IL120446A - Preparation of esters of 9-(hetero)aryl-2,3,4,5,6,9-hexahydropyrido¬2,3-f¾¬1,4¾thiazepine-8-carboxylic acid 1,1-dioxides - Google Patents

Preparation of esters of 9-(hetero)aryl-2,3,4,5,6,9-hexahydropyrido¬2,3-f¾¬1,4¾thiazepine-8-carboxylic acid 1,1-dioxides

Info

Publication number: IL120446A
Authority: IL; Israel
Prior art keywords: hexahydropyrido; dioxides; hetero; aryl; esters
Prior art date: 1990-05-03

Application number

IL12044691A

Other languages

English (en)

Original Assignee

Ortho Pharma Corp

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1990-05-03

Filing date

1991-04-29

Publication date

2000-08-31

1991-04-29 Application filed by Ortho Pharma Corp filed Critical Ortho Pharma Corp

1991-04-29 Priority to IL12704791A priority Critical patent/IL127047A/xx

2000-08-31 Publication of IL120446A publication Critical patent/IL120446A/xx

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/06—Anti-spasmodics, e.g. drugs for colics, esophagic dyskinesia
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/08—Bronchodilators
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/06—Antimigraine agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
- A61P27/06—Antiglaucoma agents or miotics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
- A61P27/14—Decongestants or antiallergics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/02—Non-specific cardiovascular stimulants, e.g. drugs for syncope, antihypotensives
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/08—Vasodilators for multiple indications
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Life Sciences & Earth Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Pharmacology & Pharmacy (AREA)
Veterinary Medicine (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Cardiology (AREA)
Heart & Thoracic Surgery (AREA)
Pulmonology (AREA)
Ophthalmology & Optometry (AREA)
Neurology (AREA)
Urology & Nephrology (AREA)
Neurosurgery (AREA)
Pain & Pain Management (AREA)
Biomedical Technology (AREA)
Hospice & Palliative Care (AREA)
Immunology (AREA)
Vascular Medicine (AREA)
Endocrinology (AREA)
Reproductive Health (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
Preparation Of Compounds By Using Micro-Organisms (AREA)
Plural Heterocyclic Compounds (AREA)
Luminescent Compositions (AREA)

IL12044691A 1990-05-03 1991-04-29 Preparation of esters of 9-(hetero)aryl-2,3,4,5,6,9-hexahydropyrido¬2,3-f¾¬1,4¾thiazepine-8-carboxylic acid 1,1-dioxides IL120446A (en)

Priority Applications (1)

Application Number	Priority Date	Filing Date	Title
IL12704791A IL127047A (en)	1990-05-03	1991-04-29	Preparation of esters of 4-aryl-1,4,10,11-tetrahydropyrido¬3,2-b¾¬1,5¾benzothiazepine-3-carboxylic acid 5,5-dioxide

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US07/518,351 US5075440A (en)	1990-05-03	1990-05-03	Novel pyrido[2,3-f](1,4)thiazepines and pyrido[3,2-b](1,5)benzothiazepines
IL97999A IL97999A (en)	1990-05-03	1991-04-29	PYRIDO £2, 3-f\| £1, 4\| THIAZEPINES AND PYRIDO £3, 2-b\| £1, 5\|- BENZOTHIAZEPINES

Publications (1)

Publication Number	Publication Date
IL120446A true IL120446A (en)	2000-08-31

Family

ID=24063558

Family Applications (6)

Application Number	Title	Priority Date	Filing Date
IL12704798A IL127047A0 (en)	1990-05-03	1991-04-29	Preparation of pyrido [3,2-b] [1,5]-benzothiazepines
IL12044691A IL120446A (en)	1990-05-03	1991-04-29	Preparation of esters of 9-(hetero)aryl-2,3,4,5,6,9-hexahydropyrido¬2,3-f¾¬1,4¾thiazepine-8-carboxylic acid 1,1-dioxides
IL12044697A IL120446A0 (en)	1990-05-03	1991-04-29	Preparation of pyrido[2,3-f][1,4]thiazepines and pyrido[3,2-b][1,5]benzothiazepines
IL12044797A IL120447A (en)	1990-05-03	1991-04-29	Pharmaceutical compositions containing pyrido [2,3-f][1,4] thiazepines and pyrido [3,2-b][1,5]-benzothiazepines
IL12704791A IL127047A (en)	1990-05-03	1991-04-29	Preparation of esters of 4-aryl-1,4,10,11-tetrahydropyrido¬3,2-b¾¬1,5¾benzothiazepine-3-carboxylic acid 5,5-dioxide
IL97999A IL97999A (en)	1990-05-03	1991-04-29	PYRIDO £2, 3-f\| £1, 4\| THIAZEPINES AND PYRIDO £3, 2-b\| £1, 5\|- BENZOTHIAZEPINES

