IL108326A0 - Lysine salt of 6-chloro-5-fluoro-3-(2-thenoyl)-2-oxindole-1-carboxamide - Google Patents

Lysine salt of 6-chloro-5-fluoro-3-(2-thenoyl)-2-oxindole-1-carboxamide

Info

Publication number: IL108326A0
Authority: IL; Israel
Prior art keywords: thenoyl; oxindole; carboxamide; fluoro; chloro
Prior art date: 1993-01-22

Application number

IL10832694A

Other languages

English (en)

Original Assignee

Pfizer

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1993-01-22

Filing date

1994-01-13

Publication date

1994-04-12

1993-01-22 Priority claimed from US08/007,217 external-priority patent/US5298522A/en

1994-01-13 Application filed by Pfizer filed Critical Pfizer

1994-04-12 Publication of IL108326A0 publication Critical patent/IL108326A0/xx

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
- C07D409/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Veterinary Medicine (AREA)
Medicinal Chemistry (AREA)
Public Health (AREA)
General Health & Medical Sciences (AREA)
Animal Behavior & Ethology (AREA)
Life Sciences & Earth Sciences (AREA)
Pharmacology & Pharmacy (AREA)
General Chemical & Material Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
Pain & Pain Management (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Neurology (AREA)
Bioinformatics & Cheminformatics (AREA)
Neurosurgery (AREA)
Biomedical Technology (AREA)
Engineering & Computer Science (AREA)
Epidemiology (AREA)
Rheumatology (AREA)
Indole Compounds (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)

IL10832694A 1993-01-22 1994-01-13 Lysine salt of 6-chloro-5-fluoro-3-(2-thenoyl)-2-oxindole-1-carboxamide IL108326A0 (en)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US08/007,217 US5298522A (en)	1993-01-22	1993-01-22	6-chloro-5-fluoro-3-(2-thenoyl)-2-oxindole-1-carboxamide as an analgesic and anti-inflammatory agent while maintaining a normal urine protein/creatinine ratio
US13827793A	1993-10-18	1993-10-18

Publications (1)

Publication Number	Publication Date
IL108326A0 true IL108326A0 (en)	1994-04-12

Family

ID=26676677

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
IL10832694A IL108326A0 (en)	1993-01-22	1994-01-13	Lysine salt of 6-chloro-5-fluoro-3-(2-thenoyl)-2-oxindole-1-carboxamide

Country Status (27)

Country	Link
EP (1)	EP0680321B1 (sh)
JP (1)	JP2711939B2 (sh)
CN (1)	CN1116822A (sh)
AP (1)	AP468A (sh)
AT (1)	ATE171373T1 (sh)
AU (1)	AU671533B2 (sh)
BG (1)	BG61966B1 (sh)
BR (1)	BR9405661A (sh)
CA (1)	CA2153050C (sh)
CZ (1)	CZ182895A3 (sh)
DE (1)	DE69413518T2 (sh)
DK (1)	DK0680321T3 (sh)
DZ (1)	DZ1748A1 (sh)
ES (1)	ES2122236T3 (sh)
FI (1)	FI940309A7 (sh)
HU (1)	HUT69687A (sh)
IL (1)	IL108326A0 (sh)
LV (1)	LV10920B (sh)
MA (1)	MA23095A1 (sh)
NO (1)	NO952904D0 (sh)
NZ (1)	NZ261449A (sh)
OA (1)	OA10173A (sh)
PL (1)	PL309957A1 (sh)
SK (1)	SK91395A3 (sh)
UY (1)	UY23723A1 (sh)
WO (1)	WO1994016694A1 (sh)
YU (1)	YU48719B (sh)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
AU7503496A (en) *	1995-12-19	1997-07-14	Pfizer Inc.	Stable, long acting salts of indole derivatives for the treatment of joint diseases
EP0826685A1 (en) *	1996-08-21	1998-03-04	Pfizer Inc.	Stable, long acting salts of carboxamides for the treatment of joint disease
DE10106852A1 (de) *	2001-02-14	2002-09-05	T Luger	Entzündungshemmende Verbindungen

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4556672A (en) *	1984-03-19	1985-12-03	Pfizer Inc.	3-Substituted 2-oxindole-1-carboxamides as analgesic and anti-inflammatory agents
US4853409A (en) *	1988-04-13	1989-08-01	Pfizer Inc.	3-substituted-2-oxindole-1-carboxamides for suppressing T-cell function
DE4111305C2 (de) *	1991-04-08	1994-12-01	Mack Chem Pharm	Pharmazeutische Zubereitung zur rektalen Applikation, die ein 2-Oxindol-l-carboxamid-derivat enthält
DE4111306C2 (de) *	1991-04-08	1994-06-01	Mack Chem Pharm	Pharmazeutische Zubereitungen, die ein 2-Oxindol-l-carboxamid-derivat enthalten und zur Injektion bestimmt sind
US5298522A (en) *	1993-01-22	1994-03-29	Pfizer Inc.	6-chloro-5-fluoro-3-(2-thenoyl)-2-oxindole-1-carboxamide as an analgesic and anti-inflammatory agent while maintaining a normal urine protein/creatinine ratio

