), (M-12052, CH₃, CH₃, F, Cl, CF₃), (M-12053, CH₃, CH₃, F, Cl, Br), (M-12054, CH₃, CH₃, F, Cl, CH₃), (M-12055, CH₃, CH₃, F, CH₃, H), (M-12056, CH₃, CH₃, F, CH₃, Cl), (M-12057, CH₃, CH₃, F, CH₃, F), (M-12058, CH₃, CH₃, F, CH₃, CF₃), (M-12059, CH₃, CH₃, F, CH₃, Br), (M-12060, CH₃, CH₃, F, CH₃, CH₃), (M-12061, CH₃, CH₃, F, Et, H), (M-12062, CH₃, CH₃, F, Et, Cl), (M-12063, CH₃, CH₃, F, Et, F), (M-12064, CH₃, CH₃, F, Et, CF₃), (M-12065, CH₃, CH₃, F, Et, Br), (M-12066, CH₃, CH₃, F, Et, CH₃), (M-12067, CH₃, CH₃, F, n-Pr, H), (M-12068, CH₃, CH₃, F, n-Pr, Cl), (M-12069, CH₃, CH₃, F, n-Pr, F), (M-12070, CH₃, CH₃, F, n-Pr, CF₃), (M-12071, CH₃, CH₃, F, n-Pr, Br), (M-12072, CH₃, CH₃, F, n-Pr, CH₃), (M-12073, CH₃, CH₃, F, c-Pr, H), (M-12074, CH₃, CH₃, F, c-Pr, Cl), (M-12075, CH₃, CH₃, F, c-Pr, F), (M-12076, CH₃, CH₃, F, c-Pr, CF₃), (M-12077, CH₃, CH₃, F, c-Pr, Br), (M-12078, CH₃, CH₃, F, c-Pr, CH₃), (M-12079, CH₃, CH₃, F, i-Pr, H), (M-12080, CH₃, CH₃, F, i-Pr, Cl), (M-12081, CH₃, CH₃, F, i-Pr, F), (M-12082, CH₃, CH₃, F, i-Pr, CF₃), (M-12083, CH₃, CH₃, F, i-Pr, Br), (M-12084, CH₃, CH₃, F, i-Pr, CH₃), (M-12085, CH₃, CH₃, F, n-Bu, H), (M-12086, CH₃, CH₃, F, n-Bu, Cl), (M-12087, CH₃, CH₃, F, n-Bu, F), (M-12088, CH₃, CH₃, F, n-Bu, CF₃), (M-12089, CH₃, CH₃, F, n-Bu, Br), (M-12090, CH₃, CH₃, F, n-Bu, CH₃), (M-12091, CH₃, CH₃, F, i-Bu, H), (M-12092, CH₃, CH₃, F, i-Bu, Cl), (M-12093, CH₃, CH₃, F, i-Bu, F), (M-12094, CH₃, CH₃, F, i-Bu, CF₃), (M-12095, CH₃, CH₃, F, i-Bu, Br), (M-12096, CH₃, CH₃, F, i-Bu, CH₃), (M-12097, CH₃, CH₃, F, sec-Bu, H), (M-12098, CH₃, CH₃, F, sec-Bu, Cl), (M-12099, CH₃, CH₃, F, sec-Bu, F), (M-12100, CH₃, CH₃, F, sec-Bu, CF₃), (M-12101, CH₃, CH₃, F, sec-Bu, Br), (M-12102, CH₃, CH₃, F, sec-Bu, CH₃), (M-12103, CH₃, CH₃, F, n-Pen, H), (M-12104, CH₃, CH₃, F, n-Pen, Cl), (M-12105, CH₃, CH₃, F, n-Pen, F), (M-12106, CH₃, CH₃, F, n-Pen, CF₃), (M-12107, CH₃, CH₃, F, n-Pen, Br), (M-12108, CH₃, CH₃, F, n-Pen, CH₃), (M-12109, CH₃, CH₃, F, c-Pen, H), (M-12110, CH₃, CH₃, F, c-Pen, Cl), (M-12111, CH₃, CH₃, F, c-Pen, F), (M-12112, CH₃, CH₃, F, c-Pen, CF₃), (M-12113, CH₃, CH₃, F, c-Pen, Br), (M-12114, CH₃, CH₃, F, c-Pen, CH₃), (M-12115, CH₃, CH₃, F, n-Hex, H), (M-12116, CH₃, CH₃, F, n-Hex, Cl), (M-12117, CH₃, CH₃, F, n-Hex, F), (M-12118, CH₃, CH₃, F, n-Hex, CF₃), (M-12119, CH₃, CH₃, F, n-Hex, Br), (M-12120, CH₃, CH₃, F, n-Hex, CH₃), (M-12121, CH₃, CH₃, F, c-Hex, H), (M-12122, CH₃, CH₃, F, c-Hex, Cl), (M-12123, CH₃, CH₃, F, c-Hex, F), (M-12124, CH₃, CH₃, F, c-Hex, CF₃), (M-12125, CH₃, CH₃, F, c-Hex, Br), (M-12126, CH₃, CH₃, F, c-Hex, CH₃), (M-12127, CH₃, CH₃, F, OH, H), (M-12128, CH₃, CH₃, F, OH, Cl), (M-12129, CH₃, CH₃, F, OH, F), (M-12130, CH₃, CH₃, F, OH, CF₃), (M-12131, CH₃, CH₃, F, OH, Br), (M-12132, CH₃, CH₃, F, OH, CH₃), (M-12133, CH₃, CH₃, F, EtO, H), (M-12134, CH₃, CH₃, F, EtO, Cl), (M-12135, CH₃, CH₃, F, EtO, F), (M-12136, CH₃, CH₃, F, EtO, CF₃), (M-12137, CH₃, CH₃, F, EtO, Br), (M-12138, CH₃, CH₃, F, EtO, CH₃), (M-12139, CH₃, CH₃, F, n-PrO, H), (M-12140, CH₃, CH₃, F, n-PrO, Cl), (M-12141, CH₃, CH₃, F, n-PrO, F), (M-12142, CH₃, CH₃, F, n-PrO, CF₃), (M-12143, CH₃, CH₃, F, n-PrO, Br), (M-12144, CH₃, CH₃, F, n-PrO, CH₃), (M-12145, CH₃, CH₃, F, PhO, H), (M-12146, CH₃, CH₃, F, PhO, Cl), (M-12147, CH₃, CH₃, F, PhO, F), (M-12148, CH₃, CH₃, F, PhO, CF₃), (M-12149, CH₃, CH₃, F, PhO, Br), (M-12150, CH₃, CH₃, F, PhO, CH₃), (M-12151, CH₃, CH₃, F, BnO, H), (M-12152, CH₃, CH₃, F, BnO, Cl), (M-12153, CH₃, CH₃, F, BnO, F), (M-12154, CH₃, CH₃, F, BnO, CF₃), (M-12155, CH₃, CH₃, F, BnO, Br), (M-12156, CH₃, CH₃, F, BnO, CH₃), (M-12157, CH₃, CH₃, F, PhCH₂CH₂O, H), (M-12158, CH₃, CH₃, F, PhCH₂CH₂O, Cl), (M-12159, CH₃, CH₃, F, PhCH₂CH₂O, F), (M-12160, CH₃, CH₃, F, PhCH₂CH₂O, CF₃), (M-12161, CH₃, CH₃, F, PhCH₂CH₂O, Br), (M-12162, CH₃, CH₃, F, PhCH₂CH₂O, CH₃), (M-12163, CH₃, CH₃, F, CF₃O, H), (M-12164, CH₃, CH₃, F, CF₃O, Cl), (M-12165, CH₃, CH₃, F, CF₃O, F), (M-12166, CH₃, CH₃, F, CF₃O, CF₃), (M-12167, CH₃, CH₃, F, CF₃O, Br), (M-12168, CH₃, CH₃, F, CF₃O, CH₃), (M-12169, CH₃, CH₃, F, Ph, H), (M-12170, CH₃, CH₃, F, Ph, Cl), (M-12171, CH₃, CH₃, F, Ph, F), (M-12172, CH₃, CH₃, F, Ph, CF₃), (M-12173, CH₃, CH₃, F, Ph, Br), (M-12174, CH₃, CH₃, F, Ph, CH₃), (M-12175, CH₃, CH₃
, F, 4-F-Ph, H), (M-12176, CH₃, CH₃, F, 4-F-Ph, Cl), (M-12177, CH₃, CH₃, F, 4-F-Ph, F), (M-12178, CH₃, CH₃, F, 4-F-Ph, CF₃), (M-12179, CH₃, CH₃, F, 4-F-Ph, Br), (M-12180, CH₃, CH₃, F, 4-F-Ph, CH₃), (M-12181, CH₃, CH₃, F, 4-CF₃-Ph, H), (M-12182, CH₃, CH₃, F, 4-CF₃-Ph, Cl), (M-12183, CH₃, CH₃, F, 4-CF₃-Ph, F), (M-12184, CH₃, CH₃, F, 4-CF₃-Ph, CF₃), (M-12185, CH₃, CH₃, F, 4-CF₃-Ph, Br), (M-12186, CH₃, CH₃, F, 4-CF₃-Ph, CH₃), (M-12187, CH₃, CH₃, F, 4-(Me)₂N-Ph, H), (M-12188, CH₃, CH₃, F, 4-(Me)₂N-Ph, Cl), (M-12189, CH₃, CH₃, F, 4-(Me)₂N-Ph, F), (M-12190, CH₃, CH₃, F, 4-(Me)₂N-Ph, CF₃), (M-12191, CH₃, CH₃, F, 4-(Me)₂N-Ph, Br), (M-12192, CH₃, CH₃, F, 4-(Me)₂N-Ph, CH₃), (M-12193, CH₃, CH₃, F, 4-OH-Ph, H), (M-12194, CH₃, CH₃, F, 4-OH-Ph, Cl), (M-12195, CH₃, CH₃, F, 4-OH-Ph, F), (M-12196, CH₃, CH₃, F, 4-OH-Ph, CF₃), (M-12197, CH₃, CH₃, F, 4-OH-Ph, Br), (M-12198, CH₃, CH₃, F, 4-OH-Ph, CH₃), (M-12199, CH₃, CH₃, F, 3,4-di-F-Ph, H), (M-12200, CH₃, CH₃, F, 3,4-di-F-Ph, Cl), (M-12201, CH₃, CH₃, F, 3,4-di-F-Ph, F), (M-12202, CH₃, CH₃, F, 3,4-di-F-Ph, CF₃), (M-12203, CH₃, CH₃, F, 3,4-di-F-Ph, Br), (M-12204, CH₃, CH₃, F, 3,4-di-F-Ph, CH₃), (M-12205, CH₃, CH₃, F, 4-COOH-Ph, H), (M-12206, CH₃, CH₃, F, 4-COOH-Ph, Cl), (M-12207, CH₃, CH₃, F, 4-COOH-Ph, F), (M-12208, CH₃, CH₃, F, 4-COOH-Ph, CF₃), (M-12209, CH₃, CH₃, F, 4-COOH-Ph, Br), (M-12210, CH₃, CH₃, F, 4-COOH-Ph, CH₃), (M-12211, CH₃, CH₃, F, Bn, H), (M-12212, CH₃, CH₃, F, Bn, Cl), (M-12213, CH₃, CH₃, F, Bn, F), (M-12214, CH₃, CH₃, F, Bn, CF₃), (M-12215, CH₃, CH₃, F, Bn, Br), (M-12216, CH₃, CH₃, F, Bn, CH₃), (M-12217, CH₃, CH₃, F, 4-F-Bn, H), (M-12218, CH₃, CH₃, F, 4-F-Bn, Cl), (M-12219, CH₃, CH₃, F, 4-F-Bn, F), (M-12220, CH₃, CH₃, F, 4-F-Bn, CF₃), (M-12221, CH₃, CH₃, F, 4-F-Bn, Br), (M-12222, CH₃, CH₃, F, 4-F-Bn, CH₃), (M-12223, CH₃, CH₃, F, 2-Py, H), (M-12224, CH₃, CH₃, F, 2-Py, Cl), (M-12225, CH₃, CH₃, F, 2-Py, F), (M-12226, CH₃, CH₃, F, 2-Py, CF₃), (M-12227, CH₃, CH₃, F, 2-Py, Br), (M-12228, CH₃, CH₃, F, 2-Py, CH₃), (M-12229, CH₃, CH₃, F, 3-Py, H), (M-12230, CH₃, CH₃, F, 3-Py, Cl), (M-12231, CH₃, CH₃, F, 3-Py, F), (M-12232, CH₃, CH₃, F, 3-Py, CF₃), (M-12233, CH₃, CH₃, F, 3-Py, Br), (M-12234, CH₃, CH₃, F, 3-Py, CH₃), (M-12235, CH₃, CH₃, F, 4-Py, H), (M-12236, CH₃, CH₃, F, 4-Py, Cl), (M-12237, CH₃, CH₃, F, 4-Py, F), (M-12238, CH₃, CH₃, F, 4-Py, CF₃), (M-12239, CH₃, CH₃, F, 4-Py, Br), (M-12240, CH₃, CH₃, F, 4-Py, CH₃), (M-12241, CH₃, CH₃, F, 2-Th, H), (M-12242, CH₃, CH₃, F, 2-Th, Cl), (M-12243, CH₃, CH₃, F, 2-Th, F), (M-12244, CH₃, CH₃, F, 2-Th, CF₃), (M-12245, CH₃, CH₃, F, 