IL142502A0 - Intermediates for the preparation of biologically active benzothiazolone ethanamines - Google Patents

Intermediates for the preparation of biologically active benzothiazolone ethanamines

Info

Publication number: IL142502A0
Authority: IL; Israel
Prior art keywords: ethanamines; intermediates; preparation; biologically active; benzothiazolone
Prior art date: 1995-12-23

Application number

IL14250296A

Other languages

English (en)

Original Assignee

Astrazeneca Ab

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1995-12-23

Filing date

1996-12-13

Publication date

2002-03-10

1996-12-13 Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab

2002-03-10 Publication of IL142502A0 publication Critical patent/IL142502A0/xx

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/60—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
- C07D277/62—Benzothiazoles
- C07D277/68—Benzothiazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/425—Thiazoles
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Pharmacology & Pharmacy (AREA)
Animal Behavior & Ethology (AREA)
Pulmonology (AREA)
Veterinary Medicine (AREA)
Public Health (AREA)
Medicinal Chemistry (AREA)
General Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
General Chemical & Material Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
Epidemiology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Thiazole And Isothizaole Compounds (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)

IL14250296A 1995-12-23 1996-12-13 Intermediates for the preparation of biologically active benzothiazolone ethanamines IL142502A0 (en)

Applications Claiming Priority (3)

Application Number	Priority Date	Filing Date	Title
GBGB9526511.2A GB9526511D0 (en)	1995-12-23	1995-12-23	Pharmaceutically active compounds
IL12499896A IL124998A0 (en)	1995-12-23	1996-12-13	Biologically active benzothiazolone ethanamines
PCT/SE1996/001650 WO1997023470A1 (en)	1995-12-23	1996-12-13	Biologically active benzothiazolone ethanamines

Publications (1)

Publication Number	Publication Date
IL142502A0 true IL142502A0 (en)	2002-03-10

Family

ID=10786064

Family Applications (2)

Application Number	Title	Priority Date	Filing Date
IL12499896A IL124998A0 (en)	1995-12-23	1996-12-13	Biologically active benzothiazolone ethanamines
IL14250296A IL142502A0 (en)	1995-12-23	1996-12-13	Intermediates for the preparation of biologically active benzothiazolone ethanamines

Family Applications Before (1)

Application Number	Title	Priority Date	Filing Date
IL12499896A IL124998A0 (en)	1995-12-23	1996-12-13	Biologically active benzothiazolone ethanamines

Country Status (27)

Country	Link
US (1)	US5929100A (et)
EP (1)	EP0918760B1 (et)
JP (1)	JP2000502681A (et)
KR (1)	KR19990076688A (et)
CN (1)	CN1072214C (et)
AR (1)	AR005008A1 (et)
AT (1)	ATE209638T1 (et)
AU (1)	AU704506B2 (et)
BR (1)	BR9612234A (et)
CA (1)	CA2238877A1 (et)
CZ (1)	CZ288704B6 (et)
DE (1)	DE69617472D1 (et)
EE (1)	EE03440B1 (et)
GB (1)	GB9526511D0 (et)
HU (1)	HUP9900100A3 (et)
IL (2)	IL124998A0 (et)
IS (1)	IS4759A (et)
MX (1)	MX9804828A (et)
NO (1)	NO982927L (et)
NZ (1)	NZ325500A (et)
PL (1)	PL327475A1 (et)
RU (1)	RU2177476C2 (et)
SK (1)	SK82098A3 (et)
TR (1)	TR199801196T2 (et)
TW (1)	TW401411B (et)
WO (1)	WO1997023470A1 (et)
ZA (1)	ZA9610354B (et)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
WO1999009018A1 (en) *	1997-08-14	1999-02-25	Kirin Beer Kabushiki Kaisha	BENZOTHIAZOLONE DERIVATIVES HAVING SELECTIVE β2 RECEPTOR AGONIST ACTIVITY
GB0218629D0 (en) *	2002-08-09	2002-09-18	Novartis Ag	Organic compounds
AR040962A1 (es) *	2002-08-09	2005-04-27	Novartis Ag	Compuestos derivados de tiazol 1,3-2-ona, composicion farmaceutica y proceso de preparacion del compuesto
DE602004021959D1 (de)	2003-11-21	2009-08-20	Theravance Inc	Verbindungen mit agonistischer wirkung am beta2-adrenergen rezeptor und am muscarinischen rezeptor
TW200738658A (en)	2005-08-09	2007-10-16	Astrazeneca Ab	Novel compounds
TW200738659A (en) *	2005-08-29	2007-10-16	Astrazeneca Ab	Novel compounds
TW200745067A (en)	2006-03-14	2007-12-16	Astrazeneca Ab	Novel compounds
TW200833670A (en)	2006-12-20	2008-08-16	Astrazeneca Ab	Novel compounds 569
GB0702458D0 (en)	2007-02-08	2007-03-21	Astrazeneca Ab	Salts 668
MX2010013477A (es)	2008-06-18	2010-12-21	Astrazeneca Ab	Derivados de benzoxazinona que actuan como agonistas de receptores adrenergicos beta2 para el tratamiento de trastornos respiratorios.