Family Applications Before (1)

Application Number	Title	Priority Date	Filing Date
IL12704798A IL127047A0 (en)	1990-05-03	1991-04-29	Preparation of pyrido [3,2-b] [1,5]-benzothiazepines

Family Applications After (4)

Application Number	Title	Priority Date	Filing Date
IL12044697A IL120446A0 (en)	1990-05-03	1991-04-29	Preparation of pyrido[2,3-f][1,4]thiazepines and pyrido[3,2-b][1,5]benzothiazepines
IL12044797A IL120447A (en)	1990-05-03	1991-04-29	Pharmaceutical compositions containing pyrido [2,3-f][1,4] thiazepines and pyrido [3,2-b][1,5]-benzothiazepines
IL12704791A IL127047A (en)	1990-05-03	1991-04-29	Preparation of esters of 4-aryl-1,4,10,11-tetrahydropyrido¬3,2-b¾¬1,5¾benzothiazepine-3-carboxylic acid 5,5-dioxide
IL97999A IL97999A (en)	1990-05-03	1991-04-29	PYRIDO £2, 3-f\| £1, 4\| THIAZEPINES AND PYRIDO £3, 2-b\| £1, 5\|- BENZOTHIAZEPINES

Country Status (25)

Country	Link
US (1)	US5075440A (xx)
EP (1)	EP0462696B1 (xx)
JP (1)	JP3296499B2 (xx)
KR (1)	KR100195345B1 (xx)
CN (2)	CN1034077C (xx)
AT (1)	ATE126231T1 (xx)
AU (1)	AU651580B2 (xx)
CA (1)	CA2041594C (xx)
DE (1)	DE69111915T2 (xx)
DK (1)	DK0462696T3 (xx)
ES (1)	ES2079570T3 (xx)
FI (1)	FI95912C (xx)
GR (1)	GR3017305T3 (xx)
HK (1)	HK51496A (xx)
HU (1)	HU218909B (xx)
IE (1)	IE68524B1 (xx)
IL (6)	IL127047A0 (xx)
MY (1)	MY106552A (xx)
NO (1)	NO179411C (xx)
NZ (1)	NZ237988A (xx)
PT (1)	PT97547B (xx)
TN (1)	TNSN91030A1 (xx)
TW (1)	TW218878B (xx)
ZA (1)	ZA913319B (xx)
ZW (1)	ZW5291A1 (xx)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US6265417B1 (en)	1997-12-18	2001-07-24	Abbott Laboratories	Potassium channel openers
CN1158259C (zh) *	1997-12-18	2004-07-21	艾博特公司	钾通道疏通剂
US6593335B1 (en) *	1997-12-18	2003-07-15	Abbott Laboratories	Potassium channel openers
JPH11193289A (ja)	1997-12-26	1999-07-21	Suntory Ltd	ピロールスルホンアミド誘導体
US6482854B1 (en) *	1999-03-25	2002-11-19	Massachusetts Eye And Ear Infirmary	Glaucoma treatment
US7015212B1 (en)	1999-05-12	2006-03-21	The United States Of America As Represented By The Department Of Health And Human Services	Thiazepine inhibitors of HIV-1 integrase
ES2207523T3 (es)	1999-06-14	2004-06-01	Ortho-Mcneil Pharmaceutical, Inc.	DITIEPINO (6,5-b)PIRIDINA Y COMPOSICIONES Y PROCEDIMIENTOS ASOCIADOS.
BR0012386A (pt) *	1999-07-12	2002-05-28	Ortho Mcneil Pharmaceutical Co	(oxatiepino-[6,5-b]-dihidropiridinas e composições e processos relacionados
AU7102700A (en) *	1999-09-22	2001-04-24	Ortho-Mcneil Pharmaceutical, Inc.	Benzo-fused dithiepino[6,5-b]pyridines, and related compositions and methods
DK1246828T3 (da) *	2000-01-12	2006-04-03	Ortho Mcneil Pharm Inc	Benzosulfoner med calciummantagonist-aktivitet
MXPA02007350A (es) *	2000-01-27	2004-06-21	Johnson & Johnson	Derivados de benzoxatiepino[3,4-b]piridina, procedimiento para su preparacion y su uso como medicamentos.
CN1247593C (zh)	2000-03-23	2006-03-29	奥索-麦克尼尔药品公司	噻庚英并[3,2－b]二氢吡啶和相关组合物及方法
US6562824B2 (en)	2000-05-30	2003-05-13	Ortho-Mcneil Pharmaceutical, Inc.	Dihydropyridine soft drugs, and related compositions and methods
KR101233139B1 (ko)	2011-04-21	2013-02-21	주식회사 한서켐	라세믹 1,4-티아제핀 화합물의 분할 방법
CN107454842A (zh) *	2014-12-30	2017-12-08	莫尔瑟瑞克斯股份有限公司	新型钙调节剂