2-Th, Br), (M-12246, CH₃, CH₃, F, 2-Th, CH₃), (M-12247, CH₃, CH₃, F, 3-Th, H), (M-12248, CH₃, CH₃, F, 3-Th, Cl), (M-12249, CH₃, CH₃, F, 3-Th, F), (M-12250, CH₃, CH₃, F, 3-Th, CF₃), (M-12251, CH₃, CH₃, F, 3-Th, Br), (M-12252, CH₃, CH₃, F, 3-Th, CH₃), (M-12253, CH₃, CH₃, F, pyrazol-2-yl, H), (M-12254, CH₃, CH₃, F, pyrazol-2-yl, Cl), (M-12255, CH₃, CH₃, F, pyrazol-2-yl, F), (M-12256, CH₃, CH₃, F, pyrazol-2-yl, CF₃), (M-12257, CH₃, CH₃, F, pyrazol-2-yl, Br), (M-12258, CH₃, CH₃, F, pyrazol-2-yl, CH₃), (M-12259, CH₃, CH₃, F, pyrazol-3-yl, H), (M-12260, CH₃, CH₃, F, pyrazol-3-yl, Cl), (M-12261, CH₃, CH₃, F, pyrazol-3-yl, F), (M-12262, CH₃, CH₃, F, pyrazol-3-yl, CF₃), (M-12263, CH₃, CH₃, F, pyrazol-3-yl, Br), (M-12264, CH₃, CH₃, F, pyrazol-3-yl, CH₃), (M-12265, CH₃, CH₃, F, pyrimidin-2-yl, H), (M-12266, CH₃, CH₃, F, pyrimidin-2-yl, Cl), (M-12267, CH₃, CH₃, F, pyrimidin-2-yl, F), (M-12268, CH₃, CH₃, F, pyrimidin-2-yl, CF₃), (M-12269, CH₃, CH₃, F, pyrimidin-2-yl, Br), (M-12270, CH₃, CH₃, F, pyrimidin-2-yl, CH₃), (M-12271, CH₃, CH₃, F, pyrimidin-4-yl, H), (M-12272, CH₃, CH₃, F, pyrimidin-4-yl, Cl), (M-12273, CH₃, CH₃, F, pyrimidin-4-yl, F), (M-12274, CH₃, CH₃, F, pyrimidin-4-yl, CF₃), (M-12275, CH₃, CH₃, F, pyrimidin-4-yl, Br), (M-12276, CH₃, CH₃, F, pyrimidin-4-yl, CH₃), (M-12277, CH₃, CH₃, F, pyrimidin-5-yl, H), (M-12278, CH₃, CH₃, F, pyrimidin-5-yl, Cl), (M-12279, CH₃, CH₃, F, pyrimidin-5-yl, F), (M-12280, CH₃, CH₃, F, pyrimidin-5-yl, CF₃), (M-12281, CH₃, CH₃, F, pyrimidin-5-yl, Br), (M-12282, CH₃, CH₃, F, pyrimidin-5-yl, CH₃), (M-12283, CH₃, CH₃, F, HOOCCH₂CH₂CH₂, H), (M-12284, CH₃, CH₃, F, HOOCCH₂CH₂CH₂, Cl), (M-12285, CH₃, CH₃, F, HOOCCH₂CH₂CH₂, F), (M-12286, CH₃, CH₃, F, HOOCCH₂CH₂CH₂, CF₃), (M-12287, CH₃, CH₃, F, HOOCCH₂CH₂CH₂, Br), (M-12288, CH₃, CH₃, F, HOOCCH₂CH₂CH₂, CH₃), (M-12289, CH₃, CH₃, F, HOOCCH₂CH₂CH₂CH₂, H), (M-12290, CH₃, CH₃, F, HOOCCH₂CH₂CH₂CH₂, Cl), (M-12291, CH₃, CH₃, F, HOOCCH₂CH₂CH₂CH₂, F), (M-12292, CH₃, CH₃, F, HOOCCH₂CH₂CH₂CH₂, CF₃), (M-12293, CH₃, CH₃, F, HOOCCH₂CH₂CH₂CH₂, Br), (M-12294, CH₃, CH₃, F, HOOCCH₂CH₂CH₂CH₂, CH₃), (M-12295, CH₃, CH₃, F, (Me)₂NCOCH₂CH₂CH₂CH₂, H), (M-12296, CH₃, CH₃, F, (Me)₂NCOCH₂CH₂CH₂CH₂, Cl), (M-12297, CH₃, CH₃, F, (Me)₂NCOCH₂CH₂CH₂CH₂, F), (M-12298, CH₃, CH₃, F, (Me)₂NCOCH₂CH₂CH₂CH₂, CF₃), (M-12299, CH₃, CH₃, F, (Me)₂NCOCH₂CH₂CH₂CH₂, Br), (M-12300, CH₃, CH₃, F, (Me)₂NCOCH₂CH₂CH₂CH₂, CH₃), (M-12301, CH₃, CH₃, F, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, H), (M-12302, CH₃, CH₃, F, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, Cl), (M-12303, CH₃, CH₃, F, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, F), (M-12304, CH₃, CH₃, F, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, CF₃), (M-12305, CH₃, CH₃, F, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, Br), (M-12306, CH₃, CH₃, F, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, CH₃), (M-12307, CH₃, CH₃, F, MeOCH₂, H), (M-12308, CH₃, CH₃, F, MeOCH₂, Cl), (M-12309, CH₃, CH₃, F, MeOCH₂, F), (M-12310, CH₃, CH₃, F, MeOCH₂, CF₃), (M-12311, CH₃
, CH₃, F, MeOCH₂, Br), (M-12312, CH₃, CH₃, F, MeOCH₂, CH₃), (M-12313, CH₃, CH₃, F, EtOCH₂, H), (M-12314, CH₃, CH₃, F, EtOCH₂, Cl), (M-12315, CH₃, CH₃, F, EtOCH₂, F), (M-12316, CH₃, CH₃, F, EtOCH₂, CF₃), (M-12317, CH₃, CH₃, F, EtOCH₂, Br), (M-12318, CH₃, CH₃, F, EtOCH₂, CH₃), (M-12319, CH₃, CH₃, F, EtOCH₂CH₂, H), (M-12320, CH₃, CH₃, F, EtOCH₂CH₂, Cl), (M-12321, CH₃, CH₃, F, EtOCH₂CH₂, F), (M-12322, CH₃, CH₃, F, EtOCH₂CH₂, CF₃), (M-12323, CH₃, CH₃, F, EtOCH₂CH₂, Br), (M-12324, CH₃, CH₃, F, EtOCH₂CH₂, CH₃), (M-12325, CH₃, CH₃, F, MeOCH₂CH₂OCH₂CH₂, H), (M-12326, CH₃, CH₃, F, MeOCH₂CH₂OCH₂CH₂, Cl), (M-12327, CH₃, CH₃, F, MeOCH₂CH₂OCH₂CH₂, F), (M-12328, CH₃, CH₃, F, MeOCH₂CH₂OCH₂CH₂, CF₃), (M-12329, CH₃, CH₃, F, MeOCH₂CH₂OCH₂CH₂, Br), (M-12330, CH₃, CH₃, F, MeOCH₂CH₂OCH₂CH₂, CH₃), (M-12331, CH₃, CH₃, F, MeOCH₂CH₂, H), (M-12332, CH₃, CH₃, F, MeOCH₂CH₂, Cl), (M-12333, CH₃, CH₃, F, MeOCH₂CH₂, F), (M-12334, CH₃, CH₃, F, MeOCH₂CH₂, CF₃), (M-12335, CH₃, CH₃, F, MeOCH₂CH₂, Br), (M-12336, CH₃, CH₃, F, MeOCH₂CH₂, CH₃), (M-12337, CH₃, CH₃, F, HOCH₂, H), (M-12338, CH₃, CH₃, F, HOCH₂, Cl), (M-12339, CH₃, CH₃, F, HOCH₂, F), (M-12340, CH₃, CH₃, F, HOCH₂, CF₃), (M-12341, CH₃, CH₃, F, HOCH₂, Br), (M-12342, CH₃, CH₃, F, HOCH₂, CH₃), (M-12343, CH₃, CH₃, F, HOCH₂CH₂, H), (M-12344, CH₃, CH₃, F, HOCH₂CH₂, Cl), (M-12345, CH₃, CH₃, F, HOCH₂CH₂, F), (M-12346, CH₃, CH₃, F, HOCH₂CH₂, CF₃), (M-12347, CH₃, CH₃, F, HOCH₂CH₂, Br), (M-12348, CH₃, CH₃, F, HOCH₂CH₂, CH₃), (M-12349, CH₃, CH₃, F, HOCH₂CH₂CH₂, H), (M-12350, CH₃, CH₃, F, HOCH₂CH₂CH₂, Cl), (M-12351, CH₃, CH₃, F, HOCH₂CH₂CH₂, F), (M-12352, CH₃, CH₃, F, HOCH₂CH₂CH₂, CF₃), (M-12353, CH₃, CH₃, F, HOCH₂CH₂CH₂, Br), (M-12354, CH₃, CH₃, F, HOCH₂CH₂CH₂, CH₃), (M-12355, CH₃, CH₃, F, HOCH₂CH₂CH₂CH₂, H), (M-12356, CH₃, CH₃, F, HOCH₂CH₂CH₂CH₂, Cl), (M-12357, CH₃, CH₃, F, HOCH₂CH₂CH₂CH₂, F), (M-12358, CH₃, CH₃, F, HOCH₂CH₂CH₂CH₂, CF₃), (M-12359, CH₃, CH₃, F, HOCH₂CH₂CH₂CH₂, Br), (M-12360, CH₃, CH₃, F, HOCH₂CH₂CH₂CH₂, CH₃), (M-12361, CH₃, CH₃, F, HOCH₂CH₂CH₂CH₂CH₂, H), (M-12362, CH₃, CH₃, F, HOCH₂CH₂CH₂CH₂CH₂, Cl), (M-12363, CH₃, CH₃, F, HOCH₂CH₂CH₂CH₂CH₂, F), (M-12364, CH₃, CH₃, F, HOCH₂CH₂CH₂CH₂CH₂, CF₃), (M-12365, CH₃, CH₃, F, HOCH₂CH₂CH₂CH₂CH₂, Br), (M-12366, CH₃, CH₃, F, HOCH₂CH₂CH₂CH₂CH₂, CH₃), (M-12367, CH₃, CH₃, F, HOCH₂CH₂OCH₂CH₂, H), (M-12368, CH₃, CH₃, F, HOCH₂CH₂OCH₂CH₂, Cl), (M-12369, CH₃, CH₃, F, HOCH₂CH₂OCH₂CH₂, F), (M-12370, CH₃, CH₃, F, HOCH₂CH₂OCH₂CH₂, CF₃), (M-12371, CH₃, CH₃, F, HOCH₂CH₂OCH₂CH₂, Br), (M-12372, CH₃, CH₃, F, HOCH₂CH₂OCH₂CH₂, CH₃), (M-12373, CH₃, CH₃, F, (Me)₂N, H), (M-12374, CH₃, CH₃, F, (Me)₂N, Cl), (M-12375, CH₃, CH₃, F, (Me)₂N, F), (M-12376, CH₃, CH₃, F, (Me)₂N, CF₃), (M-12377, CH₃, CH₃, F, (Me)₂N, Br), (M-12378, CH₃, CH₃, F, (Me)₂N, CH₃), (M-12379, CH₃, CH₃, F, piperidin-4-yl-methyl, H), (M-12380, CH₃, CH₃, F, piperidin-4-yl-methyl, Cl), (M-12381, CH₃, CH₃, F, piperidin-4-yl-methyl, F), (M-12382, CH₃, CH₃, F, piperidin-4-yl-methyl, CF₃), (M-12383, CH₃, CH₃, F, piperidin-4-yl-methyl, Br), (M-12384, CH₃, CH₃, F, piperidin-4-yl-methyl, CH₃), (M-12385, CH₃, CH₃, F, cyclohexylmethyl, H), (M-12386, CH₃, CH₃, F, cyclohexylmethyl, Cl), (M-12387, CH₃, CH₃, F, cyclohexylmethyl, F), (M-12388, CH₃, CH₃, F, cyclohexylmethyl, CF₃), (M-12389, CH₃, CH₃, F, cyclohexylmethyl, Br), (M-12390, CH₃, CH₃, F, cyclohexylmethyl, CH₃), (M-12391, CH₃, CH₃, Cl, H, H), (M-12392, CH₃, CH₃, Cl, H, Cl), (M-12393, CH₃, CH₃, Cl, H, F), (M-12394, CH₃, CH₃, Cl, H, CF₃), (M-12395, CH₃, CH₃, Cl, H, Br), (M-12396, CH₃, CH₃, Cl, H, CH₃), (M-12397, CH₃, CH₃, Cl, F, H), (M-12398, CH₃, CH₃, Cl, F, Cl), (M-12399, CH₃, CH₃, Cl, F, F), (M-12400, CH₃, CH₃, Cl, F, CF₃), (M-12401, CH₃, CH₃, Cl, F, Br), (M-12402, CH₃, CH₃, Cl, F, CH₃), (M-12403, CH₃, CH₃, Cl, Cl, H), (M-12