HRP20020881A2 - Method for the preparation of citalopram - Google Patents

Method for the preparation of citalopram

Info

Publication number: HRP20020881A2
Authority: HR; Croatia
Prior art keywords: formula; compound; image; prepared; reaction
Prior art date: 2000-05-12

Application number

Other languages

English (en)

Croatian (hr)

Inventor

Hans Petersen

Robert Dancer

Original Assignee

Lundbeck & Co As H

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2000-05-12

Filing date

2001-05-10

Publication date

2004-12-31

2001-05-10 Application filed by Lundbeck & Co As H filed Critical Lundbeck & Co As H

2004-12-31 Publication of HRP20020881A2 publication Critical patent/HRP20020881A2/hr

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
- C07D307/77—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
- C07D307/87—Benzo [c] furans; Hydrogenated benzo [c] furans
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
- C07D307/77—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
- C07D307/87—Benzo [c] furans; Hydrogenated benzo [c] furans
- C07D307/88—Benzo [c] furans; Hydrogenated benzo [c] furans with one oxygen atom directly attached in position 1 or 3

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Medicinal Chemistry (AREA)
Pharmacology & Pharmacy (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Biomedical Technology (AREA)
Neurology (AREA)
Neurosurgery (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Pain & Pain Management (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Psychiatry (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Steroid Compounds (AREA)
Furan Compounds (AREA)
Plural Heterocyclic Compounds (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)

HRP20020881 2000-05-12 2001-05-10 Method for the preparation of citalopram HRP20020881A2 (en)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
DKPA200000783		2000-05-12
PCT/DK2001/000333 WO2001085712A1 (en)	2000-05-12	2001-05-10	Method for the preparation of citalopram

Publications (1)

Publication Number	Publication Date
HRP20020881A2 true HRP20020881A2 (en)	2004-12-31

Family

ID=8159493

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
HRP20020881 HRP20020881A2 (en)	2000-05-12	2001-05-10	Method for the preparation of citalopram

Country Status (29)

Country	Link
US (1)	US6660873B2 (es)
EP (1)	EP1296970B1 (es)
JP (1)	JP2003532721A (es)
CN (1)	CN100422166C (es)
AR (1)	AR032455A1 (es)
AT (1)	ATE389645T1 (es)
AU (2)	AU5823901A (es)
BG (1)	BG65820B1 (es)
BR (1)	BR0110996A (es)
CA (1)	CA2408292C (es)
CZ (1)	CZ20024065A3 (es)
DE (1)	DE60133280T2 (es)
DK (1)	DK1296970T3 (es)
EA (1)	EA005674B1 (es)
ES (1)	ES2301541T3 (es)
HR (1)	HRP20020881A2 (es)
HU (1)	HUP0301942A2 (es)
IL (2)	IL152645A0 (es)
IS (1)	IS2586B (es)
MX (1)	MXPA02011125A (es)
NO (1)	NO327963B1 (es)
NZ (1)	NZ522475A (es)
PL (1)	PL358144A1 (es)
PT (1)	PT1296970E (es)
SI (1)	SI1296970T1 (es)
SK (1)	SK287035B6 (es)
UA (1)	UA72039C2 (es)
WO (1)	WO2001085712A1 (es)
ZA (1)	ZA200208973B (es)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
SI1173431T2 (sl)	1999-04-14	2009-12-31	Lundbeck & Co As H	Postopek za pripravo citaloprama
US6310222B1 (en)	1999-11-01	2001-10-30	Sumika Fine Chemicals Co., Ltd.	Production method of 5-phthalancarbonitrile compound, intermediate therefor and production method of the intermediate
US6433196B1 (en) *	2000-02-17	2002-08-13	Sumika Fine Chemicals Co., Ltd.	Production method of citalopram, intermediate therefor and production method of the intermediate
NL1017417C1 (nl)	2000-03-03	2001-03-16	Lundbeck & Co As H	Werkwijze voor de bereiding van Citalopram.
TR200202195T2 (tr)	2000-03-13	2002-12-23	H. Lundbeck A/S	5-Yer değiştirmiş 1-(4-florofenil)-1,3- dihidroizobenzofuran'ın adım adım alkillenmesi
IES20010206A2 (en)	2000-03-13	2002-03-06	Lundbeck & Co As H	Method for the preparation of citalopram
AR032455A1 (es)	2000-05-12	2003-11-12	Lundbeck & Co As H	Metodo para la preparacion de citalopram, un intermediario empleado en el metodo, un metodo para la preparacion del intermediario empleado en el metodo y composicion farmaceutica antidepresiva
IN192057B (es) *	2001-07-19	2004-02-14	Ranbaxy Lab Ltd
WO2004085416A1 (en) *	2003-03-24	2004-10-07	Hetero Drugs Limited	Novel crystalline forms of (s)-citalopram oxalate
AU2003278409A1 (en) *	2003-10-28	2005-05-19	Krishnaji Upadhye Bhargav	Improved process for the manufacture of citalopram hydrobromide
US20050143350A1 (en) *	2003-11-19	2005-06-30	Seed John C.	Combination drug therapy to treat obesity
KR101166280B1 (ko)	2004-08-23	2013-11-27	썬 파마 글로벌 에프제트이	시탈로프램 및 에난티오머의 제조 방법

