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JO3450B1 - أشكال جرعات تحرير جديدة معدلة لمثبطات زانثين اوكسيدوريدوكتيز أو مثبطات زانثين اوكسيديز - Google Patents

أشكال جرعات تحرير جديدة معدلة لمثبطات زانثين اوكسيدوريدوكتيز أو مثبطات زانثين اوكسيديز

Info

Publication number
JO3450B1
JO3450B1 JOP/2011/0194A JOP20110194A JO3450B1 JO 3450 B1 JO3450 B1 JO 3450B1 JO P20110194 A JOP20110194 A JO P20110194A JO 3450 B1 JO3450 B1 JO 3450B1
Authority
JO
Jordan
Prior art keywords
inhibitors
xanthine
dosage forms
release dosage
modified release
Prior art date
Application number
JOP/2011/0194A
Other languages
English (en)
Inventor
Gupte Vijay
Taneja Rajneesh
Vakilynejad Majid
Original Assignee
Takeda Pharmaceuticals Usa Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=45328897&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=JO3450(B1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Takeda Pharmaceuticals Usa Inc filed Critical Takeda Pharmaceuticals Usa Inc
Application granted granted Critical
Publication of JO3450B1 publication Critical patent/JO3450B1/ar

Links

Classifications

    • A—HUMAN NECESSITIES
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    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
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    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
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    • A61K9/167—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction with an outer layer or coating comprising drug; with chemically bound drugs or non-active substances on their surface
    • A61K9/1676—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction with an outer layer or coating comprising drug; with chemically bound drugs or non-active substances on their surface having a drug-free core with discrete complete coating layer containing drug
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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Cardiology (AREA)
  • Diabetes (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Urology & Nephrology (AREA)
  • Physiology (AREA)
  • Nutrition Science (AREA)
  • Obesity (AREA)
  • Endocrinology (AREA)
  • Hematology (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Reproductive Health (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Vascular Medicine (AREA)
  • Emergency Medicine (AREA)
  • Hospice & Palliative Care (AREA)
  • Inorganic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

يتعلق الاختراع الحالي بأشكال جرعات جديدة من مثبطات أكسيدوريداكتيز إكسانثين.
JOP/2011/0194A 2010-06-16 2011-06-15 أشكال جرعات تحرير جديدة معدلة لمثبطات زانثين اوكسيدوريدوكتيز أو مثبطات زانثين اوكسيديز JO3450B1 (ar)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US35516410P 2010-06-16 2010-06-16

Publications (1)

Publication Number Publication Date
JO3450B1 true JO3450B1 (ar) 2020-07-05

Family

ID=45328897

Family Applications (1)

Application Number Title Priority Date Filing Date
JOP/2011/0194A JO3450B1 (ar) 2010-06-16 2011-06-15 أشكال جرعات تحرير جديدة معدلة لمثبطات زانثين اوكسيدوريدوكتيز أو مثبطات زانثين اوكسيديز

Country Status (25)

Country Link
US (2) US9248119B2 (ar)
EP (1) EP2582812B1 (ar)
JP (2) JP5865904B2 (ar)
KR (1) KR101872189B1 (ar)
CN (1) CN103210084B (ar)
AU (2) AU2011268445B2 (ar)
BR (1) BR112012032033A2 (ar)
CA (1) CA2801930A1 (ar)
CL (1) CL2012003548A1 (ar)
CO (1) CO6650415A2 (ar)
EC (1) ECSP13012394A (ar)
ES (1) ES2669184T3 (ar)
IL (2) IL223455B (ar)
JO (1) JO3450B1 (ar)
MX (2) MX361138B (ar)
MY (1) MY167126A (ar)
NZ (1) NZ604646A (ar)
PE (2) PE20130574A1 (ar)
PH (1) PH12012502485A1 (ar)
RU (1) RU2602188C2 (ar)
SG (1) SG186301A1 (ar)
TW (1) TW201202249A (ar)
UA (1) UA112632C2 (ar)
WO (1) WO2011159745A1 (ar)
ZA (1) ZA201209386B (ar)

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JP5669837B2 (ja) * 2010-06-16 2015-02-18 帝人ファーマ株式会社 放出制御型の有核錠剤
MY160963A (en) * 2010-06-25 2017-03-31 Teijin Pharma Ltd Sustained-release therapeutic agent for hypertension and renal dysfunction
NZ605562A (en) * 2010-07-09 2013-11-29 Teijin Pharma Ltd Deuterated benzylbenzene derivatives and methods of use
WO2012153313A1 (en) * 2011-05-11 2012-11-15 Ranbaxy Laboratories Limited Pharmaceutical composition of febuxostat
WO2012172461A1 (en) * 2011-06-13 2012-12-20 Ranbaxy Laboratories Limited Pharmaceutical compositions of febuxostat
CA2862602A1 (en) * 2012-01-27 2013-08-01 Teijin Pharma Limited Therapeutic agent for diabetes
WO2014009817A1 (en) * 2012-07-12 2014-01-16 Alembic Pharmaceuticals Limited Pharmaceutical composition of febuxostat
CN102973530B (zh) * 2012-12-14 2016-08-03 贵州信邦制药股份有限公司 一种非布索坦双层肠溶片剂及其制备方法
WO2014125504A2 (en) * 2013-02-18 2014-08-21 Hetero Research Foundation Pharmaceutical compositions of febuxostat
SG11201509738RA (en) * 2013-05-31 2015-12-30 Takeda Pharmaceuticals Usa Inc Methods of treatment and compositions with xanthine oxidase inhibitors
EP2881116A1 (en) * 2013-12-05 2015-06-10 Ranbaxy Laboratories Limited Febuxostat composition
AU2015392441A1 (en) * 2015-04-20 2017-11-09 Twi Biotechnology, Inc. Formulations containing diacerein and methods of lowering blood levels of uric acid using the same
TWI684465B (zh) * 2015-04-22 2020-02-11 安成生物科技股份有限公司 含雙醋瑞因之製劑及使用其於降低尿酸血中濃度的方法
WO2017100559A1 (en) * 2015-12-10 2017-06-15 Cogwellin Llc Controlled release formulations of salicylate-releasing actives
CN106279024B (zh) * 2016-07-19 2018-09-14 华南理工大学 一种黄嘌呤氧化还原酶抑制剂及其制备方法与应用
CN106146419A (zh) * 2016-08-01 2016-11-23 沈阳药科大学 黄嘌呤氧化酶抑制剂
JP6861726B2 (ja) * 2016-11-28 2021-04-21 帝人ファーマ株式会社 糖尿病性腎症の治療薬または予防薬
WO2018228440A1 (zh) * 2017-06-14 2018-12-20 江苏恒瑞医药股份有限公司 一种非布司他控释组合物及其制备方法
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