404, CH₃, CH₃, Cl, Cl, Cl), (M-12405, CH₃, CH₃, Cl, Cl, F), (M-12406, CH₃, CH₃, Cl, Cl, CF₃), (M-12407, CH₃, CH₃, Cl, Cl, Br), (M-12408, CH₃, CH₃, Cl, Cl, CH₃), (M-12409, CH₃, CH₃, Cl, CH₃, H), (M-12410, CH₃, CH₃, Cl, CH₃, Cl), (M-12411, CH₃, CH₃, Cl, CH₃, F), (M-12412, CH₃, CH₃, Cl, CH₃, CF₃), (M-12413, CH₃, CH₃, Cl, CH₃, Br), (M-12414, CH₃, CH₃, Cl, CH₃, CH₃), (M-12415, CH₃, CH₃, Cl, Et, H), (M-12416, CH₃, CH₃, Cl, Et, Cl), (M-12417, CH₃, CH₃, Cl, Et, F), (M-12418, CH₃, CH₃, Cl, Et, CF₃), (M-12419, CH₃, CH₃, Cl, Et, Br), (M-12420, CH₃, CH₃, Cl, Et, CH₃), (M-12421, CH₃, CH₃, Cl, n-Pr, H), (M-12422, CH₃, CH₃, Cl, n-Pr, Cl), (M-12423, CH₃, CH₃, Cl, n-Pr, F), (M-12424, CH₃, CH₃, Cl, n-Pr, CF₃), (M-12425, CH₃, CH₃, Cl, n-Pr, Br), (M-12426, CH₃, CH₃, Cl, n-Pr, CH₃), (M-12427, CH₃, CH₃, Cl, c-Pr, H), (M-12428, CH₃, CH₃, Cl, c-Pr, Cl), (M-12429, CH₃, CH₃, Cl, c-Pr, F), (M-12430, CH₃, CH₃, Cl, c-Pr, CF₃), (M-12431, CH₃, CH₃, Cl, c-Pr, Br), (M-12432, CH₃, CH₃, Cl, c-Pr, CH₃), (M-12433, CH₃, CH₃, Cl, i-Pr, H), (M-12434, CH₃, CH₃, Cl, i-Pr, Cl), (M-12435, CH₃, CH₃, Cl, i-Pr, F), (M-12436, CH₃, CH₃, Cl, i-Pr, CF₃), (M-12437, CH₃, CH₃, Cl, i-Pr, Br), (M-12438, CH₃, CH₃, Cl, i-Pr, CH₃), (M-12439, CH₃, CH
₃, Cl, n-Bu, H), (M-12440, CH₃, CH₃, Cl, n-Bu, Cl), (M-12441, CH₃, CH₃, Cl, n-Bu, F), (M-12442, CH₃, CH₃, Cl, n-Bu, CF₃), (M-12443, CH₃, CH₃, Cl, n-Bu, Br), (M-12444, CH₃, CH₃, Cl, n-Bu, CH₃), (M-12445, CH₃, CH₃, Cl, i-Bu, H), (M-12446, CH₃, CH₃, Cl, i-Bu, Cl), (M-12447, CH₃, CH₃, Cl, i-Bu, F), (M-12448, CH₃, CH₃, Cl, i-Bu, CF₃), (M-12449, CH₃, CH₃, Cl, i-Bu, Br), (M-12450, CH₃, CH₃, Cl, i-Bu, CH₃), (M-12451, CH₃, CH₃, Cl, sec-Bu, H), (M-12452, CH₃, CH₃, Cl, sec-Bu, Cl), (M-12453, CH₃, CH₃, Cl, sec-Bu, F), (M-12454, CH₃, CH₃, Cl, sec-Bu, CF₃), (M-12455, CH₃, CH₃, Cl, sec-Bu, Br), (M-12456, CH₃, CH₃, Cl, sec-Bu, CH₃), (M-12457, CH₃, CH₃, Cl, n-Pen, H), (M-12458, CH₃, CH₃, Cl, n-Pen, Cl), (M-12459, CH₃, CH₃, Cl, n-Pen, F), (M-12460, CH₃, CH₃, Cl, n-Pen, CF₃), (M-12461, CH₃, CH₃, Cl, n-Pen, Br), (M-12462, CH₃, CH₃, Cl, n-Pen, CH₃), (M-12463, CH₃, CH₃, Cl, c-Pen, H), (M-12464, CH₃, CH₃, Cl, c-Pen, Cl), (M-12465, CH₃, CH₃, Cl, c-Pen, F), (M-12466, CH₃, CH₃, Cl, c-Pen, CF₃), (M-12467, CH₃, CH₃, Cl, c-Pen, Br), (M-12468, CH₃, CH₃, Cl, c-Pen, CH₃), (M-12469, CH₃, CH₃, Cl, n-Hex, H), (M-12470, CH₃, CH₃, Cl, n-Hex, Cl), (M-12471, CH₃, CH₃, Cl, n-Hex, F), (M-12472, CH₃, CH₃, Cl, n-Hex, CF₃), (M-12473, CH₃, CH₃, Cl, n-Hex, Br), (M-12474, CH₃, CH₃, Cl, n-Hex, CH₃), (M-12475, CH₃, CH₃, Cl, c-Hex, H), (M-12476, CH₃, CH₃, Cl, c-Hex, Cl), (M-12477, CH₃, CH₃, Cl, c-Hex, F), (M-12478, CH₃, CH₃, Cl, c-Hex, CF₃), (M-12479, CH₃, CH₃, Cl, c-Hex, Br), (M-12480, CH₃, CH₃, Cl, c-Hex, CH₃), (M-12481, CH₃, CH₃, Cl, OH, H), (M-12482, CH₃, CH₃, Cl, OH, Cl), (M-12483, CH₃, CH₃, Cl, OH, F), (M-12484, CH₃, CH₃, Cl, OH, CF₃), (M-12485, CH₃, CH₃, Cl, OH, Br), (M-12486, CH₃, CH₃, Cl, OH, CH₃), (M-12487, CH₃, CH₃, Cl, EtO, H), (M-12488, CH₃, CH₃, Cl, EtO, Cl), (M-12489, CH₃, CH₃, Cl, EtO, F), (M-12490, CH₃, CH₃, Cl, EtO, CF₃), (M-12491, CH₃, CH₃, Cl, EtO, Br), (M-12492, CH₃, CH₃, Cl, EtO, CH₃), (M-12493, CH₃, CH₃, Cl, n-PrO, H), (M-12494, CH₃, CH₃, Cl, n-PrO, Cl), (M-12495, CH₃, CH₃, Cl, n-PrO, F), (M-12496, CH₃, CH₃, Cl, n-PrO, CF₃), (M-12497, CH₃, CH₃, Cl, n-PrO, Br), (M-12498, CH₃, CH₃, Cl, n-PrO, CH₃), (M-12499, CH₃, CH₃, Cl, PhO, H), (M-12500, CH₃, CH₃, Cl, PhO, Cl), (M-12501, CH₃, CH₃, Cl, PhO, F), (M-12502, CH₃, CH₃, Cl, PhO, CF₃), (M-12503, CH₃, CH₃, Cl, PhO, Br), (M-12504, CH₃, CH₃, Cl, PhO, CH₃), (M-12505, CH₃, CH₃, Cl, BnO, H), (M-12506, CH₃, CH₃, Cl, BnO, Cl), (M-12507, CH₃, CH₃, Cl, BnO, F), (M-12508, CH₃, CH₃, Cl, BnO, CF₃), (M-12509, CH₃, CH₃, Cl, BnO, Br), (M-12510, CH₃, CH₃, Cl, BnO, CH₃), (M-12511, CH₃, CH₃, Cl, PhCH₂CH₂O, H), (M-12512, CH₃, CH₃, Cl, PhCH₂CH₂O, Cl), (M-12513, CH₃, CH₃, Cl, PhCH₂CH₂O, F), (M-12514, CH₃, CH₃, Cl, PhCH₂CH₂O, CF₃), (M-12515, CH₃, CH₃, Cl, PhCH₂CH₂O, Br), (M-12516, CH₃, CH₃, Cl, PhCH₂CH₂O, CH₃), (M-12517, CH₃, CH₃, Cl, CF₃O, H), (M-12518, CH₃, CH₃, Cl, CF₃O, Cl), (M-12519, CH₃, CH₃, Cl, CF₃O, F), (M-12520, CH₃, CH₃, Cl, CF₃O, CF₃), (M-12521, CH₃, CH₃, Cl, CF₃O, Br), (M-12522, CH₃, CH₃, Cl, CF₃O, CH₃), (M-12523, CH₃, CH₃, Cl, Ph, H), (M-12524, CH₃, CH₃, Cl, Ph, Cl), (M-12525, CH₃, CH₃, Cl, Ph, F), (M-12526, CH₃, CH₃, Cl, Ph, CF₃), (M-12527, CH₃, CH₃, Cl, Ph, Br), (M-12528, CH₃, CH₃, Cl, Ph, CH₃), (M-12529, CH₃, CH₃, Cl, 4-F-Ph, H), (M-12530, CH₃, CH₃, Cl, 4-F-Ph, Cl), (M-12531, CH₃, CH₃, Cl, 4-F-Ph, F), (M-12532, CH₃, CH₃, Cl, 4-F-Ph, CF₃), (M-12533, CH₃, CH₃, Cl, 4-F-Ph, Br), (M-12534, CH₃, CH₃, Cl, 4-F-Ph, CH₃), (M-12535, CH₃, CH₃, Cl, 4-CF₃-Ph, H), (M-12536, CH₃, CH₃, Cl, 4-CF₃-Ph, Cl), (M-12537, CH₃, CH₃, Cl, 4-CF₃-Ph, F), (M-12538, CH₃, CH₃, Cl, 4-CF₃-Ph, CF₃), (M-12539, CH₃, CH₃, Cl, 4-CF₃-Ph, Br), (M-12540, CH₃, CH₃, Cl, 4-CF₃-Ph, CH₃), (M-12541, CH₃, CH₃, Cl, 4-(Me)₂N-Ph, H), (M-12542, CH₃, CH₃, Cl, 4-(Me)₂N-Ph, Cl), (M-12543, CH₃, CH₃, Cl, 4-(Me)₂N-Ph, F), (M-12544, CH₃, CH₃, Cl, 4-(Me)₂N-Ph, CF₃), (M-12545, CH₃, CH₃, Cl, 4-(Me)₂N-Ph, Br), (M-12546, CH₃, CH₃, Cl, 4-(Me)₂N-Ph, CH₃), (M-12547, CH₃, CH₃, Cl, 4-OH-Ph, H), (M-12548, CH₃, CH₃, Cl, 4-OH-Ph, Cl), (M-12549, CH₃, CH₃, Cl, 4-OH-Ph, F), (M-12550, CH₃, CH₃, Cl, 4-OH-Ph, CF₃), (M-12551, CH₃, CH₃, Cl, 4-OH-Ph, Br), (M-12552, CH₃, CH₃, Cl, 4-OH-Ph, CH₃), (M-12553, CH₃, CH₃, Cl, 3,4-di-F-Ph, H), (M-12554, CH₃, CH₃, Cl, 3,4-di-F-Ph, Cl), (M-12555, CH₃, CH₃, Cl, 3,4-di-F-Ph, F), (M-12556, CH₃, CH₃, Cl, 3,4-di-F-Ph, CF₃), (M-12557, CH₃, CH₃, Cl, 3,4-di-F-Ph, Br), (M-12558, CH₃, CH₃, Cl, 3,4-di-F-Ph, CH₃), (M-12559, CH₃, CH₃, Cl, 4-COOH-Ph, H), (M-12560, CH₃, CH₃, Cl, 4-COOH-Ph, Cl), (M-12561, CH₃, CH₃, Cl, 4-COOH-Ph, F), (M-12562, CH₃, CH₃, Cl, 4-COOH-Ph, CF₃), (M-12563, CH₃, CH₃, Cl, 4-COOH-Ph, Br), (M-12564, CH₃, CH₃, Cl, 4-COOH-Ph, CH₃), (M-12565, CH₃, CH₃, Cl, Bn, H), (M-12566, CH₃, CH₃, Cl, Bn, Cl), (M-12567, CH₃, CH₃, Cl, Bn, F), (M-12568, CH₃, CH₃, Cl, Bn, CF₃), (M-12569, CH₃, CH₃, Cl, Bn, Br), (M-12570, CH₃, CH₃, Cl, Bn, CH₃), (M-12571, CH₃, CH₃, Cl, 4-F-Bn, H), (M-12572, CH₃, CH₃, Cl, 4-F-Bn, Cl), (M-12573, CH₃, CH₃, Cl, 4-F-Bn, F), (M-12574, CH₃, CH₃, Cl, 4-F-Bn, CF₃), (M-12575, CH₃, CH₃, Cl, 4-F-Bn, Br), (M-12576, CH₃, CH₃, Cl, 4-F-Bn, CH₃), (M-12577, CH₃, CH₃, Cl, 2-Py, H), (M-12578, CH₃, CH₃, Cl, 2-Py, Cl), (M-12579, CH₃, CH₃, Cl, 2-Py, F), (M-12580, CH₃, CH₃, Cl, 2-Py, CF₃), (M-12581, CH₃, CH₃, Cl, 2-Py, Br), (M-12582, CH₃, CH₃, Cl, 2-Py, CH₃), (M-12583, CH₃, CH₃, Cl, 3-Py, H), (M-12584, CH₃, CH₃, Cl, 3-Py, Cl), (M-12585, CH₃, CH₃, Cl, 3-Py, F), (M-12586, CH₃, CH₃, Cl, 3-Py, CF₃), (M-12587, CH₃, CH₃, Cl, 3-Py, Br), (M-12588, CH₃, CH₃, Cl, 3-Py, CH₃), (M-12589, CH₃, CH₃, Cl, 4-Py, H), (M-12590, CH₃, CH₃, Cl, 4-Py, Cl), (M-12591, CH₃, CH₃, Cl, 4-Py, F), (M-12592, CH₃, CH₃, Cl, 4-Py, CF₃), (M-12593, CH₃, CH₃, Cl, 4-Py, Br), (M-12594, CH₃, CH₃, Cl, 4-Py, CH₃), (M-12595, CH₃, CH₃, Cl, 2-Th, H), (M-12596, CH₃, CH₃, Cl, 2-Th, Cl), (M-12597, CH₃, CH₃, Cl, 2-Th, F), (M-12598, CH₃, CH₃, Cl, 2-Th, CF₃), (M-12599, CH₃, CH₃, Cl