Family Cites Families (40)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB1143702A (es)	1965-03-18
GB1526331A (en) *	1976-01-14	1978-09-27	Kefalas As	Phthalanes
GB8419963D0 (en)	1984-08-06	1984-09-12	Lundbeck & Co As H	Intermediate compound and method
GB8814057D0 (en)	1988-06-14	1988-07-20	Lundbeck & Co As H	New enantiomers & their isolation
US5296507A (en)	1990-09-06	1994-03-22	H.Lundbeck A/S	Treatment of cerbrovascular disorders
DE19626659A1 (de)	1996-07-03	1998-01-08	Basf Ag	Verfahren zur Herstellung von Phthaliden
DE19627697A1 (de)	1996-07-10	1998-01-15	Basf Ag	Verfahren zur Herstellung von Phthaliden
DK1015416T3 (da)	1997-07-08	2001-11-05	Lundbeck & Co As H	Fremgangsmåde til fremstilling af citalopram
UA62985C2 (en)	1997-11-10	2004-01-15	Lunnbeck As H	A method for the preparation of citalopram
SK283907B6 (sk) *	1997-11-11	2004-04-06	H. Lundbeck A/S	Spôsob výroby citalopramu a medziprodukty
ES2189502T3 (es)	1998-10-20	2003-07-01	Lundbeck & Co As H	Metodo para la prevencion de citalopram.
KR100454008B1 (ko)	1998-12-23	2004-10-20	하. 룬트벡 아크티에 셀스카브	5-시아노프탈리드의 제조방법
AR022329A1 (es)	1999-01-29	2002-09-04	Lundbeck & Co As H	Metodo para la preparacion de 5-cianoftalida
SI1173431T2 (sl)	1999-04-14	2009-12-31	Lundbeck & Co As H	Postopek za pripravo citaloprama
ITMI991579A1 (it)	1999-06-25	2001-01-15	Lundbeck & Co As H	Metodo per la preparazione di citalopram
ITMI991581A1 (it)	1999-06-25	2001-01-15	Lundbeck & Co As H	Metodo per la preparazione di citalopram
ITMI991486A1 (it)	1999-07-06	2001-01-06	Vis Farmaceutici S P A	Processo per la sintesi di citalopram
TR200101874T1 (tr)	1999-10-25	2002-02-21	H. Lundbeck A/S	Sitalopram hazırlanması için yöntem
AR026063A1 (es)	1999-11-01	2002-12-26	Lundbeck & Co As H	Metodo para la preparacion de 5-carboxiftalida.
US6310222B1 (en)	1999-11-01	2001-10-30	Sumika Fine Chemicals Co., Ltd.	Production method of 5-phthalancarbonitrile compound, intermediate therefor and production method of the intermediate
SI1246812T1 (en)	1999-12-28	2004-08-31	H. Lundbeck A/S	Method for the preparation of citalopram
SI1246813T1 (en)	1999-12-30	2004-08-31	H. Lundbeck A/S	Method for the preparation of citalopram
CZ20022601A3 (cs)	2000-01-14	2002-10-16	H. Lundbeck A/S	Způsob výroby 5-kyanoftalidu
IT1317729B1 (it)	2000-01-18	2003-07-15	Norpharma S P A	Procedimento per la preparazione della 5-carbossiftalide.
US6433196B1 (en)	2000-02-17	2002-08-13	Sumika Fine Chemicals Co., Ltd.	Production method of citalopram, intermediate therefor and production method of the intermediate
FR2805812A1 (fr)	2000-02-24	2001-09-07	Lundbeck & Co As H	Procede de preparation du citalopram
IES20010143A2 (en)	2000-02-24	2001-07-25	Lundbeck & Co As H	Method for the preparation of citalopram
NL1017417C1 (nl)	2000-03-03	2001-03-16	Lundbeck & Co As H	Werkwijze voor de bereiding van Citalopram.
GB0005477D0 (en)	2000-03-07	2000-04-26	Resolution Chemicals Limited	Process for the preparation of citalopram
IES20010206A2 (en)	2000-03-13	2002-03-06	Lundbeck & Co As H	Method for the preparation of citalopram
TR200202195T2 (tr)	2000-03-13	2002-12-23	H. Lundbeck A/S	5-Yer değiştirmiş 1-(4-florofenil)-1,3- dihidroizobenzofuran'ın adım adım alkillenmesi
NZ521201A (en)	2000-03-13	2004-02-27	H	Method for the preparation of citalopram
GB2357762B (en)	2000-03-13	2002-01-30	Lundbeck & Co As H	Crystalline base of citalopram
PL360107A1 (en)	2000-03-14	2004-09-06	H.Lundbeck A/S	Method for the preparation of citalopram
WO2001068632A1 (en)	2000-03-16	2001-09-20	H. Lundbeck A/S	Method for the preparation of 5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofurans
AR032455A1 (es)	2000-05-12	2003-11-12	Lundbeck & Co As H	Metodo para la preparacion de citalopram, un intermediario empleado en el metodo, un metodo para la preparacion del intermediario empleado en el metodo y composicion farmaceutica antidepresiva
CZ2002832A3 (cs)	2000-07-06	2002-05-15	H. Lundbeck A/S	Způsob výroby citalopramu
IL144816A (en)	2000-08-18	2005-09-25	Lundbeck & Co As H	Method for the preparation of citalopram
ES2228824T3 (es)	2000-12-22	2005-04-16	H. Lundbeck A/S	Metodo de preparacion de citalopram puro.
ATE222899T1 (de)	2000-12-28	2002-09-15	Lundbeck & Co As H	Verfahren zur herstellung von reinem citalopram