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB1587128A (en) *	1977-04-07	1981-04-01	Hexachimie	Benzothiazepine derivatives
US4285955A (en) *	1978-10-31	1981-08-25	Bayer Aktiengesellschaft	1,4-Dihydropyridinecarboxylic acids
NZ201395A (en) *	1981-07-30	1987-02-20	Bayer Ag	Pharmaceutical compositions containing 1,4-dihydropyridines and certain of these dihydropyridines
FR2511683A1 (fr) *	1981-08-20	1983-02-25	Hexachimie	Nouveaux derives de la pyrido (2,3-b) benzothiazepine(1,5) substituee en 5 par une carboxypiperazine, leur procede de preparation, leur application en therapeutique
EP0225175A3 (en) *	1985-11-28	1988-12-28	FISONS plc	Dihydropyridine derivatives, processes for their preparation and pharmaceutical compositions thereof

1990
- 1990-05-03 US US07/518,351 patent/US5075440A/en not_active Expired - Lifetime
1991
- 1991-04-29 NZ NZ237988A patent/NZ237988A/xx unknown
- 1991-04-29 IL IL12704798A patent/IL127047A0/xx unknown
- 1991-04-29 IL IL12044691A patent/IL120446A/xx not_active IP Right Cessation
- 1991-04-29 IL IL12044697A patent/IL120446A0/xx unknown
- 1991-04-29 IL IL12044797A patent/IL120447A/xx not_active IP Right Cessation
- 1991-04-29 IL IL12704791A patent/IL127047A/xx not_active IP Right Cessation
- 1991-04-29 IL IL97999A patent/IL97999A/xx not_active IP Right Cessation
- 1991-05-01 CA CA002041594A patent/CA2041594C/en not_active Expired - Fee Related
- 1991-05-02 ZA ZA913319A patent/ZA913319B/xx unknown
- 1991-05-02 MY MYPI91000748A patent/MY106552A/en unknown
- 1991-05-02 DK DK91303970.7T patent/DK0462696T3/da active
- 1991-05-02 JP JP13047291A patent/JP3296499B2/ja not_active Expired - Fee Related
- 1991-05-02 NO NO911723A patent/NO179411C/no unknown
- 1991-05-02 ZW ZW52/91A patent/ZW5291A1/xx unknown
- 1991-05-02 EP EP91303970A patent/EP0462696B1/en not_active Expired - Lifetime
- 1991-05-02 AU AU76354/91A patent/AU651580B2/en not_active Ceased
- 1991-05-02 IE IE148891A patent/IE68524B1/en not_active IP Right Cessation
- 1991-05-02 KR KR1019910007086A patent/KR100195345B1/ko not_active Expired - Fee Related
- 1991-05-02 FI FI912124A patent/FI95912C/fi active
- 1991-05-02 ES ES91303970T patent/ES2079570T3/es not_active Expired - Lifetime
- 1991-05-02 PT PT97547A patent/PT97547B/pt not_active IP Right Cessation
- 1991-05-02 HU HU476/91A patent/HU218909B/hu not_active IP Right Cessation
- 1991-05-02 AT AT91303970T patent/ATE126231T1/de not_active IP Right Cessation
- 1991-05-02 DE DE69111915T patent/DE69111915T2/de not_active Expired - Fee Related
- 1991-05-03 TN TNTNSN91030A patent/TNSN91030A1/fr unknown
- 1991-05-03 CN CN91103594A patent/CN1034077C/zh not_active Expired - Fee Related
- 1991-07-20 TW TW080105637A patent/TW218878B/zh active
1995
- 1995-07-29 CN CN95109346A patent/CN1039416C/zh not_active Expired - Fee Related
- 1995-09-06 GR GR950402432T patent/GR3017305T3/el unknown
1996
- 1996-03-21 HK HK51496A patent/HK51496A/en not_active IP Right Cessation