, 2-Th, Br), (M-12600, CH₃, CH₃, Cl, 2-Th, CH₃), (M-12601, CH₃, CH₃, Cl, 3-Th, H), (M-12602, CH₃, CH₃, Cl, 3-Th, Cl), (M-12603, CH₃, CH₃, Cl, 3-Th, F), (M-12604, CH₃, CH₃, Cl, 3-Th, CF₃), (M-12605, CH₃, CH₃, Cl, 3-Th, Br), (M-12606, CH₃, CH₃, Cl, 3-Th, CH₃), (M-12607, CH₃, CH₃, Cl, pyrazol-2-yl, H), (M-12608, CH₃, CH₃, Cl, pyrazol-2-yl, Cl), (M-12609, CH₃, CH₃, Cl, pyrazol-2-yl, F), (M-12610, CH₃, CH₃, Cl, pyrazol-2-yl, CF₃), (M-12611, CH₃, CH₃, Cl, pyrazol-2-yl, Br), (M-12612, CH₃, CH₃, Cl, pyrazol-2-yl, CH₃), (M-12613, CH₃, CH₃, Cl, pyrazol-3-yl, H), (M-12614, CH₃, CH₃, Cl, pyrazol-3-yl, Cl), (M-12615, CH₃, CH₃, Cl, pyrazol-3-yl, F), (M-12616, CH₃, CH₃, Cl, pyrazol-3-yl, CF₃), (M-12617, CH₃, CH₃, Cl, pyrazol-3-yl, Br), (M-12618, CH₃, CH₃, Cl, pyrazol-3-yl, CH₃), (M-12619, CH₃, CH₃, Cl, pyrimidin-2-yl, H), (M-12620, CH₃, CH₃, Cl, pyrimidin-2-yl, Cl), (M-12621, CH₃, CH₃, Cl, pyrimidin-2-yl, F), (M-12622, CH₃, CH₃, Cl, pyrimidin-2-yl, CF₃), (M-12623, CH₃, CH₃, Cl, pyrimidin-2-yl, Br), (M-12624, CH₃, CH₃, Cl, pyrimidin-2-yl, CH₃), (M-12625, CH₃, CH₃, Cl, pyrimidin-4-yl, H), (M-12626, CH₃, CH₃, Cl, pyrimidin-4-yl, Cl), (M-12627, CH₃, CH₃, Cl, pyrimidin-4-yl, F), (M-12628, CH₃, CH₃, Cl, pyrimidin-4-yl, CF₃), (M-12629, CH₃, CH₃, Cl, pyrimidin-4-yl, Br), (M-12630, CH₃, CH₃, Cl, pyrimidin-4-yl, CH₃), (M-12631, CH₃, CH₃, Cl, pyrimidin-5-yl, H), (M-12632, CH₃, CH₃, Cl, pyrimidin-5-yl, Cl), (M-12633, CH₃, CH₃, Cl, pyrimidin-5-yl, F), (M-12634, CH₃, CH₃, Cl, pyrimidin-5-yl, CF₃), (M-12635, CH₃, CH₃, Cl, pyrimidin-5-yl, Br), (M-12636, CH₃, CH₃, Cl, pyrimidin-5-yl, CH₃), (M-12637, CH₃, CH₃, Cl, HOOCCH₂CH₂CH₂, H), (M-12638, CH₃, CH₃, Cl, HOOCCH₂CH₂CH₂, Cl), (M-12639, CH₃, CH₃, Cl, HOOCCH₂CH₂CH₂, F), (M-12640, CH₃, CH₃, Cl, HOOCCH₂CH₂CH₂, CF₃), (M-12641, CH₃, CH₃, Cl, HOOCCH₂CH₂CH₂, Br), (M-12642, CH₃, CH₃, Cl, HOOCCH₂CH₂CH₂, CH₃), (M-12643, CH₃, CH₃, Cl, HOOCCH₂CH₂CH₂CH₂, H), (M-12644, CH₃, CH₃, Cl, HOOCCH₂CH₂CH₂CH₂, Cl), (M-12645, CH₃, CH₃, Cl, HOOCCH₂CH₂CH₂CH₂, F), (M-12646, CH₃, CH₃, Cl, HOOCCH₂CH₂CH₂CH₂, CF₃), (M-12647, CH₃, CH₃, Cl, HOOCCH₂CH₂CH₂CH₂, Br), (M-12648, CH₃, CH₃, Cl, HOOCCH₂CH₂CH₂CH₂, CH₃), (M-12649, CH₃, CH₃, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂, H), (M-12650, CH₃, CH₃, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂, Cl), (M-12651, CH₃, CH₃, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂, F), (M-12652, CH₃, CH₃, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂, CF₃), (M-12653, CH₃, CH₃, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂, Br), (M-12654, CH₃, CH₃, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂, CH₃), (M-12655, CH₃, CH₃, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, H), (M-12656, CH₃, CH₃, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, Cl), (M-12657, CH₃, CH₃, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, F), (M-12658, CH₃, CH₃, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, CF₃), (M-12659, CH₃, CH₃, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, Br), (M-12660, CH₃, CH₃, Cl, (Me)₂NCOCH₂CH₂CH₂CH₂CH₂, CH₃), (M-12661, CH₃, CH₃, Cl, MeOCH₂, H), (M-12662, CH₃, CH₃, Cl, MeOCH₂, Cl), (M-12663, CH₃, CH₃, Cl, MeOCH₂, F), (M-12664, CH₃, CH₃, Cl, MeOCH₂, CF₃), (M-12665, CH₃, CH₃, Cl, MeOCH₂, Br), (M-12666, CH₃, CH₃, Cl, MeOCH₂, CH₃), (M-12667, CH₃, CH₃, Cl, EtOCH₂, H), (M-12668, CH₃, CH₃, Cl, EtOCH₂, Cl), (M-12669, CH₃, CH₃, Cl, EtOCH₂, F), (M-12670, CH₃, CH₃, Cl, EtOCH₂, CF₃), (M-12671, CH₃, CH₃, Cl, EtOCH₂, Br), (M-12672, CH₃, CH₃, Cl, EtOCH₂, CH₃), (M-12673, CH₃, CH₃, Cl, EtOCH₂CH₂, H), (M-12674, CH₃, CH₃, Cl, EtOCH₂CH₂, Cl), (M-12675, CH₃, CH₃, Cl, EtOCH₂CH₂, F), (M-12676, CH₃, CH₃, Cl, EtOCH₂CH₂, CF₃), (M-12677, CH₃, CH₃, Cl, EtOCH₂CH₂, Br), (M-12678, CH₃, CH₃, Cl, EtOCH₂CH₂, CH₃), (M-12679, CH₃, CH₃, Cl, MeOCH₂CH₂OCH₂CH₂, H), (M-12680, CH₃, CH₃, Cl, MeOCH₂CH₂OCH₂CH₂, Cl), (M-12681, CH₃, CH₃, Cl, MeOCH₂CH₂OCH₂CH₂, F), (M-12682, CH₃, CH₃, Cl, MeOCH₂CH₂OCH₂CH₂, CF₃), (M-12683, CH₃, CH₃, Cl, MeOCH₂CH₂OCH₂CH₂, Br), (M-12684, CH₃, CH₃, Cl, MeOCH₂CH₂OCH₂CH₂, CH₃), (M-12685, CH₃, CH₃, Cl, MeOCH₂CH₂, H), (M-12686, CH₃, CH₃, Cl, MeOCH₂CH₂, Cl), (M-12687, CH₃, CH₃, Cl, MeOCH₂CH₂, F), (M-12688, CH₃, CH₃, Cl, MeOCH₂CH₂, CF₃), (M-12689, CH₃, CH₃, Cl, MeOCH₂CH₂, Br), (M-12690, CH₃, CH₃, Cl, MeOCH₂CH₂, CH₃), (M-12691, CH₃, CH₃, Cl, HOCH₂, H), (M-12692, CH₃, CH₃, Cl, HOCH₂, Cl), (M-12693, CH₃, CH₃, Cl, HOCH₂, F), (M-12694, CH₃, CH₃, Cl, HOCH₂, CF₃), (M-12695, CH₃, CH₃, Cl, HOCH₂, Br), (M-12696, CH₃, CH₃, Cl, HOCH₂, CH₃), (M-12697, CH₃, CH₃, Cl, HOCH₂CH₂, H), (M-12698, CH₃, CH₃, Cl, HOCH₂CH₂, Cl), (M-12699, CH₃, CH₃, Cl, HOCH₂CH₂, F), (M-12700, CH₃, CH₃, Cl, HOCH₂CH₂, CF₃), (M-12701, CH₃, CH₃, Cl, HOCH₂CH₂, Br), (M-12702, CH₃, CH₃, Cl, HOCH₂CH₂, CH₃), (M-12703, CH₃, CH₃, Cl, HOCH₂CH₂CH₂, H), (M-12704, CH₃, CH₃, Cl, HOCH₂CH₂CH₂, Cl), (M-12705, CH₃, CH₃, Cl, HOCH₂CH₂CH₂, F), (M-12706, CH₃, CH₃, Cl, HOCH₂CH₂CH₂, CF₃), (M-12707, CH₃, CH₃, Cl, HOCH₂CH₂CH₂, Br), (M-12708, CH₃, CH₃, Cl, HOCH₂CH₂CH₂, CH₃), (M-12709, CH₃, CH₃, Cl, HOCH₂CH₂CH₂CH₂, H), (M-12710, CH₃, CH₃, Cl, HOCH₂CH₂CH₂CH₂, Cl), (M-12711, CH₃, CH₃, Cl, HOCH₂CH₂CH₂CH₂, F), (M-12712, CH₃, CH₃, Cl, HOCH₂CH₂CH₂CH₂, CF₃), (M-12713, CH₃, CH₃, Cl, HOCH₂CH
₂CH₂CH₂, Br), (M-12714, CH₃, CH₃, Cl, HOCH₂CH₂CH₂CH₂, CH₃), (M-12715, CH₃, CH₃, Cl, HOCH₂CH₂CH₂CH₂CH₂, H), (M-12716, CH₃, CH₃, Cl, HOCH₂CH₂CH₂CH₂CH₂, Cl), (M-12717, CH₃, CH₃, Cl, HOCH₂CH₂CH₂CH₂CH₂, F), (M-12718, CH₃, CH₃, Cl, HOCH₂CH₂CH₂CH₂CH₂, CF₃), (M-12719, CH₃, CH₃, Cl, HOCH₂CH₂CH₂CH₂CH₂, Br), (M-12720, CH₃, CH₃, Cl, HOCH₂CH₂CH₂CH₂CH₂, CH₃), (M-12721, CH₃, CH₃, Cl, HOCH₂CH₂OCH₂CH₂, H), (M-12722, CH₃, CH₃, Cl, HOCH₂CH₂OCH₂CH₂, Cl), (M-12723, CH₃, CH₃, Cl, HOCH₂CH₂OCH₂CH₂, F), (M-12724, CH₃, CH₃, Cl, HOCH₂CH₂OCH₂CH₂, CF₃), (M-12725, CH₃, CH₃, Cl, HOCH₂CH₂OCH₂CH₂, Br), (M-12726, CH₃, CH₃, Cl, HOCH₂CH₂OCH₂CH₂, CH₃), (M-12727, CH₃, CH₃, Cl, (Me)₂N, H), (M-12728, CH₃, CH₃, Cl, (Me)₂N, Cl), (M-12729, CH₃, CH₃, Cl, (Me)₂N, F), (M-12730, CH₃, CH₃, Cl, (Me)₂N, CF₃), (M-12731, CH₃, CH₃, Cl, (Me)₂N, Br), (M-12732, CH₃, CH₃, Cl, (Me)₂N, CH₃), (M-12733, CH₃, CH₃, Cl, piperidin-4-yl-methyl, H), (M-12734, CH₃, CH₃, Cl, piperidin-4-yl-methyl, Cl), (M-12735, CH₃, CH₃, Cl, piperidin-4-yl-methyl, F), (M-12736, CH₃, CH₃, Cl, piperidin-4-yl-methyl, CF₃), (M-12737, CH₃, CH₃, Cl, piperidin-4-yl-methyl, Br), (M-12738, CH₃, CH₃, Cl, piperidin-4-yl-methyl, CH₃), (M-12739, CH₃, CH₃, Cl, cyclohexylmethyl, H), (M-12740, CH₃, CH₃, Cl, cyclohexylmethyl, Cl), (M-12741, CH₃, CH₃, Cl, cyclohexylmethyl, F), (M-12742, CH₃, CH₃, Cl, cyclohexylmethyl, CF₃), (M-12743, CH₃, CH₃, Cl, cyclohexylmethyl, Br), (M-12744, CH₃, CH₃, Cl, cyclohexylmethyl, CH₃), (M-12745, H, H, H, CF₃, H), (M-12746, H, H, H, CF₃, Cl), (M-12747, H, H, H, CF₃, F), (M-12748, H, H, H, CF₃, CF₃), (M-12749, H, H, H, CF₃, Br), (M-12750, H, H, H, CF₃, CH₃), (M-12751, H, H, F, CF₃, H), (M-12752, H, H, F, CF₃, Cl), (M-12753, H, H, F, CF₃, F), (M-12754, H, H, F, CF₃, CF₃), (M-12755, H, H, F, CF₃, Br), (M-12756, H, H, F, CF₃, CH₃), (M-12757, H, H, Cl, CF₃, H), (M-12758, H, H, Cl, CF₃, Cl), (M-12759, H, H, Cl, CF₃, F), (M-12760, H, H, Cl, CF₃, CF₃), (M-12761, H, H, Cl, CF₃, Br), (M-12762, H, H, Cl, CF₃, CH₃), (M-12763, H, F, H, CF₃, H), (M-12764, H, F, H, CF₃, Cl), (M-12765, H, F, H, CF₃, F), (M-12766, H, F, H, CF₃, CF₃), (M-12767, H, F, H, CF₃, Br), (M-12768, H, F, H, CF₃, CH₃), (M-12769, H, F, F, CF₃, H), (M-12770, H, F, F, CF₃, Cl), (M-12771, H, F, F, CF₃, F), (M-12772, H, F, F, CF₃, CF₃), (M-12773, H, F, F, CF₃, Br), (M-12774, H, F, F, CF₃, CH₃), (M-12775, H, F, Cl, CF₃, H), (M-12776, H, F, Cl, CF₃, Cl), (M-12777, H, F, Cl, CF₃, F), (M-12778, H, F, Cl, CF₃, CF₃), (M-12779, H, F, Cl, CF₃, Br), (M-12780, H, F, Cl, CF₃, CH₃), (M-12781, H, CH₃, H, CF₃, H), (M-12782, H, CH₃, H, CF₃, Cl), (M-12783, H, CH₃, H, CF₃, F), (M-12784, H, CH₃, H, CF₃, CF₃), (M-12785, H, CH₃, H, CF₃, Br), (M-12786, H, CH₃, H, CF₃, CH₃), (M-12787, H, CH₃, F, CF₃, H), (M-12788, H, CH₃, F, CF₃, Cl), (M-12789, H, CH₃, F, CF₃, F), (M-12790, H, CH₃, F, CF₃, CF₃), (M-12791, H, CH₃, F, CF₃, Br), (M-12792, H, CH₃, F, CF₃, CH₃), (M-12793, H, CH₃, Cl, CF₃, H), (M-12794, H, CH₃, Cl, CF₃, Cl), (M-12795, H, CH₃, Cl, CF₃, F), (M-12796, H, CH₃, Cl, CF₃, CF₃), (M-12797, H, CH₃, Cl, CF₃, Br), (M-12798, H, CH₃, Cl, CF₃, CH₃), (M-12799, F, H, H, CF₃, i-Pr), (M-12800, F, H, H, CF₃, Cl), (M-12801, F, H, H, CF₃, F), (M-12802, F, H, H, CF₃, CF₃), (M-12803, F, H, H, CF₃, Br), (M-12804, F, H, H, CF₃, CH₃), (M-12805, F, H, F, CF₃, H), (M-12806, F, H, F, CF₃, Cl), (M-12807, F, H, F, CF₃, F), (M-12808, F, H, F, CF₃, CF₃), (M-12809, F, H, F, CF₃, Br), (M-12810, F, H, F, CF₃, CH₃), (M-12811, F, H, Cl, CF₃, H), (M-12812, F, H, Cl, CF₃, Cl), (M-12813, F, H, Cl, CF₃, F), (M-12814, F, H, Cl, CF₃, CF₃), (M-12815, F, H, Cl, CF₃, Br), (M-12816, F, H, Cl, CF₃, CH₃), (M-12817, F, F, H, CF₃, H), (M-12818, F, F, H, CF₃, Cl), (M-12819, F, F, H, CF₃, F), (M-12820, F, F, H, CF₃, CF₃), (M-12821, F, F, H, CF₃, Br), (M-12822, F, F, H, CF₃, CH₃), (M-12823, F, F, F, CF₃, H), (M-12824, F, F, F, CF₃, Cl), (M-12825, F, F, F, CF₃, F), (M-12826, F, F, F, CF₃, CF₃), (M-12827, F, F, F, CF₃, Br), (M-12828, F, F, F, CF₃, CH₃), (M-12829, F, F, Cl, CF₃, H), (M-12830, F, F, Cl, CF₃, Cl), (M-12831, F, F, Cl, CF₃, F), (M-12832, F, F, Cl, CF₃, CF₃), (M-12833, F, F, Cl, CF₃, Br), (M-12834, F, F, Cl, CF₃, CH₃), (M-12835, F, CH₃, H, CF₃, H), (M-12836, F, CH₃, H, CF₃, Cl), (M-12837, F, CH₃, H, CF₃, F), (M-12838, F, CH₃, H, CF₃, CF₃), (M-12839, F, CH₃, H, CF₃, Br), (M-12840, F, CH₃, H, CF₃, CH₃), (M-12841, F, CH₃, F, CF₃, H), (M-12842, F, CH₃, F, CF₃, Cl), (M-12843, F, CH₃, F, CF₃, F), (M-12844, F, CH₃, F, CF₃, CF₃), (M-12845, F, CH₃, F, CF₃, Br), (M-12846, F, CH₃, F, CF₃, CH₃), (M-12847, F, CH₃, Cl, CF₃, H), (M-12848, F, CH₃, Cl, CF₃, Cl), (M-12849, F, CH₃, Cl, CF₃, F), (M-12850, F, CH₃, Cl, CF₃, CF₃), (M-12851, F, CH₃, Cl, CF₃, Br), (M-12852, F, CH₃, Cl, CF₃, CH₃), (M-12853, Cl, H, H, CF₃, i-Pr), (M-12854, Cl, H, H, CF₃, Cl), (M-12855, Cl, H, H, CF₃, F), (M-12856, Cl, H, H, CF₃, CF₃), (M-12857, Cl, H, H, CF₃, Br), (M-12858, Cl, H, H, CF₃, CH₃), (M-12859, Cl, H, F, CF₃, i-Pr), (M-12860, Cl, H, F, CF₃, Cl), (M-12861, Cl, H, F, CF₃, F), (M-12862, Cl, H, F, CF₃, CF₃), (M-12863, Cl, H, F, CF₃, Br), (M-12864, Cl, H, F, CF₃, CH₃), (M-12865, Cl, H, Cl, CF₃, H), (M-12866, Cl, H, Cl, CF₃, Cl), (M-12867, Cl, H, Cl, CF₃, F), (M-12868, Cl, H, Cl, CF₃, CF₃), (M-12869, Cl, H, Cl, CF₃, Br), (M-12870, Cl, H, Cl, CF₃, CH₃), (M-12871, Cl, F, H, CF₃, i-Pr), (M-12872, Cl, F, H, CF₃, Cl), (M-12873, Cl, F, H, CF₃, F), (M-12874, Cl, F, H, CF₃, CF₃), (M-12875, Cl, F, H, CF₃, Br), (M-12876, Cl, F, H, CF₃, CH₃), (M-12877, Cl, F, F, CF₃, H), (M-12878, Cl, F, F, CF₃, Cl), (M-12879, Cl, F, F, CF₃, F), (M-12880, Cl, F, F, CF₃, CF₃), (M-12881, Cl, F, F, CF₃, Br), (M-12882, Cl, F, F, CF₃, CH₃), (M-12883, Cl, F, Cl, CF₃, H), (M-12884, Cl, F, Cl, CF₃, Cl), (M-12885, Cl, F, Cl, CF₃, F), (M-12886, Cl, F, Cl, CF₃, CF₃), (M-12887, Cl, F, Cl, CF₃, Br), (M-12888, Cl, F, Cl, CF₃, CH₃), (M-12889, Cl, CH₃, H, CF₃, i-Pr), (M-12890, Cl, CH₃, H, CF₃, Cl), (M-12891, Cl, CH₃, H, CF₃, F), (M-12892, Cl, CH₃, H, CF₃, CF₃), (M-12893, Cl, CH₃, H, CF₃, Br), (M-12894, Cl, CH₃, H, CF₃, CH₃), (M-12895, Cl, CH₃, F, CF₃, i-Pr), (M-12896,
Cl, CH₃, F, CF₃, Cl), (M-12897, Cl, CH₃, F, CF₃, F), (M-12898, Cl, CH₃, F, CF₃, CF₃), (M-12899, Cl, CH₃, F, CF₃, Br), (M-12900, Cl, CH₃, F, CF₃, CH₃), (M-12901, Cl, CH₃, Cl, CF₃, H), (M-12902, Cl, CH₃, Cl, CF₃, Cl), (M-12903, Cl, CH₃, Cl, CF₃, F), (M-12904, Cl, CH₃, Cl, CF₃, CF₃), (M-12905, Cl, CH₃, Cl, CF₃, Br), (M-12906, Cl, CH₃, Cl, CF₃, CH₃), (M-12907, CH₃, H, H, CF₃, i-Pr), (M-12908, CH₃, H, H, CF₃, Cl), (M-12909, CH₃, H, H, CF₃, F), (M-12910, CH₃, H, H, CF₃, CF₃), (M-12911, CH₃, H, H, CF₃, Br), (M-12912, CH₃, H, H, CF₃, CH₃), (M-12913, CH₃, H, F, CF₃, H), (M-12914, CH₃, H, F, CF₃, Cl), (M-12915, CH₃, H, F, CF₃, F), (M-12916, CH₃, H, F, CF₃, CF₃), (M-12917, CH₃, H, F, CF₃, Br), (M-12918, CH₃, H, F, CF₃, CH₃), (M-12919, CH₃, H, Cl, CF₃, H), (M-12920, CH₃, H, Cl, CF₃, Cl), (M-12921, CH₃, H, Cl, CF₃, F), (M-12922, CH₃, H, Cl, CF₃, CF₃), (M-12923, CH₃, H, Cl, CF₃, Br), (M-12924, CH₃, H, Cl, CF₃, CH₃), (M-12925, CH₃, F, H, CF₃, H), (M-12926, CH₃, F, H, CF₃, Cl), (M-12927, CH₃, F, H, CF₃, F), (M-12928, CH₃, F, H, CF₃, CF₃), (M-12929, CH₃, F, H, CF₃, Br), (M-12930, CH₃, F, H, CF₃, CH₃), (M-12931, CH₃, F, F, CF₃, H), (M-12932, CH₃, F, F, CF₃, Cl), (M-12933, CH₃, F, F, CF₃, F), (M-12934, CH₃, F, F, CF₃, CF₃), (M-12935, CH₃, F, F, CF₃, Br), (M-12936, CH₃, F, F, CF₃, CH₃), (M-12937, CH₃, F, Cl, CF₃, H), (M-12938, CH₃, F, Cl, CF₃, Cl), (M-12939, CH₃, F, Cl, CF₃, F), (M-12940, CH₃, F, Cl, CF₃, CF₃), (M-12941, CH₃, F, Cl, CF₃, Br), (M-12942, CH₃, F, Cl, CF₃, CH₃), (M-12943, CH₃, CH₃, H, CF₃, H), (M-12944, CH₃, CH₃, H, CF₃, Cl), (M-12945, CH₃, CH₃, H, CF₃, F), (M-12946, CH₃, CH₃, H, CF₃, CF₃), (M-12947, CH₃, CH₃, H, CF₃, Br), (M-12948, CH₃, CH₃, H, CF₃, CH₃), (M-12949, CH₃, CH₃, F, CF₃, H), (M-12950, CH₃, CH₃, F, CF₃, Cl), (M-12951, CH₃, CH₃, F, CF₃, F), (M-12952, CH₃, CH₃, F, CF₃, CF₃), (M-12953, CH₃, CH₃, F, CF₃, Br), (M-12954, CH₃, CH₃, F, CF₃, CH₃), (M-12955, CH₃, CH₃, Cl, CF₃, H), (M-12956, CH₃, CH₃, Cl, CF₃, Cl), (M-12957, CH₃, CH₃, Cl, CF₃, F), (M-12958, CH₃, CH₃, Cl, CF₃, CF₃), (M-12959, CH₃, CH₃, Cl, CF₃, Br), (M-12960, CH₃, CH₃, Cl, CF₃, CH₃).