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4314944A (en) *	1980-08-22	1982-02-09	Smithkline Corporation	4-Aminoalkyl-7-hydroxy-2(3H)-indolones
US4452808A (en) *	1982-12-07	1984-06-05	Smithkline Beckman Corporation	4-Aminoalkyl-2(3H)-indolones
GB8426200D0 (en) *	1984-10-17	1984-11-21	Glaxo Holdings Ltd	Chemical compounds
US4554287A (en) *	1984-09-12	1985-11-19	Smithkline Beckman Corporation	Antihypertensive 7-[2-(dialkylamino)ethyl]-4-hydroxy-1,3-benzimidazol-2-ones
US4554284A (en) *	1984-09-12	1985-11-19	Smithkline Beckman Corporation	7-(2-Aminoethyl)-1,3-benzthia- or oxa-zol-2(3H)-ones
ES8606847A1 (es) *	1984-11-08	1986-05-16	Syntex Inc	Procedimiento para la preparacion de derivados de dialquila-mino-etilanilina antihipertensos
DE3728695A1 (de) *	1987-08-25	1989-03-09	Schering Ag	Neue benzimidazol-derivate
GB9210632D0 (en) *	1992-05-19	1992-07-01	Fisons Plc	Compounds
US5648370A (en) *	1990-11-20	1997-07-15	Astra Pharmaceuticals Limited	7-(2-aminoethyl) benzothiazolones
GB9211172D0 (en) *	1992-05-27	1992-07-08	Fisons Plc	Compounds
IE914003A1 (en) *	1990-11-20	1992-05-20	Astra Pharma Prod	Biologically Active Amines

1995
- 1995-12-23 GB GBGB9526511.2A patent/GB9526511D0/en active Pending
1996
- 1996-12-09 AR ARP960105568A patent/AR005008A1/es unknown
- 1996-12-09 ZA ZA9610354A patent/ZA9610354B/xx unknown
- 1996-12-11 TW TW085115316A patent/TW401411B/zh not_active IP Right Cessation
- 1996-12-13 HU HU9900100A patent/HUP9900100A3/hu unknown
- 1996-12-13 PL PL96327475A patent/PL327475A1/xx unknown
- 1996-12-13 WO PCT/SE1996/001650 patent/WO1997023470A1/en not_active Ceased
- 1996-12-13 JP JP09523560A patent/JP2000502681A/ja active Pending
- 1996-12-13 AU AU14025/97A patent/AU704506B2/en not_active Ceased
- 1996-12-13 SK SK820-98A patent/SK82098A3/sk unknown
- 1996-12-13 IL IL12499896A patent/IL124998A0/xx unknown
- 1996-12-13 AT AT96944153T patent/ATE209638T1/de not_active IP Right Cessation
- 1996-12-13 NZ NZ325500A patent/NZ325500A/xx unknown
- 1996-12-13 DE DE69617472T patent/DE69617472D1/de not_active Expired - Lifetime
- 1996-12-13 KR KR1019980704800A patent/KR19990076688A/ko not_active Withdrawn
- 1996-12-13 CZ CZ19981684A patent/CZ288704B6/cs not_active IP Right Cessation
- 1996-12-13 RU RU98114080/04A patent/RU2177476C2/ru active
- 1996-12-13 CA CA002238877A patent/CA2238877A1/en not_active Abandoned
- 1996-12-13 IL IL14250296A patent/IL142502A0/xx unknown
- 1996-12-13 TR TR1998/01196T patent/TR199801196T2/xx unknown
- 1996-12-13 EP EP96944153A patent/EP0918760B1/en not_active Expired - Lifetime
- 1996-12-13 CN CN96199237A patent/CN1072214C/zh not_active Expired - Fee Related
- 1996-12-13 EE EE9800193A patent/EE03440B1/et not_active IP Right Cessation
- 1996-12-13 BR BR9612234A patent/BR9612234A/pt not_active Application Discontinuation
- 1996-12-13 US US08/793,706 patent/US5929100A/en not_active Expired - Fee Related
1998
- 1998-05-27 IS IS4759A patent/IS4759A/is unknown
- 1998-06-16 MX MX9804828A patent/MX9804828A/es unknown
- 1998-06-23 NO NO982927A patent/NO982927L/no not_active Application Discontinuation

