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IS1869B - Afleiður af setinni 4-hýdroxýfenýlalkanósýru með gerandefnisvirkni á PPAR-gamma, lyfjaefnablöndur sem innihalda þær, notkun þeirra og aðferð til framleiðslu þeirra - Google Patents

Afleiður af setinni 4-hýdroxýfenýlalkanósýru með gerandefnisvirkni á PPAR-gamma, lyfjaefnablöndur sem innihalda þær, notkun þeirra og aðferð til framleiðslu þeirra

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Publication number
IS1869B
IS1869B IS4822A IS4822A IS1869B IS 1869 B IS1869 B IS 1869B IS 4822 A IS4822 A IS 4822A IS 4822 A IS4822 A IS 4822A IS 1869 B IS1869 B IS 1869B
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IS
Iceland
Prior art keywords
derivatives
substituted
production
pharmaceutical preparations
agonist activity
Prior art date
Application number
IS4822A
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English (en)
Other versions
IS4822A (is
Inventor
Mark Willson Timothy
Anthony Mook Jrth Robert
Kaldor Istvan
Richard Henke Brad
Norman Deaton David
Edmond Cobb Jeffrey
Jude Sharp Matthew
Alan Erickson Greg
Evan Boswell Grady
Loren Collins Jon
Brackeen Markus
Mark O'callaghan John
Original Assignee
Glaxo Group Limited
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Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=10789571&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=IS1869(B) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Glaxo Group Limited filed Critical Glaxo Group Limited
Publication of IS4822A publication Critical patent/IS4822A/is
Publication of IS1869B publication Critical patent/IS1869B/is

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    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/62—Oxygen or sulfur atoms
    • C07D213/63—One oxygen atom
    • C07D213/64—One oxygen atom attached in position 2 or 6
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    • A61K31/19—Carboxylic acids, e.g. valproic acid
    • A61K31/192—Carboxylic acids, e.g. valproic acid having aromatic groups, e.g. sulindac, 2-aryl-propionic acids, ethacrynic acid 
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    • A61K31/216—Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids of acids having aromatic rings, e.g. benactizyne, clofibrate
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    • A61K31/352—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom condensed with carbocyclic rings, e.g. methantheline 
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    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
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    • A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4439—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
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IS4822A 1996-02-28 1998-08-12 Afleiður af setinni 4-hýdroxýfenýlalkanósýru með gerandefnisvirkni á PPAR-gamma, lyfjaefnablöndur sem innihalda þær, notkun þeirra og aðferð til framleiðslu þeirra IS1869B (is)

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CN1093124C (zh) 2002-10-23
CA2247443A1 (en) 1997-09-04
HUP0004845A3 (en) 2001-07-30
RS49586B (sr) 2007-04-10
US6294580B1 (en) 2001-09-25
GB9604242D0 (en) 1996-05-01
NO983940D0 (no) 1998-08-27
DE69706658D1 (de) 2001-10-18
DK0888317T3 (da) 2002-01-21
ATE205485T1 (de) 2001-09-15
EA001403B1 (ru) 2001-02-26
WO1997031907A1 (en) 1997-09-04
HK1015369A1 (en) 1999-10-15
MY119425A (en) 2005-05-31
BR9707786B1 (pt) 2009-12-01
PL191118B1 (pl) 2006-03-31
IL125796A (en) 2001-06-14
GEP20012580B (en) 2001-11-26
NZ331381A (en) 2000-06-23
BG102792A (bg) 1999-08-31
EP0888317B1 (en) 2001-09-12

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