試験例

試験例１トロンボポエチン（TPO）の単離と精製
ヒトおよびマウスTPOは、R&D Systems社より購入した。

試験例２化合物(B-1)によるin vitro巨核球コロニー増加作用
本化合物の巨核球系細胞の増殖・分化・成熟に対する作用を、ヒト骨髄細胞を用い、メチルセルロースの半固形培養で巨核球コロニー形成法で調べた。ヒト骨髄細胞2.2x10⁵個を3 cmシャーレに播種し、10%エタノールに溶解した化合物を1%添加して37℃、5% CO₂存在下で7日間培養し、巨核球コロニー数を測定した。その結果を図1に示す。

試験例３化合物(B-1)のTPO受容体応答性
本化合物のTPO受容体応答性を、コリンスらのJ. Cell. Physiol., 137: 293-298 (1988)に記載されている方法に準じてヒトTPO受容体遺伝子をBaF-B03細胞に導入して作成した、TPO依存性細胞株BaF/hTPORを用いて測定した。トロンボポエチン受容体をコードする遺伝子の塩基配列は、ビゴンらのProc. Natl. Acad. Sci. 89:5640-5644 (1992)に記載されている。なお親株であるBaF-B03細胞にはTPOは応答しない。10%WEHI-3培養液を添加したRPMI培地にて増殖させたBAF/hTPOR細胞をPBSで1回洗浄後、WHEHI-3培養液を添加していないRPMI培地に懸濁し、96穴マイクロプレートに細胞を5x10⁴/ウェルになるように播種して、本化合物あるいはTPOを添加した。5%CO₂雰囲気下で37℃、20時間培養した後に、細胞増殖判定試薬であるWST-1試薬（宝酒造社製）を添加し、4時間後に450nmの吸収を測定した。その結果を図２に示す。また、同様の手法を用いて作成したマウスTPO受容体を発現するBaF/mTPOR細胞の応答性を調べた結果を図３に示す。ＥＤ_５０値をヒトＴＰＯの半最大応答性を示す化合物の濃度とし、それぞれの化合物のＥＤ_５０値を表３３に示した。

図１に示したように、本化合物添加により単独で巨核球コロニーが形成され、コロニー数は濃度依存的に増加した。以上の結果、本化合物は単独で巨核球前駆細胞の増殖・分化を促進し血小板産生能を有する巨核球を産生させることが明らかとなった。
図２に示したように、本化合物は濃度依存的にTPO依存性細胞株BaF/hTPOR細胞を増殖させた。図３に示したように、本化合物は、マウスTPO受容体を発現させたBaF/mTPOR細胞には応答しなかった。以上の結果より、本化合物がヒトTPO受容体に特異的に作用し、TPOアゴニストとして作用していることが明らかとなった。

製剤例

製剤例１
以下の成分を含有する顆粒剤を製造する。
成分式（Ｉ）で表わされる化合物 10 mg
乳糖 700 mg
コーンスターチ 274 mg
HPC-L 16 mg
1000 mg
式（Ｉ）で表わされる化合物と乳糖を６０メッシュのふるいに通す。コーンスターチを１２０メッシュのふるいに通す。これらをV型混合機にて混合する。混合末にＨＰＣ−Ｌ（低粘度ヒドロキシプロピルセルロース）水溶液を添加し、練合、造粒（押し出し造粒孔径０．５〜１ｍｍ）したのち、乾燥する。得られた乾燥顆粒を振動ふるい（１２／６０メッシュ）で櫛過し顆粒剤を得る。
製剤例２
以下の成分を含有するカプセル充填用散剤を製造する。
成分式（Ｉ）で表わされる化合物 10 mg
乳糖 79 mg
コーンスターチ 10 mg
ステアリン酸マグネシウム 1 mg
100 mg
式（Ｉ）で表わされる化合物、乳糖を６０メッシュのふるいに通す。コーンスターチは１２０メッシュのふるいに通す。これらとステアリン酸マグネシウムをV型混合機にて混合する。１０倍散１００ｍｇを５号硬ゼラチンカプセルに充填する。
製剤例３
以下の成分を含有するカプセル充填用顆粒剤を製造する。
成分式（Ｉ）で表わされる化合物 15 mg
乳糖 90 mg
コーンスターチ 42 mg
HPC-L 3 mg
150 mg
式（Ｉ）で表わされる化合物、乳糖を６０メッシュのふるいに通す。コーンスターチを１２０メッシュのふるいに通す。これらを混合し、混合末にＨＰＣ−Ｌ溶液を添加して練合、造粒、乾燥する。得られた乾燥顆粒を整粒後、その１５０ｍｇを４号硬ゼラチンカプセルに充填する。
製剤例４
以下の成分を含有する錠剤を製造する。
成分式（Ｉ）で表わされる化合物 10 mg
乳糖 90 mg
微結晶セルロース 30 mg
CMC-Na 15 mg
ステアリン酸マグネシウム 5 mg
150 mg
式（Ｉ）で表わされる化合物、乳糖、微結晶セルロース、ＣＭＣ−Ｎａ（カルボキシメチルセルロースナトリウム塩）を６０メッシュのふるいに通し、混合する。混合末にステアリン酸マグネシウム混合し、製錠用混合末を得る。本混合末を直打し、１５０ｍｇの錠剤を得る。
製剤例５
静脈用製剤は次のように製造する：
式（Ｉ）で表わされる化合物１００ｍｇ
飽和脂肪酸グリセリド１０００ｍｌ
上記成分の溶液は通常、１分間に１ｍｌの速度で患者に静脈内投与される。

本発明化合物は、トロンボポエチンアゴニスト作用を有し、血小板減少症等の血小板数の異常を伴う血液疾患の治療または予防剤として有効に機能し得ることを見出した。

本発明化合物によりヒト骨髄細胞より形成される巨核球コロニー数を測定し、本発明化合物の巨核球前駆細胞の増殖・分化促進作用を示したグラフである。横軸に本発明化合物の濃度、縦軸に細胞増殖の指標とした吸光度をとり、本発明化合物によるヒトTPO受容体を発現したヒトTPO依存性細胞株の細胞増殖を示したグラフである。白丸はヒトTPOによる応答を、黒丸は化合物(B-1)による応答を示している。横軸に本発明化合物の濃度、縦軸に細胞増殖の指標とした吸光度をとり、本発明化合物によるマウスTPO受容体を発現したマウスTPO依存性細胞株の細胞増殖を示したグラフである。三角はマウスTPOによる応答を、黒丸は化合物(B-1)による応答を示している。

Claims

一般式（Ｉ）：

［式中、Ｘ^１は置換されていてもよいアリール、置換されていてもよいアラルキル、置換されていてもよいヘテロアリール、または置換されていてもよいヘテロアリールアルキル；
Ｙ^１は−ＮＲ^ＡＣＯ−（ＣＲ^ＣＲ^Ｄ）_０−２−、−ＮＲ^ＡＣＯ−（ＣＨ_２）_０−２−Ｖ−、−ＮＲ^ＡＣＯ−ＣＲ^Ｃ＝ＣＲ^Ｄ−、−Ｖ−（ＣＨ_２）_１−５−ＮＲ^ＡＣＯ−（ＣＨ_２）_０−２−、−Ｖ−（ＣＨ_２）_１−５−ＣＯＮＲ^Ａ−（ＣＨ_２）_０−２−、−ＣＯＮＲ^Ａ−（ＣＨ_２）_０−２−、−（ＣＨ_２）_０−２−ＮＲ^Ａ−ＳＯ_２−（ＣＨ_２）_０−２−、−（ＣＨ_２）_０−２−ＳＯ_２−ＮＲ^Ａ−（ＣＨ_２）_０−２−、−ＮＲ^Ａ−（ＣＨ_２）_０−２−、−ＮＲ^Ａ−ＣＯ−ＮＲ^Ａ−、−ＮＲ^Ａ−ＣＳ−ＮＲ^Ａ−、−Ｎ＝Ｃ（−ＳＲ^Ａ）−ＮＲ^Ａ−、−ＮＲ^ＡＣＳＮＲ^ＡＣＯ−、−Ｎ＝Ｃ（−ＳＲ^Ａ）−ＮＲ^ＡＣＯ−、−ＮＲ^Ａ−（ＣＨ_２）_１−２−ＮＲ^Ａ−ＣＯ−、−ＮＲ^ＡＣＯＮＲ^ＡＮＲ^ＢＣＯ−、または−Ｎ＝Ｃ（−ＮＲ^ＡＲ^Ａ）−ＮＲ^ＡＣＯ−（式中、Ｒ^Ａはそれぞれ独立して水素原子または低級アルキル；Ｒ^Ｂは水素原子またはフェニル；Ｒ^ＣおよびＲ^Ｄはそれぞれ独立して、水素原子、ハロゲン、置換されていてもよい低級アルキル、置換されていてもよい低級アルキルオキシ、置換されていてもよい低級アルキルチオ、置換されていてもよい低級アルケニル、置換されていてもよい低級アルキニル、置換されていてもよいアリール、置換されていてもよいヘテロアリール、置換されていてもよいシクロアルキル、置換されていてもよいアラルキル、置換されていてもよいヘテロアリールアルキル、置換されていてもよい非芳香族複素環基、または置換されていてもよいアミノ；Ｖは酸素原子または硫黄原子）；
Ｚ^１は置換されていてもよいフェニレン、置換されていてもよい単環ヘテロアリレン、置換されていてもよい単環非芳香族複素環ジイル、または置換されていてもよい単環シクロアルカンジイル；
Ｗ^１は式：

（式中、Ｒ^１、Ｒ^２、Ｒ^３、Ｒ^４、Ｒ^７、およびＲ^８はそれぞれ独立して、水素原子、ハロゲン、置換されていてもよい低級アルキル、置換されていてもよい低級アルキルオキシ、置換されていてもよい低級アルキルチオ、置換されていてもよい低級アルケニル、置換されていてもよい低級アルキニル、置換されていてもよいアリール、置換されていてもよいヘテロアリール、置換されていてもよいシクロアルキル、置換されていてもよいアラルキル、置換されていてもよいヘテロアリールアルキル、置換されていてもよい非芳香族複素環基、または置換されていてもよいアミノ；
Ｒ^５、Ｒ^６、およびＲ^９はそれぞれ独立して、水素原子、置換されていてもよい低級アルキル、置換されていてもよい低級アルケニル、置換されていてもよい低級アルキニル、置換されていてもよいアリール、置換されていてもよいヘテロアリール、置換されていてもよいシクロアルキル、置換されていてもよいアラルキル、置換されていてもよいヘテロアリールアルキル、または置換されていてもよい非芳香族複素環基；
Ａ^１は置換されていてもよいアリールまたは置換されていてもよいヘテロアリール；
破線（−−−）は結合の存在または不存在を表わす）で表わされる基］で示される化合物、そのプロドラッグ、もしくはそれらの製薬上許容される塩、またはそれらの溶媒和物を有効成分として含有するトロンボポエチン受容体アゴニスト作用を有する医薬組成物。
Ｘ^１が置換されていてもよいヘテロアリールである請求項１記載のトロンボポエチン受容体アゴニスト作用を有する医薬組成物。
Ｘ^１が式：

（式中、Ｒ^１０およびＲ^１１はそれぞれ独立して水素原子、置換されていてもよい低級アルキル、カルボキシ、低級アルキルオキシカルボニル、ハロゲン、置換されていてもよいアミノカルボニル、置換されていてもよいヘテロアリール、または置換されていてもよいアリール；Ｒ^１２は水素原子または低級アルキル）で示される基である請求項１記載のトロンボポエチン受容体アゴニスト作用を有する医薬組成物。
Ｘ^１が式：

