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IL166307A0 - Preparation of 1h-imidazoÄ4,5-cÜquinolin-4-amines via novel 1h-imidazoÄ4,5-cÜquinolin-4-cyano and 1h-imidazo Ä4,5-cÜquinolin-4-cyano and 1h-imidazoÄ4,5-cÜquinolin-4-carboxamide intermediates - Google Patents

Preparation of 1h-imidazoÄ4,5-cÜquinolin-4-amines via novel 1h-imidazoÄ4,5-cÜquinolin-4-cyano and 1h-imidazo Ä4,5-cÜquinolin-4-cyano and 1h-imidazoÄ4,5-cÜquinolin-4-carboxamide intermediates

Info

Publication number
IL166307A0
IL166307A0 IL16630703A IL16630703A IL166307A0 IL 166307 A0 IL166307 A0 IL 166307A0 IL 16630703 A IL16630703 A IL 16630703A IL 16630703 A IL16630703 A IL 16630703A IL 166307 A0 IL166307 A0 IL 166307A0
Authority
IL
Israel
Prior art keywords
cüquinolin
imidazoä4
cyano
imidazo
quinoline
Prior art date
Application number
IL16630703A
Other languages
English (en)
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed filed Critical
Publication of IL166307A0 publication Critical patent/IL166307A0/xx

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Veterinary Medicine (AREA)
  • Immunology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Virology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Breeding Of Plants And Reproduction By Means Of Culturing (AREA)
IL16630703A 2002-07-26 2003-07-28 Preparation of 1h-imidazoÄ4,5-cÜquinolin-4-amines via novel 1h-imidazoÄ4,5-cÜquinolin-4-cyano and 1h-imidazo Ä4,5-cÜquinolin-4-cyano and 1h-imidazoÄ4,5-cÜquinolin-4-carboxamide intermediates IL166307A0 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US39859202P 2002-07-26 2002-07-26
PCT/US2003/023543 WO2004011462A1 (en) 2002-07-26 2003-07-28 Preparation of 1h-imidazo [4,5-c] quinolin-4-amines via novel 1h-imidazo [4,5-c] quinolin-4-cyano and 1h-imidazo [4,5-c] quinolin-4-carboxamide intermediates

Publications (1)

Publication Number Publication Date
IL166307A0 true IL166307A0 (en) 2006-01-15

Family

ID=31188428

Family Applications (2)

Application Number Title Priority Date Filing Date
IL16630703A IL166307A0 (en) 2002-07-26 2003-07-28 Preparation of 1h-imidazoÄ4,5-cÜquinolin-4-amines via novel 1h-imidazoÄ4,5-cÜquinolin-4-cyano and 1h-imidazo Ä4,5-cÜquinolin-4-cyano and 1h-imidazoÄ4,5-cÜquinolin-4-carboxamide intermediates
IL166307A IL166307A (en) 2002-07-26 2005-01-16 Preparation of 1h-imidazo[4,5-c]quinolin-4-amines via 1h-imidazo [4,5-c]quinolin-4-cyano and 1h-imidazo [4,5-c]quinolin-4-carboxamide intermediates

Family Applications After (1)

Application Number Title Priority Date Filing Date
IL166307A IL166307A (en) 2002-07-26 2005-01-16 Preparation of 1h-imidazo[4,5-c]quinolin-4-amines via 1h-imidazo [4,5-c]quinolin-4-cyano and 1h-imidazo [4,5-c]quinolin-4-carboxamide intermediates

Country Status (18)

Country Link
US (3) US6841678B2 (de)
EP (1) EP1539752B1 (de)
JP (1) JP2005537287A (de)
KR (1) KR20050030958A (de)
CN (1) CN100372847C (de)
AT (1) ATE357445T1 (de)
AU (1) AU2003254221A1 (de)
CA (1) CA2493158A1 (de)
DE (1) DE60312701T8 (de)
DK (1) DK1539752T3 (de)
ES (1) ES2282691T3 (de)
HR (1) HRP20050183A2 (de)
IL (2) IL166307A0 (de)
MX (1) MXPA05000997A (de)
PL (1) PL374866A1 (de)
PT (1) PT1539752E (de)
SI (1) SI1539752T1 (de)
WO (1) WO2004011462A1 (de)

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Also Published As

Publication number Publication date
US7335772B2 (en) 2008-02-26
US7166721B2 (en) 2007-01-23
IL166307A (en) 2010-04-15
PT1539752E (pt) 2007-05-31
US6841678B2 (en) 2005-01-11
CN100372847C (zh) 2008-03-05
PL374866A1 (en) 2005-11-14
SI1539752T1 (sl) 2007-08-31
US20050119294A1 (en) 2005-06-02
AU2003254221A1 (en) 2004-02-16
JP2005537287A (ja) 2005-12-08
WO2004011462A1 (en) 2004-02-05
CA2493158A1 (en) 2004-02-05
ES2282691T3 (es) 2007-10-16
DK1539752T3 (da) 2007-07-16
MXPA05000997A (es) 2005-05-16
US20040063743A1 (en) 2004-04-01
CN1684963A (zh) 2005-10-19
ATE357445T1 (de) 2007-04-15
HRP20050183A2 (en) 2005-06-30
EP1539752A1 (de) 2005-06-15
EP1539752B1 (de) 2007-03-21
US20050101627A1 (en) 2005-05-12
DE60312701D1 (de) 2007-05-03
DE60312701T2 (de) 2007-12-06
KR20050030958A (ko) 2005-03-31
DE60312701T8 (de) 2008-08-21

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