1994
- 1994-01-06 WO PCT/US1994/000096 patent/WO1994016694A1/en not_active Ceased
- 1994-01-06 NZ NZ261449A patent/NZ261449A/en unknown
- 1994-01-06 CA CA002153050A patent/CA2153050C/en not_active Expired - Fee Related
- 1994-01-06 DE DE69413518T patent/DE69413518T2/de not_active Expired - Fee Related
- 1994-01-06 ES ES94906511T patent/ES2122236T3/es not_active Expired - Lifetime
- 1994-01-06 CN CN94190974A patent/CN1116822A/zh active Pending
- 1994-01-06 JP JP6517040A patent/JP2711939B2/ja not_active Expired - Lifetime
- 1994-01-06 EP EP94906511A patent/EP0680321B1/en not_active Expired - Lifetime
- 1994-01-06 PL PL94309957A patent/PL309957A1/xx unknown
- 1994-01-06 AT AT94906511T patent/ATE171373T1/de not_active IP Right Cessation
- 1994-01-06 CZ CZ951828A patent/CZ182895A3/cs unknown
- 1994-01-06 SK SK913-95A patent/SK91395A3/sk unknown
- 1994-01-06 BR BR9405661A patent/BR9405661A/pt not_active Application Discontinuation
- 1994-01-06 DK DK94906511T patent/DK0680321T3/da active
- 1994-01-06 AU AU60198/94A patent/AU671533B2/en not_active Ceased
- 1994-01-13 IL IL10832694A patent/IL108326A0/xx unknown
- 1994-01-13 AP APAP/P/1994/000609A patent/AP468A/en active
- 1994-01-19 DZ DZ940002A patent/DZ1748A1/fr active
- 1994-01-20 UY UY23723A patent/UY23723A1/es not_active IP Right Cessation
- 1994-01-21 YU YU2394A patent/YU48719B/sh unknown
- 1994-01-21 HU HU9400176A patent/HUT69687A/hu unknown
- 1994-01-21 FI FI940309A patent/FI940309A7/fi unknown
- 1994-01-21 MA MA23401A patent/MA23095A1/fr unknown
1995
- 1995-07-05 BG BG99767A patent/BG61966B1/bg unknown
- 1995-07-21 LV LVP-95-220A patent/LV10920B/en unknown
- 1995-07-21 NO NO952904A patent/NO952904D0/no unknown
- 1995-07-21 OA OA60690A patent/OA10173A/en unknown

Also Published As

Publication number	Publication date
FI940309L (fi)	1994-07-23
EP0680321B1 (en)	1998-09-23
NO952904L (no)	1995-07-21
CN1116822A (zh)	1996-02-14
FI940309A7 (fi)	1994-07-23
YU2394A (sh)	1996-10-18
PL309957A1 (en)	1995-11-13
AU671533B2 (en)	1996-08-29
BG61966B1 (bg)	1998-11-30
MA23095A1 (fr)	1994-10-01
DE69413518D1 (en)	1998-10-29
CA2153050A1 (en)	1994-08-04
ATE171373T1 (de)	1998-10-15
WO1994016694A1 (en)	1994-08-04
NO952904D0 (no)	1995-07-21
EP0680321A1 (en)	1995-11-08
JPH08501109A (ja)	1996-02-06
DZ1748A1 (fr)	2002-02-17
DE69413518T2 (de)	1999-02-11
AP468A (en)	1996-03-05
NZ261449A (en)	1996-08-27
ES2122236T3 (es)	1998-12-16
UY23723A1 (es)	1994-06-28
CZ182895A3 (en)	1996-01-17
LV10920B (en)	1996-04-20
AU6019894A (en)	1994-08-15
JP2711939B2 (ja)	1998-02-10
AP9400609A0 (en)	1994-01-31
SK91395A3 (en)	1996-12-04
HUT69687A (en)	1995-09-28
DK0680321T3 (da)	1999-06-14
HU9400176D0 (en)	1994-05-30
BG99767A (bg)	1996-02-28
YU48719B (sh)	1999-07-28
OA10173A (en)	1996-12-18
FI940309A0 (fi)	1994-01-21
CA2153050C (en)	1998-12-29
LV10920A (lv)	1995-12-20
BR9405661A (pt)	1995-11-21

Publication	Publication Date	Title
PL313619A1 (en)	1996-07-08	Derivatives of piperydine
PL310443A1 (en)	1995-12-11	Derivatives of pyrolo-pyridine
ZA94436B (en)	1995-07-21	Lysine salt of 6-chloro-5-fluoro-3-(2-thenoyl)-2-oxindole-1-carboxamide
PL306127A1 (en)	1995-06-12	Derivatives of epi-epibathydine
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AP9400609A0 (en)	1994-01-31	Lysine salt of 6-chloro-5-fluoro-3-(2-thenoyl)-2-oxindole-1-carboxamide
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GB9326090D0 (en)	1994-02-23	Easy carry handel
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GB9313512D0 (en)	1993-08-11	Derivatives of 1-cyclohexyl-piperidine
GB9411194D0 (en)	1994-07-27	Clavulanic acid salt
PL290693A3 (en)	1992-12-28	Cosmetic preparation - bath salt
HU9300038V0 (en)	1993-05-28	Drum
GB9309401D0 (en)	1993-06-23	Preparation of flouro-compounds
NZ329141A (en)	1999-06-29	Preparation of n-cyano-dithio-iminocarbonates
GB9309794D0 (en)	1993-06-23	Preparation of flouro-nucleosides