IL142460A0 - A vitreous form of 8-[3-[n-[(e)-3-(6-acetamidopyridin-3-yl) acryloyl-glycyl] -n-methylamino] -2,6-dichlorobenzyloxy]-2-methylquinoline - Google Patents

A vitreous form of 8-[3-[n-[(e)-3-(6-acetamidopyridin-3-yl) acryloyl-glycyl] -n-methylamino] -2,6-dichlorobenzyloxy]-2-methylquinoline

Info

Publication number: IL142460A0
Authority: IL; Israel
Prior art keywords: acetamidopyridin; dichlorobenzyloxy; methylquinoline; glycyl; acryloyl
Prior art date: 1998-10-21

Application number

IL14246099A

Other languages

English (en)

Original Assignee

Fujisawa Pharmaceutical Co

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1998-10-21

Filing date

1999-10-07

Publication date

2002-03-10

1999-10-07 Application filed by Fujisawa Pharmaceutical Co filed Critical Fujisawa Pharmaceutical Co

2002-03-10 Publication of IL142460A0 publication Critical patent/IL142460A0/xx

Links

XCKWRUGRUFVXGC-NTEUORMPSA-N (e)-3-(6-acetamidopyridin-3-yl)-n-[2-[2,4-dichloro-n-methyl-3-[(2-methylquinolin-8-yl)oxymethyl]anilino]-2-oxoethyl]prop-2-enamide Chemical compound C=1C=C(Cl)C(COC=2C3=NC(C)=CC=C3C=CC=2)=C(Cl)C=1N(C)C(=O)CNC(=O)\C=C\C1=CC=C(NC(C)=O)N=C1 XCKWRUGRUFVXGC-NTEUORMPSA-N 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
- A61K31/4709—Non-condensed quinolines and containing further heterocyclic rings
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents

Landscapes

Chemical & Material Sciences (AREA)
Health & Medical Sciences (AREA)
Organic Chemistry (AREA)
Life Sciences & Earth Sciences (AREA)
Pharmacology & Pharmacy (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Engineering & Computer Science (AREA)
Immunology (AREA)
Bioinformatics & Cheminformatics (AREA)
Pulmonology (AREA)
Epidemiology (AREA)
Pain & Pain Management (AREA)
Rheumatology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)
Medicinal Preparation (AREA)
Pyridine Compounds (AREA)

IL14246099A 1998-10-21 1999-10-07 A vitreous form of 8-[3-[n-[(e)-3-(6-acetamidopyridin-3-yl) acryloyl-glycyl] -n-methylamino] -2,6-dichlorobenzyloxy]-2-methylquinoline IL142460A0 (en)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
JP29925298		1998-10-21
PCT/JP1999/005519 WO2000023439A1 (en)	1998-10-21	1999-10-07	Vitreous form of known bradykinin antagonist

Publications (1)

Publication Number	Publication Date
IL142460A0 true IL142460A0 (en)	2002-03-10

Family

ID=17870134

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
IL14246099A IL142460A0 (en)	1998-10-21	1999-10-07	A vitreous form of 8-[3-[n-[(e)-3-(6-acetamidopyridin-3-yl) acryloyl-glycyl] -n-methylamino] -2,6-dichlorobenzyloxy]-2-methylquinoline

Country Status (18)

Country	Link
US (2)	US6509468B1 (es)
EP (1)	EP1123288A1 (es)
JP (1)	JP3353784B2 (es)
KR (1)	KR100419404B1 (es)
CN (1)	CN1144801C (es)
AR (1)	AR024220A1 (es)
AU (1)	AU756479B2 (es)
BR (1)	BR9914785A (es)
CA (1)	CA2347001A1 (es)
CZ (1)	CZ20011417A3 (es)
HK (1)	HK1040245B (es)
HU (1)	HUP0104110A3 (es)
IL (1)	IL142460A0 (es)
RU (1)	RU2202550C2 (es)
TR (1)	TR200101101T2 (es)
TW (1)	TWI230158B (es)
WO (1)	WO2000023439A1 (es)
ZA (1)	ZA200102607B (es)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
WO2001092254A1 (en) *	2000-05-30	2001-12-06	Fujisawa Pharmaceutical Co., Ltd.	Method for replacing organic solvents contained in clathrate crystals
JP2005525398A (ja) *	2002-04-10	2005-08-25	オーソ−マクニール・フアーマシユーチカル・インコーポレーテツド	ブラジキニン受容体モジュレーターとして有用な新規なヘテロアリールアルキルアミド誘導体
TWI407960B (zh)	2007-03-23	2013-09-11	Jerini Ag	小分子緩激肽ｂ２受體調節劑
SMT202200154T1 (it)	2017-11-24	2022-05-12	Pharvaris Netherlands B V	Nuovi antagonisti del recettore della bradichinina b2
AR118982A1 (es)	2019-05-23	2021-11-17	Pharvaris Gmbh	Antagonistas cíclicos del receptor b2 de bradiquinina
UY38707A (es)	2019-05-23	2020-12-31	Pharvaris Gmbh	Nuevos antagonistas cíclicos del receptor b2 de bradiquinina
TW202345810A (zh)	2022-03-25	2023-12-01	瑞士商帕法瑞斯有限責任公司	包含緩激肽ｂ２受體拮抗劑之固態延長釋放組成物
EP4499038B1 (en)	2022-03-25	2025-12-03	Pharvaris GmbH	Solid composition comprising solubilised bradykinin b2-receptor antagonists
US20250268887A1 (en)	2022-03-25	2025-08-28	Pharvaris Gmbh	Therapeutic uses of bradykinin b2-receptor antagonists

