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ITMI951900A0 - Derivati idroisochinolinici sostituiti - Google Patents

Derivati idroisochinolinici sostituiti

Info

Publication number
ITMI951900A0
ITMI951900A0 ITMI951900A ITMI951900A ITMI951900A0 IT MI951900 A0 ITMI951900 A0 IT MI951900A0 IT MI951900 A ITMI951900 A IT MI951900A IT MI951900 A ITMI951900 A IT MI951900A IT MI951900 A0 ITMI951900 A0 IT MI951900A0
Authority
IT
Italy
Prior art keywords
substituted
hydroisoquinoline
derivatives
hydroisoquinoline derivatives
substituted hydroisoquinoline
Prior art date
Application number
ITMI951900A
Other languages
English (en)
Inventor
Giulio Dondio
Silvano Ronzoni
Original Assignee
Giulio Dondio
Silvano Ronzoni
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Giulio Dondio, Silvano Ronzoni filed Critical Giulio Dondio
Priority to IT1995MI001900A priority Critical patent/IT1307327B1/it
Publication of ITMI951900A0 publication Critical patent/ITMI951900A0/it
Priority to JP9511672A priority patent/JPH11512415A/ja
Priority to US09/029,621 priority patent/US5968949A/en
Priority to PCT/EP1996/004036 priority patent/WO1997010216A1/en
Priority to EP96932527A priority patent/EP0854868A1/en
Publication of ITMI951900A1 publication Critical patent/ITMI951900A1/it
Application granted granted Critical
Publication of IT1307327B1 publication Critical patent/IT1307327B1/it

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D217/00Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems
    • C07D217/02Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems with only hydrogen atoms or radicals containing only carbon and hydrogen atoms, directly attached to carbon atoms of the nitrogen-containing ring; Alkylene-bis-isoquinolines
    • C07D217/04Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems with only hydrogen atoms or radicals containing only carbon and hydrogen atoms, directly attached to carbon atoms of the nitrogen-containing ring; Alkylene-bis-isoquinolines with hydrocarbon or substituted hydrocarbon radicals attached to the ring nitrogen atom
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/30Drugs for disorders of the nervous system for treating abuse or dependence
    • A61P25/32Alcohol-abuse
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • A61P27/02Ophthalmic agents
    • A61P27/14Decongestants or antiallergics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D217/00Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems
    • C07D217/12Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems with radicals, substituted by hetero atoms, attached to carbon atoms of the nitrogen-containing ring
    • C07D217/14Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems with radicals, substituted by hetero atoms, attached to carbon atoms of the nitrogen-containing ring other than aralkyl radicals
    • C07D217/16Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems with radicals, substituted by hetero atoms, attached to carbon atoms of the nitrogen-containing ring other than aralkyl radicals substituted by oxygen atoms

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Addiction (AREA)
  • Immunology (AREA)
  • Psychiatry (AREA)
  • Ophthalmology & Optometry (AREA)
  • Pain & Pain Management (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Other In-Based Heterocyclic Compounds (AREA)
IT1995MI001900A 1995-09-12 1995-09-12 Derivati idroisochinolinici sostituiti IT1307327B1 (it)

Priority Applications (5)

Application Number Priority Date Filing Date Title
IT1995MI001900A IT1307327B1 (it) 1995-09-12 1995-09-12 Derivati idroisochinolinici sostituiti
JP9511672A JPH11512415A (ja) 1995-09-12 1996-09-12 置換されたヒドロイソキノリン誘導体および医薬としてのその使用
US09/029,621 US5968949A (en) 1995-09-12 1996-09-12 Substituted hydroisoquinoline derivatives and their use as pharmaceuticals
PCT/EP1996/004036 WO1997010216A1 (en) 1995-09-12 1996-09-12 Substituted hydroisoquinoline derivatives and their use as pharmaceuticals
EP96932527A EP0854868A1 (en) 1995-09-12 1996-09-12 Substituted hydroisoquinoline derivatives and their use as pharmaceuticals

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
IT1995MI001900A IT1307327B1 (it) 1995-09-12 1995-09-12 Derivati idroisochinolinici sostituiti

Publications (3)

Publication Number Publication Date
ITMI951900A0 true ITMI951900A0 (it) 1995-09-12
ITMI951900A1 ITMI951900A1 (it) 1997-03-12
IT1307327B1 IT1307327B1 (it) 2001-10-30

Family

ID=11372234

Family Applications (1)

Application Number Title Priority Date Filing Date
IT1995MI001900A IT1307327B1 (it) 1995-09-12 1995-09-12 Derivati idroisochinolinici sostituiti

Country Status (5)

Country Link
US (1) US5968949A (it)
EP (1) EP0854868A1 (it)
JP (1) JPH11512415A (it)
IT (1) IT1307327B1 (it)
WO (1) WO1997010216A1 (it)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2264928A1 (en) * 1997-07-09 1999-01-21 Koji Kawai Antitussives
US6103722A (en) * 1997-07-23 2000-08-15 The Medical College Of Wisconsin Research Foundation Inc. Ischemic preconditioning
CA2683097A1 (en) * 1998-03-10 1999-09-16 Research Triangle Institute Novel opiate compounds, methods of making and methods of use
EP1438304B1 (en) 2001-10-15 2006-12-06 Janssen Pharmaceutica N.V. Novel substituted 4-phenyl-4-[1h-imidazol-2-yl]-piperidine derivatives and their use as selective non-peptide delta opioid agonists
KR101255074B1 (ko) 2003-10-01 2013-04-16 아돌로 코포레이션 스피로시클릭 헤테로시클릭 유도체 및 이의 사용 방법
US7598261B2 (en) 2005-03-31 2009-10-06 Adolor Corporation Spirocyclic heterocyclic derivatives and methods of their use
US7476679B2 (en) * 2005-07-26 2009-01-13 Research Triangle Institute Octahydroisoquinoline compounds as opioid receptor modulators
US7576207B2 (en) 2006-04-06 2009-08-18 Adolor Corporation Spirocyclic heterocyclic derivatives and methods of their use
JP2010503669A (ja) 2006-09-12 2010-02-04 アドラー コーポレーション 認知機能の強化のためのn含有スピロ化合物の使用
US9604931B2 (en) 2007-01-22 2017-03-28 Gtx, Inc. Nuclear receptor binding agents
KR101763674B1 (ko) 2007-01-22 2017-08-01 지티엑스, 인코포레이티드 핵 수용체에 결합하는 물질
US9623021B2 (en) * 2007-01-22 2017-04-18 Gtx, Inc. Nuclear receptor binding agents

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2351599A1 (de) * 1972-07-20 1974-01-31 Du Pont 4a-aryl-trans-decahydrochinoline und verfahren zu ihrer herstellung
SE7509022L (sv) * 1974-09-09 1976-03-10 Du Pont Foreningar med analgetisk verkan
US4077954A (en) * 1976-02-10 1978-03-07 E. I. Du Pont De Nemours And Company N-(p-methylphenethyl)-4a-aryl-trans-decahydroisoquinolines

Also Published As

Publication number Publication date
US5968949A (en) 1999-10-19
JPH11512415A (ja) 1999-10-26
ITMI951900A1 (it) 1997-03-12
EP0854868A1 (en) 1998-07-29
IT1307327B1 (it) 2001-10-30
WO1997010216A1 (en) 1997-03-20

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