Also Published As

Publication number	Publication date
NO982927D0 (no)	1998-06-23
DE69617472D1 (de)	2002-01-10
NO982927L (no)	1998-06-23
TR199801196T2 (xx)	1998-10-21
EP0918760B1 (en)	2001-11-28
AU704506B2 (en)	1999-04-22
CZ288704B6 (cs)	2001-08-15
GB9526511D0 (en)	1996-02-28
EP0918760A1 (en)	1999-06-02
HUP9900100A3 (en)	2001-10-29
RU2177476C2 (ru)	2001-12-27
EE9800193A (et)	1998-12-15
ZA9610354B (en)	1997-06-23
AU1402597A (en)	1997-07-17
KR19990076688A (ko)	1999-10-15
SK82098A3 (en)	1998-11-04
IS4759A (is)	1998-05-27
IL124998A0 (en)	1999-01-26
PL327475A1 (en)	1998-12-07
EE03440B1 (et)	2001-06-15
CA2238877A1 (en)	1997-07-03
HUP9900100A2 (hu)	1999-05-28
ATE209638T1 (de)	2001-12-15
CN1072214C (zh)	2001-10-03
NZ325500A (en)	1999-01-28
JP2000502681A (ja)	2000-03-07
TW401411B (en)	2000-08-11
US5929100A (en)	1999-07-27
AR005008A1 (es)	1999-04-07
CN1211242A (zh)	1999-03-17
MX9804828A (es)	1998-09-30
CZ168498A3 (cs)	1998-09-16
WO1997023470A1 (en)	1997-07-03
BR9612234A (pt)	1999-07-13

Publication	Publication Date	Title
PL323152A1 (en)	1998-03-16	Derivatives of 1,3-propanodiole as biologically active compounds
EG21973A (en)	2002-05-31	A new process for the preparation of a pharmacolgically active substance
ZA9811531B (en)	1999-06-15	Novel process for the preparation of cyclosporin derivatives
HUP9602510A1 (en)	1997-05-28	Preparation of substituted thiazoles
AU4515996A (en)	1996-07-31	Methods for increasing the bioavailability of biological active agents
AU8329498A (en)	1999-02-10	Diagnosis of edema
BG98019A (en)	1994-06-30	Method for the preparation of biologically active substances
AU8758298A (en)	1999-02-16	Process for the preparation of 2'-fluoro-5-methyl-beta -l-arabinofuranosyluridine
IL142502A0 (en)	2002-03-10	Intermediates for the preparation of biologically active benzothiazolone ethanamines
AU7310896A (en)	1997-05-07	Use of nitroflavonoids for the treatment of anxiety
ZA968230B (en)	1997-04-09	Administration of biologically active material
HUP9903751A3 (en)	2001-11-28	Intermediates for the preparation of 2-imidazoline-5-ones
ZA987741B (en)	1998-10-08	Process for the preparation of oxazaphosphorine-2-amines
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AP9600854A0 (en)	1996-10-31	Polymorphs of the pro drug 6 N-(L-ALA-L-ALA) - trovafloxacin
GB9402189D0 (en)	1994-03-30	Biologically active formulations
AU4708697A (en)	1999-05-17	Process for the preparation of eberconazol and intermediates thereof
HUP9600316A3 (en)	1998-11-30	Process for the preparation of n-(ortho-alkyl-phenyl)-imides
IL132237A0 (en)	2001-03-19	Process for the preparation of 3-isochromanome
GB2287707B (en)	1998-02-25	Intermediates for biologically active products
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GB2305172B (en)	1998-11-18	Preparation of substituted thiazoles
ZA981924B (en)	1998-09-07	Process for the preparation of n-carboxylalkyl-3-fluoro-4- dialkylaminoanilines