（式中、Ｒ^１０およびＲ^１１は請求項３と同意義）で示される基である請求項１記載のトロンボポエチン受容体アゴニスト作用を有する医薬組成物。
Ｙ^１が−ＮＨＣＯ−、−ＣＯＮＨ−、−ＮＨＣＨ_２−、−ＮＨＣＯ−ＣＨ＝ＣＨ−、または−ＮＨＳＯ_２−である請求項１〜４のいずれかに記載のトロンボポエチン受容体アゴニスト作用を有する医薬組成物。
Ｙ^１が−ＮＨＣＯ−である請求項１〜４のいずれかに記載のトロンボポエチン受容体アゴニスト作用を有する医薬組成物。
Ｚ^１がハロゲンまたは低級アルキルで置換されていてもよい１，４−フェニレンである請求項１〜６のいずれかに記載のトロンボポエチン受容体アゴニスト作用を有する医薬組成物。
Ｒ^１が水素原子または低級アルキルである請求項１〜７のいずれかに記載のトロンボポエチン受容体アゴニスト作用を有する医薬組成物。
Ｒ^２が水素原子、低級アルキル、ハロゲン、低級アルキルオキシ、低級アルキルチオ、または置換されていてもよいアミノである請求項１〜８のいずれかに記載のトロンボポエチン受容体アゴニスト作用を有する医薬組成物。
Ｗ^１が式：

（式中、Ｒ^１３は水素原子、低級アルキル、低級アルキルオキシ、低級アルキルチオ、またはハロゲン；Ｒ^１４およびＲ^１５はそれぞれ独立して水素原子、またはそれぞれ以下の置換基群Ａから選択される１以上の置換基によって置換されていてもよい低級アルキル、低級アルケニル、低級アルキニル、シクロアルキル、アリール、アラルキル、ヘテロアリール、もしくはヘテロアリールアルキル；破線は請求項１と同意義；
置換基群Ａ：ハロゲン、ハロ低級アルキル、置換されていてもよいアミノ、カルボキシ、低級アルキルチオ、低級アルキルシリル、または低級アルキルオキシ）で表わされる基である、請求項１〜９のいずれかに記載のトロンボポエチン受容体アゴニスト作用を有する医薬組成物。
Ｗ^１が式：

（式中、Ｒ^１３は水素原子、低級アルキル、低級アルキルオキシ、低級アルキルチオ、またはハロゲン；Ｒ^２６は水素原子または低級アルキル；破線は請求項１と同意義）で表わされる基である、請求項１〜９のいずれかに記載のトロンボポエチン受容体アゴニスト作用を有する医薬組成物。
血小板産生調節剤である請求項１〜１１のいずれかに記載のトロンボポエチン受容体アゴニスト作用を有する医薬組成物。
一般式（ＩＩ）：

［式中、Ｘ^２は置換されていてもよい５員ヘテロアリールまたは置換されていてもよいピリジル；
Ｙ^２は−ＮＲ^ＡＣＯ−（ＣＲ^ＣＲ^Ｄ）_０−２−、−ＮＲ^ＡＣＯ−（ＣＨ_２）_０−２−Ｖ−、−ＮＲ^ＡＣＯ−ＣＲ^Ｃ＝ＣＲ^Ｄ−、−Ｖ−（ＣＨ_２）_１−５−ＮＲ^ＡＣＯ−（ＣＨ_２）_０−２−、−Ｖ−（ＣＨ_２）_１−５−ＣＯＮＲ^Ａ−（ＣＨ_２）_０−２−、−ＣＯＮＲ^Ａ−（ＣＨ_２）_０−２−、−（ＣＨ_２）_０−２−ＮＲ^Ａ−ＳＯ_２−（ＣＨ_２）_０−２−、−（ＣＨ_２）_０−２−ＳＯ_２−ＮＲ^Ａ−（ＣＨ_２）_０−２−、−ＮＲ^Ａ−（ＣＨ_２）_０−２−、−ＮＲ^Ａ−ＣＯ−ＮＲ^Ａ−、−ＮＲ^Ａ−ＣＳ−ＮＲ^Ａ−、−Ｎ＝Ｃ（−ＳＲ^Ａ）−ＮＲ^Ａ−、−ＮＲ^ＡＣＳＮＲ^ＡＣＯ−、−Ｎ＝Ｃ（−ＳＲ^Ａ）−ＮＲ^ＡＣＯ−、−ＮＲ^Ａ−（ＣＨ_２）_１−２−ＮＲ^Ａ−ＣＯ−、−ＮＲ^ＡＣＯＮＲ^ＡＮＲ^ＢＣＯ−、または−Ｎ＝Ｃ（−ＮＲ^ＡＲ^Ａ）−ＮＲ^ＡＣＯ−（式中、Ｒ^Ａはそれぞれ独立して水素原子または低級アルキル；Ｒ^Ｂは水素原子またはフェニル；Ｒ^ＣおよびＲ^Ｄはそれぞれ独立して、水素原子、ハロゲン、置換されていてもよい低級アルキル、置換されていてもよい低級アルキルオキシ、置換されていてもよい低級アルキルチオ、置換されていてもよい低級アルケニル、置換されていてもよい低級アルキニル、置換されていてもよいアリール、置換されていてもよいヘテロアリール、置換されていてもよいシクロアルキル、置換されていてもよいアラルキル、置換されていてもよいヘテロアリールアルキル、置換されていてもよい非芳香族複素環基、または置換されていてもよいアミノ；Ｖは酸素原子または硫黄原子）；
Ｚ^２は置換されていてもよいフェニレン、置換されていてもよい２，５−ピリジンジイル、置換されていてもよい２，５−チオフェンジイル、または置換されていてもよい２，５−フランジイル；
Ｗ^２は式：

（式中、Ｒ^１、Ｒ^２、Ｒ^３、Ｒ^４、Ｒ^７、およびＲ^８はそれぞれ独立して、水素原子、ハロゲン、置換されていてもよい低級アルキル、置換されていてもよい低級アルキルオキシ、置換されていてもよい低級アルキルチオ、置換されていてもよい低級アルケニル、置換されていてもよい低級アルキニル、置換されていてもよいアリール、置換されていてもよいヘテロアリール、置換されていてもよいシクロアルキル、置換されていてもよいアラルキル、置換されていてもよいヘテロアリールアルキル、置換されていてもよい非芳香族複素環基、または置換されていてもよいアミノ；
Ｒ^５、Ｒ^６、およびＲ^９はそれぞれ独立して、水素原子、置換されていてもよい低級アルキル、置換されていてもよい低級アルケニル、置換されていてもよい低級アルキニル、置換されていてもよいアリール、置換されていてもよいヘテロアリール、置換されていてもよいシクロアルキル、置換されていてもよいアラルキル、置換されていてもよいヘテロアリールアルキル、または置換されていてもよい非芳香族複素環基；
Ａ^２は置換されていてもよいアリールまたは置換されていてもよいヘテロアリール；
破線（−−−）は結合の存在または不存在を表わす）で表わされる基］で示される化合物、そのプロドラッグ、もしくはそれらの製薬上許容される塩、またはそれらの溶媒和物。
Ｘ^２が式：

（式中、Ｒ^１０およびＲ^１１はそれぞれ独立して水素原子、置換されていてもよい低級アルキル、カルボキシ、低級アルキルオキシカルボニル、ハロゲン、置換されていてもよいアミノカルボニル、置換されていてもよいヘテロアリール、または置換されていてもよいアリール）で示される基である請求項１３記載の化合物、そのプロドラッグ、もしくはそれらの製薬上許容される塩、またはそれらの溶媒和物。
Ｘ^２が式：

（式中、Ｒ^１６は水素原子、置換されていてもよい低級アルキル、カルボキシ、低級アルキルオキシカルボニル、ハロゲン、または置換されていてもよいアミノカルボニル；
Ｒ^１７、Ｒ^１８、Ｒ^１９、Ｒ^２０、Ｒ^２１、Ｒ^２２、およびＲ^２３はそれぞれ独立して水素原子、置換基群Ｂから選択される１以上の置換基によって置換されていてもよいアルキル、シクロアルキル、置換基群Ｂから選択される１以上の置換基によって置換されていてもよいアルキルオキシ、アルキルチオ、ハロゲン、置換基群Ｃから選択される１以上の置換基によって置換されていてもよいフェニル、置換基群Ｃから選択される１以上の置換基によって置換されていてもよいヘテロアリール、または置換基群Ｃから選択される１以上の置換基によって置換されていてもよい非芳香族複素環基、
置換基群Ｂ：ヒドロキシ、アルキルオキシ、ハロゲン、カルボキシ、低級アルキルオキシカルボニル、アリールオキシカルボニル、置換されていてもよいアミノ、置換基群Ｃから選択される１以上の置換基によって置換されていてもよいフェニル、非芳香族複素環基、およびヘテロアリール、
置換基群Ｃ：ヒドロキシ、アルキル、ハロゲン、ハロ低級アルキル、カルボキシ、低級アルキルオキシカルボニル、アルキルオキシ、置換されていてもよいアミノ、非芳香族複素環、およびヘテロアリール；
Ｒ^１６およびＲ^１７は一緒になって−ＣＨ_２−、−ＣＨ_２ＣＨ_２−、−ＣＨ_２ＣＨ_２ＣＨ_２−、−ＯＣＨ_２−、または−ＳＣＨ_２−を形成してもよい）で示される基である請求項１３または１４記載の化合物、そのプロドラッグ、もしくはそれらの製薬上許容される塩、またはそれらの溶媒和物。
Ｙ^２が−ＮＨＣＯ−である請求項１３〜１５のいずれかに記載の化合物、そのプロドラッグ、もしくはそれらの製薬上許容される塩、またはそれらの溶媒和物。
Ｚ^２がハロゲンまたは低級アルキルで置換されていてもよい１，４−フェニレンである請求項１３〜１６のいずれかに記載の化合物、そのプロドラッグ、もしくはそれらの製薬上許容される塩、またはそれらの溶媒和物。
Ｒ^１が水素原子または低級アルキルである請求項１３〜１７のいずれかに記載の化合物、そのプロドラッグ、もしくはそれらの製薬上許容される塩、またはそれらの溶媒和物。
Ｒ^２が水素原子、低級アルキル、ハロゲン、低級アルキルオキシ、低級アルキルチオ、または置換されていてもよいアミノである請求項１３〜１８のいずれかに記載の化合物、そのプロドラッグ、もしくはそれらの製薬上許容される塩、またはそれらの溶媒和物。
Ｗ^２が式：

（式中、Ｒ^１、Ｒ^２、Ｒ^３、Ｒ^４、Ｒ^５、Ｒ^６、Ｒ^７、Ｒ^８、およびＡ^２は請求項１３と同意義、ただし、Ｒ^２はイミダゾリル、トリアゾリル、またはテトラゾリルではない）である請求項１３〜１９のいずれかに記載の化合物、そのプロドラッグ、もしくはそれらの製薬上許容される塩、またはそれらの溶媒和物。
Ｗ^２が式：

（式中、Ｒ^１３は水素原子、低級アルキル、低級アルキルオキシ、低級アルキルチオ、またはハロゲン、Ｒ^１４およびＲ^１５はそれぞれ独立して水素原子、またはそれぞれ以下の置換基群Ａから選択される１以上の置換基によって置換されていてもよい低級アルキル、低級アルケニル、低級アルキニル、シクロアルキル、アリール、アラルキル、ヘテロアリール、ヘテロアリールアルキル、もしくは非芳香族複素環基；
置換基群Ａ：ハロゲン、ハロ低級アルキル、置換されていてもよいアミノ、カルボキシ、低級アルキルチオ、低級アルキルシリル、または低級アルキルオキシ）である請求項１３〜２０のいずれかに記載の化合物、そのプロドラッグ、もしくはそれらの製薬上許容される塩、またはそれらの溶媒和物。
Ｗ^２が式：

（式中、Ｒ^１３は水素原子、低級アルキル、低級アルキルオキシ、低級アルキルチオ、またはハロゲン；Ｒ^２６は水素原子または低級アルキル；破線は請求項１３と同意義）で表わされる基である、請求項１３〜２１のいずれかに記載の化合物、そのプロドラッグ、もしくはそれらの製薬上許容される塩、またはそれらの溶媒和物。
請求項１３〜２２のいずれかに記載の化合物を有効成分として含有する医薬組成物。
請求項１３〜２２のいずれかに記載の化合物を有効成分として含有するトロンボポエチン受容体アゴニスト作用を有する医薬組成物。
請求項１３〜２２のいずれかに記載の化合物を有効成分として含有する血小板産生調節剤。
一般式（ＩＩ）：

