[go: up one dir, main page]

IL180846A0 - 1,1,2,2-tetra (hetero) arylethanes or 1,1,2-tri (hetero) aryl-2-heterocyclylethanes as potassium channel inhibitors - Google Patents

1,1,2,2-tetra (hetero) arylethanes or 1,1,2-tri (hetero) aryl-2-heterocyclylethanes as potassium channel inhibitors

Info

Publication number
IL180846A0
IL180846A0 IL180846A IL18084607A IL180846A0 IL 180846 A0 IL180846 A0 IL 180846A0 IL 180846 A IL180846 A IL 180846A IL 18084607 A IL18084607 A IL 18084607A IL 180846 A0 IL180846 A0 IL 180846A0
Authority
IL
Israel
Prior art keywords
hetero
heterocyclylethanes
arylethanes
tetra
tri
Prior art date
Application number
IL180846A
Original Assignee
Merck & Co Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck & Co Inc filed Critical Merck & Co Inc
Publication of IL180846A0 publication Critical patent/IL180846A0/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/16Amides, e.g. hydroxamic acids
    • A61K31/18Sulfonamides
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/444Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a six-membered ring with nitrogen as a ring heteroatom, e.g. amrinone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/06Antiarrhythmics

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Cardiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
IL180846A 2004-07-29 2007-01-21 1,1,2,2-tetra (hetero) arylethanes or 1,1,2-tri (hetero) aryl-2-heterocyclylethanes as potassium channel inhibitors IL180846A0 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US59218104P 2004-07-29 2004-07-29
PCT/US2005/026334 WO2006028590A1 (en) 2004-07-29 2005-07-25 1,1,2,2-tetra (hetero) arylethanes or 1,1,2-tri (hetero) aryl-2-heterocyclylethanes as potassium channel inhibitors

Publications (1)

Publication Number Publication Date
IL180846A0 true IL180846A0 (en) 2007-06-03

Family

ID=35613661

Family Applications (1)

Application Number Title Priority Date Filing Date
IL180846A IL180846A0 (en) 2004-07-29 2007-01-21 1,1,2,2-tetra (hetero) arylethanes or 1,1,2-tri (hetero) aryl-2-heterocyclylethanes as potassium channel inhibitors

Country Status (15)

Country Link
KR (1) KR20070043985A (en)
AR (1) AR049847A1 (en)
BR (1) BRPI0513793A (en)
CR (1) CR8876A (en)
EC (1) ECSP077208A (en)
IL (1) IL180846A0 (en)
MA (1) MA28980B1 (en)
MX (1) MX2007001188A (en)
NO (1) NO20071107L (en)
PE (1) PE20060382A1 (en)
RU (1) RU2344134C2 (en)
TW (1) TW200607493A (en)
UA (1) UA88018C2 (en)
WO (1) WO2006028590A1 (en)
ZA (1) ZA200700477B (en)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN102427806B (en) * 2009-03-18 2015-11-25 麦迪库瑞国际公司 Transdermal pharmaceutical formulation and administration of tirofiban
NZ703632A (en) 2012-06-11 2016-01-29 Bristol Myers Squibb Co Phosphoramidic acid prodrugs of 5-[5-phenyl-4-(pyridin-2-ylmethylamino)quinazolin-2-yl]pyridine-3-sulfonamide

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2140865B2 (en) * 1971-08-14 1979-10-11 Bayer Ag, 5090 Leverkusen 1-imidazolyl-methanephosphonic acid ester, process for their preparation and medicaments containing them
DE19951701A1 (en) * 1999-10-27 2001-05-03 Aventis Pharma Gmbh Use of 2-imidazolyl-substituted carbinols for the manufacture of a medicament for the treatment or prophylaxis of diseases caused by ischemic conditions
ATE400551T1 (en) * 2002-01-04 2008-07-15 Neurosearch As POTASSIUM CHANNEL MODULATORS

Also Published As

Publication number Publication date
MX2007001188A (en) 2007-03-21
BRPI0513793A (en) 2008-05-13
PE20060382A1 (en) 2006-05-15
ZA200700477B (en) 2009-08-26
RU2344134C2 (en) 2009-01-20
MA28980B1 (en) 2007-11-01
RU2007107408A (en) 2008-09-10
CR8876A (en) 2007-08-28
UA88018C2 (en) 2009-09-10
ECSP077208A (en) 2007-02-28
WO2006028590A1 (en) 2006-03-16
KR20070043985A (en) 2007-04-26
TW200607493A (en) 2006-03-01
NO20071107L (en) 2007-04-19
AR049847A1 (en) 2006-09-06

Similar Documents

Publication Publication Date Title
IL163928A0 (en) Pyridinoylpiperidines as 5-htf agonists
ZA200700351B (en) Compounds, compositions and methods
ZA200502210B (en) Substrates for O6-alkylguanine-DNA alkyltansferase.
IL183706A0 (en) 2,4(4,6) pyrimidine derivatives
IL191711A0 (en) 1-orthofluorophenyl substituted 1,2,5-thiazolidinedione derivatives as ptp-as inhibitors
ZA200610142B (en) Furanopyrimidine compounds effective as potassium channel inhibitors
AP2321A (en) Quinoline derivatives for use as mycobactrial inhibitor.
EG25273A (en) Substituted dihydroquinazolines.
PL1725528T3 (en) Sulphonylpyrroles as hdac inhibitors
ZA200307420B (en) Point chisel.
EP1493437A4 (en) Compositions for diabetes
ZA200805028B (en) Arylpropionamide, arylacrylamide, arylpropynamide, or arylmethylurea analogs as factor Xla inhibitors
AU2003212310A1 (en) (4,2-disubstituted-thiazol-5-yl)amine compounds as pde7 inhibitors
ZA200704636B (en) 2-alkyl-cycloalk(en)yl-carboxamides
WO2007062308A3 (en) Homo- and heterocyclic compounds suitable as cetp inhibitors
ZA201005087B (en) 4-imidazolidinones as kv1.5 potassium channel inhibitors
IL180846A0 (en) 1,1,2,2-tetra (hetero) arylethanes or 1,1,2-tri (hetero) aryl-2-heterocyclylethanes as potassium channel inhibitors
ZA200810763B (en) Imidazolidinone Kv1.5 potassium channel inhibitors
ZA201005086B (en) 4-imidazolidinones as kv1.5 potassium channel inhibitors
ITMI20032493A1 (en) HANDLING FOR AN ALTERNATIVE COMPRESSOR.
EP1723145A4 (en) Substituted 5,12-diaza-benzoanthracene analogues
TW576286U (en) Nail-absence non-percussion device for nailing gun
AU2003301258A1 (en) Calcium channel agonists for psychotherapeutic use
AU2823P (en) P000607 Plectranthus hilliardiae x (P. saccatus x P. hilliardiae)
HK1122294A (en) Arylpropionamide, arylacrylamide, arylpropynamide, or arylmethylurea analogs as factor xia inhibitors