IL164513A0 - Pyrazolopyrimidines, pharmaceutical compositions containing them, and their use in the preparation of medicaments - Google Patents

Pyrazolopyrimidines, pharmaceutical compositions containing them, and their use in the preparation of medicaments

Info

Publication number: IL164513A0
Authority: IL; Israel
Prior art keywords: pyrazolopyrimidines; medicaments; preparation; pharmaceutical compositions; compositions containing
Prior art date: 1996-07-24

Application number

IL16451304A

Other versions

IL164513A (en

Original Assignee

Du Pont Pharm Co

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1996-07-24

Filing date

2004-10-12

Publication date

2005-12-18

1997-07-23 Priority claimed from PCT/US1997/013072 external-priority patent/WO1998003510A1/en

1997-07-23 Priority claimed from US08/899,242 external-priority patent/US6124289A/en

2004-10-12 Application filed by Du Pont Pharm Co filed Critical Du Pont Pharm Co

2005-12-18 Publication of IL164513A0 publication Critical patent/IL164513A0/en

2010-04-29 Publication of IL164513A publication Critical patent/IL164513A/en

Links

IL164513A 1996-07-24 2004-10-12 Pyrazolopyrimidines, pharmaceutical compositions containing them and their use in the preparation of medicaments IL164513A (en)

Applications Claiming Priority (4)

Application Number	Priority Date	Filing Date	Title
US2329096P	1996-07-24	1996-07-24
US68604796A	1996-07-24	1996-07-24
PCT/US1997/013072 WO1998003510A1 (en)	1996-07-24	1997-07-23	AZOLO TRIAZINES AND PYRIMIDINES
US08/899,242 US6124289A (en)	1996-07-24	1997-07-23	Azolo triazines and pyrimidines

Publications (2)

Publication Number	Publication Date
IL164513A0 true IL164513A0 (en)	2005-12-18
IL164513A IL164513A (en)	2010-04-29

Family

ID=27362048

Family Applications (4)

Application Number	Title	Priority Date	Filing Date
IL12787197A IL127871A0 (en)	1996-07-24	1997-07-23	Azolo triazines and pyrimidines
IL127871A IL127871A (en)	1996-07-24	1998-12-30	PHARMACEUTICAL COMPOSITIONS CONTAINING CRF ANTAGONIST 3-ARYL-PYRAZOLO (AND 1,2,3-TRIAZOLO) [1,5-a]-1,3,5-TRIAZINE DERIVATIVES AND SOME NEW SUCH DERIVATIVES
IL150163A IL150163A (en)	1996-07-24	2002-06-11	PHARMACEUTICAL COMPOSITIONS COMPRISING PYRAZOLO[1,5-a]PYRIMIDINE DERIVATIVES AND SOME NOVEL SUCH COMPOUNDS
IL164513A IL164513A (en)	1996-07-24	2004-10-12	Pyrazolopyrimidines, pharmaceutical compositions containing them and their use in the preparation of medicaments

Family Applications Before (3)

Application Number	Title	Priority Date	Filing Date
IL12787197A IL127871A0 (en)	1996-07-24	1997-07-23	Azolo triazines and pyrimidines
IL127871A IL127871A (en)	1996-07-24	1998-12-30	PHARMACEUTICAL COMPOSITIONS CONTAINING CRF ANTAGONIST 3-ARYL-PYRAZOLO (AND 1,2,3-TRIAZOLO) [1,5-a]-1,3,5-TRIAZINE DERIVATIVES AND SOME NEW SUCH DERIVATIVES
IL150163A IL150163A (en)	1996-07-24	2002-06-11	PHARMACEUTICAL COMPOSITIONS COMPRISING PYRAZOLO[1,5-a]PYRIMIDINE DERIVATIVES AND SOME NOVEL SUCH COMPOUNDS

Country Status (15)