［式中、Ｘ^２は置換されていてもよい５員ヘテロアリールまたは置換されていてもよいピリジル；
Ｙ^２は−ＮＲ^ＡＣＯ−（ＣＲ^ＣＲ^Ｄ）_０−２−、−ＮＲ^ＡＣＯ−（ＣＨ_２）_０−２−Ｖ−、−ＮＲ^ＡＣＯ−ＣＲ^Ｃ＝ＣＲ^Ｄ−、−Ｖ−（ＣＨ_２）_１−５−ＮＲ^ＡＣＯ−（ＣＨ_２）_０−２−、−Ｖ−（ＣＨ_２）_１−５−ＣＯＮＲ^Ａ−（ＣＨ_２）_０−２−、−ＣＯＮＲ^Ａ−（ＣＨ_２）_０−２−、−（ＣＨ_２）_０−２−ＮＲ^Ａ−ＳＯ_２−（ＣＨ_２）_０−２−、−（ＣＨ_２）_０−２−ＳＯ_２−ＮＲ^Ａ−（ＣＨ_２）_０−２−、−ＮＲ^Ａ−（ＣＨ_２）_０−２−、−ＮＲ^Ａ−ＣＯ−ＮＲ^Ａ−、−ＮＲ^Ａ−ＣＳ−ＮＲ^Ａ−、−Ｎ＝Ｃ（−ＳＲ^Ａ）−ＮＲ^Ａ−、−ＮＲ^ＡＣＳＮＲ^ＡＣＯ−、−Ｎ＝Ｃ（−ＳＲ^Ａ）−ＮＲ^ＡＣＯ−、−ＮＲ^Ａ−（ＣＨ_２）_１−２−ＮＲ^Ａ−ＣＯ−、−ＮＲ^ＡＣＯＮＲ^ＡＮＲ^ＢＣＯ−、または−Ｎ＝Ｃ（−ＮＲ^ＡＲ^Ａ）−ＮＲ^ＡＣＯ−（式中、Ｒ^Ａはそれぞれ独立して水素原子または低級アルキル；Ｒ^Ｂは水素原子またはフェニル；Ｒ^ＣおよびＲ^Ｄはそれぞれ独立して、水素原子、ハロゲン、置換されていてもよい低級アルキル、置換されていてもよい低級アルキルオキシ、置換されていてもよい低級アルキルチオ、置換されていてもよい低級アルケニル、置換されていてもよい低級アルキニル、置換されていてもよいアリール、置換されていてもよいヘテロアリール、置換されていてもよいシクロアルキル、置換されていてもよいアラルキル、置換されていてもよいヘテロアリールアルキル、置換されていてもよい非芳香族複素環基、または置換されていてもよいアミノ；Ｖは酸素原子または硫黄原子）；
Ｚ^２は置換されていてもよいフェニレン、置換されていてもよい２，５−ピリジンジイル、置換されていてもよい２，５−チオフェンジイル、または置換されていてもよい２，５−フランジイル；
Ｗ^２は式：

（式中、Ｒ^１、Ｒ^２、Ｒ^３、Ｒ^４、Ｒ^７、およびＲ^８はそれぞれ独立して、水素原子、ハロゲン、置換されていてもよい低級アルキル、置換されていてもよい低級アルキルオキシ、置換されていてもよい低級アルキルチオ、置換されていてもよい低級アルケニル、置換されていてもよい低級アルキニル、置換されていてもよいアリール、置換されていてもよいヘテロアリール、置換されていてもよいシクロアルキル、置換されていてもよいアラルキル、置換されていてもよいヘテロアリールアルキル、置換されていてもよい非芳香族複素環基、または置換されていてもよいアミノ；
Ｒ^５、Ｒ^６、およびＲ^９はそれぞれ独立して、水素原子、置換されていてもよい低級アルキル、置換されていてもよい低級アルケニル、置換されていてもよい低級アルキニル、置換されていてもよいアリール、置換されていてもよいヘテロアリール、置換されていてもよいシクロアルキル、置換されていてもよいアラルキル、置換されていてもよいヘテロアリールアルキル、または置換されていてもよい非芳香族複素環基；
Ａ^２は置換されていてもよいアリールまたは置換されていてもよいヘテロアリール；
破線（−−−）は結合の存在または不存在を表わす）で表わされる基
但し、
１）Ｘ^２がアルキルで置換されてもよいチアゾリル又はアルコキシもしくはジエチルアミノエチルで置換されてもよいベンゾチアゾリル、Ｚ^２が１，４−フェニレン、Ｗ^２が式：

の場合は、Ｒ^２は置換されていてもよいイミダゾリル、置換されていてもよいトリアゾリル、または置換されていてもよいテトラゾリルではない、
２）Ｘ^２が２−ピリジル、、Ｙ^２が−ＮＨＣＯ−ＣＨ＝ＣＨ−、または−ＮＨＣＳＮＨＣＯ−、Ｚ^２が１，４−フェニレン、Ｗ^２が式：

の場合は、Ｒ^２はトリアゾリルではない、
３）Ｘ^２がベンゾチアゾリル、Ｙ^２が−ＮＨＣＯ−ＣＨ＝ＣＨ−、Ｚ^２が１，４−フェニレン、Ｗ^２が式：

の場合は、Ｒ^２は２−ピリジルまたはカルボキシメチルではない、
４）Ｘ^２がベンゾチアゾリル、Ｙ^２が−ＮＨＣＯ−、Ｚ^２が１，４−フェニレンの場合、Ｗ^２は式：

ではない、
５）Ｘ^２がメチル、ｔ−ブチルもしくは無置換のフェニルで置換されていてもよいチアゾリル、またはアルキルもしくはジエチルアミノエチルで置換されてもよいベンゾチアゾリル、Ｚ^２が置換されていてもよいフェニレン、Ｗ^２が−ＣＨ＝Ｏである場合は、Ｙ^２は−ＮＨＣＯ−（ＣＨ_２）_０−２−、−ＮＨＣＯ−ＣＨ＝ＣＨ−、−ＮＨＣＯ−ＣＨ_２−Ｏ−、または−ＮＨＣＯ−ＣＨ_２−ＮＭｅ−ではない、
６）Ｙ^２が−ＮＨ−ＣＨ_２−、Ｚ^２が１，４−フェニレン、Ｗ^２が置換されていてもよいテトラゾリルで2位が置換されているフェニルの場合、Ｘ^２はチアジアゾリル、チアゾリル、ベンゾチアゾリル、オキサジザゾリル、イミダゾリル、またはオキサゾリルではない、
７）Ｘ^２が置換されていてもよいベンゾチアゾリル、Ｚ^２が１，４−フェニレン、Ｗ^２が式：

の場合、Ｙ^２は−ＮＨＣＯ−、−ＮＨ−ＣＨ_２−、−ＮＥｔ−ＣＨ_２−、−ＮＨ−ではない、
８）Ｘ^２が置換されていてもよいベンゾチアゾリル、Ｙ^２が−ＮＨ−、Ｚ^２が１，４−フェニレンの場合、Ｗ^２は−ＣＨ_２ＣＯＯＨまたは、−ＣＨ_２ＣＯＯＥｔではない、
９）Ｘ^２が置換されていてもよいベンゾチアゾリル、Ｙ^２が−ＮＨ−、Ｚ^２が２，５−ピリジンジイルの場合、Ｗ^２は−ＣＯＯＨまたは、−ＣＯＮＨ_２ではない、
１０）Ｘ^２が置換されていてもよいベンゾチアゾリル、Ｚ^２がメチルまたは塩素によって置換されていてもよいフェニレン、Ｗ^２が−ＣＯＯＨ、−ＣＯＯＥｔまたは、−ＣＯＮＨ_２の場合は、Ｙ^２は−ＮＨ−、−ＮＨ−ＣＨ_２−、−ＮＨ−ＣＯ−、―ＮＨ−ＳＯ_２−ではない］で示される化合物、そのプロドラッグ、もしくはそれらの製薬上許容される塩、またはそれらの溶媒和物。
Ｘ^２が式：

（式中、Ｒ^１０およびＲ^１１はそれぞれ独立して水素原子、置換されていてもよい低級アルキル、カルボキシ、低級アルキルオキシカルボニル、ハロゲン、置換されていてもよいアミノカルボニル、置換されていてもよいヘテロアリール、または置換されていてもよいアリール）で示される基である請求項２６記載の化合物、そのプロドラッグ、もしくはそれらの製薬上許容される塩、またはそれらの溶媒和物。
Ｘ^２が式：

（式中、Ｒ^１６は水素原子、置換されていてもよい低級アルキル、カルボキシ、低級アルキルオキシカルボニル、ハロゲン、または置換されていてもよいアミノカルボニル；
Ｒ^１７、Ｒ^１８、Ｒ^１９、Ｒ^２０、Ｒ^２１、Ｒ^２２、およびＲ^２３はそれぞれ独立して水素原子、置換基群Ｂから選択される１以上の置換基によって置換されていてもよいアルキル、シクロアルキル、置換基群Ｂから選択される１以上の置換基によって置換されていてもよいアルキルオキシ、アルキルチオ、ハロゲン、置換基群Ｃから選択される１以上の置換基によって置換されていてもよいフェニル、置換基群Ｃから選択される１以上の置換基によって置換されていてもよいヘテロアリール、または置換基群Ｃから選択される１以上の置換基によって置換されていてもよい非芳香族複素環基、
置換基群Ｂ：ヒドロキシ、アルキルオキシ、ハロゲン、カルボキシ、低級アルキルオキシカルボニル、アリールオキシカルボニル、置換されていてもよいアミノ、置換基群Ｃから選択される１以上の置換基によって置換されていてもよいフェニル、非芳香族複素環基、およびヘテロアリール、
置換基群Ｃ：ヒドロキシ、アルキル、ハロゲン、ハロ低級アルキル、カルボキシ、低級アルキルオキシカルボニル、アルキルオキシ、置換されていてもよいアミノ、非芳香族複素環、およびヘテロアリール；
Ｒ^１６およびＲ^１７は一緒になって−ＣＨ_２−、−ＣＨ_２ＣＨ_２−、−ＣＨ_２ＣＨ_２ＣＨ_２−、−ＯＣＨ_２−、または−ＳＣＨ_２−を形成してもよい）で示される基である請求項２６または２７記載の化合物、そのプロドラッグ、もしくはそれらの製薬上許容される塩、またはそれらの溶媒和物。
Ｙ^２が−ＮＨＣＯ−である請求項２６〜２８のいずれかに記載の化合物、そのプロドラッグ、もしくはそれらの製薬上許容される塩、またはそれらの溶媒和物。
Ｚ^２がハロゲンまたは低級アルキルで置換されていてもよい１，４−フェニレンである請求項２６〜３０のいずれかに記載の化合物、そのプロドラッグ、もしくはそれらの製薬上許容される塩、またはそれらの溶媒和物。
Ｒ^１が水素原子または低級アルキルである請求項２６〜３０のいずれかに記載の化合物、そのプロドラッグ、もしくはそれらの製薬上許容される塩、またはそれらの溶媒和物。
Ｒ^２が水素原子、低級アルキル、ハロゲン、低級アルキルオキシ、低級アルキルチオ、または置換されていてもよいアミノである請求項２６〜３１のいずれかに記載の化合物、そのプロドラッグ、もしくはそれらの製薬上許容される塩、またはそれらの溶媒和物。
Ｗ^２が式：

（式中、Ｒ^１、Ｒ^２、Ｒ^３、Ｒ^４、Ｒ^５、Ｒ^６、Ｒ^７、Ｒ^８、およびＡ^２は請求項１３と同意義、ただし、Ｒ^２はイミダゾリル、トリアゾリル、またはテトラゾリルではない）である請求項２６〜３２のいずれかに記載の化合物、そのプロドラッグ、もしくはそれらの製薬上許容される塩、またはそれらの溶媒和物。
Ｗ^２が式：

（式中、Ｒ^１３は水素原子、低級アルキル、低級アルキルオキシ、低級アルキルチオ、またはハロゲン、Ｒ^１４およびＲ^１５はそれぞれ独立して水素原子、またはそれぞれ以下の置換基群Ａから選択される１以上の置換基によって置換されていてもよい低級アルキル、低級アルケニル、低級アルキニル、シクロアルキル、アリール、アラルキル、ヘテロアリール、ヘテロアリールアルキル、もしくは非芳香族複素環基；
置換基群Ａ：ハロゲン、ハロ低級アルキル、置換されていてもよいアミノ、カルボキシ、低級アルキルチオ、低級アルキルシリル、または低級アルキルオキシ）である請求項２６〜３３のいずれかに記載の化合物、そのプロドラッグ、もしくはそれらの製薬上許容される塩、またはそれらの溶媒和物。
Ｗ^２が式：

（式中、Ｒ^１３は水素原子、低級アルキル、低級アルキルオキシ、低級アルキルチオ、またはハロゲン；Ｒ^２６は水素原子または低級アルキル；破線は請求項１３と同意義）で表わされる基である、請求項２６〜３３のいずれかに記載の化合物、そのプロドラッグ、もしくはそれらの製薬上許容される塩、またはそれらの溶媒和物。
請求項２６〜３５のいずれかに記載の化合物を有効成分として含有する医薬組成物。
請求項２６〜３５のいずれかに記載の化合物を有効成分として含有するトロンボポエチン受容体アゴニスト作用を有する医薬組成物。
請求項２６〜３５のいずれかに記載の化合物を有効成分として含有する血小板産生調節剤。