Also Published As

Publication number	Publication date
PT97547A (pt)	1992-01-31
FI912124A0 (fi)	1991-05-02
IL120447A (en)	1999-12-22
CN1056880A (zh)	1991-12-11
EP0462696A1 (en)	1991-12-27
CA2041594A1 (en)	1991-11-04
PT97547B (pt)	1998-08-31
JPH04225986A (ja)	1992-08-14
HK51496A (en)	1996-03-29
CN1118783A (zh)	1996-03-20
DE69111915D1 (de)	1995-09-14
IL127047A (en)	2000-10-31
CN1034077C (zh)	1997-02-19
MY106552A (en)	1995-06-30
NO911723D0 (no)	1991-05-02
KR100195345B1 (ko)	1999-06-15
NO179411B (no)	1996-06-24
AU651580B2 (en)	1994-07-28
FI95912C (fi)	1996-04-10
NO911723L (no)	1991-11-04
TW218878B (xx)	1994-01-11
US5075440A (en)	1991-12-24
JP3296499B2 (ja)	2002-07-02
NO179411C (no)	1996-10-02
IL127047A0 (en)	1999-09-22
KR910020019A (ko)	1991-12-19
HUT60745A (en)	1992-10-28
HU218909B (hu)	2000-12-28
IE911488A1 (en)	1991-11-06
IE68524B1 (en)	1996-06-26
FI912124A7 (fi)	1991-11-04
DE69111915T2 (de)	1996-01-04
TNSN91030A1 (fr)	1992-10-25
EP0462696B1 (en)	1995-08-09
NZ237988A (en)	1992-09-25
ES2079570T3 (es)	1996-01-16
ATE126231T1 (de)	1995-08-15
HU911476D0 (en)	1991-11-28
ZW5291A1 (en)	1993-01-06
IL97999A0 (en)	1992-06-21
DK0462696T3 (da)	1995-09-18
IL120447A0 (en)	1997-07-13
AU7635491A (en)	1991-11-07
IL120446A0 (en)	1997-07-13
GR3017305T3 (en)	1995-12-31
ZA913319B (en)	1993-01-27
CN1039416C (zh)	1998-08-05
CA2041594C (en)	2002-07-23
IL97999A (en)	1997-06-10
FI95912B (fi)	1995-12-29

Publication	Publication Date	Title
IL120446A (en)	2000-08-31	Preparation of esters of 9-(hetero)aryl-2,3,4,5,6,9-hexahydropyrido¬2,3-f¾¬1,4¾thiazepine-8-carboxylic acid 1,1-dioxides
PT86060A (en)	1987-12-01	Process for the preparation of esters of hexahydro-8-hydroxy-2,6-methano-2h-quinolizin-3(4h)-one and of related compounds
GB2235194B (en)	1992-01-29	Stereospecific process for the preparation of furo[3,4-c] pyridine enantiomers, compounds thus obtained and therapeutical compositions thereof
HUT59926A (en)	1992-07-28	Process for producing diazabicyclo-heptanes
PT84382A (en)	1987-03-01	Process for preparing substituted 1,3,4,9-tetrahydropyrano ]3,4-b" indole-1-acetic acids
PT84648A (en)	1987-05-01	Substituted thiacycloalkeno ]3,2-b" pyridines methods of preparation compositions and method of use
YU102289A (en)	1991-06-30	Process for obtaining s-enanthiomerical glutaramides
AU586074B2 (en)	1989-06-29	Substituted 1,3,4,9-tetrahydropyrano``3,4-b``indole-1-acetic acids
ATE46908T1 (de)	1989-10-15	Verfahren zur herstellung von 4,5-dihydrodithieno(3,4b:3',4'-e>-azepin-5,9-dion.
HUT51627A (en)	1990-05-28	Process for producing calcium salt of 10-propyl-2,8-bis(1h-tetrazole-5-yl)-4h,6h-benzo-(1,2-b,5,4-b')-dipyrane-4,6-dione
FI914681A0 (fi)	1991-10-04	Menetelmä terapeuttisesti käyttökelpoisten N-alkenyylibentso/b/tieno-/3,2-b/oksatsiini-2,4-dionien valmistamiseksi
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