Country	Link
JP (2)	JP4704521B2 (en)
CN (3)	CN1104432C (en)
AR (1)	AR049583A2 (en)
BR (1)	BR9710544A (en)
CA (1)	CA2259583C (en)
CZ (1)	CZ299451B6 (en)
EA (1)	EA004403B1 (en)
EE (1)	EE04316B1 (en)
HR (1)	HRP970413A2 (en)
IL (4)	IL127871A0 (en)
NO (1)	NO315610B1 (en)
NZ (1)	NZ333777A (en)
PL (1)	PL195762B1 (en)
SI (1)	SI9720045B (en)
SK (1)	SK286461B6 (en)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
ES2282401T3 (en) *	2001-03-13	2007-10-16	Bristol-Myers Squibb Pharma Company	4- (2-BUTILAMINO) -2,7-DIMETHYL-8- (2-METHYL-6-METOXIPIRID-3-IL) PIRAZOLO - 1,5-A-1,3,5-TRIAZINE, ITS ENANTIOMERS AND PHARMACEUTICALLY SALTS ACCEPTABLE AS LIGANDS OF THE RECEIVER OF THE CROTICOTROPINE RELEASE FACTOR.
WO2004110454A1 (en) *	2003-06-13	2004-12-23	Ishihara Sangyo Kaisha, Ltd.	COMPOSITION FOR TREATMENT FOR OR PREVENTION OF DISEASE NECESSITATING ADMINISTRATION OF ADENOSINE A2a RECEPTOR AGONIST
US7329662B2 (en) *	2003-10-03	2008-02-12	Hoffmann-La Roche Inc.	Pyrazolo-pyridine
GB0519957D0 (en) *	2005-09-30	2005-11-09	Sb Pharmco Inc	Chemical compound
EP2094709B1 (en) *	2006-09-20	2010-09-15	Eli Lilly And Company	Thiazole pyrazolopyrimidines as crf1 receptor antagonists
CN103694242B (en) *	2013-12-10	2016-01-06	昆明翔昊科技有限公司	Pyrazolopyrimidines and pharmaceutical composition thereof and its application in pharmacy
US20210361664A1 (en)	2017-08-14	2021-11-25	Spruce Biosciences, Inc.	Corticotropin releasing factor receptor antagonists
CN112608316B (en) *	2019-07-30	2022-10-21	厦门宝太生物科技股份有限公司	Pyrazolotriazine adenosine receptor antagonist
MX2023001688A (en)	2020-08-12	2023-02-22	Spruce Biosciences Inc	METHODS AND COMPOSITIONS TO TREAT POLYCYSTIC OVARIAN SYNDROME.
US11708372B2 (en)	2021-11-19	2023-07-25	Spruce Biosciences, Inc.	Crystalline composition of tildacerfont and methods of use and preparation thereof

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US3995039A (en) *	1975-05-27	1976-11-30	Merck & Co., Inc.	Pyrazolo [1,5-a] [1,3,5] triazines
JPS6157587A (en) *	1984-08-29	1986-03-24	Shionogi & Co Ltd	Condensed heterocyclic derivative and antiulcerative
US4824834A (en) *	1986-10-31	1989-04-25	Otsuka Pharmaceutical Company, Limited	Pyrazolotriazine compounds
JP2691317B2 (en) *	1989-08-25	1997-12-17	株式会社大塚製薬工場	4-Hydroxy-8- (3-lower alkoxy-4-phenylsulfinylphenyl) pyrazolo [1,5-a] -1,3,5-triazine optically active salts and process for producing the same
AU639615B2 (en) *	1990-10-09	1993-07-29	Otsuka Pharmaceutical Co., Ltd.	Pyrimidine derivative, production thereof, and androgen inhibitor
ES2126573T3 (en) *	1991-04-22	1999-04-01	Otsuka Pharma Co Ltd	DERIVATIVE OF PYRAZOLE (1,5-A) PIRIMIDINE AND ANTI-INFLAMMATORY AGENT CONTAINING THIS DERIVATIVE.
US5356897A (en) *	1991-09-09	1994-10-18	Fujisawa Pharmaceutical Co., Ltd.	3-(heteroaryl)-pyrazololi[1,5-a]pyrimidines