2001
- 2001-05-07 AR ARP010102152A patent/AR032455A1/es active IP Right Grant
- 2001-05-10 CZ CZ20024065A patent/CZ20024065A3/cs unknown
- 2001-05-10 SI SI200130831T patent/SI1296970T1/sl unknown
- 2001-05-10 IL IL15264501A patent/IL152645A0/xx unknown
- 2001-05-10 SK SK1754-2002A patent/SK287035B6/sk not_active IP Right Cessation
- 2001-05-10 CA CA002408292A patent/CA2408292C/en not_active Expired - Fee Related
- 2001-05-10 MX MXPA02011125A patent/MXPA02011125A/es active IP Right Grant
- 2001-05-10 HR HRP20020881 patent/HRP20020881A2/hr not_active Application Discontinuation
- 2001-05-10 DE DE60133280T patent/DE60133280T2/de not_active Expired - Fee Related
- 2001-05-10 EP EP01931469A patent/EP1296970B1/en not_active Expired - Lifetime
- 2001-05-10 ES ES01931469T patent/ES2301541T3/es not_active Expired - Lifetime
- 2001-05-10 AU AU5823901A patent/AU5823901A/xx active Pending
- 2001-05-10 PT PT01931469T patent/PT1296970E/pt unknown
- 2001-05-10 PL PL01358144A patent/PL358144A1/xx unknown
- 2001-05-10 JP JP2001582313A patent/JP2003532721A/ja not_active Withdrawn
- 2001-05-10 BR BR0110996-0A patent/BR0110996A/pt not_active Application Discontinuation
- 2001-05-10 AU AU2001258239A patent/AU2001258239B2/en not_active Ceased
- 2001-05-10 EA EA200201211A patent/EA005674B1/ru not_active IP Right Cessation
- 2001-05-10 CN CNB018125859A patent/CN100422166C/zh not_active Expired - Fee Related
- 2001-05-10 NZ NZ522475A patent/NZ522475A/en unknown
- 2001-05-10 HU HU0301942A patent/HUP0301942A2/hu unknown
- 2001-05-10 AT AT01931469T patent/ATE389645T1/de not_active IP Right Cessation
- 2001-05-10 DK DK01931469T patent/DK1296970T3/da active
- 2001-05-10 WO PCT/DK2001/000333 patent/WO2001085712A1/en not_active Ceased
- 2001-10-05 UA UA2002118821A patent/UA72039C2/uk unknown
2002
- 2002-10-31 IS IS6605A patent/IS2586B/is unknown
- 2002-11-04 IL IL152645A patent/IL152645A/en not_active IP Right Cessation
- 2002-11-05 ZA ZA200208973A patent/ZA200208973B/en unknown
- 2002-11-08 US US10/291,174 patent/US6660873B2/en not_active Expired - Fee Related
- 2002-11-12 NO NO20025423A patent/NO327963B1/no not_active IP Right Cessation
- 2002-12-03 BG BG107349A patent/BG65820B1/bg unknown