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US558455A (en) *		1896-04-14		Thomas lewty
GB8927913D0 (en) *	1989-12-11	1990-02-14	Hoffmann La Roche	Amino acid derivatives
AU680870B2 (en) *	1993-04-28	1997-08-14	Astellas Pharma Inc.	New heterocyclic compounds
JP3049648B2 (ja)	1993-12-13	2000-06-05	日立金属株式会社	加圧成形方法および加圧成形機
US5958455A (en) *	1996-02-09	1999-09-28	Quadrant Holdings Cambridge Ltd	Oral solid dosage forms, methods of making same and compositions thereof
JPH10316677A (ja)	1997-05-19	1998-12-02	Fujisawa Pharmaceut Co Ltd	結晶

1999
- 1999-10-07 HK HK02101581.1A patent/HK1040245B/zh not_active IP Right Cessation
- 1999-10-07 CN CNB998124419A patent/CN1144801C/zh not_active Expired - Fee Related
- 1999-10-07 US US09/807,421 patent/US6509468B1/en not_active Expired - Fee Related
- 1999-10-07 HU HU0104110A patent/HUP0104110A3/hu unknown
- 1999-10-07 WO PCT/JP1999/005519 patent/WO2000023439A1/en not_active Ceased
- 1999-10-07 AU AU60043/99A patent/AU756479B2/en not_active Ceased
- 1999-10-07 CA CA002347001A patent/CA2347001A1/en not_active Abandoned
- 1999-10-07 TR TR2001/01101T patent/TR200101101T2/xx unknown
- 1999-10-07 IL IL14246099A patent/IL142460A0/xx unknown
- 1999-10-07 RU RU2001113511/04A patent/RU2202550C2/ru not_active IP Right Cessation
- 1999-10-07 BR BR9914785-8A patent/BR9914785A/pt not_active IP Right Cessation
- 1999-10-07 EP EP99970660A patent/EP1123288A1/en not_active Withdrawn
- 1999-10-07 CZ CZ20011417A patent/CZ20011417A3/cs unknown
- 1999-10-07 JP JP2000577166A patent/JP3353784B2/ja not_active Expired - Fee Related
- 1999-10-07 KR KR10-2001-7003995A patent/KR100419404B1/ko not_active Expired - Fee Related
- 1999-10-12 AR ARP990105154A patent/AR024220A1/es unknown
- 1999-10-18 TW TW088117980A patent/TWI230158B/zh not_active IP Right Cessation
2001
- 2001-03-29 ZA ZA200102607A patent/ZA200102607B/en unknown
2002
- 2002-11-22 US US10/301,614 patent/US7094899B2/en not_active Expired - Fee Related

Also Published As

Publication number	Publication date
HK1040245A1 (en)	2002-05-31
RU2202550C2 (ru)	2003-04-20
TR200101101T2 (tr)	2001-09-21
ZA200102607B (en)	2002-07-01
WO2000023439A1 (en)	2000-04-27
HUP0104110A2 (hu)	2002-03-28
KR100419404B1 (ko)	2004-02-21
CA2347001A1 (en)	2000-04-27
HK1040245B (zh)	2004-10-08
CN1324354A (zh)	2001-11-28
HUP0104110A3 (en)	2003-01-28
AU756479B2 (en)	2003-01-16
US20030120076A1 (en)	2003-06-26
CN1144801C (zh)	2004-04-07
JP2002527514A (ja)	2002-08-27
US7094899B2 (en)	2006-08-22
AU6004399A (en)	2000-05-08
CZ20011417A3 (cs)	2001-09-12
BR9914785A (pt)	2001-07-03
KR20010075445A (ko)	2001-08-09
JP3353784B2 (ja)	2002-12-03
US6509468B1 (en)	2003-01-21
TWI230158B (en)	2005-04-01
AR024220A1 (es)	2002-09-25
EP1123288A1 (en)	2001-08-16

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