1997
- 1997-07-23 EE EEP199900019A patent/EE04316B1/en unknown
- 1997-07-23 PL PL97331523A patent/PL195762B1/en unknown
- 1997-07-23 EA EA199900158A patent/EA004403B1/en not_active IP Right Cessation
- 1997-07-23 CA CA002259583A patent/CA2259583C/en not_active Expired - Lifetime
- 1997-07-23 BR BR9710544A patent/BR9710544A/en not_active IP Right Cessation
- 1997-07-23 JP JP50723398A patent/JP4704521B2/en not_active Expired - Fee Related
- 1997-07-23 SK SK97-99A patent/SK286461B6/en not_active IP Right Cessation
- 1997-07-23 IL IL12787197A patent/IL127871A0/en unknown
- 1997-07-23 CN CN97196525A patent/CN1104432C/en not_active Expired - Lifetime
- 1997-07-23 SI SI9720045A patent/SI9720045B/en active Search and Examination
- 1997-07-23 CZ CZ0018499A patent/CZ299451B6/en not_active IP Right Cessation
- 1997-07-23 NZ NZ333777A patent/NZ333777A/en not_active IP Right Cessation
- 1997-07-24 HR HRP970413 patent/HRP970413A2/en not_active Application Discontinuation
1998
- 1998-12-30 IL IL127871A patent/IL127871A/en not_active IP Right Cessation
1999
- 1999-01-21 NO NO19990264A patent/NO315610B1/en not_active IP Right Cessation
2001
- 2001-05-30 CN CN 01120849 patent/CN1250223C/en not_active Expired - Lifetime
2002
- 2002-04-25 CN CN 02118589 patent/CN1388126A/en active Pending
- 2002-06-11 IL IL150163A patent/IL150163A/en not_active IP Right Cessation
2004
- 2004-07-23 JP JP2004216483A patent/JP4194539B2/en not_active Expired - Fee Related
- 2004-10-12 IL IL164513A patent/IL164513A/en not_active IP Right Cessation
2005
- 2005-07-11 AR ARP050102868A patent/AR049583A2/en not_active Application Discontinuation

Also Published As

Publication number	Publication date
JP2002513382A (en)	2002-05-08
IL164513A (en)	2010-04-29
IL127871A (en)	2010-04-29
CN1327793A (en)	2001-12-26
IL127871A0 (en)	1999-10-28
PL195762B1 (en)	2007-10-31
NZ333777A (en)	2000-07-28
JP4194539B2 (en)	2008-12-10
EE04316B1 (en)	2004-06-15
SK9799A3 (en)	2005-04-01
CZ18499A3 (en)	1999-11-17
SI9720045A (en)	1999-10-31
NO315610B3 (en)	2003-09-29
AR049583A2 (en)	2006-08-16
PL331523A1 (en)	1999-07-19
EA004403B1 (en)	2004-04-29
SK286461B6 (en)	2008-10-07
CN1225637A (en)	1999-08-11
NO315610B1 (en)	2003-09-29
CA2259583C (en)	2009-11-17
IL150163A (en)	2010-12-30
CZ299451B6 (en)	2008-07-30
CN1104432C (en)	2003-04-02
CA2259583A1 (en)	1998-01-29
NO990264D0 (en)	1999-01-21
HRP970413A2 (en)	1998-10-31
BR9710544A (en)	1999-08-17
JP4704521B2 (en)	2011-06-15
NO990264L (en)	1999-03-10
CN1388126A (en)	2003-01-01
EE9900019A (en)	1999-08-16
SI9720045B (en)	2008-02-29
CN1250223C (en)	2006-04-12
EA199900158A1 (en)	1999-10-28
JP2005097257A (en)	2005-04-14

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Legal Events

Date	Code	Title
2010-11-30	FF	Patent granted
2015-06-30	KB	Patent renewed
2018-02-28	EXP	Patent expired