Also Published As

Publication number	Publication date
DE60133280D1 (de)	2008-04-30
IS6605A (is)	2002-10-31
CA2408292C (en)	2009-11-10
NZ522475A (en)	2004-09-24
HK1056171A1 (zh)	2004-02-06
DE60133280T2 (de)	2009-04-16
CA2408292A1 (en)	2001-11-15
NO20025423D0 (no)	2002-11-12
PL358144A1 (en)	2004-08-09
EP1296970B1 (en)	2008-03-19
CZ20024065A3 (cs)	2003-03-12
NO327963B1 (no)	2009-10-26
AR032455A1 (es)	2003-11-12
BG107349A (bg)	2003-09-30
AU5823901A (en)	2001-11-20
AU2001258239B2 (en)	2005-12-08
NO20025423L (no)	2002-11-12
HUP0301942A2 (hu)	2003-09-29
MXPA02011125A (es)	2003-03-10
EA005674B1 (ru)	2005-04-28
IS2586B (is)	2010-02-15
EA200201211A1 (ru)	2003-04-24
PT1296970E (pt)	2008-06-11
ATE389645T1 (de)	2008-04-15
SK17542002A3 (sk)	2003-04-01
BG65820B1 (bg)	2010-01-29
EP1296970A1 (en)	2003-04-02
ES2301541T3 (es)	2008-07-01
SI1296970T1 (sl)	2008-08-31
BR0110996A (pt)	2003-03-18
DK1296970T3 (da)	2008-07-14
CN1441795A (zh)	2003-09-10
US20030134895A1 (en)	2003-07-17
ZA200208973B (en)	2003-11-05
IL152645A0 (en)	2003-06-24
SK287035B6 (sk)	2009-10-07
UA72039C2 (en)	2005-01-17
US6660873B2 (en)	2003-12-09
CN100422166C (zh)	2008-10-01
WO2001085712A1 (en)	2001-11-15
JP2003532721A (ja)	2003-11-05
IL152645A (en)	2009-12-24

Publication	Publication Date	Title
JP3813820B2 (ja)	2006-08-23	シタロプラムの製造方法
FI108538B (fi)	2002-02-15	Menetelmä sitalopraamin valmistamiseksi
JP3447267B2 (ja)	2003-09-16	シタロプラムの製造方法
HRP20020756A2 (en)	2004-12-31	Crystalline base of citalopram
ITMI991580A1 (it)	2001-01-15	Metodo per la preparazione di citalopram
UA72340C2 (uk)	2005-02-15	Спосіб одержання циталопраму
HRP20020743A2 (en)	2003-12-31	Method for the preparation of citalopram
HRP20020881A2 (en)	2004-12-31	Method for the preparation of citalopram
HRP20020757A2 (en)	2004-12-31	Method for the preparation of 5-cyano-1-(4-fluorophenyl)-1,3-dihydroisobenzofurans
SK9282002A3 (en)	2002-11-06	Method for the preparation of citalopram, pharmaceutical composition comprising same and intermediates
AU2001258239A1 (en)	2002-02-07	Method for the preparation of citalopram
HRP20020633A2 (en)	2004-12-31	Method for the preparation of citalopram
HRP20020744A2 (en)	2004-12-31	Method for the preparation of citalopram
HRP20020758A2 (en)	2004-12-31	Stepwise alkylation of 5-substituted 1-(4-fluorophenyl)-1,3-dihydroisobenzofurans
HRP20020741A2 (en)	2003-12-31	Method for the preparation of citalopram
KR100821912B1 (ko)	2008-04-16	시탈로프람의 제조 방법
ZA200107956B (en)	2002-11-27	Method for the preparation of citalopram.
HRP20020562A2 (en)	2003-10-31	Method for the preparation of citalopram

Legal Events

Date	Code	Title	Description
2004-12-31	A1OB	Publication of a patent application
2005-08-03	OBST	Application withdrawn
2009-05-05	ODRP	Renewal fee for the maintenance of a patent	Payment date: 20090505 Year of fee payment: 9

Date

Code

Title

Description

2004-12-31

A1OB

Publication of a patent application

2005-08-03

OBST

Application withdrawn

2009-05-05

ODRP

Renewal fee for the maintenance of a patent

Payment date: 20090505

Year of fee payment: 9